Page last updated: 2024-08-21

thiazoles and 1,4-dihydropyridine

thiazoles has been researched along with 1,4-dihydropyridine in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (50.00)29.6817
2010's2 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bihel, F; Garino, C; Kraus, JL; Laras, Y; Pietrancosta, N; Quéléver, G; Sheha, M; Wolfe, MS1
Andreani, A; Bedini, A; Budriesi, R; Chiarini, A; Cosconati, S; Di Toro, R; Ioan, P; Leoni, A; Locatelli, A; Marinelli, L; Novellino, E; Spampinato, S; Ugenti, MP1
Al-Qasoumi, SI; Al-Said, MS; Bashandy, MS; Ghorab, MM1
Fadda, AA; Refat, HM1

Other Studies

4 other study(ies) available for thiazoles and 1,4-dihydropyridine

ArticleYear
Substituted thiazolamide coupled to a redox delivery system: a new gamma-secretase inhibitor with enhanced pharmacokinetic profile.
    Organic & biomolecular chemistry, 2005, Feb-21, Volume: 3, Issue:4

    Topics: Alzheimer Disease; Amides; Amyloid Precursor Protein Secretases; Animals; Aspartic Acid Endopeptidases; Biological Availability; Blood-Brain Barrier; Dihydropyridines; Drug Delivery Systems; Endopeptidases; Enzyme Inhibitors; Humans; Male; Molecular Structure; Nicotinic Acids; Oxidation-Reduction; Rats; Rats, Sprague-Dawley; Thiazoles

2005
Imidazo[2,1-b]thiazole system: a scaffold endowing dihydropyridines with selective cardiodepressant activity.
    Journal of medicinal chemistry, 2008, Mar-27, Volume: 51, Issue:6

    Topics: Animals; Binding Sites; Computer Simulation; Dihydropyridines; Drug Design; Drug Evaluation, Preclinical; Guinea Pigs; Heart; Heart Rate; Imidazoles; Ligands; Models, Molecular; Molecular Structure; Muscle, Smooth, Vascular; Myocardial Contraction; Myocytes, Cardiac; Small Molecule Libraries; Structure-Activity Relationship; Thiazoles

2008
Anti-breast cancer activity of some novel 1,2-dihydropyridine, thiophene and thiazole derivatives.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:1

    Topics: Antineoplastic Agents; Breast Neoplasms; Cell Line, Tumor; Dihydropyridines; Humans; Inhibitory Concentration 50; Structure-Activity Relationship; Thiazoles; Thiophenes

2011
Synthesis and antimicrobial activity of some novel hydrazide, benzochromenone, dihydropyridine, pyrrole, thiazole and thiophene derivatives.
    European journal of medicinal chemistry, 2013, Volume: 70

    Topics: Anti-Bacterial Agents; Antifungal Agents; Benzopyrans; Candida albicans; Dihydropyridines; Dose-Response Relationship, Drug; Escherichia coli; Hydrazones; Microbial Sensitivity Tests; Molecular Structure; Pyrroles; Staphylococcus aureus; Structure-Activity Relationship; Thiazoles; Thiophenes

2013