Page last updated: 2024-08-23

tetradecanoylphorbol acetate and diazoxide

tetradecanoylphorbol acetate has been researched along with diazoxide in 26 studies

Research

Studies (26)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's10 (38.46)18.2507
2000's14 (53.85)29.6817
2010's2 (7.69)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Ahrén, B; Lindskog, S1
Ashcroft, SJ; Niki, I1
Detimary, P; Gao, ZY; Gembal, M; Gilon, P; Henquin, JC1
Arkhammar, P; Berggren, PO; Bokvist, K; Hallberg, A; Nilsson, T; Rorsman, P; Sjöholm, A; Welsh, M; Welsh, N1
Martin, F; Reig, JA; Soria, B1
Grapengiesser, E; Gylfe, E; Hellman, B; Liu, YJ1
Capito, K; Hansen, SE; Thams, P1
Akesson, B; Lundquist, I1
Aizawa, T; Hashizume, K; Kaneko, T; Komatsu, M; Nagai, M; Schermerhorn, T; Sharp, GW; Yajima, H1
Ahrén, B; Karlsson, S1
Fujimoto, S; Hamamoto, Y; Ishida, H; Kajikawa, M; Mukai, E; Seino, Y; Takeda, T; Tsuji, K; Tsuura, Y; Yamada, Y1
Cerasi, E; Efendic, S; Kaiser, N; Khan, A; Nesher, R; Warwar, N1
Bosco, D; Gonelle-Gispert, C; Halban, PA; Rouiller, DG; Wollheim, CB1
Fujimoto, S; Mukai, E; Nishimura, M; Seino, Y; Shen, ZP; Tsuura, Y; Yamada, Y1
Ashraf, M; Ayub, A; Takashi, E; Wang, Y; Xu, M1
Liu, H; Shao, Z; Yao, Z; Zhang, HY; Zhu, X1
Budzko, D; Miki, T; Niki, I; Niwa, T; Senda, T; Yu, W1
Galiñanes, M; Hassouna, A; Loubani, M1
Nakaya, H; Saegusa, N; Saito, T; Sato, T1
Hartelt, N; Ivannikov, MV; Mironov, SL1
Fowler, A; Galiñanes, M; Hassouna, A; Loubani, M; Matata, BM; Standen, NB1
Zawalich, KC; Zawalich, WS1
Costa, AD; Garlid, KD1
Buléon, C; Galera, P; Gérard, JL; Hanouz, JL; Lemoine, S; Massetti, M; Zhu, L1
Brennan, S; Hudman, D; Jackson, R; Lodwick, D; Norman, RI; Patel, M; Rainbow, RD; Sims, MW1

Other Studies

26 other study(ies) available for tetradecanoylphorbol acetate and diazoxide

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Studies on the mechanism by which galanin inhibits insulin secretion in islets.
    European journal of pharmacology, 1991, Nov-19, Volume: 205, Issue:1

    Topics: Animals; Bucladesine; Calcium Radioisotopes; Colforsin; Diazoxide; Galanin; Glucose; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Mice; Mice, Inbred Strains; Neuropeptides; Peptides; Permeability; Rats; Rats, Inbred Strains; Rubidium Radioisotopes; Tetradecanoylphorbol Acetate

1991
Possible involvement of protein phosphorylation in the regulation of the sulphonylurea receptor of a pancreatic beta-cell line, HIT T15.
    Biochimica et biophysica acta, 1991, Dec-03, Volume: 1133, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; ATP-Binding Cassette Transporters; Cell Line; Cell Membrane; Colforsin; Diazoxide; Glyburide; Humans; Insulin; Insulin Secretion; Islets of Langerhans; Isoquinolines; Phosphorylation; Piperazines; Potassium Channels; Potassium Channels, Inwardly Rectifying; Protein Kinase Inhibitors; Proteins; Receptors, Drug; Rubidium; Sulfonylurea Receptors; Tetradecanoylphorbol Acetate

1991
Mechanisms by which glucose can control insulin release independently from its action on adenosine triphosphate-sensitive K+ channels in mouse B cells.
    The Journal of clinical investigation, 1993, Volume: 91, Issue:3

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Diazoxide; Diterpenes; Glucose; Inositol Phosphates; Insulin; Insulin Secretion; Islets of Langerhans; Keto Acids; Kinetics; Male; Mice; Mice, Inbred Strains; Phorbol 12,13-Dibutyrate; Potassium; Potassium Channels; Protein Kinase C; Terpenes; Tetradecanoylphorbol Acetate

1993
Enhanced stimulus-secretion coupling in polyamine-depleted rat insulinoma cells. An effect involving increased cytoplasmic Ca2+, inositol phosphate generation, and phorbol ester sensitivity.
    The Journal of clinical investigation, 1993, Volume: 92, Issue:4

    Topics: Adenosine Triphosphate; Animals; Calcium; Calcium Channels; Carbachol; Cytoplasm; Diazoxide; DNA, Neoplasm; Eflornithine; Glucose; Glyburide; Inositol Phosphates; Insulin; Insulin Secretion; Insulinoma; Kinetics; Pancreatic Neoplasms; Polyamines; Potassium; Putrescine; Rats; RNA, Messenger; Spermidine; Spermine; Tetradecanoylphorbol Acetate; Theophylline; Tolbutamide; Tumor Cells, Cultured

1993
Secretagogue-induced [Ca2+]i changes in single rat pancreatic islets and correlation with simultaneously measured insulin release.
    Journal of molecular endocrinology, 1995, Volume: 15, Issue:2

    Topics: Animals; Calcium; Carbachol; Cells, Cultured; Cytosol; Diazoxide; Fluorescent Dyes; Fura-2; Glucose; Glutamine; Indoles; Inulin; Islets of Langerhans; Kinetics; Leucine; Male; Protein Kinase C; Rats; Rats, Wistar; Tetradecanoylphorbol Acetate; Time Factors; Tolbutamide

1995
Crosstalk between the cAMP and inositol trisphosphate-signalling pathways in pancreatic beta-cells.
    Archives of biochemistry and biophysics, 1996, Oct-15, Volume: 334, Issue:2

    Topics: Animals; Caffeine; Calcium; Cells, Cultured; Cyclic AMP; Cytosol; Diazoxide; Gallopamil; Glucagon; Glucose; Inositol 1,4,5-Trisphosphate; Islets of Langerhans; Kinetics; Membrane Potentials; Mice; Mice, Obese; Oscillometry; Potassium; Ryanodine; Signal Transduction; Strontium; Tetradecanoylphorbol Acetate

1996
Production of [3H]choline-labelled metabolites from endogenously 3H-labelled phosphatidylcholine in mouse pancreatic islets.
    Journal of molecular endocrinology, 1996, Volume: 17, Issue:2

    Topics: Animals; Carbachol; Cells, Cultured; Choline; Cyclohexanones; Diazoxide; Glucose; Glycerylphosphorylcholine; Insulin; Insulin Secretion; Islets of Langerhans; Isoproterenol; Kinetics; Lysophosphatidylcholines; Male; Mice; Mice, Inbred Strains; Phosphatidylcholines; Potassium Chloride; Radioisotope Dilution Technique; Rats; Sodium Fluoride; Succinates; Tetradecanoylphorbol Acetate; Tolbutamide; Tritium

1996
Evidence for nitric oxide mediated effects on islet hormone secretory phospholipase C signal transduction mechanisms.
    Bioscience reports, 1998, Volume: 18, Issue:4

    Topics: Animals; Calcium; Carbachol; Cell Membrane; Cholinergic Agonists; Diazoxide; Enzyme Inhibitors; Female; Glucagon; Hydroxylamine; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Mice; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Potassium Channels; Receptors, Muscarinic; Signal Transduction; Tetradecanoylphorbol Acetate; Type C Phospholipases

1998
cAMP enhances insulin secretion by an action on the ATP-sensitive K+ channel-independent pathway of glucose signaling in rat pancreatic islets.
    Diabetes, 1999, Volume: 48, Issue:5

    Topics: Adenosine Triphosphate; Animals; Calcium; Colforsin; Cyclic AMP; Diazoxide; Enzyme Activation; Glucose; Insulin; Insulin Secretion; Islets of Langerhans; Male; Potassium Channels; Potassium Chloride; Protein Kinase C; Rats; Rats, Wistar; Signal Transduction; Tetradecanoylphorbol Acetate

1999
Cytosolic Ca2+ oscillations by gastrin releasing peptide in single HIT-T15 cells.
    Peptides, 1999, Volume: 20, Issue:5

    Topics: Animals; Biological Transport; Calcium; Calcium Channel Blockers; Calcium Signaling; Cells, Cultured; Cytosol; Diazoxide; Dose-Response Relationship, Drug; Drug Interactions; Egtazic Acid; Gastrin-Releasing Peptide; Glucose; Ion Channel Gating; Islets of Langerhans; Mice; Nifedipine; Protein Kinase C; Tetradecanoylphorbol Acetate; Thapsigargin

1999
Augmentation of basal insulin release from rat islets by preexposure to a high concentration of glucose.
    American journal of physiology. Endocrinology and metabolism, 2000, Volume: 279, Issue:4

    Topics: Adenosine Triphosphate; Adrenergic alpha-Agonists; Animals; Calcium; Cell Membrane Permeability; Cells, Cultured; Clonidine; Colforsin; Diazoxide; Dose-Response Relationship, Drug; Electroporation; Glucose; Guanosine Diphosphate; Insulin; Insulin Secretion; Intracellular Fluid; Islets of Langerhans; Male; Mannoheptulose; Mycophenolic Acid; Oligomycins; Potassium; Rats; Rats, Wistar; Tetradecanoylphorbol Acetate; Thionucleotides

2000
Defective stimulus-secretion coupling in islets of Psammomys obesus, an animal model for type 2 diabetes.
    Diabetes, 2001, Volume: 50, Issue:2

    Topics: Animals; Colforsin; Diabetes Mellitus, Type 2; Diazoxide; Disease Models, Animal; Disease Susceptibility; Gerbillinae; Glucagon; Glucagon-Like Peptide 1; Glucose; Hyperglycemia; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Isoenzymes; Oxidation-Reduction; Peptide Fragments; Protein Kinase C; Protein Precursors; Rats; Rats, Sprague-Dawley; Reference Values; Signal Transduction; Tetradecanoylphorbol Acetate

2001
Increased intracellular calcium is required for spreading of rat islet beta-cells on extracellular matrix.
    Diabetes, 2001, Volume: 50, Issue:5

    Topics: Animals; Botulinum Toxins; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Cell Adhesion; Cell Degranulation; Cell Movement; Cell Size; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Diazoxide; Diphosphonates; Enzyme Inhibitors; Extracellular Matrix; Glucagon; Glucose; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Male; Potassium Chloride; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Signal Transduction; Tetradecanoylphorbol Acetate; Thapsigargin; Time Factors; Transfection

2001
Distinct effect of diazoxide on insulin secretion stimulated by protein kinase A and protein kinase C in rat pancreatic islets.
    Diabetes research and clinical practice, 2001, Volume: 53, Issue:1

    Topics: Animals; Bucladesine; Calcium; Cyclic AMP-Dependent Protein Kinases; Diazoxide; Dose-Response Relationship, Drug; Enzyme Activation; Glucose; Glyceraldehyde; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Male; Potassium; Protein Kinase C; Rats; Rats, Wistar; Tetradecanoylphorbol Acetate

2001
Downregulation of protein kinase C inhibits activation of mitochondrial K(ATP) channels by diazoxide.
    Circulation, 2001, Jul-03, Volume: 104, Issue:1

    Topics: Adenosine Triphosphate; Animals; Diazoxide; Dose-Response Relationship, Drug; Down-Regulation; Immunohistochemistry; In Vitro Techniques; Ischemic Preconditioning, Myocardial; Isoenzymes; L-Lactate Dehydrogenase; Male; Mitochondria; Myocardial Ischemia; Myocardium; Potassium Channel Blockers; Potassium Channels; Protein Kinase C; Protein Transport; Rats; Rats, Sprague-Dawley; Reperfusion Injury; Sarcolemma; Subcellular Fractions; Tetradecanoylphorbol Acetate; Ventricular Function, Left

2001
Preconditioning blocks cardiocyte apoptosis: role of K(ATP) channels and PKC-epsilon.
    American journal of physiology. Heart and circulatory physiology, 2002, Volume: 282, Issue:4

    Topics: Alkaloids; Animals; Apoptosis; Benzophenanthridines; Cells, Cultured; Chick Embryo; Decanoic Acids; Diazoxide; Heart; Hydroxy Acids; Ion Channel Gating; Ion Channels; Ischemic Preconditioning, Myocardial; Isoenzymes; Membrane Proteins; Myocardial Reperfusion; Myocardium; Phenanthridines; Potassium Channels; Protein Kinase C; Protein Kinase C-epsilon; Tetradecanoylphorbol Acetate

2002
Ca2+ influx does not trigger glucose-induced traffic of the insulin granules and alteration of their distribution.
    Experimental biology and medicine (Maywood, N.J.), 2003, Volume: 228, Issue:10

    Topics: Calcium; Calcium Signaling; Cell Line; Cytoplasm; Diazoxide; Dose-Response Relationship, Drug; Down-Regulation; Glucose; Insulin; Insulin Secretion; Islets of Langerhans; Myosin Light Chains; Nifedipine; Nitrendipine; Phosphorylation; Tetradecanoylphorbol Acetate; Time Factors

2003
Delayed preconditioning of the human myocardium: signal transduction and clinical implications.
    Cardiovascular research, 2004, Feb-15, Volume: 61, Issue:3

    Topics: Acetylcholine; Aged; Alkaloids; Anisomycin; Antihypertensive Agents; Benzophenanthridines; Culture Techniques; Decanoic Acids; Diazoxide; Enzyme Activation; Enzyme Inhibitors; Female; Heart Atria; Humans; Hydroxy Acids; Imidazoles; Ischemic Preconditioning, Myocardial; Male; Middle Aged; Mitogen-Activated Protein Kinases; Myocardial Ischemia; Myocardium; p38 Mitogen-Activated Protein Kinases; Phenanthridines; Phenylephrine; Potassium Channel Blockers; Potassium Channels; Protein Kinase C; Pyridines; Signal Transduction; Tetradecanoylphorbol Acetate; Time Factors

2004
Mitochondrial Ca2+-activated K+ channels in cardiac myocytes: a mechanism of the cardioprotective effect and modulation by protein kinase A.
    Circulation, 2005, Jan-18, Volume: 111, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Benzimidazoles; Carbocyanines; Cell Death; Colforsin; Cyclic AMP-Dependent Protein Kinases; Decanoic Acids; Diazoxide; Fluorescent Dyes; Guinea Pigs; Heart Ventricles; Heterocyclic Compounds, 3-Ring; Hydroxy Acids; Indoles; Intracellular Membranes; Ion Transport; Membrane Potentials; Mitochondria, Heart; Myocytes, Cardiac; Ouabain; Potassium; Potassium Channels, Calcium-Activated; Second Messenger Systems; Tetradecanoylphorbol Acetate

2005
Mitochondrial K(ATP) channels in respiratory neurons and their role in the hypoxic facilitation of rhythmic activity.
    Brain research, 2005, Feb-01, Volume: 1033, Issue:1

    Topics: Animals; Animals, Newborn; Calcium; Cell Hypoxia; Decanoic Acids; Diazoxide; Enzyme Inhibitors; Fluorescent Antibody Technique; Fluorescent Dyes; Hydroxy Acids; In Vitro Techniques; Medulla Oblongata; Mice; Mitochondria; Neurons; Periodicity; Potassium Channel Blockers; Potassium Channels; Potassium Chloride; Respiration; Staurosporine; Tetradecanoylphorbol Acetate

2005
Mitochondrial dysfunction as the cause of the failure to precondition the diabetic human myocardium.
    Cardiovascular research, 2006, Feb-01, Volume: 69, Issue:2

    Topics: Adenosine; Adrenergic alpha-Agonists; Diabetes Mellitus; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Diazoxide; Enzyme Activation; Glyburide; Heart Atria; Humans; Hypoglycemic Agents; In Vitro Techniques; Ischemic Preconditioning, Myocardial; Membrane Potentials; Metformin; Mitochondria, Heart; Myocardial Ischemia; p38 Mitogen-Activated Protein Kinases; Phenylephrine; Potassium Channels; Protein Kinase C; Reactive Oxygen Species; Tetradecanoylphorbol Acetate

2006
Enhanced activation of phospholipase C and insulin secretion from islets incubated in fatty acid-free bovine serum albumin.
    Metabolism: clinical and experimental, 2008, Volume: 57, Issue:2

    Topics: Animals; Carbachol; Cholinergic Agonists; Diazoxide; Enzyme Activation; In Vitro Techniques; Inositol; Insulin; Insulin Secretion; Islets of Langerhans; Male; Mice; Potassium Chloride; Rats; Rats, Sprague-Dawley; Serum Albumin, Bovine; Tetradecanoylphorbol Acetate; Type C Phospholipases

2008
Intramitochondrial signaling: interactions among mitoKATP, PKCepsilon, ROS, and MPT.
    American journal of physiology. Heart and circulatory physiology, 2008, Volume: 295, Issue:2

    Topics: Animals; Cyclic GMP-Dependent Protein Kinases; Diazoxide; Enzyme Activation; Feedback, Physiological; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Hydrogen Peroxide; In Vitro Techniques; Ion Channel Gating; Male; Mitochondria, Heart; Mitochondrial Membrane Transport Proteins; Mitochondrial Membranes; Mitochondrial Permeability Transition Pore; Mitochondrial Size; Nitric Oxide; Phosphorylation; Potassium Channels; Protein Kinase C-epsilon; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Signal Transduction; Superoxides; Tetradecanoylphorbol Acetate; Time Factors

2008
Mechanisms involved in the desflurane-induced post-conditioning of isolated human right atria from patients with type 2 diabetes.
    British journal of anaesthesia, 2011, Volume: 107, Issue:4

    Topics: Aged; Anesthetics, Inhalation; Blotting, Western; Decanoic Acids; Desflurane; Diabetes Mellitus, Type 2; Diazoxide; Enzyme Inhibitors; Female; Glycated Hemoglobin; Glycogen Synthase Kinase 3; Heart; Heart Atria; Humans; Hydroxy Acids; Hypoxia; Ischemic Postconditioning; Isoflurane; KATP Channels; Male; Middle Aged; Mitochondria, Heart; Myocardial Reperfusion Injury; Naphthalenes; Protein Kinase C; Proto-Oncogene Proteins c-akt; Stroke Volume; Tetradecanoylphorbol Acetate

2011
Early opening of sarcolemmal ATP-sensitive potassium channels is not a key step in PKC-mediated cardioprotection.
    Journal of molecular and cellular cardiology, 2015, Volume: 79

    Topics: Action Potentials; Adenosine; Animals; Cardiotonic Agents; Cell Separation; Diazoxide; Enzyme Activation; Heart Failure; Ion Channel Gating; Ischemic Preconditioning, Myocardial; Isoenzymes; KATP Channels; Male; Myocardial Contraction; Myocardial Reperfusion; Myocytes, Cardiac; Phenotype; Pinacidil; Protein Kinase C-epsilon; Protein Kinase Inhibitors; Rats, Wistar; Sarcolemma; Tetradecanoylphorbol Acetate; Time Factors

2015