theophylline and adenosine-5'-(n-ethylcarboxamide)

theophylline has been researched along with adenosine-5'-(n-ethylcarboxamide) in 192 studies

Research

Studies (192)

TimeframeStudies, this research(%)All Research%
pre-199067 (34.90)18.7374
1990's101 (52.60)18.2507
2000's19 (9.90)29.6817
2010's4 (2.08)24.3611
2020's1 (0.52)2.80

Authors

AuthorsStudies
Jacobson, KA; van Galen, PJ; Williams, M1
Daly, JW1
Bertin, B; Freissmuth, M; Hohenegger, M; Jockers, R; Linder, ME; Marullo, S; Nanoff, C; Strosberg, AD1
Arslan, G; Dionisotti, S; Fredholm, BB; Kull, B; Ongini, E; Zocchi, C1
Fredholm, BB; Hegler, J; Hessling, J; Klotz, KN; Kull, B; Lohse, MJ; Owman, C1
Belardinelli, L; Biaggioni, I; Feoktistov, I; Garland, EM; Goldstein, AE; Wells, JN; Zeng, D1
Calabri, FR; Catarzi, D; Colotta, V; Deflorian, F; Filacchioni, G; Lenzi, O; Martini, C; Moro, S; Trincavelli, L; Varano, F1
Borea, PA; Dalpiaz, A; Gilli, G; Gilli, P; Scatturin, A; Varani, K1
Baraldi, PG; Benini, A; Borea, PA; Cattabriga, E; Gessi, S; Klotz, KN; Lennan, SM; Leung, E; Merighi, S; Tabrizi, MA; Varani, K; Vincenzi, F1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Bertarelli, DC; Borrmann, T; Florin, NC; Hinz, S; Li, W; Müller, CE; Scheiff, AB1
Federico, S; Jacobson, KA; Jayasekara, PS; Kozma, E; Moro, S; Paoletta, S; Spalluto, G; Squarcialupi, L1
de Lera Ruiz, M; Lim, YH; Zheng, J1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Berizzi, A; Bird, L; Culurgioni, S; Navratilova, IH; Olsen, RHJ; Rawlins, PB; Robinson, S; Shepherd, C; Thompson, LEJ; Varzandeh, S1
Furlong, TJ; Pierce, KD; Selbie, LA; Shine, J1
Acevedo, CG; Contreras, E; Escalona, J; Huidobro-Toro, JP; Lewin, J1
Földes, FF; Nagano, O; Nakatsuka, H; Ohta, Y; Reich, D; Sperlagh, B; Vizi, ES1
Abramson, SB; Cronstein, BN; Hirschhorn, R; Levin, RI; Philips, M; Weissmann, G1
Martin, PL2
Gordh, T; Karlsten, R; Post, C1
Shibata, S; Tominaga, K; Watanabe, S1
Arizono, K; Brady, FO; Garrett, SH; Xiong, X1
Kurth, CD; Wagerle, LC1
Jacobson, KA; Ji, XD; Stiles, GL1
Gobran, LI; Griese, M; Rooney, SA1
Hammarström, M; Samuelson, UE; Wiklund, NP1
Amerini, S; Ledda, F; Mantelli, L; Rubino, A1
Porsius, AJ; Post, MJ; te Biesebeek, JD; van Rooij, HH; Wemer, J1
Lichtenstein, LM; Peachell, PT; Schleimer, RP1
Canonico, PL; Catania, MV; Nicoletti, F; Rampello, L; Sortino, MA1
Huddart, H; Lynch, M1
Nasir, T; Zarrindast, MR1
Aas, P; Walday, P1
Andén, NE; Casas, M; Ferré, S; Grabowska-Andén, M; Herrera-Marschitz, M; Ungerstedt, U1
Ameri, A; Jurna, I1
Arzubiaga, C; Biaggioni, I; Paul, S; Puckett, A1
Bealer, SL; Proctor, KG; Stojanov, I1
Alexander, B; Burnstock, G; Mathie, RT; Ralevic, V1
Holtzman, SG; Mumford, GK1
Brown, SJ; Evenden, JL; Gill, R; Iversen, SD; Richardson, PJ1
Wainwright, LK; Wainwright, SD1
Daly, JW; Jacobson, KA; Nikodijević, O; Sarges, R1
Aranda, JV; Beharry, K; Farri, E; Laudignon, N1
Joad, JP1
Isbrucker, R; Reid, A; Sawynok, J1
Elphick, M; Godfrey, PP; Powell, T; Taghavi, Z1
Barrett, KE; Cohn, JA; Dharmsathaphorn, K; Huott, PA; Wasserman, SI1
Gilfillan, AM; Welton, AF; Wiggan, GA1
Cronstein, BN; Salmon, JE1
Aranda, JV; Laudignon, N; Varma, DR1
Berman, RF; Lupica, CR; Rosen, JB; Whitcomb, K1
Daly, JW; Jacobson, KA; Nikodijević, O1
Barraco, RA; Stefano, GB1
Barry, SR1
Hope, W; Rose'Meyer, RB1
Franklin, PH; Murray, TF; Zhang, G1
Kitos, TE; Michaelis, ML; Mooney, T1
Anand-Srivastava, MB; Cantin, M; Gutkowska, J1
Coffin, VL; Spealman, RD1
Cederqvist, B; Gustafsson, LE; Wiklund, NP2
Fox, IH; John, D1
Dodd, PR; Johnston, GA; Watson, WE1
Belloni, FL; Gerritsen, ME; Liang, BC1
Benyon, RC; Church, MK; Hughes, PJ1
Jackman, SA; Nicholson, CD; Wilke, R1
Cushing, DJ; Mustafa, SJ; Sabouni, MH1
De Mendonça, A; Ribeiro, JA1
Lohse, MJ; Schmitz, W; Scholz, H; Scholz, J; Schwabe, U; von der Leyen, H1
Antonelli, C; Condorelli, M; Genovese, A; Marone, G; Torella, G; Vigorita, S1
Hargittai, PT; Lieberman, EM; Mustafa, SJ; Sabouni, MH1
Brod, I; Bucher, B; Illes, P; Rickmann, H; Stoclet, JC1
Durcan, MJ; Morgan, PF1
Berne, RM; Park, TS; Rubio, R; Van Wylen, DG1
Abbracchio, MP; Cattabeni, F; Clementi, F; Sher, E1
Jahnel, U; Nawrath, H1
Fredholm, BB; Lerner, UH; Sahlberg, K1
Lowenstein, JM; Ravid, K1
Cronstein, BN; Hirschhorn, R; Rose, FR; Weissmann, G1
Billig, H; Rosberg, S1
Gniess, A; Reymann, A1
Illes, P; Jackisch, R; Regenold, JT1
Kurtz, A1
Barnes, PJ; Clarke, B; McCormack, DG1
Churchill, MC; Churchill, PC1
Cronstein, BN; Hirschhorn, R; Kramer, SB; Rosenstein, ED; Weissmann, G1
Christofi, FL; Cook, MA1
Chapal, J; Loubatières-Mariani, MM; Petit, P; Roye, M1
Klotz, KN; Schirren, CG; Schwabe, U; Ukena, D1
Gustafsson, LE; Samuelson, UE; Wiklund, NP1
Böhm, M; Brückner, R; Meyer, W; Nose, M; Schmitz, W; Scholz, H; Starbatty, J1
Fredholm, BB; Jonzon, B; Lindström, K1
Sawynok, J; Sweeney, MI; White, TD1
Condorelli, M; Marone, G; Triggiani, M; Vigorita, S1
Barchowsky, A; Data, JL; Whorton, AR1
Gilfillan, AM; Rooney, SA1
Brodie, MS; Dunwiddie, TV; Fredholm, BB; Lee, K; Ståhle, L1
Spealman, RD1
Heller, LJ; Olsson, RA1
Abla, KA; Carney, JM; Daly, JW; Seale, TW; Shamim, MT1
Bartrup, JT; Stone, TW1
Craig, RH; Daluge, SM; Earl, CQ; Linden, J; Patel, A1
Finn, IB; Holtzman, SG1
Beckman, B; Brookins, J; Fisher, JW; Ueno, M1
Harper, AM; McBean, DE; Rudolphi, KA1
Granger, JP; Knox, FG; Pawlowska, D1
Della Briotta, G; Hösli, E; Hösli, L; Uhr, M1
Braunwalder, A; Ferkany, JW; Jarvis, MF; Sills, MA; Williams, M1
Bowker, HM; Chapman, AG1
Hedner, J; Hedner, T; Holmgren, M; Mellstrand, T; Nordberg, G1
Bergman, B; Hedner, J; Hedner, T; Jonason, J; Mueller, RA1
Vertes, RP; Wu, PH1
Bonnafous, JC; Chapat, JP; Francoise, MA; Levallois, C; Mani, JC; Sablayrolles, C1
Fredholm, BB; Jonzon, B1
Elfman, L; Fredholm, BB; Lindgren, E; Walum, E1
Altman, HJ; Barraco, RA; Coffin, VL; Phillis, JW; Taylor, JA1
Dobbins, JW; Forrest, JN; Laurenson, JP1
Hillyard, PA; Nials, AT; Skidmore, IF; Vardey, CJ1
Basile, AS; Dunwiddie, TV; Palmer, MR1
Carney, JM; Logan, L1
Fredholm, BB; Gazelius, B; Sidhagen, B1
Brown, C; Burnstock, G; Cusack, NJ; Meghji, P; Moody, CJ1
Hussain, T; Leigh, JH; Mustafa, SJ1
Calvo, JJ; López-Novoa, JM; Rodríguez-Nodal, F; San Román, JI1
Black, JW; Prentice, DJ; Shankley, NP1
Burnstock, G; Ralevic, V; Rubino, A1
Figarella, C; Kammouni, W; Merten, MD1
Arai, Y; Kisara, K; Nagaoka, H; Nakagawa, Y; Sakurada, S; Sakurada, T; Takeda, S1
Hargittai, PT; Lieberman, EA; Mustafa, SJ; Olanrewaju, HA1
Jarvis, JE; Reeves, JJ; Sheehan, MJ; Strong, P1
Nagy, LE1
Florio, C; Rosati, AM; Traversa, U; Vertua, R2
Modabber, M; Sabetkasai, M; Zarrindast, MR1
Coates, J; Green, MA; Sheehan, MJ; Strong, P1
Paalzow, GH1
Khoo, HE; Tan, CH; Tey, HB1
Akatsuka, Y; Egashira, K; Katsuda, Y; Narishige, T; Shimokawa, H; Takeshita, A; Ueno, H1
Martin, PL; Potts, AA1
Martin, PL; May, JM1
Nikfar, S; Zarrindast, MR1
Shafaghi, B; Zarrindast, MR1
Caussade, F; Cloarec, A1
Bass, BL; Dziki, AJ; Harmon, JW; Pennanen, MF1
Abdel-Rahman, AA; el-Mas, MM; Fahim, M; Mustafa, SJ1
Joran, ME; Murphy, DJ; Renninger, JE1
Agrawal, KC; Beckman, BS; Brookins, JW; Fisher, JW; Nakashima, J; Ohigashi, T1
Schofield, PR; Townsend-Nicholson, A1
Coates, J; Ellis, F; Evans, B; Foster, M; Gurden, MF; Hornby, E; Kennedy, I; Martin, DP; Strong, P; Vardey, CJ1
Joad, JP; Kott, KS1
Fisher, JW; Nakashima, J; Tazaki, H1
Mayfield, RD; Suzuki, F; Zahniser, NR1
Belloni, FL; Lee, HT; Linden, J; Thompson, CI1
Chauvelot-Moachon, L; Chen, YL; De Sousa, M; Florentin, I; Giroud, JP; Le Vraux, V; Masson, I1
Alexander, SP; Cooper, JA; Hill, SJ; Horn, EH; Rubin, PC1
Samini, M; Sharifzadeh, M; Zarrindast, MR1
Jen, SC; Rovainen, CM1
Harden, FA; Harrison, GJ; Headrick, J; Jordan, LR; Willis, RJ1
Konnaris, K; Lloyd, HG; Temple, DM1
Belloc, F; Boisseau, MR; Closse, C; Maurel, A; Pruvost, A; Renard, M; Seigneur, M1
Eleno, N; Lopez-Novoa, JM; MacLaughlin, M; Martinez-Salgado, C; Olivera, A1
Hourani, SM; Prentice, DJ1
Broadley, KJ; Maddock, HL1
Broadley, KJ; Ford, WR1
Chopde, CT; Ghosh, AK; Mandhane, SN1
Moghadamnia, AA; Zarrindast, MR1
Lundeberg, T; Segerdahl, M; Sjölund, KF; Sollevi, A1
Kemmotsu, O; Nakamura, I; Ohta, Y1
Caruso-Neves, C; Chagas, C; Francisco-Pedro, LG; Lopes, AG; Souza, LP1
Hourani, SM; Lewis, CD1
Hourani, SM; Nicholls, J; Skene, DJ1
Hourani, SM; Payne, SL; Prentice, DJ1
Florio, C; Frausin, F; Gaion, RM; Vertua, R1
Barahona, MV; Bustamante, S; García-Sacristán, A; Hernández, M; Orensanz, LM1
Gandolfi, O; Lucchi, R; Notari, S; Poli, A; Traversa, U; Zampacavallo, G1
Hamad, M1
Calacay, J; Cheng, K; Feighner, SD; Griffin, PR; Howard, AD; Leonard, RJ; Leong, D; Liu, K; Pomés, A; Pong, C; Schaeffer, J; Smith, AG; Smith, RG; Van der Ploeg, LH; Xu, Y1
Davis, CW; Morse, DM; Smullen, JL1
Turski, WA; Urbańska, EM; Wielosz, M; Zuchora, B1
Breschi, MC; Calderone, V; Martinotti, E; Nieri, P1
Homayoun, H; Khavandgar, S; Zarrindast, MR1
Green, TA; Schenk, S1
Rao, VS; Santos, FA1
Homayoun, H; Khavandgar, S; Torkaman-Boutorabi, A; Zarrindast, MR1
Ho, CM; Ho, ST; Peng, SC; Su, CK; Tsai, SK1
Homayounfar, H; Jamali-Raeufy, N; Sahebgharani, M; Zarrindast, MR1
Hylkema, MN; Postma, DS; Timens, W; Versluis, M1
Ben Addi, A; Boeynaems, JM; Communi, D; Hua, X; Ledent, C; Lefort, A; Libert, F; Macours, P; Robaye, B; Tilley, SL1
Kondo, Y; Morishima, T; Tsuge, M; Wada, T; Yashiro, M; Yasui, K1
Abdallah, Y; Arshad, M; Aslam, M; Becker, L; Grebe, M; Gündüz, D; Härtel, FV; Krieger, U; Noll, T; Piper, HM; Sedding, DG; Voss, RK1

Reviews

4 review(s) available for theophylline and adenosine-5'-(n-ethylcarboxamide)

ArticleYear
Adenosine receptors: pharmacology, structure-activity relationships, and therapeutic potential.
    Journal of medicinal chemistry, 1992, Feb-07, Volume: 35, Issue:3

    Topics: Adenosine; Animals; Humans; Models, Chemical; Receptors, Purinergic; Second Messenger Systems; Structure-Activity Relationship

1992
Adenosine receptors: targets for future drugs.
    Journal of medicinal chemistry, 1982, Volume: 25, Issue:3

    Topics: Adenosine; Adenosine Triphosphate; Animals; Humans; Ligands; Receptors, Cell Surface; Receptors, Purinergic; Structure-Activity Relationship; Xanthines

1982
Fluorescent ligands for adenosine receptors.
    Bioorganic & medicinal chemistry letters, 2013, Jan-01, Volume: 23, Issue:1

    Topics: Boron Compounds; Fluorescein-5-isothiocyanate; Fluorescent Dyes; Humans; Ligands; Protein Binding; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1

2013
Adenosine A2A receptor as a drug discovery target.
    Journal of medicinal chemistry, 2014, May-08, Volume: 57, Issue:9

    Topics: Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Crystallography, X-Ray; Drug Discovery; Humans; Ligands; Protein Conformation; Receptor, Adenosine A2A; Signal Transduction

2014

Other Studies

188 other study(ies) available for theophylline and adenosine-5'-(n-ethylcarboxamide)

ArticleYear
Species difference in the G protein selectivity of the human and bovine A1-adenosine receptor.
    The Journal of biological chemistry, 1994, Dec-23, Volume: 269, Issue:51

    Topics: Animals; Base Sequence; Brain; Cattle; DNA Primers; Escherichia coli; GTP-Binding Proteins; Humans; Molecular Sequence Data; Protein Binding; Receptors, Purinergic P1; Recombinant Proteins; Species Specificity

1994
Characterization of human A2A adenosine receptors with the antagonist radioligand [3H]-SCH 58261.
    British journal of pharmacology, 1997, Volume: 121, Issue:3

    Topics: Animals; Binding, Competitive; CHO Cells; Cricetinae; Cyclic AMP; Humans; Purinergic P1 Receptor Antagonists; Pyrimidines; Radioligand Assay; Rats; Receptor, Adenosine A2A; Receptors, Purinergic P1; Species Specificity; Transfection; Triazoles

1997
Comparative pharmacology of human adenosine receptor subtypes - characterization of stably transfected receptors in CHO cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 357, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Base Composition; Binding, Competitive; CHO Cells; Cricetinae; Guanylate Cyclase; Humans; Phenethylamines; Phenylisopropyladenosine; Receptors, Purinergic P1; Stereoisomerism; Structure-Activity Relationship; Transfection; Xanthines

1998
Inhibition of human mast cell activation with the novel selective adenosine A(2B) receptor antagonist 3-isobutyl-8-pyrrolidinoxanthine (IPDX)(2).
    Biochemical pharmacology, 2001, Nov-01, Volume: 62, Issue:9

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Anti-Asthmatic Agents; Cells, Cultured; Humans; Mast Cells; Purinergic P1 Receptor Antagonists; Pyrrolidinones; Receptor, Adenosine A2B; Receptors, Purinergic P1; Structure-Activity Relationship; Vasodilator Agents; Xanthine; Xanthines

2001
1,2,4-triazolo[4,3-a]quinoxalin-1-one moiety as an attractive scaffold to develop new potent and selective human A3 adenosine receptor antagonists: synthesis, pharmacological, and ligand-receptor modeling studies.
    Journal of medicinal chemistry, 2004, Jul-01, Volume: 47, Issue:14

    Topics: Adenosine A3 Receptor Antagonists; Animals; Cattle; CHO Cells; Cricetinae; Humans; Ligands; Models, Molecular; Quinoxalines; Radioligand Assay; Receptor, Adenosine A3; Structure-Activity Relationship; Triazoles

2004
Binding thermodynamics as a tool to investigate the mechanisms of drug-receptor interactions: thermodynamics of cytoplasmic steroid/nuclear receptors in comparison with membrane receptors.
    Journal of medicinal chemistry, 2005, Mar-24, Volume: 48, Issue:6

    Topics: Estradiol; Female; Humans; In Vitro Techniques; Male; Metribolone; Pregnenediones; Prostate; Receptors, Androgen; Receptors, Cell Surface; Receptors, Estrogen; Receptors, Progesterone; Receptors, Steroid; Thermodynamics; Uterus

2005
Pharmacological characterization of novel adenosine ligands in recombinant and native human A2B receptors.
    Biochemical pharmacology, 2005, Nov-25, Volume: 70, Issue:11

    Topics: Adenosine; Adenosine A2 Receptor Antagonists; Animals; Binding, Competitive; Cell Line; Cyclic AMP; Humans; Molecular Structure; Protein Binding; Receptor, Adenosine A2B; Recombinant Proteins

2005
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
1-alkyl-8-(piperazine-1-sulfonyl)phenylxanthines: development and characterization of adenosine A2B receptor antagonists and a new radioligand with subnanomolar affinity and subtype specificity.
    Journal of medicinal chemistry, 2009, Jul-09, Volume: 52, Issue:13

    Topics: Adenosine A2 Receptor Antagonists; Animals; Drug Design; Humans; Kinetics; Ligands; Mice; Protein Binding; Radioligand Assay; Rats; Receptor, Adenosine A2B; Xanthines

2009
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
Surface Plasmon Resonance Screening to Identify Active and Selective Adenosine Receptor Binding Fragments.
    ACS medicinal chemistry letters, 2022, Jul-14, Volume: 13, Issue:7

    Topics:

2022
Molecular cloning and expression of an adenosine A2b receptor from human brain.
    Biochemical and biophysical research communications, 1992, Aug-31, Volume: 187, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Amino Acid Sequence; Animals; Base Sequence; Brain Chemistry; CHO Cells; Cloning, Molecular; Cricetinae; Cyclic AMP; DNA; Gene Expression; Humans; Molecular Sequence Data; Receptors, Purinergic; Sequence Homology, Nucleic Acid; Theophylline; Transfection

1992
Pharmacological characterization of adenosine A1 and A2 receptors in the bladder: evidence for a modulatory adenosine tone regulating non-adrenergic non-cholinergic neurotransmission.
    British journal of pharmacology, 1992, Volume: 107, Issue:1

    Topics: Adenosine; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Animals; Autonomic Nervous System; Dipyridamole; Electric Stimulation; Mice; Muscle Contraction; Muscle, Smooth; Phenylisopropyladenosine; Receptors, Purinergic; Synaptic Transmission; Theophylline; Urinary Bladder

1992
Presynaptic A1-purinoceptor-mediated inhibitory effects of adenosine and its stable analogues on the mouse hemidiaphragm preparation.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 346, Issue:2

    Topics: 2-Chloroadenosine; Acetylcholine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Diaphragm; Dipyridamole; Electric Stimulation; In Vitro Techniques; Magnesium; Male; Mice; Muscle Contraction; Neuromuscular Junction; Phrenic Nerve; Purinergic Antagonists; Receptors, Purinergic; Synapses; Synaptic Transmission; Theophylline; Tritium; Tubocurarine; Xanthines

1992
Neutrophil adherence to endothelium is enhanced via adenosine A1 receptors and inhibited via adenosine A2 receptors.
    Journal of immunology (Baltimore, Md. : 1950), 1992, Apr-01, Volume: 148, Issue:7

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Antigens, CD; CD18 Antigens; Cell Adhesion; Endothelium, Vascular; Humans; Macrophage-1 Antigen; Mice; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Phenylisopropyladenosine; Receptors, Purinergic; Theophylline

1992
Relative agonist potencies of C2-substituted analogues of adenosine: evidence for adenosine A2B receptors in the guinea pig aorta.
    European journal of pharmacology, 1992, Jun-05, Volume: 216, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Aorta, Thoracic; Dose-Response Relationship, Drug; Endothelium, Vascular; Guinea Pigs; Male; Muscle, Smooth, Vascular; Phenethylamines; Receptors, Purinergic; Theophylline; Vasodilator Agents

1992
Local antinociceptive and hyperalgesic effects in the formalin test after peripheral administration of adenosine analogues in mice.
    Pharmacology & toxicology, 1992, Volume: 70, Issue:6 Pt 1

    Topics: Absorption; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Dose-Response Relationship, Drug; Drug Interactions; Extremities; Hyperalgesia; Male; Mice; Mice, Inbred Strains; Nociceptors; Pain Measurement; Phenethylamines; Phenylisopropyladenosine; Receptors, Purinergic; Theophylline

1992
A neuroprotective effect of adenosine A1-receptor agonists on ischemia-induced decrease in 2-deoxyglucose uptake in rat hippocampal slices.
    Neuroscience letters, 1992, Sep-28, Volume: 145, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Brain Ischemia; Deoxyglucose; Hippocampus; In Vitro Techniques; Male; Nervous System Diseases; Phenylisopropyladenosine; Purinergic Antagonists; Rats; Rats, Wistar; Receptors, Purinergic; Theophylline; Vasodilator Agents

1992
Evidence that adenosine receptors in the dog left atrium are not of the typical A1 or A2 adenosine receptor subtypes.
    European journal of pharmacology, 1992, Apr-22, Volume: 214, Issue:2-3

    Topics: Adenine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Dogs; Female; Heart Atria; In Vitro Techniques; Male; Myocardium; Norbornanes; Receptors, Purinergic; Theophylline; Vasodilation; Xanthines

1992
Purinergic agonist induction of metallothionein.
    Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine (New York, N.Y.), 1992, Volume: 201, Issue:1

    Topics: 2-Chloroadenosine; Adenosine; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Animals; Caffeine; Cells, Cultured; Cladribine; Deoxyadenosines; Dose-Response Relationship, Drug; Immunoblotting; Liver; Male; Metallothionein; Rats; Rats, Inbred Strains; RNA, Messenger; Theophylline; Time Factors; Transcription, Genetic; Vasodilator Agents

1992
Cerebrovascular reactivity to adenosine analogues in 0.6-0.7 gestation and near-term fetal sheep.
    The American journal of physiology, 1992, Volume: 262, Issue:5 Pt 2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Arterioles; Cerebrovascular Circulation; Female; Fetus; Gestational Age; Pregnancy; Sheep; Theophylline; Vasodilator Agents

1992
Chemical modification and irreversible inhibition of striatal A2a adenosine receptors.
    Molecular pharmacology, 1992, Volume: 42, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Affinity Labels; Amino Acid Sequence; Animals; Corpus Striatum; Diethyl Pyrocarbonate; Drug Antagonism; Hydroxylamine; Hydroxylamines; Molecular Sequence Data; Phenethylamines; Purinergic Antagonists; Rabbits; Radioligand Assay; Receptors, Purinergic; Theophylline; Xanthines

1992
A2 and P2 purine receptor interactions and surfactant secretion in primary cultures of type II cells.
    The American journal of physiology, 1991, Volume: 261, Issue:2 Pt 1

    Topics: Adenosine; Adenosine Diphosphate; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); AMP Deaminase; Animals; Cells, Cultured; Cyclic AMP; Inositol 1,4,5-Trisphosphate; Lung; Phosphatidylcholines; Pulmonary Surfactants; Receptors, Purinergic; Terbutaline; Theophylline; Thionucleotides; Xanthines

1991
Adenosine modulation of neuroeffector transmission in guinea-pig uterine smooth muscle.
    Acta physiologica Scandinavica, 1991, Volume: 143, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Muscle, Smooth; Myometrium; Synaptic Transmission; Theophylline; Uterine Contraction

1991
Adenosine receptors involved in the inhibitory control of non-adrenergic non-cholinergic neurotransmission in guinea-pig atria belong to the A1 subtype.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 344, Issue:4

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Atrial Function; Autonomic Nervous System; Electric Stimulation; Guinea Pigs; Heart; In Vitro Techniques; Male; Neurons, Afferent; Phenylisopropyladenosine; Receptors, Purinergic; Reserpine; Synaptic Transmission; Theophylline

1991
Adenosine enhances antigen-induced bronchoconstriction and histamine release in rat isolated lungs.
    Agents and actions, 1990, Volume: 30, Issue:1-2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Antigens; Bronchi; Histamine Release; In Vitro Techniques; Lung; Male; Muscle Contraction; Muscle, Smooth; Phenylisopropyladenosine; Rats; Rats, Inbred Strains; Receptors, Purinergic; Theophylline

1990
Differential regulation of human basophil and lung mast cell function by adenosine.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 256, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Basophils; Cyclic AMP; Dipyridamole; Histamine Release; Humans; Lung; Mast Cells; SRS-A; Theophylline

1991
Adenosine deaminase increases release of excitatory amino acids through a mechanism independent of adenosine depletion.
    Neuropharmacology, 1991, Volume: 30, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Adenosine; Adenosine Deaminase; Adenosine-5'-(N-ethylcarboxamide); Amino Acids; Animals; Aspartic Acid; Calcium; Calcium Radioisotopes; Cells, Cultured; Cerebellum; Female; Hydrolysis; Phosphatidylinositols; Rats; Rats, Inbred Strains; Theophylline

1991
Purinergic modulation of field stimulation responses of rat and human vas deferens smooth muscle.
    General pharmacology, 1991, Volume: 22, Issue:5

    Topics: Adenosine; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Animals; Caffeine; Electric Stimulation; Guanethidine; Humans; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Quinidine; Rats; Receptors, Purinergic; Theophylline; Urinary Bladder; Vas Deferens; Vasodilator Agents

1991
Methylxanthine-induced attenuation of pecking in chickens.
    British journal of pharmacology, 1991, Volume: 104, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Apomorphine; Behavior, Animal; Caffeine; Chickens; Dipyridamole; Female; Male; Theophylline; Xanthines

1991
Prejunctional stimulation of cholinergic nerves in rat airway smooth muscle by an adenosine analogue.
    Pulmonary pharmacology, 1991, Volume: 4, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cholinergic Fibers; In Vitro Techniques; Male; Neuromuscular Junction; Phenethylamines; Rats; Rats, Inbred Strains; Theophylline; Xanthines

1991
Postsynaptic dopamine/adenosine interaction: II. Postsynaptic dopamine agonism and adenosine antagonism of methylxanthines in short-term reserpinized mice.
    European journal of pharmacology, 1991, Jan-03, Volume: 192, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Bromocriptine; Caffeine; Dopamine; Male; Mice; Motor Activity; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Reserpine; Sulpiride; Synapses; Theophylline; Xanthines

1991
Adenosine A1 and non-A1 receptors: intracellular analysis of the actions of adenosine agonists and antagonists in rat hippocampal neurons.
    Brain research, 1991, Apr-12, Volume: 546, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Colforsin; Electric Stimulation; Electrodes; Hippocampus; Male; Membrane Potentials; Neurons; Phenylisopropyladenosine; Purinergic Antagonists; Rats; Rats, Inbred Strains; Receptors, Purinergic; Synapses; Theophylline; Xanthines

1991
Caffeine and theophylline as adenosine receptor antagonists in humans.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 258, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adult; Caffeine; Heart Rate; Humans; Male; Platelet Aggregation; Purinergic Antagonists; Receptors, Purinergic; Substance Withdrawal Syndrome; Theophylline

1991
Activation of brain adenosine receptors evokes vasodilation in skin arterioles.
    The American journal of physiology, 1991, Volume: 261, Issue:2 Pt 2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Arterioles; Brain; Cricetinae; Injections, Intraventricular; Male; Mesocricetus; Receptors, Purinergic; Skin; Theophylline; Vasodilation; Vasodilator Agents; Xanthines

1991
Adenosine-induced dilatation of the rabbit hepatic arterial bed is mediated by A2-purinoceptors.
    British journal of pharmacology, 1991, Volume: 103, Issue:1

    Topics: Acetylcholine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Antihypertensive Agents; Female; Hepatic Artery; In Vitro Techniques; Liver Circulation; Male; Phenethylamines; Phenylisopropyladenosine; Portal Vein; Rabbits; Receptors, Purinergic; Theophylline; Vasodilation

1991
Do adenosinergic substrates mediate methylxanthine effects upon reinforcement thresholds for electrical brain stimulation in the rat?
    Brain research, 1991, May-31, Volume: 550, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Brain; Carbolines; Chlordiazepoxide; Electric Stimulation; Hypothalamic Area, Lateral; Male; Midazolam; Phenylisopropyladenosine; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Purinergic; Reinforcement, Psychology; Self Stimulation; Sensory Thresholds; Theophylline; Triazoles

1991
Striatal A2 receptor regulates apomorphine-induced turning in rats with unilateral dopamine denervation.
    Psychopharmacology, 1991, Volume: 103, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Apomorphine; Brain Chemistry; Corpus Striatum; Denervation; Dopamine; Dose-Response Relationship, Drug; Hydroxydopamines; Oxidopamine; Rats; Receptors, Purinergic; Stereotyped Behavior; Substantia Nigra; Sympathectomy, Chemical; Theophylline

1991
Purinergic receptors have no major role in control of the circadian rhythm in rate of thymidine incorporation by cultured chick pineal glands.
    Journal of pineal research, 1991, Volume: 10, Issue:4

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Affinity Labels; Animals; Cells, Cultured; Chickens; Circadian Rhythm; Pineal Gland; Receptors, Purinergic; Theophylline; Thioinosine; Thymidine; Vasodilator Agents

1991
Behavioral effects of A1- and A2-selective adenosine agonists and antagonists: evidence for synergism and antagonism.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 259, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Injections, Intraperitoneal; Locomotion; Male; Mice; Phenethylamines; Receptors, Purinergic; Theophylline; Vasodilator Agents

1991
The role of adenosine in the vascular adaptation of neonatal cerebral blood flow during hypotension.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1991, Volume: 11, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Animals, Newborn; Blood Flow Velocity; Brain; Cerebrovascular Circulation; Hypotension; Hypoxanthine; Hypoxanthines; Inosine; Oxygen; Receptors, Purinergic; Swine; Theophylline; Vascular Resistance

1991
Characterization of the human peripheral lung adenosine receptor.
    American journal of respiratory cell and molecular biology, 1990, Volume: 2, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adolescent; Aged; Binding, Competitive; Cromolyn Sodium; Female; Humans; Lung; Male; Middle Aged; Receptors, Purinergic; Theophylline

1990
Adenosine mediates calcium-induced antinociception and potentiation of noradrenergic antinociception in the spinal cord.
    Brain research, 1990, Aug-06, Volume: 524, Issue:2

    Topics: 5,7-Dihydroxytryptamine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Calcium; Drug Synergism; Hot Temperature; Hydroxydopamines; Male; Methysergide; Norepinephrine; Oxidopamine; Pain; Phentolamine; Rats; Rats, Inbred Strains; Receptors, Purinergic; Serotonin; Spinal Cord; Theophylline

1990
Chronic carbamazepine down-regulates adenosine A2 receptors: studies with the putative selective adenosine antagonists PD115,199 and PD116,948.
    Psychopharmacology, 1990, Volume: 100, Issue:4

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Behavior, Animal; Brain Chemistry; Caffeine; Carbamazepine; Clonidine; Cyclic AMP; Down-Regulation; Male; Mice; Mice, Inbred C57BL; Motor Activity; Phenylisopropyladenosine; Purines; Receptors, Adrenergic; Sulfonamides; Theophylline; Xanthines

1990
Immune-related intestinal chloride secretion. II. Effect of adenosine on T84 cell line.
    The American journal of physiology, 1990, Volume: 258, Issue:5 Pt 1

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Calcium; Cell Line; Chlorides; Cyclic AMP; Cyclic GMP; Cytosol; Electrolytes; Epithelium; Histamine; Humans; Inflammation; Kinetics; Phenylisopropyladenosine; Phosphorylation; Protein Kinases; Theophylline

1990
Pertussis toxin pretreatment reveals differential effects of adenosine analogs on IgE-dependent histamine and peptidoleukotriene release from RBL-2H3 cells.
    Biochimica et biophysica acta, 1990, May-22, Volume: 1052, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Bucladesine; Cell Line; Histamine; Immunoglobulin E; Kinetics; Leukotrienes; Mast Cells; Peptides; Pertussis Toxin; Theophylline; Virulence Factors, Bordetella

1990
Fc gamma receptor-mediated functions in neutrophils are modulated by adenosine receptor occupancy. A1 receptors are stimulatory and A2 receptors are inhibitory.
    Journal of immunology (Baltimore, Md. : 1950), 1990, Oct-01, Volume: 145, Issue:7

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Antigens, Differentiation; Cell Adhesion; Cells, Cultured; Dose-Response Relationship, Drug; Flow Cytometry; Humans; In Vitro Techniques; Neutrophils; Pertussis Toxin; Phagocytosis; Phenylisopropyladenosine; Receptors, Fc; Receptors, IgG; Receptors, Purinergic; Superoxides; Theophylline; Virulence Factors, Bordetella

1990
Effects of adenosine and its analogues on isolated internal carotid arteries from newborn and adult pigs.
    Biology of the neonate, 1990, Volume: 58, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Animals, Newborn; Carotid Arteries; Dose-Response Relationship, Drug; In Vitro Techniques; Phenylisopropyladenosine; Swine; Theophylline

1990
Adenosine involvement in postictal events in amygdala-kindled rats.
    Epilepsy research, 1990, Volume: 6, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Amygdala; Animals; Anticonvulsants; Caffeine; Electric Stimulation; Electrodes, Implanted; Electroencephalography; Kindling, Neurologic; Male; Rats; Seizures; Theophylline; Time Factors

1990
Characterization of the locomotor depression produced by an A2-selective adenosine agonist.
    FEBS letters, 1990, Feb-12, Volume: 261, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Male; Mice; Molecular Structure; Motor Activity; Phenethylamines; Receptors, Purinergic; Theophylline

1990
Pharmacological evidence for the modulation of monoamine release by adenosine in the invertebrate nervous system.
    Journal of neurochemistry, 1990, Volume: 54, Issue:6

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Biogenic Amines; Bivalvia; Dopamine Antagonists; Dose-Response Relationship, Drug; Nervous System; Potassium; Serotonin Antagonists; Theophylline

1990
Adenosine depresses spontaneous transmitter release from frog motor nerve terminals by acting at an A1-like receptor.
    Life sciences, 1990, Volume: 46, Issue:19

    Topics: Acetylcholine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Membrane Potentials; Motor Neurons; Phenylisopropyladenosine; Purinergic Antagonists; Rana pipiens; Receptors, Purinergic; Theophylline; Xanthines

1990
Evidence that A2 purinoceptors are involved in endothelium-dependent relaxation of the rat thoracic aorta.
    British journal of pharmacology, 1990, Volume: 100, Issue:3

    Topics: Adenosine; Adenosine Diphosphate; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Animals; Aorta, Thoracic; Endothelium, Vascular; Hemoglobins; In Vitro Techniques; Indomethacin; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide; Norepinephrine; Phenylisopropyladenosine; Rats; Rats, Inbred Strains; Receptors, Purinergic; Theophylline

1990
Anticonvulsant effect of N-ethylcarboxamidoadenosine against kainic acid-induced behavioral seizures in the rat prepiriform cortex.
    Neuroscience letters, 1990, Jul-13, Volume: 114, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Dilazep; Kainic Acid; Limbic System; Male; Rats; Rats, Inbred Strains; Seizures; Theophylline

1990
Characteristics of adenosine binding sites in atrial sarcolemmal membranes.
    Biochimica et biophysica acta, 1985, Jun-27, Volume: 816, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Binding Sites; Binding, Competitive; Cattle; Endopeptidases; Heart Atria; Myocardium; Sarcolemma; Subcellular Fractions; Theophylline; Time Factors

1985
Adenosine-sensitive adenylate cyclase in rat anterior pituitary.
    Neuroendocrinology, 1985, Volume: 41, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adenylyl Cyclases; Animals; Cations, Divalent; Deoxyadenosines; Female; Guanine Nucleotides; In Vitro Techniques; Phenylisopropyladenosine; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains; Theophylline

1985
Modulation of the behavioral effects of chlordiazepoxide by methylxanthines and analogs of adenosine in squirrel monkeys.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Caffeine; Chlordiazepoxide; Conditioning, Psychological; Male; Phenylisopropyladenosine; Receptors, Cell Surface; Receptors, Purinergic; Saimiri; Theobromine; Theophylline; Xanthines

1985
Apparent enhancement of cholinergic transmission in rabbit bronchi via adenosine A2 receptors.
    European journal of pharmacology, 1986, Jan-21, Volume: 120, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Bronchi; Electric Stimulation; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Parasympathetic Nervous System; Phenylisopropyladenosine; Rabbits; Receptors, Cell Surface; Receptors, Purinergic; Substance P; Synaptic Transmission; Theophylline; Xanthines

1986
Characteristics of high affinity and low affinity adenosine binding sites in human cerebral cortex.
    Advances in experimental medicine and biology, 1986, Volume: 195 Pt B

    Topics: 1-Methyl-3-isobutylxanthine; 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Cell Membrane; Cerebral Cortex; Humans; Kinetics; Phenylisopropyladenosine; Receptors, Purinergic; Theophylline

1986
Adenosine receptors in post-mortem human cerebral cortex and the effect of carbamazepine.
    Clinical and experimental pharmacology & physiology, 1986, Volume: 13, Issue:10

    Topics: 1-Methyl-3-isobutylxanthine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Binding, Competitive; Carbamazepine; Cerebral Cortex; Humans; In Vitro Techniques; Kinetics; Phenylisopropyladenosine; Postmortem Changes; Receptors, Purinergic; Software; Theophylline

1986
Effects of alkylxanthines and calcium antagonists on adenosine uptake by cultured rabbit coronary microvascular endothelium.
    Pharmacology, 1987, Volume: 35, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Adenine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Calcium Channel Blockers; Cells, Cultured; Coronary Vessels; Dipyridamole; Endothelium; Ethanol; Isoproterenol; Male; Microcirculation; Rabbits; Theophylline; Trifluoperazine; Xanthines

1987
Adenosine inhibits immunoglobulin E-dependent histamine secretion from human basophil leukocytes by two independent mechanisms.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 242, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Basophils; Cyclic AMP; Dipyridamole; Dose-Response Relationship, Drug; Histamine Release; Humans; Immunoglobulin E; Methylation; Phospholipids; S-Adenosylmethionine; Theophylline; Tubercidin

1987
The ability of denbufylline to inhibit cyclic nucleotide phosphodiesterase and its affinity for adenosine receptors and the adenosine re-uptake site.
    British journal of pharmacology, 1989, Volume: 97, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; 2',3'-Cyclic-Nucleotide Phosphodiesterases; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cerebral Cortex; In Vitro Techniques; Kinetics; Male; Myocardium; Phenylisopropyladenosine; Rats; Rats, Inbred Strains; Receptors, Purinergic; Theophylline; Thioinosine; Xanthines

1989
Adenosine receptor-mediated relaxation in coronary artery: evidence for a guanyl nucleotide-binding regulatory protein involvement.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 251, Issue:3

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cattle; Cholera Toxin; Colforsin; Coronary Vessels; Ethylmaleimide; GTP-Binding Proteins; In Vitro Techniques; Receptors, Purinergic; Theophylline; Vasodilation

1989
Adenosine enhancement of adrenergic neuroeffector transmission in guinea-pig pulmonary artery.
    British journal of pharmacology, 1989, Volume: 96, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Male; Norepinephrine; Pulmonary Artery; Receptors, Purinergic; Sympathetic Nervous System; Synaptic Transmission; Theophylline; Vasoconstriction; Vasodilator Agents

1989
Diazepam enhances the inhibitory action of adenosine on transmission at the frog neuromuscular junction.
    European journal of pharmacology, 1989, May-19, Volume: 164, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Diazepam; Dipyridamole; Drug Synergism; In Vitro Techniques; Membrane Potentials; Motor Endplate; Muscle Contraction; Neuromuscular Junction; Rana ridibunda; Synaptic Transmission; Theophylline

1989
Effects of 1,3-dipropyl-8-cyclopentylxanthine (DPCPX), a highly selective adenosine receptor antagonist, on force of contraction in guinea-pig atrial and ventricular cardiac preparations.
    Naunyn-Schmiedeberg's archives of pharmacology, 1989, Volume: 340, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Female; Guinea Pigs; Heart; In Vitro Techniques; Isoenzymes; Male; Myocardial Contraction; Papillary Muscles; Phenylisopropyladenosine; Phosphoric Diester Hydrolases; Receptors, Purinergic; Theophylline; Xanthines

1989
Evidence for an adenosine A2/Ra receptor on human basophils.
    Life sciences, 1985, Jan-28, Volume: 36, Issue:4

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adenylyl Cyclases; Basophils; Biological Transport; Calcimycin; Histamine Release; Humans; Receptors, Cell Surface; Receptors, Purinergic; Structure-Activity Relationship; Theophylline; Thioinosine

1985
Evidence for adenosine receptor-mediated hyperpolarization in coronary smooth muscle.
    The American journal of physiology, 1989, Volume: 257, Issue:5 Pt 2

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cattle; Coronary Vessels; Electrophysiology; Membrane Potentials; Muscle, Smooth, Vascular; Potassium Chloride; Receptors, Purinergic; Theophylline; Vasodilator Agents

1989
Subsensitivity of presynaptic adenosine A1-receptors in caudal arteries of spontaneously hypertensive rats.
    European journal of pharmacology, 1989, Dec-19, Volume: 174, Issue:2-3

    Topics: Adenosine; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Animals; Blood Pressure; Electric Stimulation; Hypertension; In Vitro Techniques; Muscle, Smooth, Vascular; Norepinephrine; Phenylisopropyladenosine; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Rats, Inbred WKY; Receptors, Purinergic; Species Specificity; Theophylline; Vasoconstriction

1989
NECA-induced hypomotility in mice: evidence for a predominantly central site of action.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 32, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Central Nervous System; Male; Mice; Motor Activity; Receptors, Purinergic; Theophylline

1989
The effect of local infusion of adenosine and adenosine analogues on local cerebral blood flow.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1989, Volume: 9, Issue:4

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cerebrovascular Circulation; Dialysis; Injections, Intraventricular; Perfusion; Rats; Rats, Inbred Strains; Theophylline

1989
Adenosine receptors linked to adenylate cyclase activity in human neuroblastoma cells: modulation during cell differentiation.
    Neuroscience, 1989, Volume: 30, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adenylyl Cyclases; Calcium; Cell Differentiation; Cell Line; Humans; Neuroblastoma; Phenylisopropyladenosine; Receptors, Purinergic; Theophylline; Tumor Cells, Cultured

1989
Characterization of adenosine receptors in guinea-pig isolated left atria.
    British journal of pharmacology, 1989, Volume: 97, Issue:4

    Topics: Action Potentials; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Calcium Radioisotopes; Dipyridamole; Electric Stimulation; Guinea Pigs; Heart; In Vitro Techniques; Membrane Potentials; Myocardial Contraction; Myocardium; Phenylisopropyladenosine; Receptors, Purinergic; Rubidium Radioisotopes; Theophylline

1989
Characterization of adenosine receptors in bone. Studies on the effect of adenosine analogues on cyclic AMP formation and bone resorption in cultured mouse calvaria.
    Acta physiologica Scandinavica, 1987, Volume: 131, Issue:2

    Topics: 2-Chloroadenosine; Adenine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Bone and Bones; Bone Resorption; Cells, Cultured; Colforsin; Cyclic AMP; Mice; Phenylisopropyladenosine; Pyrrolidinones; Receptors, Cyclic AMP; Rolipram; Theophylline

1987
Changes in adenosine receptors during differentiation of 3T3-F442A cells to adipocytes.
    The Biochemical journal, 1988, Jan-15, Volume: 249, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adipose Tissue; Animals; Cell Differentiation; Cell Line; Colforsin; Cyclic AMP; Imidazoles; Isoproterenol; Mice; Phenylisopropyladenosine; Receptors, Purinergic; Theophylline

1988
Adenosine promotes neutrophil chemotaxis.
    The Journal of experimental medicine, 1988, Mar-01, Volume: 167, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Chemotaxis, Leukocyte; Drug Synergism; Humans; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Receptors, Purinergic; Stimulation, Chemical; Superoxides; Theophylline; Zymosan

1988
Evidence for A2 adenosine receptor-mediated effects on adenylate cyclase activity in rat ovarian membranes.
    Molecular and cellular endocrinology, 1988, Volume: 56, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adenylyl Cyclases; Animals; Cell Membrane; Cyclic AMP; Female; Follicle Stimulating Hormone; Ovary; Rats; Receptors, Purinergic; Theophylline

1988
Evidence for adenosine A1 receptor action in rat jejunal mucosa.
    European journal of pharmacology, 1988, Apr-27, Volume: 149, Issue:1-2

    Topics: Adenosine; Adenosine Deaminase; Adenosine-5'-(N-ethylcarboxamide); Animals; Colforsin; Cyclic AMP; In Vitro Techniques; Intestinal Mucosa; Jejunum; Male; Papaverine; Phenylisopropyladenosine; Rats; Rats, Inbred Strains; Receptors, Purinergic; Theophylline; Vasodilator Agents

1988
Presynaptic P1-purinoceptors in jejunal branches of the rabbit mesenteric artery and their possible function.
    The Journal of physiology, 1988, Volume: 397

    Topics: Action Potentials; Adenosine; Adenosine Deaminase; Adenosine-5'-(N-ethylcarboxamide); Animals; Female; Guanosine; In Vitro Techniques; Jejunum; Male; Mesenteric Arteries; Muscle, Smooth, Vascular; Phenylisopropyladenosine; Rabbits; Receptors, Neurotransmitter; Receptors, Purinergic; Theophylline; Thionucleosides

1988
Adenosine stimulates guanylate cyclase activity in vascular smooth muscle cells.
    The Journal of biological chemistry, 1987, May-05, Volume: 262, Issue:13

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cells, Cultured; Cyclic GMP; Enzyme Activation; Guanylate Cyclase; Male; Muscle, Smooth, Vascular; Rats; Rats, Inbred Strains; Theophylline; Time Factors

1987
Characterization of adenosine receptors in human pulmonary arteries.
    The American journal of physiology, 1989, Volume: 256, Issue:1 Pt 2

    Topics: Adenosine; Adenosine Deaminase; Adenosine-5'-(N-ethylcarboxamide); Adult; Dose-Response Relationship, Drug; Humans; Middle Aged; Phenylisopropyladenosine; Pulmonary Artery; Receptors, Purinergic; Theophylline; Vasodilation

1989
A1 and A2 adenosine receptor activation inhibits and stimulates renin secretion of rat renal cortical slices.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 232, Issue:3

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Calcium; Egtazic Acid; Gallopamil; In Vitro Techniques; Kidney Cortex; Male; Ouabain; Potassium Chloride; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Purinergic; Renin; Theophylline; Vanadates; Vanadium

1985
Adenosine; a physiologic modulator of superoxide anion generation by human neutrophils. Adenosine acts via an A2 receptor on human neutrophils.
    Journal of immunology (Baltimore, Md. : 1950), 1985, Volume: 135, Issue:2

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Binding Sites; Binding, Competitive; Humans; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Receptors, Cell Surface; Receptors, Purinergic; Superoxides; Theophylline

1985
Antagonism by theophylline of the adenosine receptor agonist 5'-N-ethylcarboxamidoadenosine at the guinea pig ileum.
    Canadian journal of physiology and pharmacology, 1985, Volume: 63, Issue:9

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Electric Stimulation; Female; Guinea Pigs; Ileum; In Vitro Techniques; Kinetics; Male; Receptors, Cell Surface; Receptors, Purinergic; Theophylline; Vasodilator Agents

1985
Evidence for an A2-subtype adenosine receptor on pancreatic glucagon secreting cells.
    British journal of pharmacology, 1985, Volume: 86, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Glucagon; In Vitro Techniques; Islets of Langerhans; Male; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Purinergic; Secretory Rate; Theophylline

1985
Evidence for an A2 adenosine receptor in guinea pig lung.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 331, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cyclic AMP; Guinea Pigs; In Vitro Techniques; Ligands; Lung; Membranes; Pyrrolidinones; Receptors, Cell Surface; Receptors, Purinergic; Rolipram; Theophylline; Time Factors

1985
Dual effects of adenosine and adenosine analogues on motor activity of the human fallopian tube.
    Acta physiologica Scandinavica, 1985, Volume: 125, Issue:3

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adult; Fallopian Tubes; Female; Humans; Lidocaine; Menstruation; Middle Aged; Muscle Contraction; Muscle, Smooth; Phenylisopropyladenosine; Receptors, Cell Surface; Receptors, Purinergic; Tetrodotoxin; Theophylline

1985
Evidence for adenosine receptor-mediated isoprenaline-antagonistic effects of the adenosine analogs PIA and NECA on force of contraction in guinea-pig atrial and ventricular cardiac preparations.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 331, Issue:2-3

    Topics: Action Potentials; Adenosine; Adenosine Deaminase; Adenosine-5'-(N-ethylcarboxamide); Adenylyl Cyclase Inhibitors; Animals; Dipyridamole; Female; Guinea Pigs; Heart Atria; Heart Ventricles; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Ouabain; Papillary Muscles; Phenylisopropyladenosine; Receptors, Cell Surface; Receptors, Purinergic; Theophylline

1985
Effect of adenosine receptor agonists and other compounds on cyclic AMP accumulation in forskolin-treated hippocampal slices.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:2

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adenylyl Cyclases; Animals; Colforsin; Cyclic AMP; Deoxyadenosines; Dideoxyadenosine; Dinoprostone; Dose-Response Relationship, Drug; Enzyme Activation; Hippocampus; Histamine; Isoproterenol; Male; Phenylisopropyladenosine; Prostaglandins E; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Purinergic; Theophylline; Xanthines

1986
Classification of adenosine receptors mediating antinociception in the rat spinal cord.
    British journal of pharmacology, 1986, Volume: 88, Issue:4

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Dose-Response Relationship, Drug; Male; Pain; Phenylisopropyladenosine; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Purinergic; Spinal Cord; Theophylline

1986
Adenosine receptors on human lymphocytes.
    Advances in experimental medicine and biology, 1986, Volume: 195 Pt B

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Alprostadil; Binding Sites; Colforsin; Cyclic AMP; Deoxyadenosines; Dideoxyadenosine; Histamine; Humans; In Vitro Techniques; Isoproterenol; Lymphocytes; Manganese; Neutrophils; Receptors, Purinergic; Theophylline; Vidarabine

1986
Inhibition of renin release by analogues of adenosine in rabbit renal cortical slices.
    Hypertension (Dallas, Tex. : 1979), 1987, Volume: 9, Issue:6

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Deoxyadenosines; Isomerism; Isoproterenol; Kidney Cortex; Male; Phenylisopropyladenosine; Rabbits; Receptors, Adrenergic, beta; Renin; Theophylline

1987
Functional evidence for adenosine A2 receptor regulation of phosphatidylcholine secretion in cultured type II pneumocytes.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:3

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cyclic AMP; Male; Phenylisopropyladenosine; Phosphatidylcholines; Pulmonary Alveoli; Rats; Rats, Inbred Strains; Receptors, Purinergic; Terbutaline; Theophylline

1987
Central versus peripheral mediation of responses to adenosine receptor agonists: evidence against a central mode of action.
    Brain research, 1987, Jul-14, Volume: 415, Issue:2

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Hippocampus; Injections, Intraperitoneal; Injections, Spinal; Phenylisopropyladenosine; Rats; Rats, Inbred Strains; Synaptic Transmission; Theophylline

1987
Psychomotor stimulant effects of methylxanthines in squirrel monkeys: relation to adenosine antagonism.
    Psychopharmacology, 1988, Volume: 95, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Caffeine; Male; Psychomotor Performance; Receptors, Purinergic; Saimiri; Stimulation, Chemical; Theophylline; Xanthines

1988
Inhibition of rat ventricular automaticity by adenosine.
    The American journal of physiology, 1985, Volume: 248, Issue:6 Pt 2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adenylyl Cyclases; Animals; Atropine; Depression, Chemical; Electric Stimulation; Electrocardiography; Heart Rate; Heart Ventricles; Male; Propranolol; Rats; Rats, Inbred Strains; Stereoisomerism; Systole; Theophylline

1985
3,7-Dimethyl-1-propargylxanthine: a potent and selective in vivo antagonist of adenosine analogs.
    Life sciences, 1988, Volume: 43, Issue:21

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Body Temperature; Caffeine; Male; Mice; Mice, Inbred DBA; Motor Activity; Reference Values; Theobromine; Theophylline

1988
Interactions of adenosine and magnesium on rat hippocampal slices.
    Brain research, 1988, Nov-01, Volume: 463, Issue:2

    Topics: 2-Chloroadenosine; Action Potentials; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Calcium; Drug Interactions; Electric Stimulation; Hippocampus; In Vitro Techniques; Magnesium; Rats; Theophylline

1988
125I-labeled 8-phenylxanthine derivatives: antagonist radioligands for adenosine A1 receptors.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:4

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adenylyl Cyclases; Affinity Labels; Algorithms; Animals; Binding, Competitive; Brain; Cattle; Humans; Iodine Radioisotopes; Iodobenzenes; Isotope Labeling; Kinetics; Ligands; Membranes; Rats; Rats, Inbred Strains; Receptors, Purinergic; Sodium Chloride; Structure-Activity Relationship; Theophylline; Xanthines

1988
Tolerance and cross-tolerance to theophylline-induced stimulation of locomotor activity in rats.
    Life sciences, 1988, Volume: 42, Issue:24

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Caffeine; Dextroamphetamine; Drug Tolerance; Male; Motor Activity; Phenylisopropyladenosine; Rats; Rats, Inbred Strains; Theophylline

1988
A1 and A2 adenosine receptor regulation of erythropoietin production.
    Life sciences, 1988, Volume: 43, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Albuterol; Animals; Erythrocytes; Erythropoietin; Female; Hypoxia; Iron Radioisotopes; Mice; Mice, Inbred ICR; Polycythemia; Receptors, Purinergic; Theophylline

1988
Effects of adenosine and its analogues on porcine basilar arteries: are only A2 receptors involved?
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1988, Volume: 8, Issue:1

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Basilar Artery; Dinoprost; Dose-Response Relationship, Drug; Phenylisopropyladenosine; Prostaglandins F; Receptors, Purinergic; Swine; Theophylline; Vasodilation; Vasodilator Agents

1988
Effects of adenosine infusion into renal interstitium on renal hemodynamics.
    The American journal of physiology, 1987, Volume: 252, Issue:4 Pt 2

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Blood Pressure; Glomerular Filtration Rate; Hemodynamics; Kidney; Male; Rats; Regional Blood Flow; Theophylline

1987
Electrophysiological evidence for adenosine receptors on astrocytes of cultured rat central nervous system.
    Neuroscience letters, 1987, Aug-18, Volume: 79, Issue:1-2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Astrocytes; Cells, Cultured; Cerebellum; Membrane Potentials; Phenylisopropyladenosine; Rats; Receptors, Purinergic; Spinal Cord; Theophylline

1987
Biochemical characterization of the antagonist actions of the xanthines, PACPX (1,3-dipropyl-8(2-amino-4-chloro)phenylxanthine) and 8-PT (8-phenyltheophylline) at adenosine A1 and A2 receptors in rat brain tissue.
    Biochemical pharmacology, 1987, Nov-15, Volume: 36, Issue:22

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Brain; In Vitro Techniques; Kinetics; Rats; Receptors, Purinergic; Theophylline; Xanthines

1987
Adenosine analogues. The temperature-dependence of the anticonvulsant effect and inhibition of 3H-D-aspartate release.
    Biochemical pharmacology, 1986, Sep-01, Volume: 35, Issue:17

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Anticonvulsants; Aspartic Acid; Body Temperature; Dose-Response Relationship, Drug; Female; Hippocampus; In Vitro Techniques; Male; Mice; Mice, Inbred DBA; Motor Activity; Potassium; Rats; Rats, Inbred Strains; Theophylline; Tritium

1986
Characterization of the antinociceptive effects of some adenosine analogues in the rat.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 334, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Analgesics; Animals; Dose-Response Relationship, Drug; Male; Phenylisopropyladenosine; Rats; Rats, Inbred Strains; Theophylline; Xanthines

1986
Characterization of adenosine-induced respiratory depression in the preterm rabbit.
    Biology of the neonate, 1985, Volume: 47, Issue:6

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Animals, Newborn; Apnea; Humans; Infant, Newborn; Infant, Newborn, Diseases; Phenylisopropyladenosine; Rabbits; Respiration Disorders; Theophylline; Tidal Volume; Time Factors

1985
Potent depressant effects of adenosine analogs on hippocampal slow-wave activity in the unanesthetized rat.
    Experimental brain research, 1985, Volume: 60, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Depression, Chemical; Electroencephalography; Hippocampus; Male; Phenylisopropyladenosine; Rats; Rats, Inbred Strains; Stereoisomerism; Theophylline

1985
Theophylline-like properties of xanthine analogs.
    Biochemical pharmacology, 1984, Jul-15, Volume: 33, Issue:14

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adenylyl Cyclases; Adult; Animals; Female; Humans; In Vitro Techniques; Male; Mice; Pyrazines; Receptors, Cell Surface; Receptors, Purinergic; Theophylline; Thymidine; Xanthines

1984
Adenosine receptor mediated inhibition of noradrenaline release from slices of the rat hippocampus.
    Life sciences, 1984, Nov-05, Volume: 35, Issue:19

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Calcium; Dipyridamole; Electric Stimulation; Hippocampus; Male; Norepinephrine; Phenylisopropyladenosine; Pyrrolidinones; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Purinergic; Rolipram; Theophylline; Xanthines

1984
Adenosine analogues stimulate cyclic AMP-accumulation in cultured neuroblastoma and glioma cells.
    Acta pharmacologica et toxicologica, 1984, Volume: 55, Issue:4

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Cell Line; Cells, Cultured; Cyclic AMP; Glioma; Humans; Kinetics; Neuroblastoma; Phenylisopropyladenosine; Phosphoric Diester Hydrolases; Pyrrolidinones; Rolipram; Theophylline; Vasodilator Agents

1984
Behavioral interaction of adenosine and methylxanthines on central purinergic systems.
    Neuroscience letters, 1984, Jun-15, Volume: 47, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Brain; Caffeine; Drug Interactions; Male; Mice; Mice, Inbred ICR; Motor Activity; Papaverine; Theophylline

1984
Adenosine and adenosine analogues stimulate adenosine cyclic 3', 5'-monophosphate-dependent chloride secretion in the mammalian ileum.
    The Journal of clinical investigation, 1984, Volume: 74, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Biological Transport; Chlorides; Cyclic AMP; Cyclic GMP; Ileum; Kinetics; Male; Phenylisopropyladenosine; Rabbits; Theophylline

1984
Characterization of the adenosine receptor responsible for the inhibition of histamine and SRS-A release from human lung fragments.
    British journal of pharmacology, 1984, Volume: 83, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Deoxyadenosines; Dideoxyadenosine; Dipyridamole; Guinea Pigs; Hexobendine; Histamine Release; Humans; In Vitro Techniques; Lung; Receptors, Cell Surface; Receptors, Purinergic; SRS-A; Theophylline; Time Factors

1984
Electrophysiological responses to adenosine analogs in rat hippocampus and cerebellum: evidence for mediation by adenosine receptors of the A1 subtype.
    Life sciences, 1984, Jan-02, Volume: 34, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cerebellum; Electrophysiology; Hippocampus; Male; Phenylisopropyladenosine; Purkinje Cells; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Purinergic; Theophylline

1984
Antagonism of the behavioral effects of L-phenylisopropyladenosine (L-PIA) by caffeine and its metabolites.
    Pharmacology, biochemistry, and behavior, 1984, Volume: 21, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Caffeine; Conditioning, Psychological; Male; Phenylisopropyladenosine; Rats; Rats, Inbred Strains; Theophylline; Xanthines

1984
Adenosine and adenosine analogues increase blood flow in oral mucosa.
    Acta physiologica Scandinavica, 1984, Volume: 120, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cats; Dipyridamole; Mouth Mucosa; Phenylisopropyladenosine; Purines; Regional Blood Flow; Theophylline; Vascular Resistance

1984
Evidence for stereospecificity of the P1-purinoceptor.
    British journal of pharmacology, 1982, Volume: 75, Issue:1

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Azides; Female; Guinea Pigs; Heart Atria; Ileum; In Vitro Techniques; Male; Receptors, Drug; Receptors, Purinergic; Stereoisomerism; Theophylline; Trachea

1982
Regulation of adenosine receptor function by theophylline in rat aorta.
    Journal of cardiovascular pharmacology, 1994, Volume: 24, Issue:1

    Topics: Acetylcholine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adrenergic beta-Agonists; Animals; Aorta; Colforsin; Endothelium, Vascular; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Norbornanes; Rats; Receptors, Purinergic P1; Theophylline

1994
Effect of adenosine and adenosine agonists on amylase release from rat pancreatic lobules.
    Life sciences, 1995, Volume: 57, Issue:17

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Amylases; Animals; Atropine; Dipyridamole; Dose-Response Relationship, Drug; Pancreatin; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Secretory Rate; Theophylline

1995
Pharmacological analysis of the interaction between purinoceptor agonists and antagonists in the guinea-pig taenia caecum.
    British journal of pharmacology, 1995, Volume: 115, Issue:4

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Binding, Competitive; Cecum; Dipyridamole; Dose-Response Relationship, Drug; Drug Interactions; Guinea Pigs; Heart Atria; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Myocardial Contraction; Phosphodiesterase Inhibitors; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Theophylline; Xanthines

1995
Contribution of P1-(A2b subtype) and P2-purinoceptors to the control of vascular tone in the rat isolated mesenteric arterial bed.
    British journal of pharmacology, 1995, Volume: 115, Issue:4

    Topics: 2-Chloroadenosine; Adenosine; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Animals; Antihypertensive Agents; Arginine; Dose-Response Relationship, Drug; Enzyme Inhibitors; In Vitro Techniques; Male; Mesenteric Arteries; Methoxamine; NG-Nitroarginine Methyl Ester; Phenethylamines; Rats; Rats, Wistar; Receptors, Purinergic P1; Receptors, Purinergic P2; Theophylline; Thionucleotides; Vasoconstriction; Vasoconstrictor Agents; Vasodilator Agents

1995
Evidence for, and characterization of, a lipopolysaccharide-inducible adenosine A2 receptor in human tracheal gland serous cells.
    FEBS letters, 1995, Aug-07, Volume: 369, Issue:2-3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Cells, Cultured; Cyclic AMP; Dipyridamole; Exocrine Glands; Humans; Lipopolysaccharides; Phenylisopropyladenosine; Proteinase Inhibitory Proteins, Secretory; Proteins; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Serine Proteinase Inhibitors; Theophylline; Trachea

1995
Theophylline-induced nociceptive behavioral response in mice: possible indirect interaction with spinal N-methyl-D-aspartate receptors.
    Neurochemistry international, 1993, Volume: 22, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Behavior, Animal; Male; Mice; Pain; Receptors, N-Methyl-D-Aspartate; Receptors, Purinergic; Spinal Cord; Substance P; Theophylline

1993
Role of endothelium in hyperpolarization of coronary smooth muscle by adenosine and its analogues.
    Journal of cardiovascular pharmacology, 1995, Volume: 25, Issue:2

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Arginine; Coronary Vessels; Dose-Response Relationship, Drug; Endothelium, Vascular; Humans; In Vitro Techniques; Indomethacin; Membrane Potentials; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide; omega-N-Methylarginine; Swine; Theophylline; Vasodilator Agents

1995
Further investigations into adenosine A1 receptor-mediated contraction in rat colonic muscularis mucosae and its augmentation by certain alkylxanthine antagonists.
    British journal of pharmacology, 1995, Volume: 114, Issue:5

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Colon; Cyclooxygenase Inhibitors; In Vitro Techniques; Indomethacin; Intestinal Mucosa; Muscle Contraction; Muscle, Smooth; Phosphodiesterase Inhibitors; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Quinazolines; Rats; Theophylline; Triazoles; Vasodilator Agents; Xanthines

1995
Role of adenosine A1 receptors in inhibition of receptor-stimulated cyclic AMP production by ethanol in hepatocytes.
    Biochemical pharmacology, 1994, Nov-29, Volume: 48, Issue:11

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cells, Cultured; Cyclic AMP; Drug Interactions; Ethanol; Glucagon; Liver; Male; Phenylisopropyladenosine; Rats; Rats, Wistar; Receptors, Purinergic P1; Theophylline

1994
Strain-related differences in adenosine receptor density and in behavioral sensitivity to adenosine analogs in mice.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 49, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Behavior, Animal; Brain; Dose-Response Relationship, Drug; Male; Membranes; Mice; Mice, Inbred CBA; Mice, Inbred Strains; Motor Activity; Platelet Aggregation Inhibitors; Radioligand Assay; Receptors, Purinergic P1; Species Specificity; Theophylline

1994
Influences of different adenosine receptor subtypes on catalepsy in mice.
    Psychopharmacology, 1993, Volume: 113, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Catalepsy; Dose-Response Relationship, Drug; Drug Interactions; Mice; Phenylisopropyladenosine; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Theophylline; Vasodilator Agents

1993
Characterization of the prejunctional adenosine receptors in the rat anococcygeus muscle.
    The Journal of pharmacy and pharmacology, 1994, Volume: 46, Issue:11

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Electric Stimulation; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle, Smooth; Phenylephrine; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Inbred Strains; Receptors, Purinergic P1; Theophylline; Vasodilator Agents; Xanthines

1994
Noradrenaline but not dopamine involved in NMDA receptor-mediated hyperalgesia induced by theophylline in awake rats.
    European journal of pharmacology, 1994, Jan-24, Volume: 252, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; alpha-Methyltyrosine; Animals; Bis(4-Methyl-1-Homopiperazinylthiocarbonyl)disulfide; Dizocilpine Maleate; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Hyperalgesia; Male; Methyltyrosines; Norepinephrine; Pain Measurement; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Reserpine; Sulpiride; Theophylline; Tyrosine 3-Monooxygenase

1994
Modulation of DNA synthesis via adenosine receptors in human epidermoid carcinoma (A431) cells.
    BioFactors (Oxford, England), 1994, Volume: 4, Issue:3-4

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Carcinoma, Squamous Cell; DNA, Neoplasm; Epidermal Growth Factor; Humans; Phenylisopropyladenosine; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Theophylline; Tumor Cells, Cultured; Xanthines

1994
ATP sensitive potassium channels are involved in adenosine A2 receptor mediated coronary vasodilatation in the dog.
    Cardiovascular research, 1994, Volume: 28, Issue:6

    Topics: Acetylcholine; Adenosine; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Animals; Colforsin; Coronary Circulation; Dogs; Dose-Response Relationship, Drug; Glyburide; Guanidines; Ion Channel Gating; Pinacidil; Potassium Channels; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P2; Theophylline; Vasodilator Agents; Xanthines

1994
The endothelium of the rat renal artery plays an obligatory role in A2 adenosine receptor-mediated relaxation induced by 5'-N-ethylcarboxamidoadenosine and N6-cyclopentyladenosine.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 270, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Arginine; Endothelium, Vascular; Glyburide; In Vitro Techniques; Indomethacin; Isoproterenol; Male; Muscle Relaxation; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitroprusside; Purinergic P1 Receptor Agonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Renal Artery; Renal Circulation; Theophylline; Vasodilator Agents; Xanthines

1994
Identification and functional characterization of A1 and A2 adenosine receptors in the rat vas deferens: a comparison with A1 receptors in guinea pig left atrium and A2 receptors in guinea pig aorta.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 269, Issue:3

    Topics: Adenine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Aorta; Guinea Pigs; Heart; In Vitro Techniques; Male; Norbornanes; Phenethylamines; Rats; Receptors, Purinergic P1; Theophylline; Vas Deferens; Xanthines

1994
Different influences of adenosine receptor agonists and antagonists on morphine antinociception in mice.
    General pharmacology, 1994, Volume: 25, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Dipyridamole; Dose-Response Relationship, Drug; Male; Mice; Morphine; Nociceptors; Phenylisopropyladenosine; Purinergic P1 Receptor Antagonists; Purinergic P2 Receptor Antagonists; Receptors, Purinergic P1; Receptors, Purinergic P2; Tail; Theophylline

1994
Effects of adenosine receptor agonists and antagonists on acquisition of passive avoidance learning.
    European journal of pharmacology, 1994, May-02, Volume: 256, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Analysis of Variance; Animals; Avoidance Learning; Caffeine; Dipyridamole; Dose-Response Relationship, Drug; Drug Interactions; Injections, Intraperitoneal; Male; Mice; Phenylisopropyladenosine; Purinergic P1 Receptor Antagonists; Theophylline; Vasodilator Agents

1994
Effect of tienoxolol, a new diuretic beta-blocking agent, on urinary prostaglandin excretion in the rat.
    British journal of pharmacology, 1993, Volume: 109, Issue:1

    Topics: 6-Ketoprostaglandin F1 alpha; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adrenergic beta-Antagonists; Animals; Brain Chemistry; Dinoprostone; Diuresis; Epoprostenol; Furosemide; Male; Natriuresis; Propanolamines; Prostaglandins; Radioimmunoassay; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Purinergic; Theophylline; Vasodilator Agents

1993
Adenosine: differential effect on blood flow to subregions of the upper gastrointestinal tract.
    The Journal of surgical research, 1994, Volume: 56, Issue:5

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Duodenum; Esophagus; Gastric Fundus; Gastric Mucosa; Ileum; Inosine; Intestine, Small; Jejunum; Mucous Membrane; Muscle, Smooth; Organ Specificity; Purinergic P1 Receptor Antagonists; Pyloric Antrum; Rabbits; Receptors, Purinergic P1; Regional Blood Flow; Theophylline; Vasodilator Agents

1994
Influence of aortic baroreceptor denervation on adenosine receptor-mediated relaxation of isolated rat aorta.
    European journal of pharmacology, 1994, Mar-11, Volume: 254, Issue:1-2

    Topics: Acetylcholine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Aorta, Thoracic; Arginine; Blood Pressure; Endothelium, Vascular; Heart Rate; In Vitro Techniques; Male; Muscle Denervation; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide; omega-N-Methylarginine; Phenylephrine; Pressoreceptors; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Theophylline

1994
Effects of adenosine agonists and antagonists on pulmonary ventilation in conscious rats.
    General pharmacology, 1993, Volume: 24, Issue:4

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Body Temperature; Bronchoconstriction; Bronchodilator Agents; Lung; Male; Naloxone; Narcotics; Phenylisopropyladenosine; Rats; Rats, Sprague-Dawley; Respiratory Mechanics; Theophylline; Vasodilator Agents; Xanthines

1993
Effects of 5'-N-ethylcarboxamideadenosine (NECA) on erythropoietin production.
    Kidney international, 1993, Volume: 44, Issue:4

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Carcinoma, Hepatocellular; Dose-Response Relationship, Drug; Erythropoietin; Female; Hypoxia; Liver Neoplasms; Mice; Mice, Inbred Strains; Osmolar Concentration; Polycythemia; Theophylline; Tumor Cells, Cultured

1993
A threonine residue in the seventh transmembrane domain of the human A1 adenosine receptor mediates specific agonist binding.
    The Journal of biological chemistry, 1994, Jan-28, Volume: 269, Issue:4

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Amino Acid Sequence; Binding Sites; Binding, Competitive; Brain; Cell Membrane; Humans; Kinetics; Mutagenesis, Site-Directed; Point Mutation; Radioligand Assay; Receptors, Purinergic P1; Recombinant Proteins; Stereoisomerism; Theophylline; Threonine; Tritium

1994
Functional characterization of three adenosine receptor types.
    British journal of pharmacology, 1993, Volume: 109, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adipose Tissue; Animals; Aorta, Thoracic; Blood Platelets; Coronary Vessels; Dogs; Female; Guinea Pigs; Heart; Humans; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Neutrophils; Norepinephrine; Phenethylamines; Rats; Receptors, Purinergic; Theophylline; Vasodilator Agents; Xanthines

1993
Effect of adenosine receptor ligands on cAMP content in human airways and peripheral lung.
    American journal of respiratory cell and molecular biology, 1993, Volume: 9, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adolescent; Adult; Aged; Child; Cromolyn Sodium; Cyclic AMP; Female; Humans; Ligands; Lung; Male; Middle Aged; Phenethylamines; Receptors, Purinergic; Respiratory System; Theophylline; Xanthines

1993
[Increase in erythropoietin secretion mediated by adenosine A2 receptors].
    Human cell, 1993, Volume: 6, Issue:1

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Carcinoma, Hepatocellular; Cell Hypoxia; Cyclic AMP; Erythropoietin; Humans; Liver Neoplasms; Receptors, Purinergic; Theophylline; Tumor Cells, Cultured

1993
Adenosine A2a receptor modulation of electrically evoked endogenous GABA release from slices of rat globus pallidus.
    Journal of neurochemistry, 1993, Volume: 60, Issue:6

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Analysis of Variance; Animals; Chromatography, High Pressure Liquid; Electric Stimulation; gamma-Aminobutyric Acid; Globus Pallidus; In Vitro Techniques; Kinetics; Male; Phenethylamines; Purinergic Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic; Theophylline; Time Factors; Xanthines

1993
Differential sensitization of cardiac actions of adenosine in rats after chronic theophylline treatment.
    The American journal of physiology, 1993, Volume: 264, Issue:5 Pt 2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Heart; Heart Atria; Male; Myocardium; Rats; Rats, Wistar; Receptors, Purinergic; Theophylline; Time Factors; Up-Regulation; Xanthines

1993
Inhibition of human monocyte TNF production by adenosine receptor agonists.
    Life sciences, 1993, Volume: 52, Issue:24

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Biological Assay; Cells, Cultured; Dexamethasone; Dipyridamole; Endotoxins; Humans; L Cells; Lipopolysaccharides; Male; Mice; Monocytes; Phenylisopropyladenosine; Rats; Rats, Inbred F344; Receptors, Purinergic; Theophylline; Tumor Necrosis Factor-alpha

1993
Adenosine receptor-induced cyclic AMP generation and inhibition of 5-hydroxytryptamine release in human platelets.
    British journal of clinical pharmacology, 1995, Volume: 40, Issue:1

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adolescent; Adult; Antihypertensive Agents; Cyclic AMP; Humans; Middle Aged; Phenethylamines; Phenylisopropyladenosine; Platelet Aggregation Inhibitors; Purinergic P1 Receptor Agonists; Purines; Receptors, Purinergic P1; Serotonin; Sulfonamides; Theophylline; Vasodilator Agents; Xanthines

1995
Effects of adenosine analogues on apomorphine-induced penile erection in rats.
    General pharmacology, 1995, Volume: 26, Issue:8

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Apomorphine; Male; Penile Erection; Rats; Receptors, Purinergic P1; Theophylline

1995
An adenosine agonist increases blood flow and density of capillary branches in the optic tectum of Xenopus laevis tadpoles.
    Microcirculation (New York, N.Y. : 1994), 1994, Volume: 1, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Caffeine; Capillaries; Microcirculation; Microscopy, Video; Neovascularization, Physiologic; Nitroglycerin; Regional Blood Flow; Superior Colliculi; Theophylline; Time Factors; Vasodilator Agents; Xenopus laevis

1994
A biphasic response to adenosine in the coronary vasculature of the K(+)-arrested perfused rat heart.
    European journal of pharmacology, 1996, Jun-20, Volume: 307, Issue:1

    Topics: Adenosine; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Animals; Coronary Vessels; Heart; Heart Arrest, Induced; In Vitro Techniques; Male; Muscle Relaxation; Perfusion; Potassium; Purinergic P1 Receptor Agonists; Rats; Rats, Wistar; Theophylline; Vasodilator Agents

1996
Release of adenosine from human sensitized lung fragments and its effect on antigen-induced mediator release.
    Pulmonary pharmacology, 1996, Volume: 9, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Antigens; Guinea Pigs; Histamine Release; Humans; Immunization; In Vitro Techniques; Leukotrienes; Lung; Mast Cells; Theophylline

1996
Effect of buflomedil on the neutrophil-endothelial cell interaction under inflammatory and hypoxia conditions.
    Haemostasis, 1996, Volume: 26 Suppl 4

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Cell Adhesion; Cell Hypoxia; Cells, Cultured; Cytokines; Endothelium, Vascular; Humans; Inflammation; Intercellular Adhesion Molecule-1; Interleukin-1; Neutrophils; P-Selectin; Pyrrolidines; Theophylline; Umbilical Veins

1996
Adenosine activates mesangial cell proliferation.
    Cellular signalling, 1997, Volume: 9, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Calcium; Cell Division; Cells, Cultured; Cyclic AMP; Glomerular Mesangium; Phenylisopropyladenosine; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Purines; Rats; Rats, Wistar; Sulfonamides; Theophylline; Thymidine; Xanthines

1997
Adenosine analogues relax guinea-pig taenia caeci via an adenosine A2B receptor and a xanthine-resistant site.
    European journal of pharmacology, 1997, Mar-26, Volume: 323, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cecum; Dose-Response Relationship, Drug; Guinea Pigs; Male; Muscle Relaxation; Muscle, Smooth; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Theophylline; Triazines; Triazoles; Vasodilator Agents; Xanthines

1997
Inhibitory and excitatory effects of adenosine antagonists on spontaneous locomotor activity in mice.
    Life sciences, 1997, Volume: 60, Issue:17

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Antineoplastic Agents; Male; Mice; Motor Activity; Purinergic P1 Receptor Agonists; Purines; Sulfonamides; Theophylline; Xanthines

1997
P1-purinoceptor-mediated vasodilatation and vasoconstriction in hypoxia.
    Journal of autonomic pharmacology, 1996, Volume: 16, Issue:6

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Guinea Pigs; Hypoxia; In Vitro Techniques; Indomethacin; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Phenethylamines; Phenylisopropyladenosine; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Theophylline; Vasoconstriction; Vasodilation

1996
Functional classification of P1-purinoceptors in guinea-pig left and right atria: anomalous characteristics of antagonism by cyclopentyltheophylline.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 355, Issue:6

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Guinea Pigs; Heart Atria; Heart Rate; In Vitro Techniques; Male; Myocardial Contraction; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Theophylline

1997
Adenosine A2 receptors modulate haloperidol-induced catalepsy in rats.
    European journal of pharmacology, 1997, Jun-11, Volume: 328, Issue:2-3

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Catalepsy; Dopamine Antagonists; Haloperidol; Male; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Scopolamine; Theobromine; Theophylline; Xanthines

1997
Adenosine receptor agents and conditioned place preference.
    General pharmacology, 1997, Volume: 29, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Conditioning, Operant; Dose-Response Relationship, Drug; Male; Mice; Phenylisopropyladenosine; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Theophylline

1997
Intrathecal adenosine analog administration reduces substance P in cerebrospinal fluid along with behavioral effects that suggest antinociception in rats.
    Anesthesia and analgesia, 1997, Volume: 85, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Analgesia; Animals; Behavior, Animal; Calcitonin Gene-Related Peptide; Dose-Response Relationship, Drug; Injections, Spinal; Male; Motor Activity; Pain Threshold; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Reaction Time; Substance P; Theophylline

1997
Characterization of adenosine receptors mediating spinal sensory transmission related to nociceptive information in the rat.
    Anesthesiology, 1997, Volume: 87, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Analgesics; Animals; Dose-Response Relationship, Drug; Female; Male; Pain; Rats; Rats, Wistar; Receptors, Purinergic P1; Reflex, Monosynaptic; Spinal Cord; Theophylline

1997
Effect of adenosine on the ouabain-insensitive Na+-ATPase activity from basolateral membrane of the proximal tubule.
    Biochimica et biophysica acta, 1997, Oct-23, Volume: 1329, Issue:2

    Topics: Adenosine; Adenosine Triphosphatases; Adenosine-5'-(N-ethylcarboxamide); Animals; Bucladesine; Cation Transport Proteins; Cell Membrane; Cholera Toxin; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Furosemide; Kidney Cortex; Kidney Tubules, Proximal; Kinetics; Ouabain; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Sodium-Potassium-Exchanging ATPase; Swine; Theophylline

1997
Involvement of functional antagonism in the effects of adenosine antagonists and L-NAME in the rat isolated heart.
    General pharmacology, 1997, Volume: 29, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adrenergic alpha-Agonists; Animals; Anti-Arrhythmia Agents; Enzyme Inhibitors; Heart; Heart Atria; In Vitro Techniques; Male; Myocardial Contraction; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Nitroprusside; Phenethylamines; Phenylephrine; Purinergic P1 Receptor Antagonists; Purines; Rats; Rats, Wistar; Sulfonamides; Theophylline; Vasodilator Agents

1997
Use of a newly developed technique to isolate rat pinealocytes and study the effects of adenosine agonists on melatonin production.
    Journal of pineal research, 1997, Volume: 23, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cell Separation; Dose-Response Relationship, Drug; Isoproterenol; Male; Melatonin; Phenethylamines; Pineal Gland; Radioimmunoassay; Rats; Rats, Wistar; Theophylline

1997
Activation of two sites by adenosine receptor agonists to cause relaxation in rat isolated mesenteric artery.
    British journal of pharmacology, 1997, Volume: 122, Issue:7

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Anti-Arrhythmia Agents; Dinucleoside Phosphates; Dose-Response Relationship, Drug; Male; Mesenteric Arteries; Purinergic P1 Receptor Agonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Theophylline; Triazines; Triazoles; Vasodilation; Vasodilator Agents

1997
Involvement of P1 receptors in the effect of forskolin on cyclic AMP accumulation and export in PC12 cells.
    Biochemical pharmacology, 1999, Feb-15, Volume: 57, Issue:4

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Colforsin; Cyclic AMP; PC12 Cells; Probenecid; Purinergic P1 Receptor Antagonists; Rats; Receptors, Purinergic P1; Theophylline; Time Factors

1999
A2B adenosine receptors mediate relaxation of the pig intravesical ureter: adenosine modulation of non adrenergic non cholinergic excitatory neurotransmission.
    British journal of pharmacology, 1999, Volume: 126, Issue:4

    Topics: Adenosine; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Animals; Dose-Response Relationship, Drug; Electric Stimulation; Female; Indomethacin; Male; Muscle Relaxation; Receptors, Purinergic P1; Swine; Synaptic Transmission; Theophylline; Ureter; Xanthines

1999
Pharmacological characterization of adenosine A1 receptors and its functional role in brown trout (Salmo trutta) brain.
    Brain research, 1999, Aug-07, Volume: 837, Issue:1-2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Binding, Competitive; Brain; Cell Membrane; Glutamic Acid; Guanosine Diphosphate; Kinetics; Neuroprotective Agents; Radioligand Assay; Receptors, Purinergic P1; Synaptosomes; Theophylline; Tritium; Trout; Xanthines

1999
The role of adenosine receptor engagement in murine fetal thymocyte development.
    APMIS : acta pathologica, microbiologica, et immunologica Scandinavica, 1999, Volume: 107, Issue:10

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Apoptosis; CD4 Antigens; CD8 Antigens; Cell Differentiation; Female; GTP-Binding Proteins; Mice; Mice, Inbred DBA; Organ Culture Techniques; Receptors, Purinergic P1; Signal Transduction; T-Lymphocyte Subsets; Theophylline; Thymus Gland

1999
Adenosine: A partial agonist of the growth hormone secretagogue receptor.
    Biochemical and biophysical research communications, 2000, Oct-05, Volume: 276, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Aequorin; Animals; Binding Sites; Cell Extracts; Cell Line; Chromatography, High Pressure Liquid; Dopamine; Humans; Hypothalamus; Indoles; Ligands; Luminescent Measurements; Mass Spectrometry; Models, Biological; Mutagenesis, Site-Directed; Neurons; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Receptors, Ghrelin; Spiro Compounds; Swine; Theophylline

2000
Differential effects of UTP, ATP, and adenosine on ciliary activity of human nasal epithelial cells.
    American journal of physiology. Cell physiology, 2001, Volume: 280, Issue:6

    Topics: Adenosine; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Antineoplastic Agents; Cilia; Cyclic AMP; Dose-Response Relationship, Drug; Epithelial Cells; Humans; Nasal Mucosa; Purinergic P2 Receptor Antagonists; Receptors, Purinergic P2; Receptors, Purinergic P2Y1; Receptors, Purinergic P2Y2; Theophylline; Uridine Triphosphate

2001
Protective effect of adenosine receptor agonists in a new model of epilepsy--seizures evoked by mitochondrial toxin, 3-nitropropionic acid, in mice.
    Neuroscience letters, 2001, Jun-08, Volume: 305, Issue:2

    Topics: 2-Chloroadenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Convulsants; Epilepsy; Hormone Antagonists; Male; Mice; Mitochondria; Neuroprotective Agents; Nitro Compounds; Phenylisopropyladenosine; Propionates; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Theophylline

2001
Adenosine-mediated hypotension in in vivo guinea-pig: receptors involved and role of NO.
    British journal of pharmacology, 2001, Volume: 134, Issue:4

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Blood Pressure; Diphenhydramine; Dose-Response Relationship, Drug; Enzyme Inhibitors; Guinea Pigs; Heart Rate; Hypotension; Male; Methylene Blue; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Theophylline; Triazines; Triazoles; Vasodilator Agents; Xanthines

2001
Effects of adenosine receptor agonists and antagonists on pentylenetetrazole-induced amnesia.
    European journal of pharmacology, 2001, Nov-02, Volume: 430, Issue:2-3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Amnesia; Analysis of Variance; Animals; Avoidance Learning; Convulsants; Dose-Response Relationship, Drug; Male; Mice; Pentylenetetrazole; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Retention, Psychology; Theophylline

2001
Dopaminergic mechanism for caffeine-produced cocaine seeking in rats.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2002, Volume: 26, Issue:4

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Benzazepines; Caffeine; Central Nervous System Stimulants; Cocaine-Related Disorders; Conditioning, Operant; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Male; Motor Activity; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Reinforcement Schedule; Salicylamides; Self Administration; Theophylline; Vasodilator Agents

2002
Possible role of mast cells in cineole-induced scratching behavior in mice.
    Food and chemical toxicology : an international journal published for the British Industrial Biological Research Association, 2002, Volume: 40, Issue:10

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Behavior, Animal; Cyclohexanols; Cyproheptadine; Diphenhydramine; Eucalyptol; Histamine H1 Antagonists; Male; Mast Cells; Mice; Monoterpenes; Naloxone; p-Methoxy-N-methylphenethylamine; Purinergic P1 Receptor Agonists; Serotonin Antagonists; Terpenes; Theophylline

2002
The effects of adenosine receptor agonists and antagonists on morphine state-dependent memory of passive avoidance.
    Neurobiology of learning and memory, 2002, Volume: 78, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Analgesics, Opioid; Animals; Learning; Male; Memory; Mice; Morphine; Receptors, Purinergic P1; Theophylline; Vasodilator Agents

2002
The role of intraspinal adenosine A1 receptors in sympathetic regulation.
    European journal of pharmacology, 2004, May-10, Volume: 492, Issue:1

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine A3 Receptor Agonists; Adenosine A3 Receptor Antagonists; Adenosine-5'-(N-ethylcarboxamide); Animals; Dihydropyridines; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Spinal Cord; Splanchnic Nerves; Sympathetic Nervous System; Synaptic Transmission; Theobromine; Theophylline; Triazines; Triazoles

2004
Adenosine receptor mediates nicotine-induced antinociception in formalin test.
    Pharmacological research, 2005, Volume: 51, Issue:3

    Topics: Adenosine-5'-(N-ethylcarboxamide); Analgesics; Animals; Dose-Response Relationship, Drug; Male; Mice; Nicotine; Pain Measurement; Purinergic P1 Receptor Agonists; Receptors, Purinergic P1; Theophylline

2005
Effects of IL-4 and IL-13 on adenosine receptor expression and responsiveness of the human mast cell line 1.
    International immunopharmacology, 2008, Volume: 8, Issue:6

    Topics: Adenosine Monophosphate; Adenosine-5'-(N-ethylcarboxamide); Bronchoconstriction; Cell Line, Tumor; Histamine Release; Humans; Interleukin-13; Interleukin-4; Interleukin-8; Mast Cells; Receptor, Adenosine A2A; Receptor, Adenosine A2B; Theophylline; Vasodilator Agents

2008
Modulation of murine dendritic cell function by adenine nucleotides and adenosine: involvement of the A(2B) receptor.
    European journal of immunology, 2008, Volume: 38, Issue:6

    Topics: Acetamides; Adenine Nucleotides; Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine-5'-(N-ethylcarboxamide); Animals; Antigens, Surface; Arginase; Cyclic AMP; Cytokines; Dendritic Cells; Gene Expression; Gene Expression Profiling; Interleukin-12; Lipopolysaccharides; Mice; Mice, Inbred C57BL; Mice, Knockout; Nitrites; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Purines; Receptor, Adenosine A2A; Receptor, Adenosine A2B; Receptors, Purinergic P1; Signal Transduction; Theophylline

2008
Theophylline inhibits the differentiation of human monocyte into dendritic cell potentially via adenosine receptor antagonism.
    Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology, 2009, Volume: 39, Issue:12

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine Deaminase; Adenosine-5'-(N-ethylcarboxamide); Adult; Apoptosis; Caspase 3; CD11c Antigen; Cell Differentiation; Dendritic Cells; Granulocyte-Macrophage Colony-Stimulating Factor; HLA-DR Antigens; Humans; Interleukin-4; Male; Monocytes; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptor, Adenosine A1; Receptors, Purinergic P1; Recombinant Proteins; RNA, Small Interfering; Rolipram; Theophylline; Xanthines

2009
Opposing effects of ATP and adenosine on barrier function of rat coronary microvasculature.
    Journal of molecular and cellular cardiology, 2012, Volume: 52, Issue:5

    Topics: Actin Cytoskeleton; Adenosine; Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Animals; Cadherins; Cells, Cultured; Coronary Vessels; Edema, Cardiac; Endothelial Cells; Male; Myocardium; Permeability; Protein Transport; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Purinergic P2 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Theophylline; Venules

2012