tetrahydrodeoxycorticosterone has been researched along with gamma-aminobutyric acid in 47 studies
*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]
*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 16 (34.04) | 18.2507 |
2000's | 23 (48.94) | 29.6817 |
2010's | 8 (17.02) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Gee, KW; Lan, NC | 1 |
Blakeman, DP; Im, WB | 1 |
Ayer, DE; Blakeman, DP; Davis, JP; Im, WB | 1 |
Costa, E; Paul, SM; Pritchett, DB; Puia, G; Purdy, RH; Santi, MR; Seeburg, PH; Vicini, S | 1 |
Finn, DA; Gee, KW | 1 |
Acosta-Burruel, M; Goodnough, DB; Hawkinson, JE; Kimbrough, CL; Wood, PL | 1 |
Biscardi, R; Wilson, MA | 1 |
Vicini, S; Zhu, WJ | 1 |
Reith, CA; Sillar, KT | 1 |
Chapell, R; Leidenheimer, NJ | 1 |
Alvarez-Hernandez, X; Bueno, OF; Leidenheimer, NJ; Robinson, LC | 1 |
Banerjee, PK; Brailowsky, S; Olsen, RW; Snead, OC; Tillakaratne, NJ; Tobin, AJ | 1 |
Banerjee, PK; Liu, CC; Snead, OC | 1 |
Deisz, RA; Holsboer, F; Vedder, H; Wetzel, CH; Zieglgänsberger, W | 1 |
Amin, J; Moorefield, CN; Morris, KD | 1 |
Breese, GR; Criswell, HE; McCown, TJ; Ming, Z; Mueller, RA | 1 |
Biggio, G; Littera, M; Papi, G; Pisu, MG; Purdy, RH; Sanna, E; Serra, M; Tuveri, F; Usala, L | 1 |
Carroll, SS; Li, YH; McEwen, BS; Orchinik, M; Weiland, NG | 1 |
Hevers, W; Korpi, ER; Lüddens, H | 1 |
Bianchi, MT; Macdonald, RL; Wohlfarth, KM | 1 |
Bianchi, MT; Haas, KF; Macdonald, RL | 1 |
Homanics, GE; Huguenard, JR; Huntsman, MM; Mihalek, RM; Porcello, DM | 1 |
Bianchi, MT; Macdonald, RL | 1 |
Bäckström, T; Lundgren, P; Strömberg, J | 1 |
Bíró, T; Maksay, G | 1 |
Bäckström, T; Johansson, IM; Lindblad, C; Rahman, M; Wang, MD | 1 |
Mashimo, T; Takahashi, A; Uchida, I | 1 |
Barrett-Jolley, R; Pyner, S; Womack, MD | 1 |
Amin, J; Hadley, SH | 1 |
Poisbeau, P; Schlichter, R; Vergnano, AM | 1 |
Sedelnikova, A; Weiss, DS; Zheleznova, N | 1 |
Dósa, Z; Drasbek, KR; Jensen, K; Vardya, I | 1 |
Han, SM; Youn, DH | 1 |
De Sarro, G; Dore, R; Maciocco, E; Mostallino, MC; Mura, ML; Pisu, MG; Russo, E; Serra, M | 1 |
Meera, P; Olsen, RW; Otis, TS; Wallner, M | 1 |
Deuchars, J; Deuchars, SA; Spary, E; Wang, L | 1 |
Baur, R; Kaur, KH; Sigel, E | 2 |
Chang, JL; Chen, MJ; Lin, TB; Lu, HT; Pan, SF; Peng, HY; Wu, HC | 1 |
Bonin, RP; De Koninck, Y; Eng, DG; Labrakakis, C; Orser, BA; Whissell, PD | 1 |
Cho, CH; Han, SK; Jeon, BH; Jeong, JA; Jo, JY; Kim, HW; Lee, SK; Lee, SY; Pandit, S; Park, JB; Ryu, PD; Stern, JE | 1 |
Cho, KH; Jang, HJ; Kim, MJ; Rhie, DJ; Yoon, SH | 1 |
Anton, F; Darbon, P; Hanesch, U; Juif, PÉ; Poisbeau, P; Zell, V | 1 |
Smart, TG; Villumsen, IS; Wellendorph, P | 1 |
Baur, R; Sigel, E; Wongsamitkul, N | 1 |
Endres, T; Lessmann, V; Meis, S; Munsch, T | 1 |
47 other study(ies) available for tetrahydrodeoxycorticosterone and gamma-aminobutyric acid
Article | Year |
---|---|
Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Gamma-aminobutyric acidA receptor complexes in rat frontal cortex and spinal cord show differential responses to steroid modulation.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Desoxycorticosterone; Diazepam; gamma-Aminobutyric Acid; Ionophores; Male; Pentobarbital; Pregnanediol; Pregnanolone; Rats; Rats, Inbred Strains; Receptors, GABA-A; Spinal Cord; Steroids; Sulfur Radioisotopes | 1991 |
Correlation between gamma-aminobutyric acidA receptor ligand-induced changes in t-butylbicyclophosphoro[35S]thionate binding and 36Cl- uptake in rat cerebrocortical membranes.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cerebral Cortex; Chloride Channels; Chlorides; Desoxycorticosterone; Diazepam; Ethanol; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Ligands; Membrane Proteins; Pentobarbital; Pregnanolone; Rats; Receptors, GABA-A; Synaptosomes | 1991 |
Studies on the mechanism of interactions between anesthetic steroids and gamma-aminobutyric acidA receptors.
Topics: Anesthetics; Animals; Chlorides; Desoxycorticosterone; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Nipecotic Acids; Pentobarbital; Pregnanolone; Progesterone; Proline; Rats; Receptors, GABA-A; Synaptic Membranes | 1990 |
Neurosteroids act on recombinant human GABAA receptors.
Topics: Benzodiazepines; Cell Line, Transformed; Cell Membrane Permeability; Chlorides; Desoxycorticosterone; Electric Conductivity; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Ion Channel Gating; Kidney; Membrane Potentials; Pentobarbital; Pregnanolone; Receptors, GABA-A; Recombinant Proteins; Transfection | 1990 |
The influence of estrus cycle on neurosteroid potency at the gamma-aminobutyric acidA receptor complex.
Topics: Animals; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Desoxycorticosterone; Estrus; Female; gamma-Aminobutyric Acid; Male; Pregnanolone; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sex Factors | 1993 |
Steroid inhibition of [3H]SR 95531 binding to the GABAA recognition site.
Topics: Allosteric Regulation; Androstanes; Animals; Azasteroids; Cell Membrane; Cerebral Cortex; Desoxycorticosterone; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Pregnanolone; Pregnenolone; Protein Binding; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA; Steroids | 1996 |
Influence of gender and brain region on neurosteroid modulation of GABA responses in rats.
Topics: Amygdala; Androgens; Androsterone; Animals; Brain; Cerebellum; Cerebral Cortex; Chlorides; Desoxycorticosterone; Dose-Response Relationship, Drug; Female; gamma-Aminobutyric Acid; Hippocampus; Male; Pregnanolone; Rats; Sex Characteristics | 1997 |
Neurosteroid prolongs GABAA channel deactivation by altering kinetics of desensitized states.
Topics: Age Factors; Animals; Anti-Anxiety Agents; Cerebellum; Desoxycorticosterone; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Ion Channel Gating; Kinetics; Organ Culture Techniques; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Sensitivity and Specificity; Taurine | 1997 |
Pre- and postsynaptic modulation of spinal GABAergic neurotransmission by the neurosteroid, 5 beta-pregnan-3 alpha-ol-20-one.
Topics: Anesthetics; Animals; Desoxycorticosterone; Electrophysiology; gamma-Aminobutyric Acid; Larva; Motor Neurons; Neural Inhibition; Neurotransmitter Agents; Pregnanediones; Pregnanes; Receptors, GABA-A; Spinal Cord; Synaptic Transmission; Tetrodotoxin; Xenopus laevis | 1997 |
Effects of PKC activation and receptor desensitization on neurosteroid modulation of GABA(A) receptors.
Topics: Animals; Anti-Anxiety Agents; Chloride Channels; Desoxycorticosterone; Enzyme Activation; Female; gamma-Aminobutyric Acid; Humans; Kinetics; Oocytes; Phorbol Esters; Pregnenolone; Protein Kinase C; Receptors, GABA-A; Recombinant Proteins; Staurosporine; Tetradecanoylphorbol Acetate; Xenopus laevis | 1997 |
Functional characterization and visualization of a GABAA receptor-GFP chimera expressed in Xenopus oocytes.
Topics: Anesthetics; Animals; Bicuculline; Cell Membrane; Desoxycorticosterone; Dose-Response Relationship, Drug; Electrophysiology; Female; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Gene Expression; Genes, Reporter; Green Fluorescent Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Indicators and Reagents; Ion Channel Gating; Luminescent Proteins; Membrane Potentials; Microscopy, Confocal; Midazolam; Oocytes; Pentobarbital; Picrotoxin; Receptors, GABA-A; Recombinant Fusion Proteins; Xenopus laevis | 1998 |
Absence seizures decrease steroid modulation of t-[35S]butylbicyclophosphorothionate binding in thalamic relay nuclei.
Topics: Action Potentials; Animals; Binding Sites; Bridged Bicyclo Compounds, Heterocyclic; Desoxycorticosterone; Epilepsy, Absence; gamma-Aminobutyric Acid; Hydroxybutyrates; Male; Pentobarbital; Pregnanediones; Rats; Rats, Sprague-Dawley; Sulfur Radioisotopes; Thalamic Nuclei | 1998 |
Steroid-inhibition of [3H]gamma-hydroxybutyric acid (GHB) binding in thalamic relay nuclei increases during absence seizures.
Topics: Anesthetics; Animals; Binding, Competitive; Cerebral Cortex; Desoxycorticosterone; Epilepsy, Absence; gamma-Aminobutyric Acid; Male; Neurons; Parietal Lobe; Pregnanediones; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Thalamus; Tritium; Up-Regulation | 1998 |
Bidirectional effects of the neuroactive steroid tetrahydrodeoxycorticosterone on GABA-activated Cl- currents in cultured rat hypothalamic neurons.
Topics: Animals; Cells, Cultured; Chloride Channels; Desoxycorticosterone; gamma-Aminobutyric Acid; Hypothalamus; Rats; Synapses | 1999 |
Differential modulation of the gamma-aminobutyric acid type C receptor by neuroactive steroids.
Topics: 5-alpha-Dihydroprogesterone; Animals; Anti-Inflammatory Agents; Desoxycorticosterone; gamma-Aminobutyric Acid; Humans; Oocytes; Patch-Clamp Techniques; Pregnanediones; Pregnanolone; Receptors, GABA; Receptors, Purinergic P1; Xenopus laevis | 1999 |
Interactive role for neurosteroids in ethanol enhancement of gamma-aminobutyric acid-gated currents from dissociated substantia nigra reticulata neurons.
Topics: Anesthetics; Animals; Cells, Cultured; Central Nervous System Depressants; Desoxycorticosterone; Electrophysiology; Ethanol; gamma-Aminobutyric Acid; Ion Channel Gating; Neurons; Patch-Clamp Techniques; Pregnanediones; Rats; Steroids; Substantia Nigra | 1999 |
Social isolation-induced decreases in both the abundance of neuroactive steroids and GABA(A) receptor function in rat brain.
Topics: Animals; Anxiety; Brain; Cerebral Cortex; Conflict, Psychological; Corticosterone; Dehydroepiandrosterone; Desoxycorticosterone; Electroshock; Female; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Male; Oocytes; Pregnanolone; Pregnenolone; Progesterone; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Social Isolation; Steroids; Synaptosomes; Time Factors; Xenopus laevis | 2000 |
Heterogeneity of hippocampal GABA(A) receptors: regulation by corticosterone.
Topics: Allosteric Regulation; Animals; Autoradiography; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Corticosterone; Dendrites; Desoxycorticosterone; Drug Implants; Flunitrazepam; gamma-Aminobutyric Acid; Hippocampus; Ligands; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA-A | 2001 |
Assembly of functional alpha6beta3gamma2delta GABA(A) receptors in vitro.
Topics: Affinity Labels; Anesthetics; Animals; Anticonvulsants; Azides; Benzodiazepines; Binding Sites; Cells, Cultured; Desoxycorticosterone; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Membrane Potentials; Muscimol; Protein Structure, Tertiary; Rats; Receptors, GABA-A; Transfection; Triazoles; Tritium | 2000 |
Enhanced neurosteroid potentiation of ternary GABA(A) receptors containing the delta subunit.
Topics: Allosteric Regulation; Animals; Cell Line; Desoxycorticosterone; Dose-Response Relationship, Drug; Fibroblasts; gamma-Aminobutyric Acid; Gene Expression; Humans; Ion Channel Gating; Kidney; Patch-Clamp Techniques; Protein Isoforms; Protein Subunits; Rats; Receptors, GABA-A; Transfection | 2002 |
Alpha1 and alpha6 subunits specify distinct desensitization, deactivation and neurosteroid modulation of GABA(A) receptors containing the delta subunit.
Topics: Amino Acid Sequence; Animals; Desoxycorticosterone; Electric Stimulation; Electrophysiology; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Isomerism; Membrane Potentials; Molecular Sequence Data; Neurotransmitter Agents; Patch-Clamp Techniques; Rats; Receptors, GABA-A; Recombinant Fusion Proteins; Recombinant Proteins | 2002 |
Intact synaptic GABAergic inhibition and altered neurosteroid modulation of thalamic relay neurons in mice lacking delta subunit.
Topics: Anesthetics; Animals; Desoxycorticosterone; Evoked Potentials; Female; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neural Inhibition; Neural Pathways; Pregnenolone; Receptors, GABA-A; Synapses; Thalamus | 2003 |
Neurosteroids shift partial agonist activation of GABA(A) receptor channels from low- to high-efficacy gating patterns.
Topics: Allosteric Regulation; beta-Alanine; Cell Line; Desoxycorticosterone; Fibroblasts; GABA Agonists; gamma-Aminobutyric Acid; Humans; Ion Channel Gating; Kidney; Mutagenesis, Site-Directed; Patch-Clamp Techniques; Receptors, GABA-A; Steroids; Taurine; Transfection | 2003 |
Rapid non-genomic effect of glucocorticoid metabolites and neurosteroids on the gamma-aminobutyric acid-A receptor.
Topics: Animals; Cerebral Cortex; Chlorides; Desoxycorticosterone; Dose-Response Relationship, Drug; Drug Interactions; gamma-Aminobutyric Acid; Glucocorticoids; Male; Neurons; Pregnanolone; Rats; Rats, Wistar; Receptors, GABA-A; Synaptosomes | 2005 |
High affinity, heterogeneous displacement of [3H]EBOB binding to cerebellar GABA A receptors by neurosteroids and GABA agonists.
Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Desoxycorticosterone; Dose-Response Relationship, Drug; Drug Interactions; GABA Agonists; gamma-Aminobutyric Acid; Hippocampus; Male; Pregnanolone; Protein Binding; Radioligand Assay; Rats; Rats, Wistar; Receptors, GABA-A | 2005 |
Neurosteroid modulation of recombinant rat alpha5beta2gamma2L and alpha1beta2gamma2L GABA(A) receptors in Xenopus oocyte.
Topics: Androstane-3,17-diol; Animals; Desoxycorticosterone; Dose-Response Relationship, Drug; Female; GABA Agonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Male; Membrane Potentials; Microinjections; Oocytes; Patch-Clamp Techniques; Pregnanediol; Pregnanes; Pregnenolone; Protein Subunits; Pyridines; Rats; Rats, Wistar; Receptors, GABA-A; RNA, Messenger; Steroids; Xenopus laevis; Zolpidem | 2006 |
GABAergic tonic inhibition of substantia gelatinosa neurons in mouse spinal cord.
Topics: Action Potentials; Anesthetics; Animals; Bicuculline; Desoxycorticosterone; Drug Interactions; Furosemide; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Mice; Neural Inhibition; Neurons; Patch-Clamp Techniques; Receptors, GABA-A; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sodium Potassium Chloride Symporter Inhibitors; Spinal Cord; Substantia Gelatinosa | 2006 |
Inhibition by alpha-tetrahydrodeoxycorticosterone (THDOC) of pre-sympathetic parvocellular neurones in the paraventricular nucleus of rat hypothalamus.
Topics: Action Potentials; Animals; Bicuculline; Desoxycorticosterone; Dose-Response Relationship, Drug; Drug Synergism; Female; GABA Antagonists; gamma-Aminobutyric Acid; Hypothalamus; Ion Channel Gating; Kinetics; Male; Neurons; Paraventricular Hypothalamic Nucleus; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, GABA-A; Sympathetic Nervous System; Synaptic Transmission | 2006 |
Rat alpha6beta2delta GABAA receptors exhibit two distinct and separable agonist affinities.
Topics: Action Potentials; Animals; beta-Alanine; Bicuculline; Crotonates; Desoxycorticosterone; Dose-Response Relationship, Drug; Female; Furosemide; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Imidazoles; Microinjections; Mutation; Neural Inhibition; Neurons; Oocytes; Picrotoxin; Pyridazines; Rats; Receptors, GABA-A; Sesterterpenes; Taurine; Xenopus laevis; Zinc | 2007 |
PKC activation sets an upper limit to the functional plasticity of GABAergic transmission induced by endogenous neurosteroids.
Topics: Alkaloids; Animals; Benzophenanthridines; Desoxycorticosterone; Drug Interactions; Enzyme Activation; Enzyme Inhibitors; Finasteride; GABA Agents; gamma-Aminobutyric Acid; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Interneurons; Isoquinolines; Membrane Potentials; Patch-Clamp Techniques; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Rats, Wistar; Spinal Cord; Steroids | 2007 |
alpha1beta2delta, a silent GABAA receptor: recruitment by tracazolate and neurosteroids.
Topics: Animals; Desoxycorticosterone; Dose-Response Relationship, Drug; Electrophysiology; gamma-Aminobutyric Acid; Gene Expression; Oocytes; Patch-Clamp Techniques; Protein Isoforms; Protein Subunits; Pyrazoles; Rats; Receptors, GABA-A; Xenopus laevis | 2008 |
Cell type-specific GABA A receptor-mediated tonic inhibition in mouse neocortex.
Topics: Anesthetics; Animals; Animals, Newborn; Desoxycorticosterone; Drug Interactions; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Isoxazoles; Mice; Neocortex; Neural Inhibition; Neurons; Patch-Clamp Techniques; Reaction Time; Receptors, GABA-A | 2008 |
GABAA receptor-mediated tonic currents in substantia gelatinosa neurons of rat spinal trigeminal nucleus pars caudalis.
Topics: Animals; Anti-Anxiety Agents; Desoxycorticosterone; Female; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Ion Channels; Male; Membrane Potentials; Neural Inhibition; Neurons; Organ Culture Techniques; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Glutamate; Receptors, Glycine; Substantia Gelatinosa; Synaptic Transmission; Trigeminal Caudal Nucleus | 2008 |
Neuroactive steroids and GABAA receptor plasticity in the brain of the WAG/Rij rat, a model of absence epilepsy.
Topics: Aging; Animals; Animals, Genetically Modified; Brain; Brain Chemistry; Cerebral Cortex; Desoxycorticosterone; Disease Models, Animal; Down-Regulation; Epilepsy, Absence; gamma-Aminobutyric Acid; Male; Neuronal Plasticity; Pregnanolone; Protein Subunits; Rats; Rats, Wistar; Receptors, GABA-A; Steroids; Stress, Psychological; Synapses; Synaptic Transmission; Thalamus; Up-Regulation | 2008 |
Etomidate, propofol and the neurosteroid THDOC increase the GABA efficacy of recombinant alpha4beta3delta and alpha4beta3 GABA A receptors expressed in HEK cells.
Topics: Cell Line, Transformed; Central Nervous System Depressants; Desoxycorticosterone; Dose-Response Relationship, Drug; Drug Synergism; Electric Stimulation; Ethanol; Etomidate; gamma-Aminobutyric Acid; Gene Expression; Humans; Hypnotics and Sedatives; Patch-Clamp Techniques; Propofol; Receptors, GABA-A; Recombinant Proteins; Transfection | 2009 |
Tonic GABAergic inhibition of sympathetic preganglionic neurons: a novel substrate for sympathetic control.
Topics: Anesthetics; Animals; Animals, Newborn; Autonomic Fibers, Preganglionic; Desoxycorticosterone; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Electric Stimulation; Female; GABA Agents; gamma-Aminobutyric Acid; Glycine Agents; In Vitro Techniques; Male; Membrane Potentials; Neural Inhibition; Neurons; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Rats; Sodium Channel Blockers; Strychnine; Tetrodotoxin | 2008 |
Unanticipated structural and functional properties of delta-subunit-containing GABAA receptors.
Topics: Animals; Anti-Anxiety Agents; Central Nervous System Depressants; Desoxycorticosterone; Dose-Response Relationship, Drug; Ethanol; GABA Agents; GABA Agonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Gene Expression; Humans; Oocytes; Protein Structure, Quaternary; Receptors, GABA-A; Recombinant Fusion Proteins; Structure-Activity Relationship; Xenopus; Zinc | 2009 |
Structure of alpha6 beta3 delta GABA(A) receptors and their lack of ethanol sensitivity.
Topics: Animals; Anti-Anxiety Agents; Biophysical Phenomena; Central Nervous System Depressants; Desoxycorticosterone; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Ethanol; GABA Agonists; gamma-Aminobutyric Acid; Isoxazoles; Membrane Potentials; Oocytes; Patch-Clamp Techniques; Protein Subunits; Receptors, GABA-A; Transfection; Xenopus | 2009 |
Acute neurosteroids inhibit the spinal reflex potentiation via GABAergic neurotransmission.
Topics: Action Potentials; Animals; Bicuculline; Desoxycorticosterone; Electric Stimulation; Electromyography; Female; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Injections, Spinal; Neuronal Plasticity; Neurotransmitter Agents; Pregnanolone; Progesterone; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Reflex; Spinal Nerves; Synaptic Transmission; Time Factors; Urethra | 2010 |
Pharmacological enhancement of δ-subunit-containing GABA(A) receptors that generate a tonic inhibitory conductance in spinal neurons attenuates acute nociception in mice.
Topics: Action Potentials; Analgesics; Anesthetics; Animals; Bicuculline; Desoxycorticosterone; Dose-Response Relationship, Drug; Electric Stimulation; Formaldehyde; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hindlimb Suspension; In Vitro Techniques; Isoxazoles; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neural Inhibition; Pain Measurement; Psychomotor Performance; Receptors, GABA-A; Sensory Receptor Cells; Spinal Cord | 2011 |
Neurosteroid modulation of benzodiazepine-sensitive GABAA tonic inhibition in supraoptic magnocellular neurons.
Topics: Animals; Benzodiazepines; Desoxycorticosterone; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Imidazoles; Inhibitory Postsynaptic Potentials; Male; Models, Animal; Neurons; Neurotransmitter Agents; Pregnanolone; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Supraoptic Nucleus | 2011 |
Layer- and cell-type-specific tonic GABAergic inhibition of pyramidal neurons in the rat visual cortex.
Topics: Animals; Desoxycorticosterone; Female; gamma-Aminobutyric Acid; Male; Neurons; Pyramidal Cells; Rats; Receptors, GABA-A; Visual Cortex | 2013 |
Corticosterone analgesia is mediated by the spinal production of neuroactive metabolites that enhance GABAergic inhibitory transmission on dorsal horn rat neurons.
Topics: Animals; Blood Chemical Analysis; Corticosterone; Desoxycorticosterone; gamma-Aminobutyric Acid; Microelectrodes; Neural Inhibition; Nociceptive Pain; Pain Measurement; Patch-Clamp Techniques; Physical Stimulation; Posterior Horn Cells; Radioimmunoassay; Rats; Receptors, GABA-A; Synaptic Transmission; Tissue Culture Techniques | 2015 |
Pharmacological characterisation of murine α4β1δ GABAA receptors expressed in Xenopus oocytes.
Topics: Animals; Cations, Divalent; Copper; Desoxycorticosterone; Dose-Response Relationship, Drug; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Mice; Oocytes; Patch-Clamp Techniques; Rats; Receptors, GABA-A; Xenopus laevis; Zinc | 2015 |
Toward Understanding Functional Properties and Subunit Arrangement of α4β2δ γ-Aminobutyric Acid, Type A (GABAA) Receptors.
Topics: Animals; Benzamides; Desoxycorticosterone; gamma-Aminobutyric Acid; Imidazoles; Rats; Receptors, GABA-A; Xenopus | 2016 |
Presynaptic Regulation of Tonic Inhibition by Neuromodulatory Transmitters in the Basal Amygdala.
Topics: Adrenergic alpha-1 Receptor Antagonists; Amygdala; Animals; Desoxycorticosterone; Fear; gamma-Aminobutyric Acid; Ion Channel Gating; Male; Memory; Mice, Inbred C57BL; Neural Inhibition; Neurons; Neurotransmitter Agents; Nicotine; Norepinephrine; Presynaptic Terminals; Serotonin | 2018 |