Page last updated: 2024-08-16

tetraethylammonium and verapamil

tetraethylammonium has been researched along with verapamil in 95 studies

Research

Studies (95)

TimeframeStudies, this research(%)All Research%
pre-199021 (22.11)18.7374
1990's40 (42.11)18.2507
2000's27 (28.42)29.6817
2010's7 (7.37)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dresser, MJ; Giacomini, KM; Gray, AT; Terashita, S; Yost, SC; Zhang, L1
Giacomini, KM; Schaner, ME; Zhang, L1
Nezu, J; Oku, A; Sai, Y; Sakamoto, K; Shimane, M; Tamai, I; Tsuji, A; Yabuuchi, H1
Nezu, JI; Ohashi, R; Oku, A; Sai, Y; Shimane, M; Tamai, I; Tsuji, A; Yabuuchi, H1
Conway, SJ; Ganapathy, V; George, RL; Huang, W; Leibach, FH; Wang, H; Wu, X1
Desir, GV; Lang, R; Lee, G; Liu, W; Orias, M; Rafi, H; Segal, AS; Tian, S1
Blom-Roosemalen, MC; Breimer, DD; de Boer, AG; van der Sandt, IC1
Hashimoto, N; Nezu Ji, J; Nikaido, H; Ohashi, R; Oku, A; Sai, Y; Shimane, M; Tamai, I; Tsuji, A1
Arieff, Z; Bardien-Kruger, S; Brink, P; Chandy, KG; Corfield, V; Wulff, H1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Benet, LZ; Brouwer, KL; Chu, X; Dahlin, A; Evers, R; Fischer, V; Giacomini, KM; Hillgren, KM; Hoffmaster, KA; Huang, SM; Ishikawa, T; Keppler, D; Kim, RB; Lee, CA; Niemi, M; Polli, JW; Sugiyama, Y; Swaan, PW; Tweedie, DJ; Ware, JA; Wright, SH; Yee, SW; Zamek-Gliszczynski, MJ; Zhang, L1
Ahlin, G; Bergström, F; Bredberg, U; Fridén, M; Hammarlund-Udenaes, M; Rehngren, M; Wan, H1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Niu, GB; Pei, JM; Zang, YM; Zhou, SS; Zhu, MZ1
Haseley, TS; Hosford, M; Lesniak, ME; McKinney, TD; Scheller, MB1
Frank, C; Sagratella, S; Scotti de Carolis, A1
Ferrier, J; Richter, C1
Amigorena, S; Choquet, D; Fridman, WH; Korn, H; Teillaud, JL1
Felix, D; Hirt, A; Huwyler, T; Morell, A1
Carpenter, FG1
Dreyer, F; Penner, R1
Gupta, S1
Shuba, MF; Smirnov, SV1
Boutin, L; Derosiers, J; Schanne, OF1
Aubin, JE; Ferrier, J; Heersche, JN; Ward-Kesthely, A1
Gemba, M; Hori, M1
Wali, FA1
Mitchell, HW1
Ballerini, P; Caciagli, F; Ciccarelli, R; Di Iorio, P; Tacconelli, L1
Lambert, CR; Pepine, CJ1
Asano, T; Kasuya, Y; Shigenobu, K1
Lazcano, C; Marín, J; Recio, L; Salaices, M; Sanchez-Ferrer, CF1
Dascal, N; Landau, EM; Lass, Y1
Jamieson, DD; Lander, J1
Barták, F; Jezek, K; Králícek, P; Pucelík, P1
Atarashi, H; Elharrar, V; Surawicz, B1
Foster, RW; Okpalugo, BI; Small, RC1
Downing, OA; Louttit, JB; Wilson, KA1
Sperelakis, N; Zelcer, E1
Kawamura, A; Solaro, RJ; Wahler, GM1
Cook, DI; Hayashi, T; Hirono, C; Young, JA1
Miller, DS1
Cook, DI; Ishikawa, T1
Santos, DE; Takeuchi, H1
Renfro, JL; Sussman-Turner, C1
Fricker, G; Miller, DS; Schramm, U; Wenger, R1
Delbono, O; Kotsias, BA1
Ortiz-Miranda, SI; Pappone, PA1
Ito, Y; Takagi, K; Tomita, T1
Cheng, PM; Donnelly, DF1
Lopatin, AN; Nichols, CG; Romano, C; Sha, Q1
Ağar, E; Green, GG; Sanders, DJ1
Irimajiri, A; Kakigi, A; Saito, H; Takeda, T; Takeuchi, S1
García-Segoviano, JA; Naranjo-Rodríguez, EB; Prieto-Gómez, B; Reyes-Vázquez, C; Trujillo-Santana, JT1
Das, P; Schurman, DJ; Smith, RL1
Hu, Q; Huang, F; Shi, Y1
Eusebi, F; Giovannelli, A; Lorenzon, P; Ragozzino, D; Ruzzier, F1
Dantzler, WH; Kim, YK1
Advenier, C; Bessard, G; Corompt, E; Devillier, P; Lantuejoul, S; Naline, E1
Ando, M; Takeuchi, S2
Kang, BS; Lee, YH; Seo, JH1
Atchison, WD; Hewett, SJ; Xu, YF1
Duff, HJ; Exner, DV; Feng, ZP; Geonzon, R; Wang, L; Woodman, RC1
Miller, DS; Pritchard, JB; Villalobos, AR1
Clauss, W; Heinke, B1
Adams, DJ; Catacuzzeno, L; Franciolini, F; Hogg, RC; Petris, A; Trequattrini, C1
Catacuzzeno, L; Franciolini, F; Petris, A; Trequattrini, C1
Hein, W; Wohlrab, D1
Kostyuk, PG; Lemonnier, L; Mauroy, B; Prevarskaya, N; Shuba, YM; Skryma, R; Van Coppenolle, F1
Le Bourhis, X; Legrand, G; Lemonnier, L; Prevarskaya, N; Rybalchenko, V; Skryma, R; Van Coppenolle, F1
Cosgrove, DJ; Spalding, EP1
Tyerman, SD; Zhang, WH1
Chang, JP; Johnson, JD; Kwong, P; Wong, CJ; Yunker, WK1
Krüger, T; Lebek, S; Reichel, H; Wohlrab, D1
Chan, CB; Joseph, JW; MacDonald, PE; Sakellaropoulos, G; Salapatek, AM; Saleh, MC; Sewing, S; Smukler, SR; Tsushima, RG; Wang, J; Wheeler, MB1
Andrinolo, D; Fraga, S; Gomes, P; Lagos, N; Soares-da-Silva, P1
Davenport, RJ; White, PJ1
Diss, JK; Djamgoz, MB; Dolly, JO; Fraser, SP; Grimes, JA; Stewart, D1
Darling, IM; Kamath, AV; Morris, ME1
Besson, P; Le Guennec, JY; Roger, S1
O'Donnell, MJ; Rheault, MR1
Dohgu, S; Higuchi, S; Katamine, S; Kataoka, Y; Naito, M; Niwa, M; Sawada, Y; Shirabe, S; Takata, F; Tsuruo, T; Yamauchi, A1
Gorji, A; Köhling, R; Rüschenschmidt, C; Siep, E; Speckmann, EJ; Straub, H1
Dorange, G; Droguet, M; Gioux, M; Giroux-Metgès, MA; Pennec, JP; Talarmin, H1
Fukami, T; Furuishi, T; Moriki, Y; Suzuki, T; Tomono, K; Watanabe, J1
Leader, JP; O'Donnell, MJ1
Cao, LH; Choi, DH; Kang, DG; Kim, JS; Kim, SJ; Lee, H; Lee, HS; Lee, JK1
Kato, Y; Kubo, Y; Sugiura, T; Tsuji, A1
Bendhack, LM; Rocha, ML1
Hayashi, M; Kishimoto, H; Takizawa, Y; Tomita, M1
Bieger, D; Ford, CA; Tabrizchi, R1
Kaddoumi, A; Mohamed, LA1
Fukui, T; Iwai, H; Juge, N; Kawakami, M; Miyaji, T; Moriyama, S; Moriyama, Y; Nelson, N; Omote, H1
Lucetti, LT; Magalhães, PJ; Ribeiro-Filho, HV; Vasconcelos, TB1

Reviews

1 review(s) available for tetraethylammonium and verapamil

ArticleYear
Membrane transporters in drug development.
    Nature reviews. Drug discovery, 2010, Volume: 9, Issue:3

    Topics: Animals; Computer Simulation; Decision Trees; Drug Approval; Drug Discovery; Drug Evaluation, Preclinical; Drug Interactions; Humans; Membrane Transport Proteins; Mice; Mice, Knockout; Prescription Drugs

2010

Other Studies

94 other study(ies) available for tetraethylammonium and verapamil

ArticleYear
Cloning and functional expression of a human liver organic cation transporter.
    Molecular pharmacology, 1997, Volume: 51, Issue:6

    Topics: Amino Acid Sequence; Animals; Base Sequence; Carrier Proteins; Cloning, Molecular; DNA, Complementary; Humans; Liver; Membrane Proteins; Molecular Sequence Data; Oocytes; Organic Cation Transporter 1; Polymerase Chain Reaction; Rats; RNA, Messenger; Sequence Homology, Amino Acid; Species Specificity; Tissue Distribution; Xenopus laevis

1997
Functional characterization of an organic cation transporter (hOCT1) in a transiently transfected human cell line (HeLa).
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 286, Issue:1

    Topics: Carrier Proteins; Corticosterone; HeLa Cells; Humans; Membrane Proteins; Midazolam; Organic Cation Transporter 1; Permeability; Recombinant Proteins; Structure-Activity Relationship; Tetraethylammonium Compounds; Transfection

1998
Novel membrane transporter OCTN1 mediates multispecific, bidirectional, and pH-dependent transport of organic cations.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 289, Issue:2

    Topics: Animals; Biological Transport, Active; Carrier Proteins; Cell Line; Gene Expression; Humans; Hydrogen-Ion Concentration; Membrane Potentials; Membrane Proteins; Membrane Transport Proteins; Oocytes; Organic Cation Transport Proteins; Quinidine; RNA, Messenger; Symporters; Tetraethylammonium Compounds; Xenopus laevis

1999
Na(+)-dependent carnitine transport by organic cation transporter (OCTN2): its pharmacological and toxicological relevance.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 291, Issue:2

    Topics: Biological Transport, Active; Carnitine; Carrier Proteins; Cations; Cells, Cultured; Dose-Response Relationship, Drug; Embryo, Mammalian; Humans; Hydrogen-Ion Concentration; Kidney; Membrane Proteins; Organic Cation Transport Proteins; Sodium; Solute Carrier Family 22 Member 5; Stereoisomerism

1999
Structural and functional characteristics and tissue distribution pattern of rat OCTN1, an organic cation transporter, cloned from placenta.
    Biochimica et biophysica acta, 2000, Jun-01, Volume: 1466, Issue:1-2

    Topics: Amino Acid Sequence; Animals; Base Sequence; Carnitine; Carrier Proteins; Cloning, Molecular; DNA, Complementary; Humans; Membrane Proteins; Membrane Transport Proteins; Molecular Sequence Data; Organic Cation Transport Proteins; Placenta; Rats; RNA, Messenger; Solute Carrier Proteins; Structure-Activity Relationship; Symporters; Tetraethylammonium; Tissue Distribution

2000
KCNA10: a novel ion channel functionally related to both voltage-gated potassium and CNG cation channels.
    American journal of physiology. Renal physiology, 2000, Volume: 278, Issue:6

    Topics: Animals; Base Sequence; Cyclic Nucleotide-Gated Cation Channels; DNA Primers; Female; Humans; In Vitro Techniques; Ion Channel Gating; Ion Channels; Membrane Potentials; Oocytes; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Voltage-Gated; Rabbits; Recombinant Proteins; Second Messenger Systems; Shaker Superfamily of Potassium Channels; Xenopus laevis

2000
Specificity of doxorubicin versus rhodamine-123 in assessing P-glycoprotein functionality in the LLC-PK1, LLC-PK1:MDR1 and Caco-2 cell lines.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2000, Volume: 11, Issue:3

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Caco-2 Cells; Cell Line; Cell Polarity; Cimetidine; Cyclosporine; Doxorubicin; Drug Resistance, Multiple; Epithelial Cells; Humans; Kinetics; LLC-PK1 Cells; Rhodamine 123; Swine; Tumor Cells, Cultured; Verapamil

2000
Molecular and physiological evidence for multifunctionality of carnitine/organic cation transporter OCTN2.
    Molecular pharmacology, 2001, Volume: 59, Issue:2

    Topics: Animals; Biological Transport; Carbon Radioisotopes; Carnitine; Carrier Proteins; Cells, Cultured; Embryo, Mammalian; Fibroblasts; Humans; Male; Membrane Proteins; Mice; Mice, Inbred C3H; Organic Cation Transport Proteins; Solute Carrier Family 22 Member 5; Tetraethylammonium; Tissue Distribution; Tritium

2001
Characterisation of the human voltage-gated potassium channel gene, KCNA7, a candidate gene for inherited cardiac disorders, and its exclusion as cause of progressive familial heart block I (PFHBI).
    European journal of human genetics : EJHG, 2002, Volume: 10, Issue:1

    Topics: Amino Acid Sequence; Animals; Base Sequence; Cloning, Molecular; COS Cells; DNA; Heart Block; Heart Diseases; Humans; Mice; Molecular Sequence Data; Potassium Channels; Potassium Channels, Voltage-Gated; Shaker Superfamily of Potassium Channels; Trinucleotide Repeats

2002
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Measurement of unbound drug exposure in brain: modeling of pH partitioning explains diverging results between the brain slice and brain homogenate methods.
    Drug metabolism and disposition: the biological fate of chemicals, 2011, Volume: 39, Issue:3

    Topics: Animals; Biological Transport; Brain; Chemical Phenomena; Dialysis; Hydrogen-Ion Concentration; In Vitro Techniques; Lysosomes; Male; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Tissue Distribution

2011
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
[Effects of tetraethylammonium chloride and verapamil on the effective refractory period of ischemic myocardium in rabbits].
    Yao xue xue bao = Acta pharmaceutica Sinica, 1992, Volume: 27, Issue:10

    Topics: Animals; Female; Male; Myocardial Ischemia; Rabbits; Refractory Period, Electrophysiological; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1992
Basolateral transport of tetraethylammonium by a clone of LLC-PK1 cells.
    Journal of the American Society of Nephrology : JASN, 1992, Volume: 2, Issue:10

    Topics: Animals; Basement Membrane; Biological Transport, Active; Cimetidine; Clone Cells; Kidney; Kinetics; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1992
Effects of calcium and potassium extracellular ionic concentration changes on the hippocampal CA1 activity of purinergic drugs.
    General pharmacology, 1991, Volume: 22, Issue:2

    Topics: 4-Aminopyridine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Calcium; Cesium; Chlorides; Evoked Potentials; Hippocampus; In Vitro Techniques; Male; Phenylisopropyladenosine; Potassium; Rats; Rats, Inbred Strains; Receptors, Purinergic; Synapses; Synaptic Transmission; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1991
Continuously active sodium channels in osteoblastic ROS 17/2.8 cells.
    Bone and mineral, 1991, Volume: 15, Issue:1

    Topics: Animals; Calcium; Conductometry; Membrane Potentials; Nifedipine; Osteoblasts; Osteosarcoma; Rats; Sodium; Sodium Channels; Tetraethylammonium; Tetraethylammonium Compounds; Tumor Cells, Cultured; Verapamil

1991
Ion channel blockers inhibit B cell activation at a precise stage of the G1 phase of the cell cycle. Possible involvement of K+ channels.
    Journal of immunology (Baltimore, Md. : 1950), 1990, Mar-15, Volume: 144, Issue:6

    Topics: 4-Aminopyridine; Animals; Antibodies, Monoclonal; B-Lymphocytes; Cell Cycle; Electric Conductivity; Lipopolysaccharides; Lymphocyte Activation; Mice; Potassium Channels; Quaternary Ammonium Compounds; Quinine; Tetraethylammonium; Tetraethylammonium Compounds; Thymidine; Time Factors; Verapamil

1990
Effect of cations and cation channel blockers on human natural killer cells.
    International journal of immunopharmacology, 1985, Volume: 7, Issue:4

    Topics: Anesthetics, Local; Calcium; Cytotoxicity, Immunologic; Dose-Response Relationship, Immunologic; Humans; Ion Channels; Killer Cells, Natural; Magnesium; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Verapamil

1985
Potentiation of nerve-induced bladder contractions after calcium channel blockade.
    The American journal of physiology, 1985, Volume: 249, Issue:4 Pt 2

    Topics: Animals; Calcium; Carbachol; Elasticity; Ion Channels; Male; Muscle Contraction; Muscle, Smooth; Potassium; Rats; Stimulation, Chemical; Tetraethylammonium; Tetraethylammonium Compounds; Urinary Bladder; Verapamil

1985
Two different presynaptic calcium currents in mouse motor nerve terminals.
    Pflugers Archiv : European journal of physiology, 1986, Volume: 406, Issue:2

    Topics: 4-Aminopyridine; Amifampridine; Aminopyridines; Animals; Barium; Cadmium; Calcium; Diltiazem; In Vitro Techniques; Ion Channels; Kinetics; Manganese; Mice; Motor Neurons; Neuromuscular Junction; Potassium; Strontium; Synapses; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1986
Autologous mixed-lymphocyte reaction in man. XVII. In vitro effect of ion channel-blocking agents on the autologous mixed-lymphocyte response.
    Cellular immunology, 1987, Volume: 104, Issue:2

    Topics: 4-Aminopyridine; Aminopyridines; Dose-Response Relationship, Drug; Humans; Interleukin-2; Ion Channels; Lymphocyte Activation; Lymphocyte Culture Test, Mixed; Quaternary Ammonium Compounds; Quinine; Receptors, Immunologic; Receptors, Interleukin-2; Recombinant Proteins; T-Lymphocytes; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1987
Potential-dependent calcium inward current in a single isolated smooth muscle cell of the guinea-pig taenia caeci.
    The Journal of physiology, 1986, Volume: 380

    Topics: Action Potentials; Animals; Calcium; Cesium; Guinea Pigs; In Vitro Techniques; Ion Channels; Kinetics; Muscle, Smooth; Potassium; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1986
Effects of K-channel blockers, calcium, and verapamil suggest different pacemaker mechanisms in cultured neonatal rat and embryonic chick ventricle cells.
    Canadian journal of physiology and pharmacology, 1989, Volume: 67, Issue:7

    Topics: Animals; Calcium; Cells, Cultured; Cesium; Chick Embryo; Heart Rate; Heart Ventricles; Membrane Potentials; Potassium Channels; Rats; Rats, Inbred Strains; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1989
Membrane potential changes, cAMP stimulation and contraction in osteoblast-like UMR 106 cells in response to calcitonin and parathyroid hormone.
    Bone and mineral, 1988, Volume: 4, Issue:2

    Topics: Animals; Bucladesine; Calcimycin; Calcitonin; Cell Line; Dinoprostone; Isoproterenol; Membrane Potentials; Osteoblasts; Parathyroid Hormone; Potassium Channels; Quinine; Rats; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1988
Effect of barium ion on p-aminohippurate transport in basolateral membrane vesicles isolated from rat kidney cortex.
    Archives internationales de pharmacodynamie et de therapie, 1985, Volume: 275, Issue:2

    Topics: Acid Phosphatase; Alkaline Phosphatase; Aminohippuric Acids; Animals; Barium; Biological Transport, Active; Cations; Glucose-6-Phosphatase; In Vitro Techniques; Kidney Cortex; L-Lactate Dehydrogenase; Male; Membranes; Onium Compounds; p-Aminohippuric Acid; Rats; Rats, Inbred Strains; Sodium-Potassium-Exchanging ATPase; Succinate Dehydrogenase; Tetraethylammonium; Tetraethylammonium Compounds; Trityl Compounds; Verapamil

1985
Interaction of verapamil with d-tubocurarine and cholinergic agonists at the avian neuromuscular junction.
    Acta anaesthesiologica Scandinavica, 1987, Volume: 31, Issue:1

    Topics: Acetylcholine; Animals; Chickens; Drug Interactions; In Vitro Techniques; Neuromuscular Junction; Synaptic Transmission; Tetraethylammonium; Tetraethylammonium Compounds; Tubocurarine; Verapamil

1987
Electromechanical effects of tetraethylammonium and K+ on histamine-induced contraction in pig isolated tracheal smooth muscle.
    Lung, 1987, Volume: 165, Issue:3

    Topics: Acetylcholine; Airway Resistance; Animals; Calcium; Histamine; Histamine Antagonists; In Vitro Techniques; Potassium; Sucrose; Swine; Tetraethylammonium; Tetraethylammonium Compounds; Trachea; Verapamil

1987
Cultures of glial cells release purines under field electrical stimulation: the possible ionic mechanisms.
    Pharmacological research communications, 1988, Volume: 20, Issue:11

    Topics: Adenosine; Adenosine Deaminase Inhibitors; Animals; Animals, Newborn; Brain; Cells, Cultured; Coformycin; Electric Stimulation; Neuroglia; Nucleotides; Pentostatin; Pharmacology; Rats; Reference Values; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Verapamil

1988
Tetraethylammonium-induced phasic arterial constriction: temporal and spatial characteristics.
    The American journal of physiology, 1986, Volume: 251, Issue:2 Pt 2

    Topics: Animals; Dogs; Femoral Artery; Physiology; Tetraethylammonium; Tetraethylammonium Compounds; Time Factors; Vasoconstriction; Verapamil

1986
TEA prevents the decline of the duration of the action potential in hypoxic cardiac muscle.
    Japanese journal of pharmacology, 1985, Volume: 38, Issue:1

    Topics: Action Potentials; Animals; Calcimycin; Calcium Chloride; Guinea Pigs; Heart; Hypoxia; In Vitro Techniques; Male; Myocardial Contraction; Tetraethylammonium; Tetraethylammonium Compounds; Time Factors; Verapamil

1985
Effect of tetraethylammonium and verapamil on noradrenaline release induced by field electrical stimulation and potassium from cat cerebral and femoral arteries.
    General pharmacology, 1985, Volume: 16, Issue:3

    Topics: Animals; Calcium; Cats; Cerebral Arteries; Electric Stimulation; Female; Femoral Artery; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Norepinephrine; Potassium; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Verapamil

1985
Xenopus oocyte resting potential, muscarinic responses and the role of calcium and guanosine 3',5'-cyclic monophosphate.
    The Journal of physiology, 1984, Volume: 352

    Topics: Acetylcholine; Action Potentials; Animals; Calcium; Cell Membrane Permeability; Chlorides; Cyclic GMP; Female; In Vitro Techniques; Membrane Potentials; Oocytes; Ouabain; Potassium; Sodium; Tetraethylammonium; Tetraethylammonium Compounds; Time Factors; Verapamil; Xenopus laevis

1984
Investigation of the mode of action of the anaesthetic agent, ketamine, in the heart of the bivalve mollusc Tapes watlingi.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1984, Volume: 77, Issue:1

    Topics: Acetylcholine; Amphetamine; Animals; Dose-Response Relationship, Drug; Heart; Heart Rate; Ketamine; Methysergide; Metoclopramide; Mollusca; Phentolamine; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1984
An analysis of the postnatal development of the action potential repolarization process in the working ventricular myocardium of albino rats (effect of tea, frequency, verapamil and adrenaline).
    Physiologia Bohemoslovaca, 1983, Volume: 32, Issue:5

    Topics: Action Potentials; Age Factors; Animals; Animals, Newborn; Calcium; Electric Stimulation; Epinephrine; Female; Heart; Heart Ventricles; Ion Channels; Male; Myocardial Contraction; Potassium; Rats; Rats, Inbred Strains; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1983
Cycle length-dependent action potential duration in canine cardiac Purkinje fibers.
    The American journal of physiology, 1984, Volume: 247, Issue:6 Pt 2

    Topics: Action Potentials; Animals; Cobalt; Dogs; Female; Heart Conduction System; Homeostasis; In Vitro Techniques; Isoproterenol; Kinetics; Lidocaine; Male; Purkinje Fibers; Reaction Time; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Verapamil

1984
Antagonism of Ca2+ and other actions of verapamil in guinea-pig isolated trachealis.
    British journal of pharmacology, 1984, Volume: 81, Issue:3

    Topics: Acetylcholine; Action Potentials; Airway Resistance; Animals; Calcium Channel Blockers; Dinoprostone; Electrophysiology; Female; Guinea Pigs; Histamine; In Vitro Techniques; Male; Potassium Chloride; Prostaglandins E; Tetraethylammonium; Tetraethylammonium Compounds; Trachea; Verapamil

1984
Differential effects of strychnine on two types of vascular muscle.
    European journal of pharmacology, 1984, Feb-17, Volume: 98, Issue:2

    Topics: 4-Aminopyridine; Aminopyridines; Animals; Aorta, Thoracic; Cardiovascular Agents; Male; Muscle Contraction; Muscle, Smooth, Vascular; Portal Vein; Prazosin; Rats; Rats, Inbred Strains; Strychnine; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Verapamil

1984
Angiotensin induction of active responses in cultured reaggregates of rat aortic smooth muscle cells.
    Blood vessels, 1981, Volume: 18, Issue:6

    Topics: Angiotensin II; Animals; Aorta, Thoracic; Barium; Barium Compounds; Cell Aggregation; Cells, Cultured; Chlorides; Electric Stimulation; Electrophysiology; Male; Membrane Potentials; Muscle, Smooth, Vascular; Rats; Rats, Inbred Strains; Sodium; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1981
RWJ-24517, a positive inotropic agent, has novel effects on action potentials in guinea pig myocardium.
    Journal of cardiovascular pharmacology, 1993, Volume: 22, Issue:4

    Topics: Actin Cytoskeleton; Action Potentials; Adenosine Triphosphatases; Animals; Cardiotonic Agents; Dose-Response Relationship, Drug; Electrophysiology; Female; Guinea Pigs; Male; Mercaptopurine; Papillary Muscles; Piperazines; Potassium Channel Blockers; Sodium Channels; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1993
The ACh-induced whole-cell currents in sheep parotid secretory cells. Do BK channels really carry the ACh-evoked whole-cell K+ current?
    The Journal of membrane biology, 1995, Volume: 144, Issue:2

    Topics: 4-Aminopyridine; Acetylcholine; Animals; Barium; Cell Membrane; Chlorides; Parotid Gland; Patch-Clamp Techniques; Potassium; Potassium Channel Blockers; Potassium Channels; Quinidine; Quinine; Sensitivity and Specificity; Sheep; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1995
Daunomycin secretion by killfish renal proximal tubules.
    The American journal of physiology, 1995, Volume: 269, Issue:2 Pt 2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Buffers; Cyclosporine; Daunorubicin; Hydrogen-Ion Concentration; Image Processing, Computer-Assisted; Kidney Tubules, Proximal; Killifishes; Microscopy, Fluorescence; Television; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1995
Effects of K+ channel blockers on inwardly and outwardly rectifying whole-cell K+ currents in sheep parotid secretory cells.
    The Journal of membrane biology, 1993, Volume: 133, Issue:1

    Topics: Animals; Barium; Cesium; Charybdotoxin; In Vitro Techniques; Lidocaine; Membrane Potentials; Parotid Gland; Potassium; Potassium Channels; Quinidine; Quinine; Scorpion Venoms; Sheep; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1993
Influence of the drugs for membrane excitability modification on the excitation caused by achatin-I.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1993, Volume: 105, Issue:2

    Topics: Amino Acid Sequence; Animals; Concanavalin A; Drug Interactions; Ion Channels; Membrane Potentials; Molecular Sequence Data; Neurons; Neuropeptides; Picrotoxin; Snails; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Tyrosine; Verapamil

1993
Heat-shock-stimulated transepithelial daunomycin secretion by flounder renal proximal tubule primary cultures.
    The American journal of physiology, 1995, Volume: 268, Issue:1 Pt 2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cells, Cultured; Cycloheximide; Cyclosporine; Daunorubicin; Epithelial Cells; Epithelium; Flounder; Hot Temperature; Immunohistochemistry; Kidney Tubules, Proximal; Kinetics; Microvilli; p-Aminohippuric Acid; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil; Vinblastine

1995
P-glycoprotein-mediated secretion of a fluorescent cyclosporin analogue by teleost renal proximal tubules.
    The American journal of physiology, 1995, Volume: 268, Issue:1 Pt 2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cyclosporine; Fluorescent Dyes; Kidney Tubules, Proximal; Killifishes; Kinetics; Microscopy, Fluorescence; p-Aminohippuric Acid; Potassium Cyanide; Quinine; Tetraethylammonium; Tetraethylammonium Compounds; Time Factors; Verapamil; Vinblastine

1995
Effect of aminophylline-Ca2+ blocker interaction on membrane potential of rat diaphragm fibers.
    Journal of applied physiology (Bethesda, Md. : 1985), 1993, Volume: 74, Issue:6

    Topics: Aminophylline; Animals; Apamin; Diaphragm; Drug Interactions; In Vitro Techniques; Membrane Potentials; Nifedipine; Rats; Rats, Wistar; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1993
Blockers of voltage-gated K channels inhibit proliferation of cultured brown fat cells.
    The American journal of physiology, 1993, Volume: 264, Issue:4 Pt 1

    Topics: Adipose Tissue, Brown; Animals; Animals, Newborn; Calcium; Cell Division; Cells, Cultured; Kinetics; Membrane Potentials; Nifedipine; Norepinephrine; Potassium Channels; Quinine; Rats; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1993
Relaxant actions of isoprenaline on guinea-pig isolated tracheal smooth muscle.
    British journal of pharmacology, 1995, Volume: 116, Issue:6

    Topics: Adrenergic beta-Agonists; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Female; Guinea Pigs; In Vitro Techniques; Indoles; Isoproterenol; Male; Membrane Potentials; Muscle Relaxation; Muscle Tonus; Muscle, Smooth; Potassium Channels; Tetraethylammonium; Tetraethylammonium Compounds; Trachea; Verapamil

1995
Relationship between changes of glomus cell current and neural response of rat carotid body.
    Journal of neurophysiology, 1995, Volume: 74, Issue:5

    Topics: Afferent Pathways; Animals; Apamin; Carotid Body; Cell Hypoxia; Charybdotoxin; Membrane Potentials; Neural Inhibition; Patch-Clamp Techniques; Potassium Channels; Rats; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1995
Spermidine release from xenopus oocytes. Electrodiffusion through a membrane channel.
    The Journal of biological chemistry, 1996, Feb-16, Volume: 271, Issue:7

    Topics: Animals; Calcium; Cells, Cultured; Diffusion; Female; Kinetics; Oocytes; Patch-Clamp Techniques; Potassium; Potassium Channels; Recombinant Proteins; Spermidine; Tetraethylammonium; Tetraethylammonium Compounds; Tritium; Verapamil; Xenopus laevis

1996
Membrane properties of complex spike firing neurons of the mouse dorsal cochlear nucleus in vitro.
    Journal of basic and clinical physiology and pharmacology, 1996, Volume: 7, Issue:2

    Topics: 4-Aminopyridine; Action Potentials; Animals; Auditory Pathways; Calcium Channel Blockers; Cochlear Nucleus; In Vitro Techniques; Mice; Mice, Inbred BALB C; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Verapamil

1996
Intravascularly applied K(+)-channel blockers suppress differently the positive endocochlear potential maintained by vascular perfusion.
    Hearing research, 1996, Nov-01, Volume: 101, Issue:1-2

    Topics: Analgesics, Non-Narcotic; Animals; Barium; Calcium Channel Blockers; Cerebellum; Cochlear Microphonic Potentials; Guinea Pigs; Potassium Channel Blockers; Quinine; Stria Vascularis; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1996
Apamin blocks the direct relaxant effect of melatonin on rat ileal smooth muscle.
    Journal of pineal research, 1997, Volume: 22, Issue:1

    Topics: 4-Aminopyridine; Adrenergic alpha-Antagonists; Animals; Apamin; Calcium; Calcium Channel Blockers; Carbachol; Cholinergic Antagonists; Glyburide; Hexamethonium; Humans; Ileum; Male; Melatonin; Muscarinic Antagonists; Muscle Contraction; Neuromuscular Depolarizing Agents; Nitrendipine; Phentolamine; Rats; Rats, Wistar; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Verapamil

1997
Nitric oxide and G proteins mediate the response of bovine articular chondrocytes to fluid-induced shear.
    Journal of orthopaedic research : official publication of the Orthopaedic Research Society, 1997, Volume: 15, Issue:1

    Topics: Animals; Calcium Channel Blockers; Cartilage, Articular; Cattle; Enzyme Inhibitors; Glycosaminoglycans; GTP-Binding Proteins; Neomycin; Nitric Oxide; Nitric Oxide Synthase; omega-N-Methylarginine; Ornithine; Pertussis Toxin; Protein Synthesis Inhibitors; Signal Transduction; Stress, Mechanical; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil; Virulence Factors, Bordetella; Weight-Bearing

1997
Inhibition of Toosendanin on the delayed rectifier potassium current in neuroblastoma x glioma NG108-15 cells.
    Brain research, 1997, Mar-14, Volume: 751, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Delayed Rectifier Potassium Channels; Dose-Response Relationship, Drug; Drugs, Chinese Herbal; Glioma; Hybrid Cells; Mice; Neuroblastoma; Neuromuscular Blocking Agents; Nifedipine; Patch-Clamp Techniques; Potassium; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Voltage-Gated; Rats; Tetraethylammonium; Tetraethylammonium Compounds; Verapamil

1997
Spontaneous and repetitive calcium transients in C2C12 mouse myotubes during in vitro myogenesis.
    The European journal of neuroscience, 1997, Volume: 9, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenosine Triphosphate; Animals; Apamin; Caffeine; Calcium; Cell Differentiation; Cell Line; Cytosol; Egtazic Acid; Kinetics; Membrane Potentials; Mice; Microscopy, Confocal; Microscopy, Video; Muscle, Skeletal; Oscillometry; Potassium Chloride; Tetraethylammonium; Tetraethylammonium Compounds; Tetrodotoxin; Verapamil

1997
Ca2+ and Ba2+ effects on basolateral tetraethylammonium transport in isolated snake renal proximal tubules.
    Pflugers Archiv : European journal of physiology, 1997, Volume: 435, Issue:1

    Topics: Animals; Barium; Biological Transport; Calcium; Colubridae; Egtazic Acid; Kidney Tubules, Proximal; Lanthanum; Membrane Potentials; Tetraethylammonium; Tritium; Verapamil

1997
Inhibitory effects of large Ca2+-activated K+ channel blockers on beta-adrenergic- and NO-donor-mediated relaxations of human and guinea-pig airway smooth muscles.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 357, Issue:1

    Topics: Adrenergic beta-Agonists; Adult; Aged; Aged, 80 and over; Albuterol; Animals; Benzimidazoles; Bronchi; Calcium; Calcium Channel Blockers; Charybdotoxin; Guinea Pigs; Humans; Male; Middle Aged; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nitric Oxide; Nitroprusside; Peptides; Potassium Channels; Tetraethylammonium; Vasodilator Agents; Verapamil

1998
Inwardly rectifying K+ currents in intermediate cells in the cochlea of gerbils: a possible contribution to the endocochlear potential.
    Neuroscience letters, 1998, May-15, Volume: 247, Issue:2-3

    Topics: 4-Aminopyridine; Animals; Barium; Cadmium; Cesium; Cochlear Microphonic Potentials; Endolymph; Gerbillinae; Ion Transport; Models, Neurological; Nerve Tissue Proteins; Patch-Clamp Techniques; Potassium; Potassium Channels; Potassium Channels, Inwardly Rectifying; Quinine; Stria Vascularis; Tetraethylammonium; Verapamil

1998
Effects of hypoxia on pulmonary vascular contractility.
    Yonsei medical journal, 1998, Volume: 39, Issue:3

    Topics: Animals; Blood Vessels; Calcium Channel Blockers; Cyclooxygenase Inhibitors; Enzyme Inhibitors; Hypoxia; Indomethacin; Nitroarginine; Pulmonary Circulation; Rats; Tetraethylammonium; Vasoconstriction; Verapamil

1998
Passive transfer of Lambert-Eaton myasthenic syndrome induces dihydropyridine sensitivity of ICa in mouse motor nerve terminals.
    Journal of neurophysiology, 1998, Volume: 80, Issue:3

    Topics: Animals; Autoantibodies; Binding, Competitive; Calcium; Calcium Channel Blockers; Dihydropyridines; Immunization, Passive; Lambert-Eaton Myasthenic Syndrome; Male; Mice; Mice, Inbred ICR; Motor Neurons; Nifedipine; omega-Agatoxin IVA; omega-Conotoxins; Peptides; Plasma; Potassium Channel Blockers; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Spider Venoms; Synaptosomes; Tetraethylammonium; Verapamil

1998
A high affinity binding site for [3H]-Dofetilide on human leukocytes.
    Journal of molecular and cellular cardiology, 1998, Volume: 30, Issue:9

    Topics: Animals; Anti-Arrhythmia Agents; Binding Sites; Charybdotoxin; Guinea Pigs; Humans; Kinetics; Leukocytes; Neuropeptides; Neutrophils; Phenethylamines; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Voltage-Gated; Shaw Potassium Channels; Sulfonamides; Tetraethylammonium; Verapamil

1998
Organic cation transport in rat choroid plexus cells studied by fluorescence microscopy.
    The American journal of physiology, 1999, Volume: 276, Issue:4

    Topics: Animals; Animals, Newborn; Biological Transport; Cations; Choroid Plexus; Kinetics; Microscopy, Confocal; Microscopy, Fluorescence; Monensin; Neurons; Potassium Cyanide; Quinacrine; Rats; Rats, Inbred F344; Tetraethylammonium; Verapamil; Video Recording

1999
Potassium conductances in isolated single cells from Xenopus laevis colonic epithelium.
    Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology, 1999, Volume: 169, Issue:2

    Topics: Animals; Barium; Cesium; Colon; Epithelial Cells; Female; Hydrogen-Ion Concentration; Ion Transport; Lidocaine; Membrane Potentials; Patch-Clamp Techniques; Potassium; Potassium Channel Blockers; Potassium Channels; Quinidine; Quinine; Tetraethylammonium; Verapamil; Xenopus laevis

1999
Mechanisms of verapamil inhibition of action potential firing in rat intracardiac ganglion neurons.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 289, Issue:3

    Topics: 4-Aminopyridine; Acetylcholine; Action Potentials; Animals; Animals, Newborn; Apamin; Cells, Cultured; Charybdotoxin; Electric Stimulation; Ganglia, Parasympathetic; Heart; Membrane Potentials; Muscarine; Neurons; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Rats; Tetraethylammonium; Verapamil

1999
Mechanism of verapamil block of a neuronal delayed rectifier K channel: active form of the blocker and location of its binding domain.
    British journal of pharmacology, 1999, Volume: 126, Issue:8

    Topics: Animals; Binding Sites; Binding, Competitive; Biotransformation; Calcium Channel Blockers; Chick Embryo; Electrophysiology; Gallopamil; Ganglia, Spinal; Kinetics; Neurons; Potassium Channel Blockers; Potassium Channels; Tetraethylammonium; Verapamil

1999
Voltage-dependent outward K(+) current in intermediate cell of stria vascularis of gerbil cochlea.
    The American journal of physiology, 1999, Volume: 277, Issue:1

    Topics: Animals; Barium; Calcium; Electric Conductivity; Electrophysiology; Patch-Clamp Techniques; Potassium; Potassium Channel Blockers; Potassium Channels; Quinine; Stria Vascularis; Tetraethylammonium; Verapamil

1999
[Effect of ion channel modulators on the membrane potential of human chondrocytes].
    Der Orthopade, 2000, Volume: 29, Issue:2

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4-Aminopyridine; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Cell Division; Cells, Cultured; Chondrocytes; Flow Cytometry; Humans; Ion Channels; Membrane Potentials; Tetraethylammonium; Verapamil

2000
Volume-regulated chloride conductance in the LNCaP human prostate cancer cell line.
    American journal of physiology. Cell physiology, 2000, Volume: 279, Issue:4

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; 8-Bromo Cyclic Adenosine Monophosphate; Adenosine Triphosphate; Anions; Calcium; Calcium Channel Blockers; Carcinoma; Cell Membrane Permeability; Chloride Channels; Electric Stimulation; Humans; Hypotonic Solutions; Ion Transport; Male; Membrane Potentials; Nitrobenzoates; Patch-Clamp Techniques; Potassium; Prostatic Neoplasms; Protein-Tyrosine Kinases; Substrate Specificity; Tetraethylammonium; Tumor Cells, Cultured; Verapamil

2000
Verapamil inhibits proliferation of LNCaP human prostate cancer cells influencing K+ channel gating.
    Molecular pharmacology, 2001, Volume: 59, Issue:6

    Topics: Antineoplastic Agents; Binding Sites; Binding, Competitive; Calcium Channel Blockers; Cell Division; Dose-Response Relationship, Drug; Electrophysiology; Humans; Male; Potassium Channel Blockers; Potassium Channels; Prostatic Neoplasms; Tetraethylammonium; Tumor Cells, Cultured; Verapamil

2001
Mechanism of blue-light-induced plasma-membrane depolarization in etiolated cucumber hypocotyls.
    Planta, 1992, Volume: 188, Issue:2

    Topics: Adenosine Triphosphate; Cell Membrane; Cucumis sativus; Egtazic Acid; Enzyme Activation; Hypocotyl; Ion Channels; Light; Membrane Potentials; Potassium Channel Blockers; Proton-Translocating ATPases; Tetraethylammonium; Tetraethylammonium Compounds; Vanadates; Verapamil

1992
Effect of low oxygen concentration on the electrical properties of cortical cells of wheat roots.
    Journal of plant physiology, 1997, Volume: 150, Issue:5

    Topics: Calcium Channel Blockers; Cell Hypoxia; Endoplasmic Reticulum; Membrane Potentials; Microelectrodes; Oxygen; Plant Roots; Potassium Acetate; Potassium Chloride; Tetraethylammonium; Triticum; Verapamil

1997
Modulation of gonadotropin II release by K+ channel blockers in goldfish gonadotropes: a novel stimulatory action of 4-aminopyridine.
    Journal of neuroendocrinology, 2001, Volume: 13, Issue:11

    Topics: 4-Aminopyridine; Animals; Caffeine; Calcium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Fluorescent Dyes; Fura-2; Goldfish; Gonadotropins, Pituitary; Phosphodiesterase Inhibitors; Pituitary Gland; Potassium Channel Blockers; Tetraethylammonium; Verapamil

2001
Influence of ion channels on the proliferation of human chondrocytes.
    Biorheology, 2002, Volume: 39, Issue:1-2

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4-Aminopyridine; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Adult; Aged; Calcium Channel Blockers; Cartilage, Articular; Cell Cycle; Cell Division; Chloride Channels; Chondrocytes; Female; Flow Cytometry; Humans; Ion Channel Gating; Lidocaine; Male; Membrane Potentials; Middle Aged; Osteoarthritis, Knee; Potassium Channel Blockers; Sodium Channel Blockers; Tetraethylammonium; Verapamil

2002
Inhibition of Kv2.1 voltage-dependent K+ channels in pancreatic beta-cells enhances glucose-dependent insulin secretion.
    The Journal of biological chemistry, 2002, Nov-22, Volume: 277, Issue:47

    Topics: Animals; Calcium; Calcium Channel Blockers; Delayed Rectifier Potassium Channels; Diazoxide; Female; Glucose; Humans; In Vitro Techniques; Insulin; Insulin Secretion; Insulinoma; Islets of Langerhans; Membrane Potentials; Mice; Pancreas; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Voltage-Gated; Recombinant Fusion Proteins; Shab Potassium Channels; Tetraethylammonium; Tumor Cells, Cultured; Verapamil

2002
Transport of the organic cations gonyautoxin 2/3 epimers, a paralytic shellfish poison toxin, through the human and rat intestinal epitheliums.
    Toxicon : official journal of the International Society on Toxinology, 2002, Volume: 40, Issue:10

    Topics: Adenosine; Animals; Biological Transport; Biological Transport, Active; Caco-2 Cells; Cations; Dinitrophenols; Humans; Intestinal Mucosa; Marine Toxins; Rats; Saxitoxin; Sodium; Stereoisomerism; Tetraethylammonium; Verapamil

2002
The voltage-independent cation channel in the plasma membrane of wheat roots is permeable to divalent cations and may be involved in cytosolic Ca2+ homeostasis.
    Plant physiology, 2002, Volume: 130, Issue:3

    Topics: Barium; Calcium; Calcium Channels; Calcium Radioisotopes; Cell Membrane; Cytosol; Gadolinium; Homeostasis; Plant Roots; Potassium; Potassium Channels, Voltage-Gated; Signal Transduction; Sodium; Sodium Channels; Tetraethylammonium; Triticum; Verapamil

2002
Predominant expression of Kv1.3 voltage-gated K+ channel subunit in rat prostate cancer cell lines: electrophysiological, pharmacological and molecular characterisation.
    Pflugers Archiv : European journal of physiology, 2003, Volume: 446, Issue:5

    Topics: 4-Aminopyridine; Animals; Blotting, Western; Calcium Channel Blockers; Cell Line, Tumor; Charybdotoxin; Gene Expression Regulation, Neoplastic; Kv1.3 Potassium Channel; Male; Membrane Potentials; Molecular Sequence Data; Neurotoxins; Patch-Clamp Techniques; Potassium; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Voltage-Gated; Prostatic Neoplasms; Rats; Reverse Transcriptase Polymerase Chain Reaction; Scorpion Venoms; Tetraethylammonium; Verapamil

2003
Choline uptake in human intestinal Caco-2 cells is carrier-mediated.
    The Journal of nutrition, 2003, Volume: 133, Issue:8

    Topics: Caco-2 Cells; Carrier Proteins; Choline; Daunorubicin; Humans; Intestinal Mucosa; Intestines; Kinetics; Membrane Transport Proteins; Niacinamide; Sodium; Tetraethylammonium; Time Factors; Verapamil

2003
Particular sensitivity to calcium channel blockers of the fast inward voltage-dependent sodium current involved in the invasive properties of a metastastic breast cancer cell line.
    British journal of pharmacology, 2004, Volume: 141, Issue:4

    Topics: Breast Neoplasms; Calcium Channel Blockers; Cell Division; Cell Line, Tumor; Cell Survival; Diltiazem; Electrophysiology; Female; Humans; Nifedipine; Potassium Channel Blockers; Sodium Channels; Tetraethylammonium; Tetrodotoxin; Verapamil

2004
Organic cation transport by Malpighian tubules of Drosophila melanogaster: application of two novel electrophysiological methods.
    The Journal of experimental biology, 2004, Volume: 207, Issue:Pt 12

    Topics: Animals; Biological Transport, Active; Cimetidine; Drosophila melanogaster; Electrophysiology; Ion Transport; Malpighian Tubules; Microelectrodes; Potassium; Quinidine; Tetraethylammonium; Tetraphenylborate; Verapamil; Vinblastine

2004
Uptake and efflux of quinacrine, a candidate for the treatment of prion diseases, at the blood-brain barrier.
    Cellular and molecular neurobiology, 2004, Volume: 24, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blood-Brain Barrier; Cation Transport Proteins; Cell Line; Cell Membrane; Cell Polarity; Cimetidine; Cyclosporine; Endothelial Cells; Fluorescein; Membrane Potentials; Mice; Prion Diseases; Quinacrine; Tetraethylammonium; Verapamil

2004
Reduction of human neocortical and guinea pig CA1-neuron A-type currents by organic calcium channel blockers.
    Neuroscience letters, 2004, Sep-16, Volume: 368, Issue:1

    Topics: Adolescent; Adult; Aged; Anesthetics, Local; Animals; Calcium Channel Blockers; Child; Epilepsy; Female; Guinea Pigs; Humans; In Vitro Techniques; Male; Middle Aged; Neocortex; Neural Conduction; Neurons; Nifedipine; Potassium Channel Blockers; Pyramidal Cells; Stereoisomerism; Tetraethylammonium; Tetrodotoxin; Verapamil

2004
Characterization of the voltage-activated currents in cultured atrial myocytes isolated from the heart of the common oyster Crassostrea gigas.
    The Journal of experimental biology, 2004, Volume: 207, Issue:Pt 22

    Topics: 4-Aminopyridine; Animals; Cadmium; Calcium; Cells, Cultured; Charybdotoxin; Cobalt; Electrophysiology; Heart Atria; Ion Channels; Membrane Potentials; Myocytes, Cardiac; Ostreidae; Patch-Clamp Techniques; Potassium; Sodium; Tetraethylammonium; Verapamil

2004
In vivo evidence for the efflux transport of pentazocine from the brain across the blood-brain barrier using the brain efflux index method.
    Journal of drug targeting, 2005, Volume: 13, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blood-Brain Barrier; Brain; Carbon Radioisotopes; Carnitine; Dose-Response Relationship, Drug; Drug Carriers; Drug Evaluation, Preclinical; Half-Life; Inulin; Male; Microinjections; Pentazocine; Quinidine; Rats; Rats, Wistar; Tetraethylammonium; Tritium; Verapamil

2005
Transepithelial transport of fluorescent p-glycoprotein and MRP2 substrates by insect Malpighian tubules: confocal microscopic analysis of secreted fluid droplets.
    The Journal of experimental biology, 2005, Volume: 208, Issue:Pt 23

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Daunorubicin; Drosophila melanogaster; Epithelium; Fluorescent Dyes; Gryllidae; Malpighian Tubules; Microscopy, Confocal; Multidrug Resistance-Associated Proteins; Probenecid; Propionates; Quinacrine; Quinolines; Tetraethylammonium; Verapamil

2005
Endothelium-dependent induction of vasorelaxation by the butanol extract of Phellinus igniarius in isolated rat aorta.
    The American journal of Chinese medicine, 2006, Volume: 34, Issue:4

    Topics: Animals; Aorta; Atropine; Butanols; Cyclic GMP; Diltiazem; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Glyburide; In Vitro Techniques; Indomethacin; Male; Methylene Blue; NG-Nitroarginine Methyl Ester; Oxadiazoles; Polyporaceae; Propranolol; Quinoxalines; Rats; Rats, Sprague-Dawley; Tetraethylammonium; Vasodilation; Vasodilator Agents; Verapamil

2006
Mutation in an adaptor protein PDZK1 affects transport activity of organic cation transporter OCTNs and oligopeptide transporter PEPT2.
    Drug metabolism and pharmacokinetics, 2006, Volume: 21, Issue:5

    Topics: Adaptor Protein Complex gamma Subunits; Biological Transport; Carbon Radioisotopes; Carnitine; Carrier Proteins; Cell Line; Cell Membrane; Dipeptides; Humans; Membrane Proteins; Mutation; Organic Cation Transport Proteins; Organic Cation Transporter 1; Protein Binding; Pyrilamine; Solute Carrier Family 22 Member 5; Symporters; Tetraethylammonium; Transfection; Tritium; Two-Hybrid System Techniques; Verapamil

2006
Spontaneous oscillatory contractions in aortas of rats with arterial pressure lability caused by sinoaortic denervation.
    Clinical and experimental pharmacology & physiology, 2007, Volume: 34, Issue:8

    Topics: Animals; Aorta, Thoracic; Autonomic Denervation; Blood Pressure; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Chloride; Male; Oscillometry; Pinacidil; Potassium; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Tetraethylammonium; Time Factors; Vasoconstriction; Vasodilator Agents; Verapamil

2007
Effects of intestinal ischemia/reperfusion on P-glycoprotein mediated biliary and renal excretion of rhodamine123 in rat.
    Drug metabolism and pharmacokinetics, 2009, Volume: 24, Issue:5

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biliary Tract; Cimetidine; Cyclosporine; Kidney; Liver; Male; Nitric Oxide Synthase Type I; Nitric Oxide Synthase Type II; Rats; Rats, Wistar; Reperfusion Injury; Rhodamine 123; Tetraethylammonium; Verapamil

2009
Potassium-induced intermittent vasomotion in rat isolated pulmonary artery.
    Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi, 2011, Volume: 47, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 4-Aminopyridine; Animals; Barium; Indoles; Male; Mibefradil; Nicardipine; Niflumic Acid; Potassium; Potassium Channels; Pulmonary Artery; Rats; Rats, Sprague-Dawley; Tetraethylammonium; Verapamil

2011
Tacrine sinusoidal uptake and biliary excretion in sandwich-cultured primary rat hepatocytes.
    Journal of pharmacy & pharmaceutical sciences : a publication of the Canadian Society for Pharmaceutical Sciences, Societe canadienne des sciences pharmaceutiques, 2014, Volume: 17, Issue:3

    Topics: Animals; Cells, Cultured; Cimetidine; Dose-Response Relationship, Drug; Hepatocytes; Male; Rats; Rats, Sprague-Dawley; Tacrine; Tetraethylammonium; Tissue Distribution; Verapamil

2014
Plasmodium falciparum chloroquine resistance transporter is a H+-coupled polyspecific nutrient and drug exporter.
    Proceedings of the National Academy of Sciences of the United States of America, 2015, Mar-17, Volume: 112, Issue:11

    Topics: Amino Acids; Biological Transport; Chloroquine; Drug Resistance; Membrane Transport Proteins; Protons; Protozoan Proteins; Tetraethylammonium; Verapamil

2015
β-Citronellol, an alcoholic monoterpene with inhibitory properties on the contractility of rat trachea.
    Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas, 2016, Volume: 49, Issue:2

    Topics: Acyclic Monoterpenes; Analysis of Variance; Animals; Calcium Channel Blockers; Enzyme Inhibitors; Indomethacin; Inhibitory Concentration 50; Male; Monoterpenes; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Parasympatholytics; Rats, Wistar; Tetraethylammonium; Thapsigargin; Trachea; Verapamil

2016