tetraethylammonium has been researched along with verapamil in 95 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 21 (22.11) | 18.7374 |
1990's | 40 (42.11) | 18.2507 |
2000's | 27 (28.42) | 29.6817 |
2010's | 7 (7.37) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Dresser, MJ; Giacomini, KM; Gray, AT; Terashita, S; Yost, SC; Zhang, L | 1 |
Giacomini, KM; Schaner, ME; Zhang, L | 1 |
Nezu, J; Oku, A; Sai, Y; Sakamoto, K; Shimane, M; Tamai, I; Tsuji, A; Yabuuchi, H | 1 |
Nezu, JI; Ohashi, R; Oku, A; Sai, Y; Shimane, M; Tamai, I; Tsuji, A; Yabuuchi, H | 1 |
Conway, SJ; Ganapathy, V; George, RL; Huang, W; Leibach, FH; Wang, H; Wu, X | 1 |
Desir, GV; Lang, R; Lee, G; Liu, W; Orias, M; Rafi, H; Segal, AS; Tian, S | 1 |
Blom-Roosemalen, MC; Breimer, DD; de Boer, AG; van der Sandt, IC | 1 |
Hashimoto, N; Nezu Ji, J; Nikaido, H; Ohashi, R; Oku, A; Sai, Y; Shimane, M; Tamai, I; Tsuji, A | 1 |
Arieff, Z; Bardien-Kruger, S; Brink, P; Chandy, KG; Corfield, V; Wulff, H | 1 |
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM | 1 |
Benet, LZ; Brouwer, KL; Chu, X; Dahlin, A; Evers, R; Fischer, V; Giacomini, KM; Hillgren, KM; Hoffmaster, KA; Huang, SM; Ishikawa, T; Keppler, D; Kim, RB; Lee, CA; Niemi, M; Polli, JW; Sugiyama, Y; Swaan, PW; Tweedie, DJ; Ware, JA; Wright, SH; Yee, SW; Zamek-Gliszczynski, MJ; Zhang, L | 1 |
Ahlin, G; Bergström, F; Bredberg, U; Fridén, M; Hammarlund-Udenaes, M; Rehngren, M; Wan, H | 1 |
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR | 1 |
Niu, GB; Pei, JM; Zang, YM; Zhou, SS; Zhu, MZ | 1 |
Haseley, TS; Hosford, M; Lesniak, ME; McKinney, TD; Scheller, MB | 1 |
Frank, C; Sagratella, S; Scotti de Carolis, A | 1 |
Ferrier, J; Richter, C | 1 |
Amigorena, S; Choquet, D; Fridman, WH; Korn, H; Teillaud, JL | 1 |
Felix, D; Hirt, A; Huwyler, T; Morell, A | 1 |
Carpenter, FG | 1 |
Dreyer, F; Penner, R | 1 |
Gupta, S | 1 |
Shuba, MF; Smirnov, SV | 1 |
Boutin, L; Derosiers, J; Schanne, OF | 1 |
Aubin, JE; Ferrier, J; Heersche, JN; Ward-Kesthely, A | 1 |
Gemba, M; Hori, M | 1 |
Wali, FA | 1 |
Mitchell, HW | 1 |
Ballerini, P; Caciagli, F; Ciccarelli, R; Di Iorio, P; Tacconelli, L | 1 |
Lambert, CR; Pepine, CJ | 1 |
Asano, T; Kasuya, Y; Shigenobu, K | 1 |
Lazcano, C; Marín, J; Recio, L; Salaices, M; Sanchez-Ferrer, CF | 1 |
Dascal, N; Landau, EM; Lass, Y | 1 |
Jamieson, DD; Lander, J | 1 |
Barták, F; Jezek, K; Králícek, P; Pucelík, P | 1 |
Atarashi, H; Elharrar, V; Surawicz, B | 1 |
Foster, RW; Okpalugo, BI; Small, RC | 1 |
Downing, OA; Louttit, JB; Wilson, KA | 1 |
Sperelakis, N; Zelcer, E | 1 |
Kawamura, A; Solaro, RJ; Wahler, GM | 1 |
Cook, DI; Hayashi, T; Hirono, C; Young, JA | 1 |
Miller, DS | 1 |
Cook, DI; Ishikawa, T | 1 |
Santos, DE; Takeuchi, H | 1 |
Renfro, JL; Sussman-Turner, C | 1 |
Fricker, G; Miller, DS; Schramm, U; Wenger, R | 1 |
Delbono, O; Kotsias, BA | 1 |
Ortiz-Miranda, SI; Pappone, PA | 1 |
Ito, Y; Takagi, K; Tomita, T | 1 |
Cheng, PM; Donnelly, DF | 1 |
Lopatin, AN; Nichols, CG; Romano, C; Sha, Q | 1 |
Ağar, E; Green, GG; Sanders, DJ | 1 |
Irimajiri, A; Kakigi, A; Saito, H; Takeda, T; Takeuchi, S | 1 |
García-Segoviano, JA; Naranjo-Rodríguez, EB; Prieto-Gómez, B; Reyes-Vázquez, C; Trujillo-Santana, JT | 1 |
Das, P; Schurman, DJ; Smith, RL | 1 |
Hu, Q; Huang, F; Shi, Y | 1 |
Eusebi, F; Giovannelli, A; Lorenzon, P; Ragozzino, D; Ruzzier, F | 1 |
Dantzler, WH; Kim, YK | 1 |
Advenier, C; Bessard, G; Corompt, E; Devillier, P; Lantuejoul, S; Naline, E | 1 |
Ando, M; Takeuchi, S | 2 |
Kang, BS; Lee, YH; Seo, JH | 1 |
Atchison, WD; Hewett, SJ; Xu, YF | 1 |
Duff, HJ; Exner, DV; Feng, ZP; Geonzon, R; Wang, L; Woodman, RC | 1 |
Miller, DS; Pritchard, JB; Villalobos, AR | 1 |
Clauss, W; Heinke, B | 1 |
Adams, DJ; Catacuzzeno, L; Franciolini, F; Hogg, RC; Petris, A; Trequattrini, C | 1 |
Catacuzzeno, L; Franciolini, F; Petris, A; Trequattrini, C | 1 |
Hein, W; Wohlrab, D | 1 |
Kostyuk, PG; Lemonnier, L; Mauroy, B; Prevarskaya, N; Shuba, YM; Skryma, R; Van Coppenolle, F | 1 |
Le Bourhis, X; Legrand, G; Lemonnier, L; Prevarskaya, N; Rybalchenko, V; Skryma, R; Van Coppenolle, F | 1 |
Cosgrove, DJ; Spalding, EP | 1 |
Tyerman, SD; Zhang, WH | 1 |
Chang, JP; Johnson, JD; Kwong, P; Wong, CJ; Yunker, WK | 1 |
Krüger, T; Lebek, S; Reichel, H; Wohlrab, D | 1 |
Chan, CB; Joseph, JW; MacDonald, PE; Sakellaropoulos, G; Salapatek, AM; Saleh, MC; Sewing, S; Smukler, SR; Tsushima, RG; Wang, J; Wheeler, MB | 1 |
Andrinolo, D; Fraga, S; Gomes, P; Lagos, N; Soares-da-Silva, P | 1 |
Davenport, RJ; White, PJ | 1 |
Diss, JK; Djamgoz, MB; Dolly, JO; Fraser, SP; Grimes, JA; Stewart, D | 1 |
Darling, IM; Kamath, AV; Morris, ME | 1 |
Besson, P; Le Guennec, JY; Roger, S | 1 |
O'Donnell, MJ; Rheault, MR | 1 |
Dohgu, S; Higuchi, S; Katamine, S; Kataoka, Y; Naito, M; Niwa, M; Sawada, Y; Shirabe, S; Takata, F; Tsuruo, T; Yamauchi, A | 1 |
Gorji, A; Köhling, R; Rüschenschmidt, C; Siep, E; Speckmann, EJ; Straub, H | 1 |
Dorange, G; Droguet, M; Gioux, M; Giroux-Metgès, MA; Pennec, JP; Talarmin, H | 1 |
Fukami, T; Furuishi, T; Moriki, Y; Suzuki, T; Tomono, K; Watanabe, J | 1 |
Leader, JP; O'Donnell, MJ | 1 |
Cao, LH; Choi, DH; Kang, DG; Kim, JS; Kim, SJ; Lee, H; Lee, HS; Lee, JK | 1 |
Kato, Y; Kubo, Y; Sugiura, T; Tsuji, A | 1 |
Bendhack, LM; Rocha, ML | 1 |
Hayashi, M; Kishimoto, H; Takizawa, Y; Tomita, M | 1 |
Bieger, D; Ford, CA; Tabrizchi, R | 1 |
Kaddoumi, A; Mohamed, LA | 1 |
Fukui, T; Iwai, H; Juge, N; Kawakami, M; Miyaji, T; Moriyama, S; Moriyama, Y; Nelson, N; Omote, H | 1 |
Lucetti, LT; Magalhães, PJ; Ribeiro-Filho, HV; Vasconcelos, TB | 1 |
1 review(s) available for tetraethylammonium and verapamil
Article | Year |
---|---|
Membrane transporters in drug development.
Topics: Animals; Computer Simulation; Decision Trees; Drug Approval; Drug Discovery; Drug Evaluation, Preclinical; Drug Interactions; Humans; Membrane Transport Proteins; Mice; Mice, Knockout; Prescription Drugs | 2010 |
94 other study(ies) available for tetraethylammonium and verapamil
Article | Year |
---|---|
Cloning and functional expression of a human liver organic cation transporter.
Topics: Amino Acid Sequence; Animals; Base Sequence; Carrier Proteins; Cloning, Molecular; DNA, Complementary; Humans; Liver; Membrane Proteins; Molecular Sequence Data; Oocytes; Organic Cation Transporter 1; Polymerase Chain Reaction; Rats; RNA, Messenger; Sequence Homology, Amino Acid; Species Specificity; Tissue Distribution; Xenopus laevis | 1997 |
Functional characterization of an organic cation transporter (hOCT1) in a transiently transfected human cell line (HeLa).
Topics: Carrier Proteins; Corticosterone; HeLa Cells; Humans; Membrane Proteins; Midazolam; Organic Cation Transporter 1; Permeability; Recombinant Proteins; Structure-Activity Relationship; Tetraethylammonium Compounds; Transfection | 1998 |
Novel membrane transporter OCTN1 mediates multispecific, bidirectional, and pH-dependent transport of organic cations.
Topics: Animals; Biological Transport, Active; Carrier Proteins; Cell Line; Gene Expression; Humans; Hydrogen-Ion Concentration; Membrane Potentials; Membrane Proteins; Membrane Transport Proteins; Oocytes; Organic Cation Transport Proteins; Quinidine; RNA, Messenger; Symporters; Tetraethylammonium Compounds; Xenopus laevis | 1999 |
Na(+)-dependent carnitine transport by organic cation transporter (OCTN2): its pharmacological and toxicological relevance.
Topics: Biological Transport, Active; Carnitine; Carrier Proteins; Cations; Cells, Cultured; Dose-Response Relationship, Drug; Embryo, Mammalian; Humans; Hydrogen-Ion Concentration; Kidney; Membrane Proteins; Organic Cation Transport Proteins; Sodium; Solute Carrier Family 22 Member 5; Stereoisomerism | 1999 |
Structural and functional characteristics and tissue distribution pattern of rat OCTN1, an organic cation transporter, cloned from placenta.
Topics: Amino Acid Sequence; Animals; Base Sequence; Carnitine; Carrier Proteins; Cloning, Molecular; DNA, Complementary; Humans; Membrane Proteins; Membrane Transport Proteins; Molecular Sequence Data; Organic Cation Transport Proteins; Placenta; Rats; RNA, Messenger; Solute Carrier Proteins; Structure-Activity Relationship; Symporters; Tetraethylammonium; Tissue Distribution | 2000 |
KCNA10: a novel ion channel functionally related to both voltage-gated potassium and CNG cation channels.
Topics: Animals; Base Sequence; Cyclic Nucleotide-Gated Cation Channels; DNA Primers; Female; Humans; In Vitro Techniques; Ion Channel Gating; Ion Channels; Membrane Potentials; Oocytes; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Voltage-Gated; Rabbits; Recombinant Proteins; Second Messenger Systems; Shaker Superfamily of Potassium Channels; Xenopus laevis | 2000 |
Specificity of doxorubicin versus rhodamine-123 in assessing P-glycoprotein functionality in the LLC-PK1, LLC-PK1:MDR1 and Caco-2 cell lines.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Caco-2 Cells; Cell Line; Cell Polarity; Cimetidine; Cyclosporine; Doxorubicin; Drug Resistance, Multiple; Epithelial Cells; Humans; Kinetics; LLC-PK1 Cells; Rhodamine 123; Swine; Tumor Cells, Cultured; Verapamil | 2000 |
Molecular and physiological evidence for multifunctionality of carnitine/organic cation transporter OCTN2.
Topics: Animals; Biological Transport; Carbon Radioisotopes; Carnitine; Carrier Proteins; Cells, Cultured; Embryo, Mammalian; Fibroblasts; Humans; Male; Membrane Proteins; Mice; Mice, Inbred C3H; Organic Cation Transport Proteins; Solute Carrier Family 22 Member 5; Tetraethylammonium; Tissue Distribution; Tritium | 2001 |
Characterisation of the human voltage-gated potassium channel gene, KCNA7, a candidate gene for inherited cardiac disorders, and its exclusion as cause of progressive familial heart block I (PFHBI).
Topics: Amino Acid Sequence; Animals; Base Sequence; Cloning, Molecular; COS Cells; DNA; Heart Block; Heart Diseases; Humans; Mice; Molecular Sequence Data; Potassium Channels; Potassium Channels, Voltage-Gated; Shaker Superfamily of Potassium Channels; Trinucleotide Repeats | 2002 |
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship | 2008 |
Measurement of unbound drug exposure in brain: modeling of pH partitioning explains diverging results between the brain slice and brain homogenate methods.
Topics: Animals; Biological Transport; Brain; Chemical Phenomena; Dialysis; Hydrogen-Ion Concentration; In Vitro Techniques; Lysosomes; Male; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Tissue Distribution | 2011 |
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection | 2012 |
[Effects of tetraethylammonium chloride and verapamil on the effective refractory period of ischemic myocardium in rabbits].
Topics: Animals; Female; Male; Myocardial Ischemia; Rabbits; Refractory Period, Electrophysiological; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil | 1992 |
Basolateral transport of tetraethylammonium by a clone of LLC-PK1 cells.
Topics: Animals; Basement Membrane; Biological Transport, Active; Cimetidine; Clone Cells; Kidney; Kinetics; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil | 1992 |
Effects of calcium and potassium extracellular ionic concentration changes on the hippocampal CA1 activity of purinergic drugs.
Topics: 4-Aminopyridine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Calcium; Cesium; Chlorides; Evoked Potentials; Hippocampus; In Vitro Techniques; Male; Phenylisopropyladenosine; Potassium; Rats; Rats, Inbred Strains; Receptors, Purinergic; Synapses; Synaptic Transmission; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil | 1991 |
Continuously active sodium channels in osteoblastic ROS 17/2.8 cells.
Topics: Animals; Calcium; Conductometry; Membrane Potentials; Nifedipine; Osteoblasts; Osteosarcoma; Rats; Sodium; Sodium Channels; Tetraethylammonium; Tetraethylammonium Compounds; Tumor Cells, Cultured; Verapamil | 1991 |
Ion channel blockers inhibit B cell activation at a precise stage of the G1 phase of the cell cycle. Possible involvement of K+ channels.
Topics: 4-Aminopyridine; Animals; Antibodies, Monoclonal; B-Lymphocytes; Cell Cycle; Electric Conductivity; Lipopolysaccharides; Lymphocyte Activation; Mice; Potassium Channels; Quaternary Ammonium Compounds; Quinine; Tetraethylammonium; Tetraethylammonium Compounds; Thymidine; Time Factors; Verapamil | 1990 |
Effect of cations and cation channel blockers on human natural killer cells.
Topics: Anesthetics, Local; Calcium; Cytotoxicity, Immunologic; Dose-Response Relationship, Immunologic; Humans; Ion Channels; Killer Cells, Natural; Magnesium; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Verapamil | 1985 |
Potentiation of nerve-induced bladder contractions after calcium channel blockade.
Topics: Animals; Calcium; Carbachol; Elasticity; Ion Channels; Male; Muscle Contraction; Muscle, Smooth; Potassium; Rats; Stimulation, Chemical; Tetraethylammonium; Tetraethylammonium Compounds; Urinary Bladder; Verapamil | 1985 |
Two different presynaptic calcium currents in mouse motor nerve terminals.
Topics: 4-Aminopyridine; Amifampridine; Aminopyridines; Animals; Barium; Cadmium; Calcium; Diltiazem; In Vitro Techniques; Ion Channels; Kinetics; Manganese; Mice; Motor Neurons; Neuromuscular Junction; Potassium; Strontium; Synapses; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil | 1986 |
Autologous mixed-lymphocyte reaction in man. XVII. In vitro effect of ion channel-blocking agents on the autologous mixed-lymphocyte response.
Topics: 4-Aminopyridine; Aminopyridines; Dose-Response Relationship, Drug; Humans; Interleukin-2; Ion Channels; Lymphocyte Activation; Lymphocyte Culture Test, Mixed; Quaternary Ammonium Compounds; Quinine; Receptors, Immunologic; Receptors, Interleukin-2; Recombinant Proteins; T-Lymphocytes; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil | 1987 |
Potential-dependent calcium inward current in a single isolated smooth muscle cell of the guinea-pig taenia caeci.
Topics: Action Potentials; Animals; Calcium; Cesium; Guinea Pigs; In Vitro Techniques; Ion Channels; Kinetics; Muscle, Smooth; Potassium; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil | 1986 |
Effects of K-channel blockers, calcium, and verapamil suggest different pacemaker mechanisms in cultured neonatal rat and embryonic chick ventricle cells.
Topics: Animals; Calcium; Cells, Cultured; Cesium; Chick Embryo; Heart Rate; Heart Ventricles; Membrane Potentials; Potassium Channels; Rats; Rats, Inbred Strains; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil | 1989 |
Membrane potential changes, cAMP stimulation and contraction in osteoblast-like UMR 106 cells in response to calcitonin and parathyroid hormone.
Topics: Animals; Bucladesine; Calcimycin; Calcitonin; Cell Line; Dinoprostone; Isoproterenol; Membrane Potentials; Osteoblasts; Parathyroid Hormone; Potassium Channels; Quinine; Rats; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil | 1988 |
Effect of barium ion on p-aminohippurate transport in basolateral membrane vesicles isolated from rat kidney cortex.
Topics: Acid Phosphatase; Alkaline Phosphatase; Aminohippuric Acids; Animals; Barium; Biological Transport, Active; Cations; Glucose-6-Phosphatase; In Vitro Techniques; Kidney Cortex; L-Lactate Dehydrogenase; Male; Membranes; Onium Compounds; p-Aminohippuric Acid; Rats; Rats, Inbred Strains; Sodium-Potassium-Exchanging ATPase; Succinate Dehydrogenase; Tetraethylammonium; Tetraethylammonium Compounds; Trityl Compounds; Verapamil | 1985 |
Interaction of verapamil with d-tubocurarine and cholinergic agonists at the avian neuromuscular junction.
Topics: Acetylcholine; Animals; Chickens; Drug Interactions; In Vitro Techniques; Neuromuscular Junction; Synaptic Transmission; Tetraethylammonium; Tetraethylammonium Compounds; Tubocurarine; Verapamil | 1987 |
Electromechanical effects of tetraethylammonium and K+ on histamine-induced contraction in pig isolated tracheal smooth muscle.
Topics: Acetylcholine; Airway Resistance; Animals; Calcium; Histamine; Histamine Antagonists; In Vitro Techniques; Potassium; Sucrose; Swine; Tetraethylammonium; Tetraethylammonium Compounds; Trachea; Verapamil | 1987 |
Cultures of glial cells release purines under field electrical stimulation: the possible ionic mechanisms.
Topics: Adenosine; Adenosine Deaminase Inhibitors; Animals; Animals, Newborn; Brain; Cells, Cultured; Coformycin; Electric Stimulation; Neuroglia; Nucleotides; Pentostatin; Pharmacology; Rats; Reference Values; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Verapamil | 1988 |
Tetraethylammonium-induced phasic arterial constriction: temporal and spatial characteristics.
Topics: Animals; Dogs; Femoral Artery; Physiology; Tetraethylammonium; Tetraethylammonium Compounds; Time Factors; Vasoconstriction; Verapamil | 1986 |
TEA prevents the decline of the duration of the action potential in hypoxic cardiac muscle.
Topics: Action Potentials; Animals; Calcimycin; Calcium Chloride; Guinea Pigs; Heart; Hypoxia; In Vitro Techniques; Male; Myocardial Contraction; Tetraethylammonium; Tetraethylammonium Compounds; Time Factors; Verapamil | 1985 |
Effect of tetraethylammonium and verapamil on noradrenaline release induced by field electrical stimulation and potassium from cat cerebral and femoral arteries.
Topics: Animals; Calcium; Cats; Cerebral Arteries; Electric Stimulation; Female; Femoral Artery; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Norepinephrine; Potassium; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Verapamil | 1985 |
Xenopus oocyte resting potential, muscarinic responses and the role of calcium and guanosine 3',5'-cyclic monophosphate.
Topics: Acetylcholine; Action Potentials; Animals; Calcium; Cell Membrane Permeability; Chlorides; Cyclic GMP; Female; In Vitro Techniques; Membrane Potentials; Oocytes; Ouabain; Potassium; Sodium; Tetraethylammonium; Tetraethylammonium Compounds; Time Factors; Verapamil; Xenopus laevis | 1984 |
Investigation of the mode of action of the anaesthetic agent, ketamine, in the heart of the bivalve mollusc Tapes watlingi.
Topics: Acetylcholine; Amphetamine; Animals; Dose-Response Relationship, Drug; Heart; Heart Rate; Ketamine; Methysergide; Metoclopramide; Mollusca; Phentolamine; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil | 1984 |
An analysis of the postnatal development of the action potential repolarization process in the working ventricular myocardium of albino rats (effect of tea, frequency, verapamil and adrenaline).
Topics: Action Potentials; Age Factors; Animals; Animals, Newborn; Calcium; Electric Stimulation; Epinephrine; Female; Heart; Heart Ventricles; Ion Channels; Male; Myocardial Contraction; Potassium; Rats; Rats, Inbred Strains; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil | 1983 |
Cycle length-dependent action potential duration in canine cardiac Purkinje fibers.
Topics: Action Potentials; Animals; Cobalt; Dogs; Female; Heart Conduction System; Homeostasis; In Vitro Techniques; Isoproterenol; Kinetics; Lidocaine; Male; Purkinje Fibers; Reaction Time; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Verapamil | 1984 |
Antagonism of Ca2+ and other actions of verapamil in guinea-pig isolated trachealis.
Topics: Acetylcholine; Action Potentials; Airway Resistance; Animals; Calcium Channel Blockers; Dinoprostone; Electrophysiology; Female; Guinea Pigs; Histamine; In Vitro Techniques; Male; Potassium Chloride; Prostaglandins E; Tetraethylammonium; Tetraethylammonium Compounds; Trachea; Verapamil | 1984 |
Differential effects of strychnine on two types of vascular muscle.
Topics: 4-Aminopyridine; Aminopyridines; Animals; Aorta, Thoracic; Cardiovascular Agents; Male; Muscle Contraction; Muscle, Smooth, Vascular; Portal Vein; Prazosin; Rats; Rats, Inbred Strains; Strychnine; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Verapamil | 1984 |
Angiotensin induction of active responses in cultured reaggregates of rat aortic smooth muscle cells.
Topics: Angiotensin II; Animals; Aorta, Thoracic; Barium; Barium Compounds; Cell Aggregation; Cells, Cultured; Chlorides; Electric Stimulation; Electrophysiology; Male; Membrane Potentials; Muscle, Smooth, Vascular; Rats; Rats, Inbred Strains; Sodium; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil | 1981 |
RWJ-24517, a positive inotropic agent, has novel effects on action potentials in guinea pig myocardium.
Topics: Actin Cytoskeleton; Action Potentials; Adenosine Triphosphatases; Animals; Cardiotonic Agents; Dose-Response Relationship, Drug; Electrophysiology; Female; Guinea Pigs; Male; Mercaptopurine; Papillary Muscles; Piperazines; Potassium Channel Blockers; Sodium Channels; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil | 1993 |
The ACh-induced whole-cell currents in sheep parotid secretory cells. Do BK channels really carry the ACh-evoked whole-cell K+ current?
Topics: 4-Aminopyridine; Acetylcholine; Animals; Barium; Cell Membrane; Chlorides; Parotid Gland; Patch-Clamp Techniques; Potassium; Potassium Channel Blockers; Potassium Channels; Quinidine; Quinine; Sensitivity and Specificity; Sheep; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil | 1995 |
Daunomycin secretion by killfish renal proximal tubules.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Buffers; Cyclosporine; Daunorubicin; Hydrogen-Ion Concentration; Image Processing, Computer-Assisted; Kidney Tubules, Proximal; Killifishes; Microscopy, Fluorescence; Television; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil | 1995 |
Effects of K+ channel blockers on inwardly and outwardly rectifying whole-cell K+ currents in sheep parotid secretory cells.
Topics: Animals; Barium; Cesium; Charybdotoxin; In Vitro Techniques; Lidocaine; Membrane Potentials; Parotid Gland; Potassium; Potassium Channels; Quinidine; Quinine; Scorpion Venoms; Sheep; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil | 1993 |
Influence of the drugs for membrane excitability modification on the excitation caused by achatin-I.
Topics: Amino Acid Sequence; Animals; Concanavalin A; Drug Interactions; Ion Channels; Membrane Potentials; Molecular Sequence Data; Neurons; Neuropeptides; Picrotoxin; Snails; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Tyrosine; Verapamil | 1993 |
Heat-shock-stimulated transepithelial daunomycin secretion by flounder renal proximal tubule primary cultures.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cells, Cultured; Cycloheximide; Cyclosporine; Daunorubicin; Epithelial Cells; Epithelium; Flounder; Hot Temperature; Immunohistochemistry; Kidney Tubules, Proximal; Kinetics; Microvilli; p-Aminohippuric Acid; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil; Vinblastine | 1995 |
P-glycoprotein-mediated secretion of a fluorescent cyclosporin analogue by teleost renal proximal tubules.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cyclosporine; Fluorescent Dyes; Kidney Tubules, Proximal; Killifishes; Kinetics; Microscopy, Fluorescence; p-Aminohippuric Acid; Potassium Cyanide; Quinine; Tetraethylammonium; Tetraethylammonium Compounds; Time Factors; Verapamil; Vinblastine | 1995 |
Effect of aminophylline-Ca2+ blocker interaction on membrane potential of rat diaphragm fibers.
Topics: Aminophylline; Animals; Apamin; Diaphragm; Drug Interactions; In Vitro Techniques; Membrane Potentials; Nifedipine; Rats; Rats, Wistar; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil | 1993 |
Blockers of voltage-gated K channels inhibit proliferation of cultured brown fat cells.
Topics: Adipose Tissue, Brown; Animals; Animals, Newborn; Calcium; Cell Division; Cells, Cultured; Kinetics; Membrane Potentials; Nifedipine; Norepinephrine; Potassium Channels; Quinine; Rats; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil | 1993 |
Relaxant actions of isoprenaline on guinea-pig isolated tracheal smooth muscle.
Topics: Adrenergic beta-Agonists; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Female; Guinea Pigs; In Vitro Techniques; Indoles; Isoproterenol; Male; Membrane Potentials; Muscle Relaxation; Muscle Tonus; Muscle, Smooth; Potassium Channels; Tetraethylammonium; Tetraethylammonium Compounds; Trachea; Verapamil | 1995 |
Relationship between changes of glomus cell current and neural response of rat carotid body.
Topics: Afferent Pathways; Animals; Apamin; Carotid Body; Cell Hypoxia; Charybdotoxin; Membrane Potentials; Neural Inhibition; Patch-Clamp Techniques; Potassium Channels; Rats; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil | 1995 |
Spermidine release from xenopus oocytes. Electrodiffusion through a membrane channel.
Topics: Animals; Calcium; Cells, Cultured; Diffusion; Female; Kinetics; Oocytes; Patch-Clamp Techniques; Potassium; Potassium Channels; Recombinant Proteins; Spermidine; Tetraethylammonium; Tetraethylammonium Compounds; Tritium; Verapamil; Xenopus laevis | 1996 |
Membrane properties of complex spike firing neurons of the mouse dorsal cochlear nucleus in vitro.
Topics: 4-Aminopyridine; Action Potentials; Animals; Auditory Pathways; Calcium Channel Blockers; Cochlear Nucleus; In Vitro Techniques; Mice; Mice, Inbred BALB C; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Verapamil | 1996 |
Intravascularly applied K(+)-channel blockers suppress differently the positive endocochlear potential maintained by vascular perfusion.
Topics: Analgesics, Non-Narcotic; Animals; Barium; Calcium Channel Blockers; Cerebellum; Cochlear Microphonic Potentials; Guinea Pigs; Potassium Channel Blockers; Quinine; Stria Vascularis; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil | 1996 |
Apamin blocks the direct relaxant effect of melatonin on rat ileal smooth muscle.
Topics: 4-Aminopyridine; Adrenergic alpha-Antagonists; Animals; Apamin; Calcium; Calcium Channel Blockers; Carbachol; Cholinergic Antagonists; Glyburide; Hexamethonium; Humans; Ileum; Male; Melatonin; Muscarinic Antagonists; Muscle Contraction; Neuromuscular Depolarizing Agents; Nitrendipine; Phentolamine; Rats; Rats, Wistar; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Verapamil | 1997 |
Nitric oxide and G proteins mediate the response of bovine articular chondrocytes to fluid-induced shear.
Topics: Animals; Calcium Channel Blockers; Cartilage, Articular; Cattle; Enzyme Inhibitors; Glycosaminoglycans; GTP-Binding Proteins; Neomycin; Nitric Oxide; Nitric Oxide Synthase; omega-N-Methylarginine; Ornithine; Pertussis Toxin; Protein Synthesis Inhibitors; Signal Transduction; Stress, Mechanical; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil; Virulence Factors, Bordetella; Weight-Bearing | 1997 |
Inhibition of Toosendanin on the delayed rectifier potassium current in neuroblastoma x glioma NG108-15 cells.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Delayed Rectifier Potassium Channels; Dose-Response Relationship, Drug; Drugs, Chinese Herbal; Glioma; Hybrid Cells; Mice; Neuroblastoma; Neuromuscular Blocking Agents; Nifedipine; Patch-Clamp Techniques; Potassium; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Voltage-Gated; Rats; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil | 1997 |
Spontaneous and repetitive calcium transients in C2C12 mouse myotubes during in vitro myogenesis.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenosine Triphosphate; Animals; Apamin; Caffeine; Calcium; Cell Differentiation; Cell Line; Cytosol; Egtazic Acid; Kinetics; Membrane Potentials; Mice; Microscopy, Confocal; Microscopy, Video; Muscle, Skeletal; Oscillometry; Potassium Chloride; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Verapamil | 1997 |
Ca2+ and Ba2+ effects on basolateral tetraethylammonium transport in isolated snake renal proximal tubules.
Topics: Animals; Barium; Biological Transport; Calcium; Colubridae; Egtazic Acid; Kidney Tubules, Proximal; Lanthanum; Membrane Potentials; Tetraethylammonium; Tritium; Verapamil | 1997 |
Inhibitory effects of large Ca2+-activated K+ channel blockers on beta-adrenergic- and NO-donor-mediated relaxations of human and guinea-pig airway smooth muscles.
Topics: Adrenergic beta-Agonists; Adult; Aged; Aged, 80 and over; Albuterol; Animals; Benzimidazoles; Bronchi; Calcium; Calcium Channel Blockers; Charybdotoxin; Guinea Pigs; Humans; Male; Middle Aged; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nitric Oxide; Nitroprusside; Peptides; Potassium Channels; Tetraethylammonium; Vasodilator Agents; Verapamil | 1998 |
Inwardly rectifying K+ currents in intermediate cells in the cochlea of gerbils: a possible contribution to the endocochlear potential.
Topics: 4-Aminopyridine; Animals; Barium; Cadmium; Cesium; Cochlear Microphonic Potentials; Endolymph; Gerbillinae; Ion Transport; Models, Neurological; Nerve Tissue Proteins; Patch-Clamp Techniques; Potassium; Potassium Channels; Potassium Channels, Inwardly Rectifying; Quinine; Stria Vascularis; Tetraethylammonium; Verapamil | 1998 |
Effects of hypoxia on pulmonary vascular contractility.
Topics: Animals; Blood Vessels; Calcium Channel Blockers; Cyclooxygenase Inhibitors; Enzyme Inhibitors; Hypoxia; Indomethacin; Nitroarginine; Pulmonary Circulation; Rats; Tetraethylammonium; Vasoconstriction; Verapamil | 1998 |
Passive transfer of Lambert-Eaton myasthenic syndrome induces dihydropyridine sensitivity of ICa in mouse motor nerve terminals.
Topics: Animals; Autoantibodies; Binding, Competitive; Calcium; Calcium Channel Blockers; Dihydropyridines; Immunization, Passive; Lambert-Eaton Myasthenic Syndrome; Male; Mice; Mice, Inbred ICR; Motor Neurons; Nifedipine; omega-Agatoxin IVA; omega-Conotoxins; Peptides; Plasma; Potassium Channel Blockers; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Spider Venoms; Synaptosomes; Tetraethylammonium; Verapamil | 1998 |
A high affinity binding site for [3H]-Dofetilide on human leukocytes.
Topics: Animals; Anti-Arrhythmia Agents; Binding Sites; Charybdotoxin; Guinea Pigs; Humans; Kinetics; Leukocytes; Neuropeptides; Neutrophils; Phenethylamines; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Voltage-Gated; Shaw Potassium Channels; Sulfonamides; Tetraethylammonium; Verapamil | 1998 |
Organic cation transport in rat choroid plexus cells studied by fluorescence microscopy.
Topics: Animals; Animals, Newborn; Biological Transport; Cations; Choroid Plexus; Kinetics; Microscopy, Confocal; Microscopy, Fluorescence; Monensin; Neurons; Potassium Cyanide; Quinacrine; Rats; Rats, Inbred F344; Tetraethylammonium; Verapamil; Video Recording | 1999 |
Potassium conductances in isolated single cells from Xenopus laevis colonic epithelium.
Topics: Animals; Barium; Cesium; Colon; Epithelial Cells; Female; Hydrogen-Ion Concentration; Ion Transport; Lidocaine; Membrane Potentials; Patch-Clamp Techniques; Potassium; Potassium Channel Blockers; Potassium Channels; Quinidine; Quinine; Tetraethylammonium; Verapamil; Xenopus laevis | 1999 |
Mechanisms of verapamil inhibition of action potential firing in rat intracardiac ganglion neurons.
Topics: 4-Aminopyridine; Acetylcholine; Action Potentials; Animals; Animals, Newborn; Apamin; Cells, Cultured; Charybdotoxin; Electric Stimulation; Ganglia, Parasympathetic; Heart; Membrane Potentials; Muscarine; Neurons; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Rats; Tetraethylammonium; Verapamil | 1999 |
Mechanism of verapamil block of a neuronal delayed rectifier K channel: active form of the blocker and location of its binding domain.
Topics: Animals; Binding Sites; Binding, Competitive; Biotransformation; Calcium Channel Blockers; Chick Embryo; Electrophysiology; Gallopamil; Ganglia, Spinal; Kinetics; Neurons; Potassium Channel Blockers; Potassium Channels; Tetraethylammonium; Verapamil | 1999 |
Voltage-dependent outward K(+) current in intermediate cell of stria vascularis of gerbil cochlea.
Topics: Animals; Barium; Calcium; Electric Conductivity; Electrophysiology; Patch-Clamp Techniques; Potassium; Potassium Channel Blockers; Potassium Channels; Quinine; Stria Vascularis; Tetraethylammonium; Verapamil | 1999 |
[Effect of ion channel modulators on the membrane potential of human chondrocytes].
Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4-Aminopyridine; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Cell Division; Cells, Cultured; Chondrocytes; Flow Cytometry; Humans; Ion Channels; Membrane Potentials; Tetraethylammonium; Verapamil | 2000 |
Volume-regulated chloride conductance in the LNCaP human prostate cancer cell line.
Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; 8-Bromo Cyclic Adenosine Monophosphate; Adenosine Triphosphate; Anions; Calcium; Calcium Channel Blockers; Carcinoma; Cell Membrane Permeability; Chloride Channels; Electric Stimulation; Humans; Hypotonic Solutions; Ion Transport; Male; Membrane Potentials; Nitrobenzoates; Patch-Clamp Techniques; Potassium; Prostatic Neoplasms; Protein-Tyrosine Kinases; Substrate Specificity; Tetraethylammonium; Tumor Cells, Cultured; Verapamil | 2000 |
Verapamil inhibits proliferation of LNCaP human prostate cancer cells influencing K+ channel gating.
Topics: Antineoplastic Agents; Binding Sites; Binding, Competitive; Calcium Channel Blockers; Cell Division; Dose-Response Relationship, Drug; Electrophysiology; Humans; Male; Potassium Channel Blockers; Potassium Channels; Prostatic Neoplasms; Tetraethylammonium; Tumor Cells, Cultured; Verapamil | 2001 |
Mechanism of blue-light-induced plasma-membrane depolarization in etiolated cucumber hypocotyls.
Topics: Adenosine Triphosphate; Cell Membrane; Cucumis sativus; Egtazic Acid; Enzyme Activation; Hypocotyl; Ion Channels; Light; Membrane Potentials; Potassium Channel Blockers; Proton-Translocating ATPases; Tetraethylammonium; Tetraethylammonium Compounds; Vanadates; Verapamil | 1992 |
Effect of low oxygen concentration on the electrical properties of cortical cells of wheat roots.
Topics: Calcium Channel Blockers; Cell Hypoxia; Endoplasmic Reticulum; Membrane Potentials; Microelectrodes; Oxygen; Plant Roots; Potassium Acetate; Potassium Chloride; Tetraethylammonium; Triticum; Verapamil | 1997 |
Modulation of gonadotropin II release by K+ channel blockers in goldfish gonadotropes: a novel stimulatory action of 4-aminopyridine.
Topics: 4-Aminopyridine; Animals; Caffeine; Calcium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Fluorescent Dyes; Fura-2; Goldfish; Gonadotropins, Pituitary; Phosphodiesterase Inhibitors; Pituitary Gland; Potassium Channel Blockers; Tetraethylammonium; Verapamil | 2001 |
Influence of ion channels on the proliferation of human chondrocytes.
Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4-Aminopyridine; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Adult; Aged; Calcium Channel Blockers; Cartilage, Articular; Cell Cycle; Cell Division; Chloride Channels; Chondrocytes; Female; Flow Cytometry; Humans; Ion Channel Gating; Lidocaine; Male; Membrane Potentials; Middle Aged; Osteoarthritis, Knee; Potassium Channel Blockers; Sodium Channel Blockers; Tetraethylammonium; Verapamil | 2002 |
Inhibition of Kv2.1 voltage-dependent K+ channels in pancreatic beta-cells enhances glucose-dependent insulin secretion.
Topics: Animals; Calcium; Calcium Channel Blockers; Delayed Rectifier Potassium Channels; Diazoxide; Female; Glucose; Humans; In Vitro Techniques; Insulin; Insulin Secretion; Insulinoma; Islets of Langerhans; Membrane Potentials; Mice; Pancreas; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Voltage-Gated; Recombinant Fusion Proteins; Shab Potassium Channels; Tetraethylammonium; Tumor Cells, Cultured; Verapamil | 2002 |
Transport of the organic cations gonyautoxin 2/3 epimers, a paralytic shellfish poison toxin, through the human and rat intestinal epitheliums.
Topics: Adenosine; Animals; Biological Transport; Biological Transport, Active; Caco-2 Cells; Cations; Dinitrophenols; Humans; Intestinal Mucosa; Marine Toxins; Rats; Saxitoxin; Sodium; Stereoisomerism; Tetraethylammonium; Verapamil | 2002 |
The voltage-independent cation channel in the plasma membrane of wheat roots is permeable to divalent cations and may be involved in cytosolic Ca2+ homeostasis.
Topics: Barium; Calcium; Calcium Channels; Calcium Radioisotopes; Cell Membrane; Cytosol; Gadolinium; Homeostasis; Plant Roots; Potassium; Potassium Channels, Voltage-Gated; Signal Transduction; Sodium; Sodium Channels; Tetraethylammonium; Triticum; Verapamil | 2002 |
Predominant expression of Kv1.3 voltage-gated K+ channel subunit in rat prostate cancer cell lines: electrophysiological, pharmacological and molecular characterisation.
Topics: 4-Aminopyridine; Animals; Blotting, Western; Calcium Channel Blockers; Cell Line, Tumor; Charybdotoxin; Gene Expression Regulation, Neoplastic; Kv1.3 Potassium Channel; Male; Membrane Potentials; Molecular Sequence Data; Neurotoxins; Patch-Clamp Techniques; Potassium; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Voltage-Gated; Prostatic Neoplasms; Rats; Reverse Transcriptase Polymerase Chain Reaction; Scorpion Venoms; Tetraethylammonium; Verapamil | 2003 |
Choline uptake in human intestinal Caco-2 cells is carrier-mediated.
Topics: Caco-2 Cells; Carrier Proteins; Choline; Daunorubicin; Humans; Intestinal Mucosa; Intestines; Kinetics; Membrane Transport Proteins; Niacinamide; Sodium; Tetraethylammonium; Time Factors; Verapamil | 2003 |
Particular sensitivity to calcium channel blockers of the fast inward voltage-dependent sodium current involved in the invasive properties of a metastastic breast cancer cell line.
Topics: Breast Neoplasms; Calcium Channel Blockers; Cell Division; Cell Line, Tumor; Cell Survival; Diltiazem; Electrophysiology; Female; Humans; Nifedipine; Potassium Channel Blockers; Sodium Channels; Tetraethylammonium; Tetrodotoxin; Verapamil | 2004 |
Organic cation transport by Malpighian tubules of Drosophila melanogaster: application of two novel electrophysiological methods.
Topics: Animals; Biological Transport, Active; Cimetidine; Drosophila melanogaster; Electrophysiology; Ion Transport; Malpighian Tubules; Microelectrodes; Potassium; Quinidine; Tetraethylammonium; Tetraphenylborate; Verapamil; Vinblastine | 2004 |
Uptake and efflux of quinacrine, a candidate for the treatment of prion diseases, at the blood-brain barrier.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blood-Brain Barrier; Cation Transport Proteins; Cell Line; Cell Membrane; Cell Polarity; Cimetidine; Cyclosporine; Endothelial Cells; Fluorescein; Membrane Potentials; Mice; Prion Diseases; Quinacrine; Tetraethylammonium; Verapamil | 2004 |
Reduction of human neocortical and guinea pig CA1-neuron A-type currents by organic calcium channel blockers.
Topics: Adolescent; Adult; Aged; Anesthetics, Local; Animals; Calcium Channel Blockers; Child; Epilepsy; Female; Guinea Pigs; Humans; In Vitro Techniques; Male; Middle Aged; Neocortex; Neural Conduction; Neurons; Nifedipine; Potassium Channel Blockers; Pyramidal Cells; Stereoisomerism; Tetraethylammonium; Tetrodotoxin; Verapamil | 2004 |
Characterization of the voltage-activated currents in cultured atrial myocytes isolated from the heart of the common oyster Crassostrea gigas.
Topics: 4-Aminopyridine; Animals; Cadmium; Calcium; Cells, Cultured; Charybdotoxin; Cobalt; Electrophysiology; Heart Atria; Ion Channels; Membrane Potentials; Myocytes, Cardiac; Ostreidae; Patch-Clamp Techniques; Potassium; Sodium; Tetraethylammonium; Verapamil | 2004 |
In vivo evidence for the efflux transport of pentazocine from the brain across the blood-brain barrier using the brain efflux index method.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blood-Brain Barrier; Brain; Carbon Radioisotopes; Carnitine; Dose-Response Relationship, Drug; Drug Carriers; Drug Evaluation, Preclinical; Half-Life; Inulin; Male; Microinjections; Pentazocine; Quinidine; Rats; Rats, Wistar; Tetraethylammonium; Tritium; Verapamil | 2005 |
Transepithelial transport of fluorescent p-glycoprotein and MRP2 substrates by insect Malpighian tubules: confocal microscopic analysis of secreted fluid droplets.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Daunorubicin; Drosophila melanogaster; Epithelium; Fluorescent Dyes; Gryllidae; Malpighian Tubules; Microscopy, Confocal; Multidrug Resistance-Associated Proteins; Probenecid; Propionates; Quinacrine; Quinolines; Tetraethylammonium; Verapamil | 2005 |
Endothelium-dependent induction of vasorelaxation by the butanol extract of Phellinus igniarius in isolated rat aorta.
Topics: Animals; Aorta; Atropine; Butanols; Cyclic GMP; Diltiazem; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Glyburide; In Vitro Techniques; Indomethacin; Male; Methylene Blue; NG-Nitroarginine Methyl Ester; Oxadiazoles; Polyporaceae; Propranolol; Quinoxalines; Rats; Rats, Sprague-Dawley; Tetraethylammonium; Vasodilation; Vasodilator Agents; Verapamil | 2006 |
Mutation in an adaptor protein PDZK1 affects transport activity of organic cation transporter OCTNs and oligopeptide transporter PEPT2.
Topics: Adaptor Protein Complex gamma Subunits; Biological Transport; Carbon Radioisotopes; Carnitine; Carrier Proteins; Cell Line; Cell Membrane; Dipeptides; Humans; Membrane Proteins; Mutation; Organic Cation Transport Proteins; Organic Cation Transporter 1; Protein Binding; Pyrilamine; Solute Carrier Family 22 Member 5; Symporters; Tetraethylammonium; Transfection; Tritium; Two-Hybrid System Techniques; Verapamil | 2006 |
Spontaneous oscillatory contractions in aortas of rats with arterial pressure lability caused by sinoaortic denervation.
Topics: Animals; Aorta, Thoracic; Autonomic Denervation; Blood Pressure; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Chloride; Male; Oscillometry; Pinacidil; Potassium; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Tetraethylammonium; Time Factors; Vasoconstriction; Vasodilator Agents; Verapamil | 2007 |
Effects of intestinal ischemia/reperfusion on P-glycoprotein mediated biliary and renal excretion of rhodamine123 in rat.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biliary Tract; Cimetidine; Cyclosporine; Kidney; Liver; Male; Nitric Oxide Synthase Type I; Nitric Oxide Synthase Type II; Rats; Rats, Wistar; Reperfusion Injury; Rhodamine 123; Tetraethylammonium; Verapamil | 2009 |
Potassium-induced intermittent vasomotion in rat isolated pulmonary artery.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 4-Aminopyridine; Animals; Barium; Indoles; Male; Mibefradil; Nicardipine; Niflumic Acid; Potassium; Potassium Channels; Pulmonary Artery; Rats; Rats, Sprague-Dawley; Tetraethylammonium; Verapamil | 2011 |
Tacrine sinusoidal uptake and biliary excretion in sandwich-cultured primary rat hepatocytes.
Topics: Animals; Cells, Cultured; Cimetidine; Dose-Response Relationship, Drug; Hepatocytes; Male; Rats; Rats, Sprague-Dawley; Tacrine; Tetraethylammonium; Tissue Distribution; Verapamil | 2014 |
Plasmodium falciparum chloroquine resistance transporter is a H+-coupled polyspecific nutrient and drug exporter.
Topics: Amino Acids; Biological Transport; Chloroquine; Drug Resistance; Membrane Transport Proteins; Protons; Protozoan Proteins; Tetraethylammonium; Verapamil | 2015 |
β-Citronellol, an alcoholic monoterpene with inhibitory properties on the contractility of rat trachea.
Topics: Acyclic Monoterpenes; Analysis of Variance; Animals; Calcium Channel Blockers; Enzyme Inhibitors; Indomethacin; Inhibitory Concentration 50; Male; Monoterpenes; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Parasympatholytics; Rats, Wistar; Tetraethylammonium; Thapsigargin; Trachea; Verapamil | 2016 |