thiazoles has been researched along with 1-(2',6'-difluorophenyl)-1h,3h-thiazolo(3,4-a)benzimidazole in 9 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 6 (66.67) | 18.2507 |
| 2000's | 2 (22.22) | 29.6817 |
| 2010's | 1 (11.11) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Allen, LB; Buckheit, RW; Decker, WD; Germany-Decker, J; Hollingshead, MG; McMahon, JB; Ross, LJ; Shannon, WM; Westbrook, L; White, EL | 1 |
| Anderson, BD; Hoesterey, BL; Lim, K; Tinwalla, AY; Xiang, TX | 1 |
| Chimirri, A; Grasso, S; Molica, C; Monforte, AM; Monforte, P; Scopelliti, R; Zappalà, M | 1 |
| Boyer, PL; Buckheit, RW; Hughes, SH; Michejda, CJ; Morningstar, ML; Roth, T | 1 |
| Chimirri, A; D'Alessandro, N; Gancitano, RA; Grimaudo, S; Tolomeo, M; Zappala, M | 1 |
| Barreca, ML; Calace, MP; Carotti, A; Carrieri, A; Chimirri, A; Monforte, AM; Rao, A | 1 |
| Capone, F; Chimirri, A; Grimaudo, S; Monforte, AM; Poretto, F; Raimondi, MV; Simoni, D; Tolomeo, M | 1 |
| Bergmann, M; Canard, B; Chimirri, A; Coutard, B; De Clercq, E; De Palma, AM; Heggermont, W; Lanke, K; Monforte, AM; Neyts, J; Pürstinger, G; Rohayem, J; van Kuppeveld, F | 1 |
| Andreoli, F; Coppola, F; Farran, D; Kaid-Slimane, R; Roussel, C; Vanthuyne, N | 1 |
9 other study(ies) available for thiazoles and 1-(2',6'-difluorophenyl)-1h,3h-thiazolo(3,4-a)benzimidazole
| Article | Year |
|---|---|
Thiazolobenzimidazole: biological and biochemical anti-retroviral activity of a new nonnucleoside reverse transcriptase inhibitor.
Topics: Antiviral Agents; Base Sequence; Benzimidazoles; Cell Line; Didanosine; DNA, Single-Stranded; Drug Synergism; HIV Reverse Transcriptase; HIV-1; Humans; Leukemia Virus, Murine; Molecular Sequence Data; Molecular Structure; Reverse Transcriptase Inhibitors; Thiazoles; Zidovudine | 1993 |
Solubilization of thiazolobenzimidazole using a combination of pH adjustment and complexation with 2-hydroxypropyl-beta-cyclodextrin.
Topics: 2-Hydroxypropyl-beta-cyclodextrin; Benzimidazoles; beta-Cyclodextrins; Chromatography, High Pressure Liquid; Computer Simulation; Cyclodextrins; Hydrogen-Ion Concentration; Magnetic Resonance Spectroscopy; Models, Chemical; Regression Analysis; Solubility; Solvents; Thiazoles | 1993 |
Anti-HIV agents. IV. Synthesis and in vitro anti-HIV activity of novel 1-(2,6-difluorophenyl)-1H,3H-thiazolo[3,4-a]benzimidazoles.
Topics: Antiviral Agents; Benzimidazoles; HIV-1; Structure-Activity Relationship; Thiazoles | 1996 |
Synthesis and biological activity of novel nonnucleoside inhibitors of HIV-1 reverse transcriptase. 2-Aryl-substituted benzimidazoles.
Topics: Anti-HIV Agents; Benzimidazoles; Cell Line; Cytoprotection; Drug Design; Drug Resistance, Microbial; HIV Reverse Transcriptase; HIV-1; Humans; Magnetic Resonance Spectroscopy; Models, Molecular; Molecular Structure; Reverse Transcriptase Inhibitors; Structure-Activity Relationship; Thiazoles | 1997 |
Selective induction of apoptosis in multidrug resistant HL60R cells by the thiazolobenzoimidazole derivative 1-(2,6-difluorophenyl)-1H,3H-thiazolo [3,4-a] benzimidazole (TBZ).
Topics: Anti-HIV Agents; Apoptosis; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Flow Cytometry; HL-60 Cells; Humans; Proto-Oncogene Proteins c-bcl-2; Thiazoles; Tumor Suppressor Protein p53 | 1998 |
Comparative molecular field analysis (CoMFA) and docking studies of non-nucleoside HIV-1 RT inhibitors (NNIs).
Topics: Benzimidazoles; Benzodiazepines; Crystallography, X-Ray; HIV Reverse Transcriptase; Imidazoles; Models, Chemical; Models, Molecular; Protein Conformation; Reverse Transcriptase Inhibitors; Structure-Activity Relationship; Thiazoles | 1999 |
Apoptotic effects of thiazolobenzimidazole derivatives on sensitive and multidrug resistant leukaemic cells.
Topics: Antineoplastic Agents; Apoptosis; Benzimidazoles; Caspase Inhibitors; Cell Cycle; Drug Resistance, Multiple; Drug Resistance, Neoplasm; fas Receptor; HL-60 Cells; Humans; Leukemia; Thiazoles | 2001 |
The thiazolobenzimidazole TBZE-029 inhibits enterovirus replication by targeting a short region immediately downstream from motif C in the nonstructural protein 2C.
Topics: Adenosine Triphosphatases; Amino Acid Motifs; Amino Acid Substitution; Animals; Antiviral Agents; Benzimidazoles; Carrier Proteins; Chlorocebus aethiops; Drug Resistance, Viral; Enterovirus B, Human; Guanidine; Molecular Structure; Mutation, Missense; Pyridines; RNA, Viral; Thiazoles; Vero Cells; Viral Nonstructural Proteins; Virus Replication | 2008 |
Access to N-thioalkenyl and N-(o-thio)aryl-benzimidazol-2-ones by ring opening of thiazolobenzimidazolium and benzimidazobenzothiazolium salts and C-O bond cleavage of an alkoxide.
Topics: Benzimidazoles; Molecular Structure; Oxides; Salts; Thiazoles | 2015 |