Page last updated: 2024-08-23

tetradecanoylphorbol acetate and rolipram

tetradecanoylphorbol acetate has been researched along with rolipram in 21 studies

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's9 (42.86)18.2507
2000's8 (38.10)29.6817
2010's4 (19.05)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Carmody, LC; Dandapani, S; Donckele, E; Feng, Y; Fernandez, C; Germain, AR; Gupta, PB; Lander, ES; Morgan, B; Munoz, B; Nag, PP; Palmer, M; Perez, JR; Schreiber, SL; Verplank, L1
Alfonso, A; Botana, LM; Botana, MA; Cabado, AG; Louzao, MC; Vieytes, MR1
Schultz, RM1
Turner, NC; Wood, LJ1
Boeckh, C; Gebicke-Härter, P; Meyer, DK; Olenik, C; Theodoridu, A; Ziefer, P1
Bansbach, CC; Caccese, RG; Heaslip, RJ; Lewis, GM1
Koch, B; Lutz-Bucher, B1
Akaike, N; Furukawa, K; Kogure, K1
Angel, JB; Dinarello, CA; Endres, S; Greten, TF; Saget, BM; Skolnik, PR; Walsh, SP1
Carr, DW; Davey, MP; Kasyapa, CS; Stentz, CL1
Blandizzi, C; Colucci, R; Del Tacca, M; Tognetti, M1
Busse, R; Herkert, O; Kuhl, H; Schini-Kerth, VB1
Ahmed, S; Brennan, FM; Feldmann, M; Field, S; Foey, AD; Jain, A; Williams, R1
Irifune, M; Nishikawa, T; Ohnishi, Y; Sato, T; Tanaka, K; Teramoto, T1
Al-Ayadhi, LY; Al-Tuwajri, AS1
Astier, A; Bertrand, C; Jacob, C; Lagente, V; Martin-Chouly, CA; Pruniaux, MP1
Ezeamuzie, CI; Taslim, N1
Baillie, GS; Bird, RJ; Yarwood, SJ1
Adderley, SP; Bowles, EA; Ellsworth, ML; Sprague, RS; Sridharan, M; Stephenson, AH1
Jing, Y; Liao, F; Rao, J; Xi, L; Yang, X; Zou, M1

Other Studies

21 other study(ies) available for tetradecanoylphorbol acetate and rolipram

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells.
    Bioorganic & medicinal chemistry letters, 2013, Mar-15, Volume: 23, Issue:6

    Topics: Amides; Breast Neoplasms; Cell Line, Tumor; Drug Screening Assays, Antitumor; Female; Humans; Neoplastic Stem Cells; Small Molecule Libraries; Structure-Activity Relationship

2013
Influence of protein kinase C, cAMP and phosphatase activity on histamine release produced by compound 48/80 and sodium fluoride on rat mast cells.
    Agents and actions, 1992, Volume: 37, Issue:1-2

    Topics: Animals; Colforsin; Cyclic AMP; Enzyme Activation; Ethers, Cyclic; Histamine Release; In Vitro Techniques; Mast Cells; Okadaic Acid; p-Methoxy-N-methylphenethylamine; Phosphodiesterase Inhibitors; Phosphoprotein Phosphatases; Protein Kinase C; Protein Kinases; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Rolipram; Sodium Fluoride; Tetradecanoylphorbol Acetate

1992
Effect of recombinant human granulocyte/macrophage colony-stimulating factor on neutrophil superoxide production.
    Immunopharmacology and immunotoxicology, 1991, Volume: 13, Issue:1-2

    Topics: Adult; Alkaloids; Cytochalasin B; Granulocyte-Macrophage Colony-Stimulating Factor; Humans; In Vitro Techniques; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Phosphodiesterase Inhibitors; Protein Kinase C; Pyrrolidinones; Rolipram; Signal Transduction; Staurosporine; Superoxides; Tetradecanoylphorbol Acetate

1991
Superoxide generation by guinea-pig peritoneal macrophages is inhibited by rolipram, staurosporine and mepacrine in an agonist-dependent manner.
    Cellular signalling, 1994, Volume: 6, Issue:8

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Alkaloids; Animals; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Guinea Pigs; Macrophages, Peritoneal; Male; N-Formylmethionine Leucyl-Phenylalanine; Phospholipases A; Phospholipases A2; Phosphoric Diester Hydrolases; Platelet Activating Factor; Protein Kinase C; Pyrrolidinones; Quinacrine; Respiratory Burst; Rolipram; Staurosporine; Superoxides; Tetradecanoylphorbol Acetate; Zymosan

1994
Interaction of protein kinases A and C in their effects on the proenkephalin gene in astroglial cells.
    Neurochemistry international, 1994, Volume: 25, Issue:4

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Astrocytes; Cholera Toxin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cycloheximide; Drug Synergism; Enkephalins; Enzyme Activation; Gene Expression Regulation; Protein Kinase C; Protein Precursors; Pyrrolidinones; Rats; RNA, Messenger; Rolipram; Tetradecanoylphorbol Acetate

1994
Effects of rolipram and CI-930 on IL-2 mRNA transcription in human Jurkat cells.
    Agents and actions, 1993, Volume: 39 Spec No

    Topics: Animals; Cell Survival; Humans; Interleukin-2; Lymphocyte Activation; Mice; Mice, Inbred C57BL; Phosphodiesterase Inhibitors; Pyridazines; Pyrrolidinones; RNA, Messenger; Rolipram; Spleen; T-Lymphocytes; Tetradecanoylphorbol Acetate; Transcription, Genetic; Tumor Cells, Cultured

1993
Vasopressin, unlike phorbol ester, fails to synergistically interact with pituitary adenylate cyclase activating polypeptide (PACAP) in stimulating cyclic AMP formation and ACTH secretion in cultured anterior pituitary cells.
    Molecular and cellular endocrinology, 1993, Volume: 92, Issue:2

    Topics: Adrenocorticotropic Hormone; Animals; Arginine Vasopressin; Cells, Cultured; Colforsin; Corticotropin-Releasing Hormone; Cyclic AMP; Drug Interactions; Male; Neuropeptides; Pituitary Adenylate Cyclase-Activating Polypeptide; Pituitary Gland, Anterior; Protein Kinase C; Pyrrolidinones; Rats; Rats, Wistar; Rolipram; Signal Transduction; Tetradecanoylphorbol Acetate

1993
Rolipram enhances the development of voltage-dependent Ca2+ current and serotonin-induced current in rat pheochromocytoma cells.
    Brain research, 1993, Aug-20, Volume: 620, Issue:1

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Acetylcholine; Animals; Calcium; Electrophysiology; Nerve Growth Factors; PC12 Cells; Phosphodiesterase Inhibitors; Pyrrolidinones; Rats; Rolipram; Serotonin; Tetradecanoylphorbol Acetate

1993
Rolipram, a specific type IV phosphodiesterase inhibitor, is a potent inhibitor of HIV-1 replication.
    AIDS (London, England), 1995, Volume: 9, Issue:10

    Topics: Cell Line; Cells, Cultured; HIV Core Protein p24; HIV-1; Humans; Leukocytes, Mononuclear; Lipopolysaccharides; Monocytes; Pentoxifylline; Phosphodiesterase Inhibitors; Pyrrolidinones; RNA, Viral; Rolipram; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha; Virus Replication

1995
Regulation of IL-15-stimulated TNF-alpha production by rolipram.
    Journal of immunology (Baltimore, Md. : 1950), 1999, Sep-01, Volume: 163, Issue:5

    Topics: Adjuvants, Immunologic; Anti-Inflammatory Agents, Non-Steroidal; Antigens, CD; Antigens, Differentiation, T-Lymphocyte; Cells, Cultured; Coculture Techniques; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Humans; Intercellular Adhesion Molecule-1; Interleukin-15; Lectins, C-Type; Lymphocyte Activation; Lymphocyte Function-Associated Antigen-1; Macrophages; Pyrrolidinones; Rolipram; T-Lymphocytes; Tetradecanoylphorbol Acetate; Thionucleotides; Tumor Necrosis Factor-alpha; U937 Cells

1999
Histamine H(3) receptors mediate inhibition of noradrenaline release from intestinal sympathetic nerves.
    British journal of pharmacology, 2000, Volume: 129, Issue:7

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 4-Aminopyridine; Adrenergic alpha-Antagonists; Animals; Calcium; Colforsin; Dose-Response Relationship, Drug; Ethylmaleimide; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Ileum; In Vitro Techniques; Intestinal Mucosa; Intestines; Male; Muscle, Smooth; Myenteric Plexus; Nifedipine; Norepinephrine; omega-Conotoxins; Pertussis Toxin; Phenols; Receptors, Histamine H3; Rolipram; Sympathetic Nervous System; Tetradecanoylphorbol Acetate; Tetraethylammonium; Tetrodotoxin; Virulence Factors, Bordetella; Yohimbine

2000
The progestin levonorgestrel induces endothelium-independent relaxation of rabbit jugular vein via inhibition of calcium entry and protein kinase C: role of cyclic AMP.
    British journal of pharmacology, 2000, Volume: 130, Issue:8

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Calcium; Calcium Chloride; Chlormadinone Acetate; Cyclic AMP; Cyclic GMP; Desogestrel; Dose-Response Relationship, Drug; Endothelium, Vascular; Ethinyl Estradiol; In Vitro Techniques; Jugular Veins; Levonorgestrel; Male; Norpregnenes; Potassium Chloride; Progesterone Congeners; Protein Kinase C; Rabbits; Rolipram; Tetradecanoylphorbol Acetate; Thionucleotides; Vasodilation

2000
Impact of VIP and cAMP on the regulation of TNF-alpha and IL-10 production: implications for rheumatoid arthritis.
    Arthritis research & therapy, 2003, Volume: 5, Issue:6

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Arthritis, Rheumatoid; Bucladesine; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinase Type II; Cyclic AMP-Dependent Protein Kinases; Cyclic Nucleotide Phosphodiesterases, Type 4; Gene Expression Regulation; Humans; Interferon-gamma; Interleukin-10; Ionomycin; Lipopolysaccharides; Macrophages; Monocytes; Phosphodiesterase Inhibitors; Protein Kinase C; Rolipram; Synovial Membrane; T-Lymphocytes; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha; Vasoactive Intestinal Peptide

2003
Inhibitory effects of group II mGluR-related drugs on memory performance in mice.
    Physiology & behavior, 2004, Volume: 80, Issue:5

    Topics: Amino Acids; Animals; Anticonvulsants; Avoidance Learning; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclopropanes; Dose-Response Relationship, Drug; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Glycine; Isoquinolines; Male; Memory; Mice; Reaction Time; Receptors, Metabotropic Glutamate; Rolipram; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Xanthenes

2004
The synergistic effect of adenosine A2A receptors agonist, type IV phosphodiestease inhibitor and ATP-sensitive K channels activation on free radicals production and aggregation of human polymorphoneuclear leukocytes.
    Pharmacological research, 2004, Volume: 50, Issue:2

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenosine; Adenosine A2 Receptor Agonists; Cell Aggregation; Cell Survival; Cromakalim; Cyclic Nucleotide Phosphodiesterases, Type 4; Dose-Response Relationship, Drug; Drug Synergism; Free Radicals; Humans; Luminescent Measurements; Luminol; Neutrophils; Phenethylamines; Phosphodiesterase Inhibitors; Potassium Channels, Inwardly Rectifying; Reactive Oxygen Species; Receptor, Adenosine A2A; Respiratory Burst; Rolipram; Tetradecanoylphorbol Acetate

2004
Modulation of matrix metalloproteinase production from human lung fibroblasts by type 4 phosphodiesterase inhibitors.
    Life sciences, 2004, Jul-02, Volume: 75, Issue:7

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Azepines; Blotting, Western; Bronchodilator Agents; Carboxylic Acids; Cell Line; Cyclic Nucleotide Phosphodiesterases, Type 4; Cyclohexanecarboxylic Acids; Drug Interactions; Drug Therapy, Combination; Fibroblasts; Humans; Isoenzymes; Lung; Matrix Metalloproteinase 1; Matrix Metalloproteinase 2; Metalloproteases; Niacinamide; Nitriles; Phosphodiesterase Inhibitors; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Rolipram; Tetradecanoylphorbol Acetate; Transforming Growth Factor beta; Transforming Growth Factor beta1; Tumor Necrosis Factor-alpha

2004
Protein kinase C- and reactive oxygen species-dependent stimulation of intracellular cAMP in human eosinophils. The role of extracellular signal-regulated protein kinases.
    Medical principles and practice : international journal of the Kuwait University, Health Science Centre, 2008, Volume: 17, Issue:6

    Topics: Cyclic AMP; Eosinophils; Extracellular Signal-Regulated MAP Kinases; Humans; In Vitro Techniques; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Phosphorylation; Protein Kinase C; Reactive Oxygen Species; Rolipram; Signal Transduction; Tetradecanoylphorbol Acetate

2008
Interaction with receptor for activated C-kinase 1 (RACK1) sensitizes the phosphodiesterase PDE4D5 towards hydrolysis of cAMP and activation by protein kinase C.
    The Biochemical journal, 2010, Nov-15, Volume: 432, Issue:1

    Topics: Binding Sites; Blotting, Western; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 3; Cyclic Nucleotide Phosphodiesterases, Type 4; Enzyme Activation; GTP-Binding Proteins; HEK293 Cells; Humans; Hydrolysis; Intracellular Space; Isoproterenol; Kinetics; Mutation; Neoplasm Proteins; Phosphodiesterase 4 Inhibitors; Phosphorylation; Protein Binding; Protein Kinase C; Protein Kinase C-alpha; Protein Transport; Receptors for Activated C Kinase; Receptors, Cell Surface; Rolipram; Tetradecanoylphorbol Acetate; Transfection

2010
Inhibition of ATP release from erythrocytes: a role for EPACs and PKC.
    Microcirculation (New York, N.Y. : 1994), 2011, Volume: 18, Issue:2

    Topics: Adenine; Adenosine Triphosphate; Cilostazol; Colforsin; Cyclic AMP; Enzyme Activation; Erythrocytes; Guanine Nucleotide Exchange Factors; Humans; Iloprost; In Vitro Techniques; Isoproterenol; Models, Biological; Naphthalenes; Phosphodiesterase Inhibitors; Protein Kinase C; Rolipram; Signal Transduction; Tetradecanoylphorbol Acetate; Tetrazoles; Thionucleotides

2011
[Optimization and evaluation of an inflammatory cell model in LPS-stimulated PMA-differentiated THP-1 cells].
    Xi bao yu fen zi mian yi xue za zhi = Chinese journal of cellular and molecular immunology, 2017, Volume: 33, Issue:11

    Topics: Anti-Inflammatory Agents; Cell Differentiation; Humans; Inflammation Mediators; Interleukin-6; Leukemia, Monocytic, Acute; Lipopolysaccharides; Macrophages; Models, Biological; Phosphodiesterase 4 Inhibitors; Rolipram; Tetradecanoylphorbol Acetate; THP-1 Cells; Tumor Necrosis Factor-alpha

2017