tetradecanoylphorbol acetate has been researched along with h 89 in 93 studies
Timeframe | Studies, this research(%) | All Research% |
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pre-1990 | 0 (0.00) | 18.7374 |
1990's | 46 (49.46) | 18.2507 |
2000's | 37 (39.78) | 29.6817 |
2010's | 9 (9.68) | 24.3611 |
2020's | 1 (1.08) | 2.80 |
Authors | Studies |
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Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J | 1 |
Hidaka, H; Kanda, K; Matsui, N; Miyamoto, N; Seo, H | 1 |
Iwanaga, M; Sano, M | 1 |
Geilen, CC; Reutter, W; Wieder, T; Wieprecht, M | 1 |
Allen, JM; Balbi, D | 1 |
Azarani, A; Goltzman, D; Orlowski, J | 1 |
Catravas, JD; Ganapathy, V; Leibach, FH; Papapetropoulos, A; Ramamoorthy, JD; Ramamoorthy, S | 1 |
Alvaro, D; Bini, A; Capocaccia, L; Della Guardia, P; Furfaro, S; Gigliozzi, A; La Rosa, T; Piat, C | 1 |
Deleu, L; Faisst, S; Kherrouche, Z; Perros, M; Rommelaere, J; Spruyt, N; Vanacker, JM | 1 |
Abe, M; Furuno, T; Hara, N; Hidaka, K; Mitsuyama, T; Takeshige, K; Tanaka, T | 1 |
Agell, N; Bachs, O; Bosch, M; López-Girona, A | 1 |
Chan, KF; Loh, TT; Lok, CN | 1 |
De Lisle, RC; Howell, GW | 1 |
Baldi, G; Bevilacqua, M; Dallegri, F; Norbiato, G; Renesto, E; Vago, T | 1 |
Linder, S; Shoshan, MC | 1 |
Fujimura, S; Kato, N; Miya, T; Sato, K; Tagawa, M; Takahashi, K | 1 |
Kubota, C; Murata, Y; Shinagawa, T; Shinohara, O | 1 |
Kessels, GC; Krause, KH; Verhoeven, AJ | 1 |
Fujihara, M; Ito, N; Muroi, M; Muroi, Y; Suzuki, T | 1 |
Muroi, M; Suzuki, T | 1 |
Ikeda, K; Takasaka, T; Wu, D | 1 |
Bosche, MC; Levine, RA; Nandi, J; Rotker, JD; Strapko, A | 1 |
Dittrich, C; Grill, S; Harant, H; Huber, H; Hulla, W; Krupitza, G; Szekeres, T | 1 |
Benz, D; Möller, K; Perrin, D; Söling, HD | 1 |
Nishikawa, T; Omura, M; Sasano, H; Suematsu, S | 1 |
Linder, S; Ljungdahl, S; Shoshan, MC | 1 |
Carson, DD; Ding, ZM; Kuo, MT; Wegner, CC; Zhou, X | 1 |
Downing, JR; Garcia, JV; Luo, T | 1 |
Body, JJ; Lacroix, M | 1 |
Chen, C; Clarke, IJ; Wu, D | 1 |
Böl, GF; Hülster, A; Pfeuffer, T | 1 |
Feltkamp, D; Gustafsson, JA; Huang, CJ; Nilsson, S | 1 |
Attardi, B; Winters, SJ | 1 |
Greene, RM; Lloyd, MR; Potchinsky, MB; Weston, WM | 1 |
Reenstra, WW; Yurko-Mauro, KA | 1 |
Kimura, M; Ogihara, M | 2 |
Kobayashi, M; Kuroda, A; Maruyama, M; Mino, T; Sugiyama, E; Taki, H; Yamashita, N | 1 |
Solem, ML; Thomas, AP | 1 |
Had-Aissouni, L; Kerkerian-Le Goff, L; Lortet, S; Masmejean, F; Pisano, P; Samuel, D | 1 |
Fukuda, J; Kagabu, S; Karube, A; Kodama, H; Murata, M; Tanaka, T | 1 |
Davis, JR; Ray, DW; Reem, GH | 1 |
Abad, C; Delgado, M; Ganea, D; Gomariz, RP; Leceta, J; Martinez, C | 1 |
Brown, EJ; Wang, J | 1 |
Barratt, MJ; Clayton, AL; Hazzalin, CA; Mahadevan, LC; Rose, S; Thomson, S | 1 |
Huang, YT; Lee, MT; Lin, JK | 1 |
Lesslauer, W; Mary, JL; Tomás-Zuber, M | 1 |
Dunkerley, HA; Jimmo, SL; Liu, H; Maurice, DH; Palmer, D; Pang, SC; Tilley, DG | 1 |
Kataoka, K; Nakamura, Y; Si, Q | 1 |
Chang, CH; Chang, TM; Chey, WY | 1 |
Kubo, Y; Miyashita, T | 1 |
Fujita, N; Higashiyama, M; Honda, K; Ishikawa, S; Kusaka, I; Okada, K; Saito, T | 1 |
Hermans, E; Maloteaux, JM; Najimi, M; Page, G; Peeters, M | 1 |
Hontela, A; Lacroix, M | 1 |
Bauer, CK; Schledermann, W; Schwarz, JR; Wulfsen, I | 1 |
Låg, M; Refsnes, M; Schwarze, PE; Thoresen, GH; Thrane, EV | 1 |
Ding, WQ; Holicky, E; Miller, LJ | 1 |
Beckmann, JD; Kai, M; Keeton, TP; Stewart, A | 1 |
Arima, N; Hamada, T; Kimura, S; Murata, Y; Nomaguchi, M; Sasaguri, Y; Tanimoto, A; Xu, H | 1 |
Dudas, PL; Gocek-Sutterlin, G; Laverty, G; Renfro, JL; Villalobos, AR | 1 |
Bachteeva, VT; Fock, EM; Lavrova, EA; Naboka, EV; Parnova, RG | 1 |
Cho, YJ; Jeong, SW; Kim, JY; Kim, ON; Lee, SB | 1 |
Hsu, CC; Huang, BM; Huang, YL; Tsai, SJ | 1 |
Pacheco, MA; Pastoor, TE; Wecker, L | 1 |
Carlson, RR; Dudman, JT; Konradi, C; Macías, W | 1 |
Irifune, M; Nishikawa, T; Ohnishi, Y; Sato, T; Tanaka, K; Teramoto, T | 1 |
Cho, YW; Hahm, ET; Lee, JJ; Min, BI | 1 |
Diniz, C; Fresco, P; Gonçalves, J | 1 |
Bretschneider, E; Censarek, P; Fischer, JW; Meyer-Kirchrath, J; Pape, R; Rabausch, K; Sarbia, M; Schrör, K; Weber, AA | 1 |
Amsterdam, A; Fukuda, S; Kotsuji, F; Miyamoto, K; Orisaka, M; Tajima, K; Yoshii, K | 1 |
Allagnat, F; Condorelli, DF; Haefliger, JA; Martin, D; Waeber, G | 1 |
Canaff, L; Chihara, K; Hendy, GN; Kaji, H; Naito, J; Sowa, H; Sugimoto, T; Tobimatsu, T | 1 |
Ikewaki, N; Inoko, H; Kulski, JK | 1 |
Linsdell, P; McDonald, TF; Missan, S | 1 |
Chen, YH; Tsai, MC | 1 |
Jo, Y; Manna, PR; Stocco, DM | 1 |
Carlson, AE; Franceschi, RT; Gopalakrishnan, R; Suttamanatwong, S | 1 |
Becu-Villalobos, D; Díaz-Torga, G; Pérez-Millán, MI; Vela, J | 1 |
Avkiran, M; Cuello, F; Haworth, RS; Roberts, NA | 1 |
Bode, AM; Cho, YY; Dong, Z; Kang, NJ; Kim, HG; Lee, KW; Oh, SM | 1 |
Garcia, N; Lanuza, MA; Santafé, MM; Tomàs, J; Tomàs, M | 1 |
Ackermann, TF; Bhandaru, M; Boini, KM; Lang, F; Rotte, A | 1 |
Fei, XW; He, YL; Mei, YA; Yang, G; Zhang, M | 1 |
Miao, Y; Wang, Z; Yang, XL; Zhang, M; Zhao, WJ | 1 |
Ceballos, NR; Volonteri, MC | 1 |
Arun, SN; Bollag, WB; Dodd, ME; Xie, D; Zhong, X | 1 |
Cao, AL; Liu, HY; Zeng, WD; Zhang, CQ | 1 |
Chouinard, L; Gallo-Payet, N; Pinard, S; Roy, S | 1 |
Aguiar, JF; Costa, RR; Reis, RI; Varanda, WA | 1 |
Akamatsu, T; Azlina, A; Hasegawa, T; Hosoi, K; Javkhlan, P; Yao, C | 1 |
Akaaboune, M; Martinez-Pena y Valenzuela, I; Pires-Oliveira, M | 1 |
Liu, C; Shu, L; Su, G; Xu, J; Zhang, J; Zhang, W | 1 |
Adewumi, I; Beacon, TH; Davie, JR; Hu, P; Jia, S; López, C; Sharma, KL; Xu, W | 1 |
93 other study(ies) available for tetradecanoylphorbol acetate and h 89
Article | Year |
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Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection | 2009 |
A 3',5'-cyclic adenosine monophosphate-dependent pathway is responsible for a rapid increase in c-fos messenger ribonucleic acid by adrenocorticotropin.
Topics: Adrenal Glands; Adrenocorticotropic Hormone; Animals; Bucladesine; Cells, Cultured; Corticosterone; Cyclic AMP; Cycloheximide; Gene Expression; Genes, fos; Isoquinolines; Kinetics; Male; Potassium; Protein Kinase Inhibitors; Protein Kinases; Rats; Rats, Inbred Strains; RNA, Messenger; Sulfonamides; Tetradecanoylphorbol Acetate | 1992 |
Requirement for specific protein kinase activities during the rapid redistribution of F-actin that precedes the outgrowth of neurites in PC12D cells.
Topics: Actins; Animals; Bucladesine; Carbazoles; Colchicine; Cytochalasin B; Cytoskeleton; Epidermal Growth Factor; Fibroblast Growth Factor 2; Indole Alkaloids; Isoquinolines; Nerve Growth Factors; Neurons; Protein Kinases; Rats; Sulfonamides; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1992 |
A selective inhibitor of cyclic AMP-dependent protein kinase, N-[2-bromocinnamyl(amino)ethyl]-5-isoquinolinesulfonamide (H-89), inhibits phosphatidylcholine biosynthesis in HeLa cells.
Topics: Colforsin; HeLa Cells; Humans; Isoquinolines; Kinetics; Phosphatidylcholines; Protein Kinase Inhibitors; Sulfonamides; Tetradecanoylphorbol Acetate | 1992 |
Role of protein kinase C in mediating NGF effect on neuropeptide Y expression in PC12 cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Base Sequence; Binding Sites; Blotting, Northern; Bucladesine; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cycloheximide; Gene Expression; Isoquinolines; Kinetics; Molecular Sequence Data; Naphthalenes; Nerve Growth Factors; Neuropeptide Y; Oligodeoxyribonucleotides; PC12 Cells; Piperazines; Polycyclic Compounds; Promoter Regions, Genetic; Protein Kinase C; RNA, Messenger; Sulfonamides; Tetradecanoylphorbol Acetate; Transcription, Genetic | 1994 |
Parathyroid hormone and parathyroid hormone-related peptide activate the Na+/H+ exchanger NHE-1 isoform in osteoblastic cells (UMR-106) via a cAMP-dependent pathway.
Topics: Animals; Bone Neoplasms; Cell Line; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cytosol; Enzyme Inhibitors; Humans; Isoquinolines; Kinetics; Osteosarcoma; Parathyroid Hormone; Parathyroid Hormone-Related Protein; Protein Kinase C; Proteins; Rats; Recombinant Proteins; Second Messenger Systems; Sodium-Hydrogen Exchangers; Sulfonamides; Tetradecanoylphorbol Acetate; Transfection; Tumor Cells, Cultured | 1995 |
Cyclic AMP-independent up-regulation of the human serotonin transporter by staurosporine in choriocarcinoma cells.
Topics: Alkaloids; Carrier Proteins; Cholera Toxin; Choriocarcinoma; Cocaine; Cyclic AMP; Cyclic GMP; Cycloheximide; Dactinomycin; Female; Humans; Isoquinolines; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Pregnancy; RNA, Messenger; Serotonin; Serotonin Plasma Membrane Transport Proteins; Staurosporine; Sulfonamides; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Up-Regulation | 1995 |
Effect of glucagon on intracellular pH regulation in isolated rat hepatocyte couplets.
Topics: Animals; Antiporters; Bicarbonates; Bile; Bucladesine; Cells, Cultured; Chloride-Bicarbonate Antiporters; Chlorides; Cholagogues and Choleretics; Colchicine; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Glucagon; Hydrogen-Ion Concentration; Intracellular Fluid; Isoquinolines; Liver; Male; Nitrobenzoates; Rats; Rats, Wistar; Sodium; Sodium-Hydrogen Exchangers; Sulfonamides; Tetradecanoylphorbol Acetate; Thionucleotides | 1995 |
Upstream CREs participate in the basal activity of minute virus of mice promoter P4 and in its stimulation in ras-transformed cells.
Topics: Alkaloids; Animals; Base Sequence; Bucladesine; Cell Line; Cell Line, Transformed; Cell Nucleus; Cyclic AMP-Dependent Protein Kinases; DNA, Viral; Gene Expression Regulation, Viral; Genes, ras; Isoquinolines; Kinetics; Minute Virus of Mice; Molecular Sequence Data; Nucleic Acid Conformation; Plasmids; Promoter Regions, Genetic; Rats; Rats, Inbred F344; Regulatory Sequences, Nucleic Acid; Staurosporine; Sulfonamides; TATA Box; Tetradecanoylphorbol Acetate; Transcription Factors; Transcription, Genetic; Viral Nonstructural Proteins | 1995 |
An inhibitor of cyclic AMP-dependent protein kinase enhances the superoxide production of human neutrophils stimulated by N-formyl-methionyl-leucyl-phenylalanine.
Topics: Bucladesine; Calcium; Cell Membrane Permeability; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Isoquinolines; Male; N-Formylmethionine Leucyl-Phenylalanine; Neutrophil Activation; Neutrophils; Respiratory Burst; Signal Transduction; Sodium Dodecyl Sulfate; Sulfonamides; Superoxides; Tetradecanoylphorbol Acetate | 1995 |
Protein kinase C regulates calmodulin expression in NRK cells activated to proliferate from quiescence.
Topics: Alkaloids; Animals; Calmodulin; Cattle; Cell Division; Cell Line; Contact Inhibition; Culture Media; Culture Media, Serum-Free; Cyclic AMP-Dependent Protein Kinases; DNA Replication; Epithelial Cells; Epithelium; Fetal Blood; Gene Expression Regulation; Ionomycin; Isoquinolines; Kidney; Protein Kinase C; Rats; RNA, Messenger; Staurosporine; Sulfonamides; Tetradecanoylphorbol Acetate; Transcription, Genetic | 1994 |
Effects of protein kinase modulators on transferrin receptor expression in human leukaemic HL-60 cells.
Topics: Alkaloids; Bucladesine; Cell Division; Cell Line; Cyclic AMP-Dependent Protein Kinases; DNA, Neoplasm; Enzyme Activation; Gene Expression; Humans; Indoles; Isoquinolines; Leukemia, Promyelocytic, Acute; Maleimides; Protein Kinase C; Protein Kinases; Receptors, Transferrin; RNA, Messenger; Staurosporine; Sulfonamides; Tetradecanoylphorbol Acetate; Thymidine; Tumor Cells, Cultured | 1995 |
Evidence of heterotrimeric G-protein involvement in regulated exocytosis from permeabilized pancreatic acini.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Bacterial Proteins; Calcium; Cell Membrane Permeability; Cholera Toxin; Cyclic AMP; Exocytosis; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Intercellular Signaling Peptides and Proteins; Isoquinolines; Macromolecular Substances; Mice; Pancreas; Peptides; Pertussis Toxin; Protein Kinase Inhibitors; Streptolysins; Sulfonamides; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella; Wasp Venoms | 1995 |
Nimesulide decreases superoxide production by inhibiting phosphodiesterase type IV.
Topics: Adenylyl Cyclases; Anti-Inflammatory Agents, Non-Steroidal; Blood Platelets; Cell Membrane; Chemotaxis, Leukocyte; Cyclic AMP; Humans; In Vitro Techniques; Isoquinolines; N-Formylmethionine Leucyl-Phenylalanine; NADH, NADPH Oxidoreductases; Neutrophils; Oxygen Consumption; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Protein Kinase Inhibitors; Sulfonamides; Superoxides; Tetradecanoylphorbol Acetate | 1994 |
Induction of the collagenase phorbol ester response element by staurosporine.
Topics: Alkaloids; Animals; Cell Line; Cell Line, Transformed; Collagen; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Edetic Acid; Fibroblasts; Gene Expression; Genes, jun; Genes, ras; Isoquinolines; Kinetics; Oncogene Protein p65(gag-jun); Promoter Regions, Genetic; Protein Kinase C; Proto-Oncogene Proteins c-jun; Rats; Regulatory Sequences, Nucleic Acid; RNA, Messenger; Staurosporine; Sulfonamides; Tetradecanoylphorbol Acetate | 1994 |
Prostaglandin E2/parathyroid hormone-induced suppression of alkaline phosphatase activity is mediated by protein kinase C.
Topics: Alkaline Phosphatase; Alkaloids; Animals; Bucladesine; Calcimycin; Cyclic AMP; Cycloheximide; Dinoprostone; Isoquinolines; Osteoblasts; Osteosarcoma; Parathyroid Hormone; Protein Kinase C; Rats; Staurosporine; Sulfonamides; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1994 |
Protein kinase C inhibitors enhance differentiation of rat adipocyte precursor cells in serum-free culture.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adipose Tissue; Alkaloids; Animals; Cell Differentiation; Cells, Cultured; Culture Media, Serum-Free; Glycerolphosphate Dehydrogenase; Isoquinolines; Male; Piperazines; Protein Kinase C; Rats; Staurosporine; Sulfonamides; Tetradecanoylphorbol Acetate | 1994 |
Protein kinase C activity is not involved in N-formylmethionyl-leucyl-phenylalanine-induced phospholipase D activation in human neutrophils, but is essential for concomitant NADPH oxidase activation: studies with a staurosporine analogue with improved sel
Topics: Alkaloids; Bucladesine; Enzyme Activation; Humans; In Vitro Techniques; Isoquinolines; Kinetics; N-Formylmethionine Leucyl-Phenylalanine; NADH, NADPH Oxidoreductases; NADPH Oxidases; Neutrophils; Phospholipase D; Protein Kinase C; Staurosporine; Sulfonamides; Superoxides; Tetradecanoylphorbol Acetate | 1993 |
Mechanism of lipopolysaccharide-triggered junB activation in a mouse macrophage-like cell line (J774).
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Base Sequence; Cell Line; Cyclic AMP; Female; Isoquinolines; Lipopolysaccharides; Macrophages; Mice; Mice, Inbred BALB C; Molecular Sequence Data; Oligodeoxyribonucleotides; Piperazines; Protein Kinase C; Proto-Oncogene Proteins c-jun; RNA, Messenger; Sulfonamides; Tetradecanoylphorbol Acetate | 1993 |
Role of protein kinase A in LPS-induced activation of NF-kappa B proteins of a mouse macrophage-like cell line, J774.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amino Acid Sequence; Animals; Base Sequence; Bucladesine; Cholera Toxin; Colforsin; Consensus Sequence; Cyclic AMP; Dinoprostone; Female; Gene Expression Regulation, Neoplastic; Isoquinolines; Lipopolysaccharides; Macrophage Activation; Macrophages; Mice; Mice, Inbred BALB C; Molecular Sequence Data; Neoplasm Proteins; NF-kappa B; Phosphorylation; Piperazines; Protein Kinases; Protein Processing, Post-Translational; Proto-Oncogene Proteins; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Transcription Factor RelB; Transcription Factors; Transcription, Genetic; Tumor Cells, Cultured | 1993 |
Cellular mechanisms in activation of Na-K-Cl cotransport in nasal gland acinar cells of guinea pigs.
Topics: Acetylcholine; Alkaloids; Animals; Benzophenanthridines; Biological Transport; Bucladesine; Bumetanide; Calcium; Calmodulin; Carrier Proteins; Charybdotoxin; Cholinergic Fibers; Cyclic AMP; Cyclic GMP; Enzyme Inhibitors; Exocrine Glands; Furosemide; Guinea Pigs; Ionomycin; Ionophores; Isoquinolines; Nasal Cavity; Phenanthridines; Protein Kinase Inhibitors; Protein Kinases; Second Messenger Systems; Signal Transduction; Sodium; Sodium-Potassium-Chloride Symporters; Sulfonamides; Tetradecanoylphorbol Acetate; Trifluoperazine; Vasoactive Intestinal Peptide | 1995 |
Effects of cyclic adenosine monophosphate-dependent protein kinase and calcium-dependent protein kinase modulators on stimulated gastric acid secretion in the perfused rat stomach.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Administration, Oral; Animals; Calcium; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Gastric Acid; Histamine; Injections, Intravenous; Isoquinolines; Male; Naphthalenes; Pentagastrin; Piperazines; Protein Kinase C; Rats; Rats, Sprague-Dawley; Sulfonamides; Tetradecanoylphorbol Acetate | 1995 |
Genes related to growth and invasiveness are repressed by sodium butyrate in ovarian carcinoma cells.
Topics: Adenylyl Cyclases; Butyrates; Butyric Acid; Cell Division; Cell Line; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cyclin D1; Cyclins; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Gene Expression Regulation, Neoplastic; Humans; Intercellular Signaling Peptides and Proteins; Isoquinolines; Neoplasm Invasiveness; Oncogene Proteins; Oncogenes; Ovarian Neoplasms; Protein Kinase C; Proteins; RNA, Messenger; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Transcription, Genetic; Tumor Cells, Cultured; Urokinase-Type Plasminogen Activator | 1996 |
The role of protein kinase C in carbachol-induced and of cAMP-dependent protein kinase in isoproterenol-induced secretion in primary cultured guinea pig parotid acinar cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; alpha-Amylases; Animals; Calcium; Carbachol; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Down-Regulation; Enzyme Inhibitors; Exocytosis; Guinea Pigs; Immunoblotting; Isoproterenol; Isoquinolines; Male; Parotid Gland; Phorbol 12,13-Dibutyrate; Piperazines; Protein Binding; Protein Kinase C; Sulfonamides; Tetradecanoylphorbol Acetate | 1996 |
Regulation of expression of the steroidogenic acute regulatory (StAR) protein by ACTH in bovine adrenal fasciculata cells.
Topics: Adrenocorticotropic Hormone; Animals; Bucladesine; Calcimycin; Cattle; Cells, Cultured; Colforsin; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gene Expression Regulation; Hydrocortisone; Immunohistochemistry; Isoquinolines; Kinetics; Naphthalenes; Phosphoproteins; Quinazolines; Sulfonamides; Tetradecanoylphorbol Acetate; Zona Fasciculata | 1996 |
H-89 inhibits collagenase induction by phorbol ester through a mechanism that does not involve protein kinase A.
Topics: Animals; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line, Transformed; Collagenases; Cyclic AMP-Dependent Protein Kinases; Genes, jun; Isoquinolines; Matrix Metalloproteinase Inhibitors; Rats; RNA, Messenger; Sulfonamides; Tetradecanoylphorbol Acetate | 1996 |
Tyrosine kinase inhibition decreases Muc-1 expression in mouse epithelial cells.
Topics: 1-Methyl-3-isobutylxanthine; Amino Acid Sequence; Animals; Antibodies; Base Sequence; Cell Line; Cells, Cultured; Conserved Sequence; DNA Primers; Enzyme Inhibitors; Epithelium; Female; Gene Expression; Genistein; Isoflavones; Isoquinolines; Kinetics; Mammary Glands, Animal; Mice; Molecular Sequence Data; Mucin-1; Naphthalenes; Peptide Fragments; Polymerase Chain Reaction; Pregnancy; Protein Biosynthesis; Protein-Tyrosine Kinases; Recombinant Fusion Proteins; RNA, Messenger; Staurosporine; Sulfonamides; Tetradecanoylphorbol Acetate; Transcription, Genetic; Transfection; Uterus | 1997 |
Induction of phosphorylation of human immunodeficiency virus type 1 Nef and enhancement of CD4 downregulation by phorbol myristate acetate.
Topics: CD4 Antigens; CD4-Positive T-Lymphocytes; Cyclic AMP-Dependent Protein Kinases; Down-Regulation; Enzyme Inhibitors; Gene Products, nef; HIV-1; Humans; Indoles; Isoquinolines; Maleimides; nef Gene Products, Human Immunodeficiency Virus; Phosphorylation; Phytohemagglutinins; Protein Kinase C; Recombinant Fusion Proteins; Serine; Sulfonamides; Tetradecanoylphorbol Acetate | 1997 |
Regulation of c-fos and c-jun expression by calcitonin in human breast cancer cells.
Topics: Blotting, Northern; Breast Neoplasms; Calcitonin; Carcinogens; Cell Division; Colforsin; Dose-Response Relationship, Drug; Drug Interactions; Epidermal Growth Factor; Female; Gene Expression Regulation, Neoplastic; Genes, fos; Genes, jun; Glycoproteins; Humans; Insulin; Isoquinolines; Metalloendopeptidases; Protein Biosynthesis; Protein Kinase Inhibitors; Proteins; Receptors, Calcitonin; RNA, Messenger; Sulfonamides; Tetradecanoylphorbol Acetate; Tissue Inhibitor of Metalloproteinase-2; Tissue Inhibitor of Metalloproteinases; Tumor Cells, Cultured | 1997 |
The role of protein kinase C in GH secretion induced by GH-releasing factor and GH-releasing peptides in cultured ovine somatotrophs.
Topics: Alkaloids; Animals; Benzophenanthridines; Carcinogens; Cell Membrane; Cells, Cultured; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cytosol; Dose-Response Relationship, Drug; Enzyme Inhibitors; Growth Hormone; Growth Hormone-Releasing Hormone; Isoquinolines; Naphthalenes; Oligopeptides; Phenanthridines; Pituitary Gland; Protein Kinase C; Second Messenger Systems; Sheep; Staurosporine; Sulfonamides; Tetradecanoylphorbol Acetate; Time Factors | 1997 |
Adenylyl cyclase type II is stimulated by PKC via C-terminal phosphorylation.
Topics: Adenylyl Cyclases; Cell Line; Enzyme Inhibitors; Humans; Isoenzymes; Isoquinolines; Kidney; Macromolecular Substances; Peptide Fragments; Phosphates; Phosphorylation; Protein Kinase C; Protein Kinase Inhibitors; Protein Kinases; Recombinant Proteins; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Transfection | 1997 |
Synergistic activation of RLD-1 by agents triggering PKA and PKC dependent signalling.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; CHO Cells; Colforsin; Cricetinae; Cyclic AMP-Dependent Protein Kinases; Dinoprostone; DNA-Binding Proteins; Drug Synergism; Enzyme Inhibitors; Genes, Reporter; Hydroxycholesterols; Indoles; Isoquinolines; Liver X Receptors; Maleimides; Orphan Nuclear Receptors; Protein Kinase C; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Receptors, Thyroid Hormone; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Transfection | 1998 |
Transcriptional regulation of the glycoprotein hormone alpha-subunit gene by pituitary adenylate cyclase-activating polypeptide (PACAP) in alphaT3-1 cells.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Base Sequence; Cell Line; Cyclic AMP-Dependent Protein Kinases; DNA; Enzyme Inhibitors; Genes, Reporter; Glycoprotein Hormones, alpha Subunit; Gonadotropin-Releasing Hormone; Isoquinolines; Luciferases; Mice; Neuropeptides; Pituitary Adenylate Cyclase-Activating Polypeptide; Promoter Regions, Genetic; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Transcriptional Activation; Transfection | 1998 |
Selective modulation of MAP kinase in embryonic palate cells.
Topics: Animals; Calcimycin; Carcinogens; Cells, Cultured; Cholera Toxin; Cyclic AMP; Endothelial Growth Factors; Enzyme Activation; Enzyme Inhibitors; Fetus; Flavonoids; Ionophores; Isoquinolines; MAP Kinase Kinase 1; MAP Kinase Kinase 2; Mice; Mice, Inbred ICR; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase Kinases; Palate; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Transforming Growth Factor beta | 1998 |
Prostaglandin F2alpha stimulates CFTR activity by PKA- and PKC-dependent phosphorylation.
Topics: 3T3 Cells; Animals; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cystic Fibrosis Transmembrane Conductance Regulator; Dinoprost; Enzyme Inhibitors; Inositol 1,4,5-Trisphosphate; Iodides; Isoquinolines; Kinetics; Mice; Phosphopeptides; Phosphorylation; Protein Kinase C; Recombinant Proteins; Staurosporine; Sulfonamides; Tetradecanoylphorbol Acetate; Transfection | 1998 |
Effects of insulin-like growth factor I and II on DNA synthesis and proliferation in primary cultures of adult rat hepatocytes.
Topics: Animals; Brimonidine Tartrate; Cell Count; Cell Division; Cyclic AMP; DNA; Dose-Response Relationship, Drug; Drug Interactions; Insulin-Like Growth Factor I; Insulin-Like Growth Factor II; Isoquinolines; Liver; Male; Metaproterenol; Phenylephrine; Quinoxalines; Rats; Rats, Wistar; Signal Transduction; Sphingosine; Sulfonamides; Tetradecanoylphorbol Acetate; Time Factors | 1998 |
Interleukin-1alpha and tumor necrosis factor alpha synergistically stimulate prostaglandin E2-dependent production of interleukin-11 in rheumatoid synovial fibroblasts.
Topics: Arthritis, Rheumatoid; Carcinogens; Cells, Cultured; Dinoprostone; Drug Synergism; Enzyme Inhibitors; Fibroblasts; Gene Expression Regulation, Enzymologic; Humans; Indoles; Interleukin-1; Interleukin-11; Isoquinolines; Maleimides; Protein Kinase C; Signal Transduction; Sulfonamides; Synovial Membrane; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha | 1998 |
Modulation of cardiac Ca2+ channels by IGF1.
Topics: Animals; Calcium; Calcium Channels; Carbazoles; Cells, Cultured; Chromones; Cytosol; Enzyme Inhibitors; Heart; Humans; Indoles; Insulin-Like Growth Factor I; Isoquinolines; Kinetics; Male; Manganese; Morpholines; Protein Kinase C; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Sarcolemma; Sulfonamides; Tetradecanoylphorbol Acetate | 1998 |
Effects of PKA and PKC modulators on high affinity glutamate uptake in primary neuronal cell cultures from rat cerebral cortex.
Topics: Alkaloids; Animals; Benzophenanthridines; Biological Transport; Cells, Cultured; Cerebral Cortex; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Fetus; Glutamic Acid; Isoquinolines; Kinetics; Neurons; Phenanthridines; Protein Kinase C; Rats; Rats, Wistar; Sulfonamides; Tetradecanoylphorbol Acetate | 1999 |
Inhibitory effects of nitric oxide on the expression and activity of aromatase in human granulosa cells.
Topics: Adult; Aromatase; Aromatase Inhibitors; Cells, Cultured; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Female; Gene Expression Regulation; Granulosa Cells; Humans; Isoquinolines; Nitrates; Nitric Oxide; Penicillamine; Protein Kinase C; Sodium Nitrite; Sulfonamides; Tetradecanoylphorbol Acetate; Transcription, Genetic | 1999 |
The human prolactin gene upstream promoter is regulated in lymphoid cells by activators of T-cells and by cAMP.
Topics: Base Sequence; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Cyclosporine; DNA Primers; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gene Expression Regulation; Humans; Isoquinolines; Jurkat Cells; Lymphocyte Activation; Phosphoprotein Phosphatases; Phytohemagglutinins; Prolactin; Promoter Regions, Genetic; Protein Binding; Sulfonamides; Tetradecanoylphorbol Acetate; Transfection | 1999 |
Regulation of VIP production and secretion by murine lymphocytes.
Topics: Animals; Carcinogens; Cell Division; Cells, Cultured; Colforsin; Dexamethasone; Enzyme Inhibitors; Enzyme-Linked Immunosorbent Assay; Feedback; Flow Cytometry; Glucocorticoids; Granulocytes; Interleukin-1; Interleukin-2; Interleukin-6; Isoquinolines; Lymph Nodes; Macrophages, Peritoneal; Male; Mast Cells; Mitogens; Neuroimmunomodulation; Peritoneum; Rats; Rats, Wistar; Retinaldehyde; Sensitivity and Specificity; Spleen; Sulfonamides; Tetradecanoylphorbol Acetate; Thymus Gland; Tumor Necrosis Factor-alpha; Vasoactive Intestinal Peptide | 1999 |
Immune complex-induced integrin activation and L-plastin phosphorylation require protein kinase A.
Topics: Amino Acid Sequence; Antigen-Antibody Complex; Carbazoles; Cell Adhesion; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Indoles; Isoquinolines; Macrophage-1 Antigen; Membrane Glycoproteins; Microfilament Proteins; Molecular Sequence Data; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Phosphatidylinositol 3-Kinases; Phosphoproteins; Phosphorylation; Pyrroles; Receptors, IgG; Serine; Sulfonamides; Tetradecanoylphorbol Acetate | 1999 |
The nucleosomal response associated with immediate-early gene induction is mediated via alternative MAP kinase cascades: MSK1 as a potential histone H3/HMG-14 kinase.
Topics: Animals; Anisomycin; Blotting, Western; Calcium-Calmodulin-Dependent Protein Kinases; Cells, Cultured; Enzyme Inhibitors; Fibroblasts; Gene Expression Regulation, Enzymologic; Genes, Immediate-Early; High Mobility Group Proteins; Histones; Isoquinolines; Mice; Mice, Inbred C3H; Mitogen-Activated Protein Kinases; Models, Biological; Nucleosomes; Phosphorylation; Protein Synthesis Inhibitors; Proto-Oncogene Proteins c-fos; Proto-Oncogene Proteins c-jun; Ribosomal Protein S6 Kinases, 90-kDa; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Time Factors; Transcriptional Activation | 1999 |
Stimulation by transforming growth factor-alpha of DNA synthesis and proliferation of adult rat hepatocytes in primary cultures: modulation by alpha- and beta-adrenoceptor agonists.
Topics: Adrenergic alpha-Agonists; Adrenergic Antagonists; Adrenergic beta-Agonists; Animals; Anti-Inflammatory Agents; Antibodies, Monoclonal; Brimonidine Tartrate; Cell Division; Cells, Cultured; Dexamethasone; DNA; Dose-Response Relationship, Drug; Drug Interactions; ErbB Receptors; Isoquinolines; Liver; Male; Metaproterenol; Mitogen-Activated Protein Kinase Kinases; Phenylephrine; Phosphatidylinositol 3-Kinases; Protein Kinase C; Protein Kinases; Quinoxalines; Rats; Rats, Wistar; Receptor Protein-Tyrosine Kinases; Ribosomal Protein S6 Kinases; Signal Transduction; Sphingosine; Sulfonamides; Tetradecanoylphorbol Acetate; Time Factors; Transforming Growth Factor alpha; Type C Phospholipases | 1999 |
Inhibition of 12-O-tetradecanoylphorbol-13-acetate induction of c-fos mRNA by the protein kinase A inhibitor N-[2-(p-bromocinnamylamino)ethyl]-5-isoquinoline sulfonamide.
Topics: 3T3 Cells; Animals; Carcinogens; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Drug Interactions; Enzyme Inhibitors; Isoquinolines; Mice; Proto-Oncogene Proteins c-fos; RNA, Messenger; Sulfonamides; Tetradecanoylphorbol Acetate; Transcription, Genetic | 1999 |
Control sites of ribosomal S6 kinase B and persistent activation through tumor necrosis factor.
Topics: Amino Acid Sequence; Catalytic Domain; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Inhibitors; Epidermal Growth Factor; HeLa Cells; Humans; Indoles; Insulin; Ionomycin; Isoquinolines; Mitogen-Activated Protein Kinases; Molecular Sequence Data; Phosphorylation; Protein Binding; Protein Kinase C; Protein Structure, Tertiary; Recombinant Proteins; Ribosomal Protein S6 Kinases; Serine; Signal Transduction; Substrate Specificity; Sulfonamides; Tetradecanoylphorbol Acetate; Threonine; Tumor Necrosis Factor-alpha | 2000 |
Expression of phosphodiesterase 4D (PDE4D) is regulated by both the cyclic AMP-dependent protein kinase and mitogen-activated protein kinase signaling pathways. A potential mechanism allowing for the coordinated regulation of PDE4D activity and expression
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; 8-Bromo Cyclic Adenosine Monophosphate; Angiotensin II; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclic Nucleotide Phosphodiesterases, Type 4; Cycloheximide; Dactinomycin; Enzyme Inhibitors; Isoquinolines; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Muscle, Smooth, Vascular; Protein Kinase C; Protein Synthesis Inhibitors; Proto-Oncogene Proteins c-raf; Rats; RNA, Messenger; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate | 2000 |
Differential regulation of microglial NO production by protein kinase C inhibitors.
Topics: Animals; Carbazoles; Drug Synergism; Enzyme Induction; Enzyme Inhibitors; Indoles; Isoquinolines; Lipopolysaccharides; Microglia; Nerve Tissue Proteins; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Protein Isoforms; Protein Kinase C; Pyrroles; Rats; Signal Transduction; Staurosporine; Sulfonamides; Tetradecanoylphorbol Acetate | 2001 |
Cellular mechanism of sodium oleate-stimulated secretion of cholecystokinin and secretin.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Biological Transport; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Cell Fractionation; Cells, Cultured; Chelating Agents; Cholecystokinin; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Duodenum; Egtazic Acid; Enzyme Inhibitors; Intestinal Mucosa; Isoquinolines; Oleic Acid; Phosphodiesterase Inhibitors; Protein Kinase C; Rats; Secretin; Sulfonamides; Tetradecanoylphorbol Acetate | 2000 |
Extracellular Ca2+ sensitivity of mGluR1alpha induces an increase in the basal cAMP level by direct coupling with Gs protein in transfected CHO cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Actins; Animals; Calcium; Cell Size; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Flavonoids; Fluorescent Dyes; Glutamic Acid; GTP-Binding Protein alpha Subunits, Gs; Isoquinolines; MAP Kinase Signaling System; Protein Kinase C; Receptors, Metabotropic Glutamate; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Transfection; Type C Phospholipases | 2000 |
Inhibition by adrenomedullin of arginine vasopressin-activated mitogen-activated protein kinase in rat glomerular mesangial cells via cAMP production.
Topics: Adrenomedullin; Animals; Antihypertensive Agents; Arginine Vasopressin; Blotting, Western; Calcium; Carcinogens; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Inhibitors; Glomerular Mesangium; Isoquinolines; Male; Mitogen-Activated Protein Kinases; Peptides; Rats; Rats, Sprague-Dawley; Sulfonamides; Tetradecanoylphorbol Acetate; Vasoconstrictor Agents | 1996 |
Modulation of the neuronal dopamine transporter activity by the metabotropic glutamate receptor mGluR5 in rat striatal synaptosomes through phosphorylation mediated processes.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Carrier Proteins; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Glycine; Indoles; Isoquinolines; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Neurons; Phosphorylation; Pyridines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; Staurosporine; Sulfonamides; Synaptosomes; Tetradecanoylphorbol Acetate | 2001 |
Regulation of acute cortisol synthesis by cAMP-dependent protein kinase and protein kinase C in a teleost species, the rainbow trout (Oncorhynchus mykiss).
Topics: Adrenocorticotropic Hormone; Analysis of Variance; Animals; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Inhibitors; Female; Hydrocortisone; Isoquinolines; Kidney; Male; Oncorhynchus mykiss; Pregnenolone; Protein Kinase C; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate | 2001 |
Modulation of rat erg1, erg2, erg3 and HERG K+ currents by thyrotropin-releasing hormone in anterior pituitary cells via the native signal cascade.
Topics: Animals; Arachidonic Acid; Cation Transport Proteins; Cells, Cultured; Cholecystokinin; Colforsin; DNA-Binding Proteins; Enzyme Inhibitors; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Flavonoids; Humans; Indoles; Isoquinolines; Kinetics; Maleimides; Membrane Potentials; Membrane Transport Proteins; Patch-Clamp Techniques; Pituitary Gland, Anterior; Potassium Channels; Potassium Channels, Voltage-Gated; Protein Kinase Inhibitors; Protein Kinases; Rats; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Thyrotropin-Releasing Hormone; Trans-Activators; Transcriptional Regulator ERG; Tyrphostins; Vasoactive Intestinal Peptide | 2001 |
Mechanisms in fluoride-induced interleukin-8 synthesis in human lung epithelial cells.
Topics: Androstadienes; Benzylamines; Cell Line; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Egtazic Acid; Epithelial Cells; Flavonoids; Genistein; Humans; Indoles; Interleukin-8; Isoquinolines; Lung; Maleimides; Okadaic Acid; Pertussis Toxin; Protein Kinase C; Signal Transduction; Sodium Fluoride; Sulfonamides; Tetradecanoylphorbol Acetate; Vanadates; Virulence Factors, Bordetella; Wortmannin | 2001 |
Glucose and forskolin regulate IAPP gene expression through different signal transduction pathways.
Topics: Adenylyl Cyclase Inhibitors; Amyloid; Blotting, Northern; Carcinoma, Pancreatic Ductal; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Inhibitors; Gene Expression Regulation; Glucose; Humans; Islet Amyloid Polypeptide; Isoquinolines; Pancreatic Neoplasms; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 2001 |
Controls of EGF-induced morphological transformation of human bronchial epithelial cells.
Topics: Bronchi; Bucladesine; Cell Line; Cells, Cultured; Dose-Response Relationship, Drug; Drug Antagonism; Enzyme Inhibitors; Epidermal Growth Factor; Epithelial Cells; ErbB Receptors; Humans; Isoquinolines; Kinetics; Phosphorylation; Pseudopodia; Respiratory Mucosa; Sulfonamides; Tetradecanoylphorbol Acetate; Transforming Growth Factor beta | 2001 |
Histamine increases the expression of LOX-1 via H2 receptor in human monocytic THP-1 cells.
Topics: Bucladesine; Cell Differentiation; Colforsin; CREB-Binding Protein; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cytokines; Dinoprostone; Enzyme Inhibitors; Gene Expression Regulation; Histamine; Humans; Isoquinolines; Macrophages; Monocytes; Nuclear Proteins; Promoter Regions, Genetic; Prostaglandin D2; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, LDL; Receptors, Oxidized LDL; RNA, Messenger; Scavenger Receptors, Class E; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Trans-Activators; Tumor Cells, Cultured; Up-Regulation | 2001 |
Regulation of transepithelial phosphate transport by PTH in chicken proximal tubule epithelium.
Topics: Animals; Biological Transport; Carcinogens; Cells, Cultured; Chickens; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Epithelial Cells; Indoles; Isoquinolines; Kidney Tubules, Proximal; Maleimides; Parathyroid Hormone; Phosphates; Protein Kinase C; Sodium-Phosphate Cotransporter Proteins; Sulfonamides; Symporters; Tetradecanoylphorbol Acetate | 2002 |
Regulation of urea permeability in frog urinary bladder by prostaglandin E(2).
Topics: Algorithms; Animals; Biological Transport, Active; Cyclic AMP; Dinoprostone; In Vitro Techniques; Indicators and Reagents; Isoquinolines; Male; Osmolar Concentration; Phloretin; Rana temporaria; Receptors, Prostaglandin; Sulfonamides; Tetradecanoylphorbol Acetate; Urea; Urinary Bladder; Vasotocin | 2002 |
Cyclic AMP induces activation of extracellular signal-regulated kinases in HL-60 cells: role in cAMP-induced differentiation.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Cell Differentiation; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Inhibitors; Flavonoids; HL-60 Cells; Humans; Isoquinolines; Lipopolysaccharide Receptors; MAP Kinase Kinase 1; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Neoplasm Proteins; Phenotype; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins B-raf; Proto-Oncogene Proteins c-raf; Second Messenger Systems; Sulfonamides; Superoxides; Tetradecanoylphorbol Acetate | 2003 |
Regulatory mechanism of Cordyceps sinensis mycelium on mouse Leydig cell steroidogenesis.
Topics: Androstenedione; Animals; Cells, Cultured; Colforsin; Cordyceps; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Hydroxycholesterols; Isoquinolines; Leydig Cells; Male; Mice; Mice, Inbred C57BL; Mycelium; Progestins; Protein Kinase C; Staurosporine; Sulfonamides; Testosterone; Tetradecanoylphorbol Acetate | 2003 |
Phosphorylation of the alpha4 subunit of human alpha4beta2 nicotinic receptors: role of cAMP-dependent protein kinase (PKA) and protein kinase C (PKC).
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Bucladesine; Carcinogens; Cell Line; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Humans; Indoles; Isoquinolines; Neurons; Phosphorylation; Protein Kinase C; Receptors, Nicotinic; Sulfonamides; Tetradecanoylphorbol Acetate; Thionucleotides; Transfection | 2003 |
Striatal proenkephalin gene induction: coordinated regulation by cyclic AMP and calcium pathways.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Antihypertensive Agents; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Carcinogens; Cells, Cultured; Colforsin; Corpus Striatum; Cyclic AMP; Drug Interactions; Embryo, Mammalian; Enkephalins; Enzyme Inhibitors; Gene Expression Regulation, Developmental; Humans; Isoquinolines; Neurons; Nifedipine; Protein Precursors; Pyrroles; Rats; Rats, Sprague-Dawley; Sulfonamides; Tetradecanoylphorbol Acetate; Transcriptional Activation; Transfection | 2003 |
Inhibitory effects of group II mGluR-related drugs on memory performance in mice.
Topics: Amino Acids; Animals; Anticonvulsants; Avoidance Learning; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclopropanes; Dose-Response Relationship, Drug; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Glycine; Isoquinolines; Male; Memory; Mice; Reaction Time; Receptors, Metabotropic Glutamate; Rolipram; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Xanthenes | 2004 |
Activation of protein kinase C antagonizes the opioid inhibition of calcium current in rat spinal dorsal horn neurons.
Topics: Analgesics, Opioid; Animals; Animals, Newborn; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Colforsin; Drug Interactions; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enzyme Activation; Enzyme Inhibitors; Female; Indoles; Isoquinolines; Male; Maleimides; Membrane Potentials; Narcotics; Patch-Clamp Techniques; Posterior Horn Cells; Potassium Channel Blockers; Protein Kinase C; Rats; Rats, Sprague-Dawley; Sulfonamides; Tetradecanoylphorbol Acetate; Tetraethylammonium; Tetrodotoxin | 2004 |
Facilitation of noradrenaline release by activation of adenosine A(2A) receptors triggers both phospholipase C and adenylate cyclase pathways in rat tail artery.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Adenylyl Cyclases; Animals; Arteries; Cyclic AMP-Dependent Protein Kinases; Endothelium, Vascular; Enzyme Activation; Indoles; Isoquinolines; Male; Norepinephrine; Phenethylamines; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptor, Adenosine A2A; Signal Transduction; Sulfonamides; Tail; Tetradecanoylphorbol Acetate; Triazoles; Tritium; Type C Phospholipases | 2004 |
Regulation of thrombomodulin expression in human vascular smooth muscle cells by COX-2-derived prostaglandins.
Topics: Alprostadil; Blood Coagulation; Bucladesine; Carotid Artery Diseases; Carotid Artery, Internal; Cells, Cultured; Colforsin; Coronary Vessels; Culture Media, Serum-Free; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Diclofenac; Dinoprostone; Epoprostenol; Etoricoxib; Gene Expression Profiling; Gene Expression Regulation; Humans; Iloprost; Isoquinolines; Mammary Arteries; Membrane Proteins; Models, Biological; Myocytes, Smooth Muscle; Oligonucleotide Array Sequence Analysis; Prostaglandin-Endoperoxide Synthases; Prostaglandins; Pyridines; Receptors, Prostaglandin; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP3 Subtype; RNA, Messenger; Saphenous Vein; Second Messenger Systems; Sulfonamides; Sulfones; Tetradecanoylphorbol Acetate; Thrombomodulin; Thrombophilia; Vasodilator Agents | 2005 |
Luteinizing hormone-induced extracellular-signal regulated kinase activation differently modulates progesterone and androstenedione production in bovine theca cells.
Topics: Androstenedione; Animals; Butadienes; Cattle; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Inhibitors; Extracellular Signal-Regulated MAP Kinases; Female; Fibroblast Growth Factor 2; Isoquinolines; Luteinizing Hormone; Nitriles; Phosphoproteins; Phosphoric Monoester Hydrolases; Phosphorylation; Progesterone; Protein Kinase Inhibitors; RNA, Messenger; Steroid 17-alpha-Hydroxylase; Sulfonamides; Tetradecanoylphorbol Acetate; Theca Cells | 2005 |
Glucose represses connexin36 in insulin-secreting cells.
Topics: Animals; Base Sequence; Cell Line, Tumor; Colforsin; Connexins; Cyclic AMP; Cyclic AMP Response Element Modulator; Cyclic AMP-Dependent Protein Kinases; DNA-Binding Proteins; Down-Regulation; Flavonoids; Gap Junction delta-2 Protein; Glucose; Humans; Insulin-Secreting Cells; Isoquinolines; Mitogen-Activated Protein Kinases; Nifedipine; Promoter Regions, Genetic; Rats; Response Elements; RNA, Messenger; Sequence Deletion; Sulfonamides; Tetradecanoylphorbol Acetate | 2005 |
Parathyroid hormone increases beta-catenin levels through Smad3 in mouse osteoblastic cells.
Topics: Animals; Apoptosis; beta Catenin; Bone and Bones; Bone Development; Cell Line, Tumor; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Dexamethasone; Enzyme Inhibitors; Etoposide; Gene Expression Regulation; Isoquinolines; Lithium Chloride; Luciferases; Mice; Naphthalenes; NIH 3T3 Cells; Osteoblasts; Parathyroid Hormone; Protein Kinase C; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Smad3 Protein; Staurosporine; Sulfonamides; Tetradecanoylphorbol Acetate; Time Factors; Transfection; Transforming Growth Factor beta | 2006 |
Regulation of CD93 cell surface expression by protein kinase C isoenzymes.
Topics: Acetophenones; Benzopyrans; Benzoquinones; Carbazoles; Down-Regulation; Endothelial Cells; Flow Cytometry; Humans; Immunoenzyme Techniques; Indoles; Interferon-gamma; Interleukin-8; Isoenzymes; Isoquinolines; Lactams, Macrocyclic; Membrane Glycoproteins; Monocytes; Protein Kinase C; Protein Kinase Inhibitors; Quinones; Receptors, Complement; Rifabutin; Sulfonamides; Tetradecanoylphorbol Acetate; U937 Cells; Up-Regulation | 2006 |
Role of kinases and G-proteins in the hyposmotic stimulation of cardiac IKs.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Cell Line; Chromans; Colforsin; Cricetinae; Cyclic AMP-Dependent Protein Kinases; Cytochalasin D; Cytoskeleton; GTP-Binding Proteins; Guinea Pigs; Indoles; Isoquinolines; KCNQ1 Potassium Channel; Maleimides; Mitogen-Activated Protein Kinases; Myocytes, Cardiac; Osmotic Pressure; Phosphatidylinositol 3-Kinases; Potassium Channels; Protein Kinase C; Protein-Tyrosine Kinases; Sulfonamides; Tetradecanoylphorbol Acetate; Tyrphostins | 2006 |
(+/-)3,4-Methylenedioxyamphetamine elicits action potential bursts in a central snail neuron.
Topics: Action Potentials; Alkaloids; Animals; Benzophenanthridines; Calcium; Carbazoles; Electrophysiology; Enzyme Inhibitors; Estrenes; Ganglia, Invertebrate; Hallucinogens; In Vitro Techniques; Indoles; Isoquinolines; Magnesium; N-Methyl-3,4-methylenedioxyamphetamine; Neurons; Patch-Clamp Techniques; Phosphodiesterase Inhibitors; Protein Kinase C; Pyrroles; Pyrrolidinones; Snails; Sulfonamides; Tetradecanoylphorbol Acetate | 2007 |
Regulation of Leydig cell steroidogenesis by extracellular signal-regulated kinase 1/2: role of protein kinase A and protein kinase C signaling.
Topics: Animals; Blotting, Western; Bucladesine; Butadienes; Cell Line, Tumor; Chorionic Gonadotropin; Cyclic AMP-Dependent Protein Kinases; DAX-1 Orphan Nuclear Receptor; DNA-Binding Proteins; Enzyme Activation; Extracellular Signal-Regulated MAP Kinases; Isoquinolines; Leydig Cells; Male; Mice; Nitriles; Phosphoproteins; Phosphorylation; Progesterone; Protein Kinase C; Receptors, Retinoic Acid; Repressor Proteins; Reverse Transcriptase Polymerase Chain Reaction; Scavenger Receptors, Class B; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate | 2007 |
Regulation of matrix Gla protein by parathyroid hormone in MC3T3-E1 osteoblast-like cells involves protein kinase A and extracellular signal-regulated kinase pathways.
Topics: 3T3 Cells; Animals; Butadienes; Calcium-Binding Proteins; Colforsin; Cyclic AMP-Dependent Protein Kinases; Extracellular Matrix Proteins; Extracellular Signal-Regulated MAP Kinases; Gene Expression Regulation; Indoles; Isoquinolines; Maleimides; Matrix Gla Protein; Mice; Nitriles; Osteoblasts; Parathyroid Hormone; Promoter Regions, Genetic; Protein Kinase C; Recombinant Proteins; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate | 2007 |
Different kinases regulate activation of voltage-dependent calcium channels by depolarization in GH3 cells.
Topics: Animals; Calcium; Calcium Channels, L-Type; Carcinogens; Cell Line; Cell Line, Tumor; Cyclic AMP-Dependent Protein Kinases; ErbB Receptors; Female; Fluorescent Dyes; Fura-2; Isoquinolines; Membrane Potentials; Pituitary Gland; Pituitary Neoplasms; Potassium Chloride; Protein Kinase C; Protein Kinase Inhibitors; Protein Kinases; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Proto-Oncogene Proteins pp60(c-src); Rats; Rats, Inbred WF; Sulfonamides; Tetradecanoylphorbol Acetate | 2007 |
Regulation of protein kinase D activity in adult myocardium: novel counter-regulatory roles for protein kinase Cepsilon and protein kinase A.
Topics: Animals; Colforsin; Cyclic AMP-Dependent Protein Kinases; Endothelin-1; Enzyme Activation; Heart Ventricles; Isoproterenol; Isoquinolines; Male; Mice; Myocardium; Myocytes, Cardiac; Phosphorylation; Protein Kinase C; Protein Kinase C-epsilon; Protein Transport; Rats; Rats, Wistar; Sulfonamides; Tetradecanoylphorbol Acetate; Troponin I | 2007 |
Mitogen- and stress-activated kinase 1-mediated histone H3 phosphorylation is crucial for cell transformation.
Topics: Animals; Cell Growth Processes; Cell Transformation, Neoplastic; Enzyme Activation; Epidermal Growth Factor; G1 Phase; Histones; Isoquinolines; Mice; Phosphorylation; Protein Kinase Inhibitors; Ribosomal Protein S6 Kinases, 90-kDa; RNA, Small Interfering; Skin; Sulfonamides; Tetradecanoylphorbol Acetate; Transcription Factor AP-1 | 2008 |
Interaction between protein kinase C and protein kinase A can modulate transmitter release at the rat neuromuscular synapse.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Acetylcholine; Analysis of Variance; Animals; Cyclic AMP-Dependent Protein Kinases; Isoquinolines; Membrane Potentials; Naphthalenes; Neuromuscular Junction; Protein Kinase C; Protein Kinase Inhibitors; Rats; Rats, Sprague-Dawley; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Thionucleotides | 2009 |
Role of PDK1 in regulation of gastric acid secretion.
Topics: 3-Phosphoinositide-Dependent Protein Kinases; Animals; Carbachol; Colforsin; Extracellular Space; Gastric Acid; Hydrogen-Ion Concentration; Isoquinolines; Mice; Omeprazole; Parietal Cells, Gastric; Potassium; Protein Serine-Threonine Kinases; Quaternary Ammonium Compounds; Sulfonamides; Tetradecanoylphorbol Acetate | 2008 |
Bradykinin inhibits the transient outward K+ current in mouse Schwann cells via the cAMP/PKA pathway.
Topics: Adamantane; Animals; Benzenesulfonates; Bradykinin; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclic CMP; Enzyme Activators; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Guanosine 5'-O-(3-Thiotriphosphate); Isoquinolines; Membrane Potentials; Mice; Mice, Inbred ICR; Potassium; Potassium Channels, Voltage-Gated; Protein Kinase C; Protein Kinase Inhibitors; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Schwann Cells; Sciatic Nerve; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Time Factors | 2009 |
Melatonin potentiates glycine currents through a PLC/PKC signalling pathway in rat retinal ganglion cells.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Bridged-Ring Compounds; Calcium; Carbazoles; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Egtazic Acid; Estrenes; Glycine; Guanosine Diphosphate; Indoles; Isoquinolines; Male; Maleimides; Melatonin; Norbornanes; Pertussis Toxin; Protein Kinase C; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Receptor, Melatonin, MT2; Retinal Ganglion Cells; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Tetrahydronaphthalenes; Thiocarbamates; Thiones; Type C Phospholipases | 2010 |
Mechanism of hCG-induced spermiation in the toad Rhinella arenarum (Amphibia, Anura).
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Amiloride; Animals; Bufo arenarum; Chorionic Gonadotropin; Cyclic AMP-Dependent Protein Kinases; Indoles; Isoquinolines; Male; Maleimides; Ouabain; Protein Kinase C; Sertoli Cells; Sodium-Potassium-Exchanging ATPase; Spermatozoa; Staurosporine; Sulfonamides; Tetradecanoylphorbol Acetate | 2010 |
The potential use of protein kinase D inhibitors for prevention/treatment of epidermal tumors.
Topics: Animals; Anticarcinogenic Agents; Carbazoles; Cell Differentiation; Cell Proliferation; Cells, Cultured; Epidermis; Isoquinolines; Keratinocytes; Mice; Protein Kinase C; Protein Kinase Inhibitors; Resveratrol; Skin Neoplasms; Stilbenes; Sulfonamides; Tetradecanoylphorbol Acetate | 2010 |
Follicle-stimulating hormone promotes proliferation of cultured chicken ovarian germ cells through protein kinases A and C activation.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Cell Proliferation; Cells, Cultured; Chickens; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Follicle Stimulating Hormone; Isoquinolines; Ovum; Protein Kinase C; Receptors, FSH; Sulfonamides; Tetradecanoylphorbol Acetate | 2010 |
Adrenocorticotropin hormone (ACTH) effects on MAPK phosphorylation in human fasciculata cells and in embryonic kidney 293 cells expressing human melanocortin 2 receptor (MC2R) and MC2R accessory protein (MRAP)β.
Topics: Adrenocorticotropic Hormone; Cyclic AMP; Endocytosis; Enzyme Activators; HEK293 Cells; Humans; Isoquinolines; Membrane Proteins; Mitogen-Activated Protein Kinase 3; Models, Biological; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Receptor, Melanocortin, Type 2; Sulfonamides; Tetradecanoylphorbol Acetate; Time Factors; Zona Fasciculata | 2011 |
Luteinizing hormone (LH) acts through PKA and PKC to modulate T-type calcium currents and intracellular calcium transients in mice Leydig cells.
Topics: Animals; Benzophenanthridines; Calcium; Calcium Channels, T-Type; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Electrophysiological Phenomena; Isoquinolines; Leydig Cells; Luteinizing Hormone; Male; Mice; Peptides; Protein Kinase C; Staurosporine; Sulfonamides; Tetradecanoylphorbol Acetate | 2011 |
Novel phosphorylation of aquaporin-5 at its threonine 259 through cAMP signaling in salivary gland cells.
Topics: Amino Acid Substitution; Animals; Antibodies; Antibody Specificity; Aquaporin 5; Calcimycin; Cell Line, Tumor; Cell Membrane; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Detergents; Humans; Isoproterenol; Isoquinolines; Male; Mice; Mice, Inbred ICR; Parotid Gland; Phosphorylation; Pilocarpine; Protein Kinase Inhibitors; Protein Transport; Salivary Glands; Signal Transduction; Submandibular Gland; Sulfonamides; Tetradecanoylphorbol Acetate; Threonine; Transfection | 2011 |
PKC and PKA regulate AChR dynamics at the neuromuscular junction of living mice.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cyclic AMP-Dependent Protein Kinases; Enzyme Activators; Female; Isoquinolines; Mice; Muscle Denervation; Naphthalenes; Neuromuscular Junction; Post-Synaptic Density; Protein Kinase C; Protein Kinase Inhibitors; Protein Transport; Receptors, Cholinergic; Sulfonamides; Synaptic Transmission; Tetradecanoylphorbol Acetate; Time-Lapse Imaging | 2013 |
Modulation of HERG K+ channels by chronic exposure to activators and inhibitors of PKA and PKC: actions independent of PKA and PKC phosphorylation.
Topics: Colforsin; Cyclic AMP-Dependent Protein Kinases; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; HEK293 Cells; Humans; Indoles; Isoquinolines; Maleimides; Membrane Potential, Mitochondrial; Metalloporphyrins; Patch-Clamp Techniques; Phosphorylation; Protein Kinase C; Reactive Oxygen Species; Sulfonamides; Tetradecanoylphorbol Acetate | 2013 |
Mitogen-induced transcriptional programming in human fibroblasts.
Topics: Cell Line; Cyclic AMP; Epidermal Growth Factor; Fibroblasts; Gene Expression Profiling; Gene Expression Regulation; Genes, Immediate-Early; Humans; Isoquinolines; Mitogens; Reproducibility of Results; Ribosomal Protein S6 Kinases, 90-kDa; Sulfonamides; Tetradecanoylphorbol Acetate; Thionucleotides | 2021 |