tetradecanoylphorbol acetate has been researched along with bisindolylmaleimide i in 294 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 125 (42.52) | 18.2507 |
2000's | 150 (51.02) | 29.6817 |
2010's | 19 (6.46) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Alcami, J; Bessia, C; Hay, RT; Paya, CV; Ten, RM; Virelizier, JL | 1 |
Imre, K; Jacobson, PB; Kuchera, SL; Metz, A; Schächtele, C; Schrier, DJ | 1 |
Loh, TT; Zhu, WH | 1 |
Falet, H; Rendu, F | 1 |
Corvol, M; Friedlander, G; Garabédian, M; Menaa, C; Vrtovsnik, F | 1 |
Baldo, A; Cianflone, K; Sniderman, AD; St Luce, S; Zhang, XJ | 1 |
King, GL; Kramer, RM; Xia, P | 1 |
Cox, AJ; Lee, RK; Nitsch, RM; Wurtman, RJ | 1 |
Ausiello, DA; Breuer, W; Cabantchik, IZ; Glickstein, H; Kartner, N; Riordan, JR | 1 |
Hori, M; Itoh, T; Iwakura, K; Kitakaze, M; Komamura, K; Minamino, T; Morioka, T; Node, K; Okazaki, Y; Takashima, S | 1 |
Laughlin, KV; Marano, CW; Mullin, JM; Russo, LM | 1 |
Araki, R; Komada, T; Naka, M; Nakatani, K; Shima, T; Tanaka, T | 1 |
Chan, KF; Loh, TT; Lok, CN | 1 |
Deli, E; Kiss, Z | 1 |
Brass, LF; Hagège, J; He, CJ; Rondeau, E; Sraer, JD; Xu, Y; Zacharias, U | 1 |
Anderson, WH; Kiss, Z; Phillips, H | 1 |
Bouchard, B; Coulomb, B; Dubertret, L; Le Panse, R; Lebreton, C; Mitev, V | 1 |
Leslie, CC; Qiu, ZH | 1 |
Finkenzeller, G; Häussinger, D; Lang, F; Newsome, W | 1 |
Dautrevaux, M; Formstecher, P; Lefebvre, P; Tahayato, A | 1 |
Bi, N; Mamrack, MD | 1 |
Brecha, N; Corey, JL; Davidson, N; Lester, HA; Quick, MW | 1 |
Schächtele, C; Seifert, R; Wenzel-Seifert, K | 1 |
Dwyer, LD; Jaken, S; Malkinson, AM; Miller, AC; Parks, AL | 1 |
Burn, P; Camoin, L; Fagard, R; Fischer, S; Guillaume, JL; Meggio, F; Rothhut, B; Soula, M; Strosberg, D; Vorherr, T | 1 |
Barth, H; Jacobson, P; Kuchera, S; Metz, A; Schaechtele, C; Schrier, D | 1 |
Bonev, AD; Nelson, MT | 1 |
Eriksson, K; Heikkilä, J; Jalava, A | 1 |
Ben-Av, P; Eli, Y; Liscovitch, M; Schmidt, US; Tobias, KE | 1 |
Blumberg, PM; Goodnight, JA; Kazanietz, MG; Kolch, W; Martiny-Baron, G; Mischak, H; Mushinski, JF; Pierce, JH; Schaechtle, C | 1 |
Dadgar, J; Hundle, B; McMahon, T; Messing, RO | 1 |
Erusalimsky, JD; Hong, Y; Martin, JF; Vainchenker, W | 1 |
Haimovich, B; Ji, P; Kaneshiki, N | 1 |
Bhatia, M; Kirkland, JB; Meckling-Gill, KA | 1 |
Carey, JO; deVente, JE; Pettit, GR; Posekany, KJ; Ways, DK | 1 |
Alexandrov, IA; Hilbert, DM; Mushinski, JF; Nordan, RP; Romanova, LY; Schwab, G | 1 |
Bouchard, B; Coulomb, B; Le Panse, R; Lebreton, C | 1 |
Granot, Y; Isakov, N; Tamir, A | 1 |
Fagerström, S; Gestblom, C; Nånberg, E; Påhlman, S | 1 |
Carpentier, G; Lagord, C; Leibovitch, MP; Leibovitch, SA; Martelly, I | 1 |
Kurata, S; Matsumoto, M; Nakajima, H | 1 |
Kiss, Z | 1 |
Gercken, G; Radloff, M | 1 |
Driessens, MH; Roos, E; Soede, RD; van Hulten, PE; van Rijthoven, EA | 1 |
Dubois, T; Geny, B; Lukowski, S; Mira, JP; Oudinet, JP; Russo-Marie, F | 1 |
Hakeda, Y; Kameda, T; Kumegawa, M; Mano, H; Raisz, LG; Shiokawa, M | 1 |
Hori, M; Inoue, M; Kamada, T; Kitakaze, M; Minamino, T; Node, K; Tada, M | 1 |
Evans, R; Fuller, JA; Kamdar, SJ | 1 |
Classen, S; Eissner, G; Fichter, M; Hinrichs, R; Scheffer, B; Ueffing, M | 1 |
Benna, JE; Dang, PM; Fay, M; Gaudry, M; Gougerot-Pocidalo, MA; Hakim, J; Morel, F | 1 |
Ferrante, A; Hii, CS; Huang, ZH; Murray, AW; Poulos, A; Rathjen, DA | 1 |
Fukuda, K; Kato, S; Mori, K; Morikawa, H; Shoda, T | 1 |
Hakeda, Y; Hanada, K; Kakudo, S; Kameda, T; Kumegawa, M; Mano, H; Miyazawa, K; Mori, Y; Nakamaru, Y; Shiokawa-Sawada, M; Yuasa, T | 1 |
Courage, C; Gescher, A; Hubbard, A; Jones, T | 1 |
Boucheix, C; Francastel, C; Lantz, O; Le Naour, F; Prenant, M; Rubinstein, E | 1 |
Jorcano, JL; Paramio, JM | 1 |
Evans, R; Fuller, JA; Kamdar, SJ; Nishikawa, SI | 1 |
Cox, ME; Parsons, SJ | 1 |
Brunet, C; Cabanis, A; Cazin, JC; Cazin, M; Dine, T; Gressier, B; Luyckx, M | 1 |
Byers, SW; Crockett, C; Jensen, JP; Orford, K; Weissman, AM | 1 |
Häussinger, D; Kurz, AK; Schliess, F; vom Dahl, S | 1 |
Gilad, E; Matzkin, H; Zisapel, N | 1 |
Funaya, H; Hori, M; Kitakaze, M; Kuzuya, T; Minamino, T; Node, K; Okuyama, Y; Sato, H; Ueda, Y; Yoshida, K | 1 |
Acs, P; Bíró, T; Blumberg, PM; Bögi, K; Lorenzo, PS; Marquez, AM; Mushinski, JF; Szállási, Z; Wang, QJ | 1 |
Stepan, VM; Takeuchi, Y; Todisco, A; Urumov, A; Yamada, J; Yamada, T | 1 |
García, LJ; González, A; Jensen, RT; Rosado, JA | 1 |
Jensen, RT; Kusui, T; Tsuda, T | 1 |
Almazan, G; Larocca, JN | 1 |
Liu, J; Marcus, DC; Scofield, MA; Shen, Z; Sunose, H | 1 |
Chang, WC; Chen, BK; Liaw, YW; Liu, YW | 1 |
Friedman, LM; Lazarovici, P; Matsuda, Y | 1 |
Kucera, GL; Stadheim, TA | 1 |
Gohda, E; Iwao, M; Okauchi, H; Yamamoto, I | 1 |
Alexandrov, IA; Blagosklonny, MV; Mushinski, JF; Nordan, RP; Romanova, LY | 1 |
de Jonge, HR; Dorrestijn, J; Maassen, JA; Narumiya, S; Tilly, BC; van der Wijk, T | 1 |
Aaronson, DS; Crespo, P; Font de Mora, J; Gutkind, JS; Santos, E | 1 |
Alameda, F; Batlle, E; de Herreros, AG; del Mont Llosas, M; Díaz, V; Domínguez, D; Loukili, N; Paciucci, R; Verdú, J | 1 |
Amar, LS; Forest, N; Martin, N; Oboeuf, M | 1 |
Chow, SC; Jondal, M; Osorio, LM; Rottenberg, M | 1 |
Bond, JA; Dawson, TP; Eccles, NG; Gescher, A; Hall-Jackson, CA; Jones, T; Wynford-Thomas, D | 1 |
Andersson, G; Onyango, I; Pihlgren, U; Rask, L; Setterblad, N | 1 |
Kobayashi, M; Kuroda, A; Maruyama, M; Mino, T; Sugiyama, E; Taki, H; Yamashita, N | 1 |
Costa, LG; Guizzetti, M; Wei, M | 1 |
Nagarkatti, DS; Sha'afi, RI | 1 |
Fukunaga, T; Ishibashi, S; Nigorikawa, K; Okamura, N; Yaname, H | 1 |
Conn, PM; Lin, X | 1 |
Albright, JA; Kolomytkin, OV; Marino, AA; Sadasivan, KK; Wolf, RE | 1 |
Blank, U; David, B; Guérin-Marchand, C; Iannascoli, B; Marchand, F; Pelletier, C; Weyer, A | 1 |
Hayashi, R; Kobayashi, M; Maruyama, M; Matsui, S; Sugiyama, E; Sugiyama, S; Yamashita, N | 1 |
Guo, YL; Kang, B; Williamson, JR | 1 |
Aboud, M; Mor-Vaknin, N; Torgeman, A | 1 |
Barboule, N; Chadebech, P; Lafon, C; Valette, A; Vidal, S | 1 |
Lan, L; Wong, NS | 1 |
Brown, JF; Chang, Q; Soper, BD; Tepperman, BL | 1 |
Abe, N; Habu, S; Iwakabe, K; Kitamura, H; Matsuki, N; Nakui, M; Nishimura, T; Ohmi, Y; Ohta, A; Sato, M; Yagita, H; Yahata, C; Yahata, T | 1 |
Bissonnette, M; Brasitus, TA; Khare, S; Scaglione-Sewell, B; Sitrin, MD; Wali, RK | 1 |
Acs, P; Alexandrov, IA; Blagosklonny, MV; Blumberg, PM; Garfield, S; Mushinski, JF; Nguyen, P; Nordan, RP; Romanova, LY; Trepel, J | 1 |
Conn, PM; Han, XB | 1 |
Shibuya, M; Takahashi, T; Ueno, H | 1 |
Oldenborg, PA; Sehlin, J | 1 |
Nishioka, M; Okumura, K; Sasazuki, T; Shirasawa, S | 1 |
Akasaki, T; Koga, H; Sumimoto, H | 1 |
Akiba, S; Hayama, M; Kume, K; Mizunaga, S; Sato, T | 1 |
Christoffersen, T; Dajani, OF; Melien, O; Nilssen, LS; Rezvani, F; Sandnes, D; Thoresen, GH | 1 |
Brass, LF; Cichowski, K; Orsini, MJ | 1 |
Barańska, J; Czajkowski, R | 1 |
Boland, RL; Capiati, DA; Limbozzi, F; Téllez-Iñón, MT | 1 |
Backendorf, C; Borgstein, AM; Medema, JP; Sark, MW; van de Putte, P | 1 |
Amar, LS; Forest, N; Martin, N; Oboeuf, M; Shabana, AH | 1 |
Anema, SM; Arthur, JR; Beckett, GJ; Howie, AF; Nicol, F; Walker, SW | 1 |
Leupen, SM; Levine, JE | 1 |
Akamatsu, N; Higaki, T; Imamura, H; Komatsu, S; Kono, Y; Nakagawa, M; Sato, T; Sawada, S; Tada, Y; Tamagaki, T; Toratani, A; Tsuda, Y; Tsuji, H; Yamasaki, S | 1 |
Karnes, WE; Klein, IK; Penington, RC; Weller, SG | 1 |
Libermann, TA; Petersen, N; Prinz, S; Sallmann, S; Schneider, A; Schwaninger, M; Spranger, M | 1 |
Ferris, HA; García, LJ; Jensen, RT; Tapia, JA | 1 |
Becker, K; Brodde, OE; Heinroth-Hoffmann, I; Osten, B; Pönicke, K | 1 |
Palmer, TM; Stiles, GL | 1 |
Barnes, PJ; Giembycz, MA; Hellewell, PG; Lindsay, MA; Lynch, OT | 1 |
Chang, Q; Soper, BD; Tepperman, BL | 2 |
Behrens, MM; Choi, DW; Gwag, BJ; Koh, JY; Strasser, U | 1 |
Hamad, AM; Knox, AJ | 1 |
Gear, AR; Polanowska-Grabowska, R | 1 |
Becker, M; Cato, AC; Klocker, H; Mink, S; Peterziel, H; Schonert, A | 1 |
Farokhzad, OC; Hrnjez, BJ; Matthews, JB; Song, JC | 1 |
Alessi, DR; Fahlman, R; Krook, A; Ryder, JW; Wallberg-Henriksson, H; Zierath, JR | 1 |
Costa, LG; Guizzetti, M; Wei, M; Yost, M | 1 |
Cafferata, EG; Giordano, L; González-Guerrico, AM; Pivetta, OH; Santa-Coloma, TA | 1 |
Chiu, CT; Huang, SC; Lin, CC; Pan, SL; Tsai, YJ; Wang, CC; Wu, WB; Yang, CM | 1 |
Han, B; Logsdon, CD | 1 |
Bourgeade, MF; Cayre, YE; Thang, MN; Ye, F | 1 |
Chen, Y; Deng, J; Wu, R | 1 |
Slack, BE | 1 |
Bao, HF; Eaton, DC; Malik, B; Middleton, P; Schenck, J; Schlanger, LE; Stockand, JD | 1 |
Tai, HH; Tong, M | 1 |
Chaudhuri, S; Raha, S | 1 |
Aquino, A; Barrera, G; Dianzani, MU; Farace, MG; Fazio, VM; Pizzimenti, S; Rinaldi, M; Spinsanti, P | 1 |
Kapfhammer, JP; Metzger, F | 1 |
Dunzendorfer, S; Wiedermann, CJ | 1 |
Barańska, J; Bobeszko, M; Dygas, A; Nalepa, I | 1 |
Bao, HF; Eaton, DC; Edinger, RS; Johnson, JP; Yue, G | 1 |
Almas, J; Rubin, E; Solem, M; Thomas, A | 1 |
Auberger, P; Baier, G; Bertolotto, C; Filippa, N; Maulon, L | 1 |
Fujimoto, S; Hayakawa, T; Kawakami, N; Kita, K; Yamaguchi, T | 1 |
Chae, SW; Cho, CH; Jo, SH; Lee, CO | 1 |
Bruni, P; Cencetti, F; Donati, C; Meacci, E; Romiti, E | 1 |
Cunningham, FM; Goode, NT; Greenaway, EC | 1 |
Brodbeck, K; Häring, HU; Pfeiffer, A; Sauer, U; Schleicher, ED; Weigert, C | 1 |
Aoki, T; Etoh, T; Hashimoto, T; Imamura, M; Inoguchi, T; Kakimoto, M; Li, P; Naruse, M; Nawata, H; Sano, H; Umeda, F; Utsumi, H; Yu, HY | 1 |
Hasse, A; Kuger, P; Meyer-Kirchrath, J; Nilius, SM; Schrör, K | 1 |
Doggett, TA; Lemker, JL; Partridge, NC; Swarthout, JT | 1 |
Aguilera, J; Gil, C; Najib, A; Pelliccioni, P | 1 |
Meinhardt, G; Roth, J; Totok, G | 1 |
Courtois, G; Kuiperij, HB; van der Eb, AJ; Vertegaal, AC; Yamaoka, S; Zantema, A | 1 |
Jang, MA; Kwon, TK; Lee, YH; Park, JW; Passaniti, A | 1 |
Wenner, CE; Yan, S | 1 |
Kaneda, N; Murata, T; Niimi, Y | 1 |
Boland, R; Buitrago, C; de Boland, AR; Morelli, S | 1 |
Giardina, JB; Khalil, RA; Tanner, DJ | 1 |
Akimoto, K; Hattori, Y; Kakishita, H; Kasai, K; Matsumura, M | 1 |
Grant, S; Vrana, JA | 1 |
Bauer, CK; Schledermann, W; Schwarz, JR; Wulfsen, I | 1 |
Aizawa, T; Hashizume, K; Ikeo, S; Nakajima, K; Shigematsu, S; Yamauchi, K | 1 |
Hashimoto, M; Hsu, L; Mallory, M; Masliah, E; Rockenstein, E | 1 |
Banan, A; Fields, JZ; Keshavarzian, A; Zhang, Y | 1 |
Hamada, H; Shimizu, T; Sugibayashi, R; Suzuki, T; Takeda, K; Yamamoto, N | 1 |
Massoumi, R; Sjölander, A | 1 |
Avruch, J; Gonçalves, D; Lenz, G; Luo, Z; Neary, JT; Rodnight, R | 1 |
Haye, B; Huet, E; Legue, O; Martiny, L; Petitfrère, E; Sartelet, H | 1 |
Hashimoto, T; Imamura, M; Inoguchi, T; Kakimoto, M; Nakashima, N; Nawata, H; Umeda, F; Yu, HY | 1 |
Kanda, Y; Kuroki, Y; Mizuno, K; Nishio, E; Watanabe, Y | 1 |
Chaby, R; Girard, R; Pédron, T | 1 |
Chen, JS; Song, JG | 1 |
Chibalin, AV; Féraille, E; Kovalenko, MV; Ryder, JW; Wallberg-Henriksson, H; Zierath, JR | 1 |
Crow, T; Neary, JT; Siddiqi, V; Xue-Bian, JJ | 1 |
Cruciani, V; Husøy, T; Mikalsen, SO | 1 |
Costa, LG; Guizzetti, M; Lu, H | 1 |
Gant, TW; Gescher, A; Gill, PK | 1 |
Matthews, JB; Mun, EC; Nichols, A; Song, JC; Yoo, J | 1 |
Higashi, T; Horiuchi, H; Kita, T; Nishioka, H; Ozaki, H; Shirakawa, R; Tabuchi, A; Yamamoto, A; Yoshioka, A | 1 |
Andreeva, AY; Blasig, IE; Krause, E; Müller, EC; Utepbergenov, DI | 1 |
Låg, M; Refsnes, M; Schwarze, PE; Thoresen, GH; Thrane, EV | 1 |
Denys, A; Hichami, A; Khan, NA; Maume, B | 1 |
Bayguinov, O; Hagen, B; Kenyon, JL; Sanders, KM | 1 |
Hur, SY; Ki, IK; Kim, JW; Kim, TE; Kim, YW; Lee, JM; Namkoong, SE | 1 |
Frey, BM; Frey, FJ; Heiniger, CD; Rochat, MK | 1 |
Kwak, JY; Lee, MJ; Oh, JY; Park, HT; Uhlinger, DJ | 1 |
Cho, W; Han, JM; Jung, YW; Kim, JH; Kim, Y; Kuroki, T; Lee, BD; Lee, S; Lee, SD; Ohba, M; Ryu, SH; Suh, PG | 1 |
Hung, AC; Sun, SH | 1 |
Chandrasekhar, S; Halladay, D; Martin, TJ; Onyia, JE; Yang, X | 1 |
Bander, E; Faragó, A; Sipeki, S; Ways, DK | 1 |
Fujitani, Y; Gorogawa, S; Hori, M; Kajimoto, Y; Kawamori, D; Kuroda, A; Ohtoshi, K; Umayahara, Y; Yamasaki, Y; Yasuda, T; Yoshida, S | 1 |
Surmacz, L; Wiejak, J; Wyroba, E | 1 |
Barritault, D; Crépin, M; Ledoux, D; Liu, JF; Liu, JM | 1 |
Auberger, P; Bottero, V; Busuttil, V; Frelin, C; Imbert, V; Peyron, JF; Ricci, JE | 1 |
Baker, HW; Dunlop, ME; Garrett, C; Grkovic, I; Liu, DY; Martic, M | 1 |
Joseph, SR; Le, TL; Stow, JL; Yap, AS | 1 |
Fukuta, H; Kito, Y; Suzuki, H; Yamamoto, Y | 1 |
Bragado, MJ; García-Marin, LJ; Jensen, RT; Pace, A; Tapia, JA | 1 |
Banerji, L; Glassford, J; Holman, M; Kadowaki, T; Klaus, GG; Koyasu, S; Lam, EW; Skarell, SM; Soeiro, I | 1 |
Bacon, BR; Britton, RS; Li, L; O'Neill, R; Ramm, GA | 1 |
Bhugra, P; Dhalla, NS; Rathi, S; Xu, YJ | 1 |
Briaud, I; Dickson, LM; Lingohr, MK; Rhodes, CJ; Wrede, CE | 1 |
Cruciani, V; Leithe, E; Mikalsen, SO; Rivedal, E; Sanner, T | 1 |
Cohen, GM; Farrow, SN; Harper, N; Hughes, MA; MacFarlane, M | 1 |
Chain, BM; Cho, JY; Katz, DR | 1 |
Alemany, S; Caivano, M; Cohen, P; Rodriguez, C | 1 |
Chang, YY; Sun, SH; Wang, CM | 1 |
Charkaoui-Malki, M; Cherkaoui-Malki, M; Hichami, A; Khan, NA; Madani, S | 1 |
Dutta, S; Häussinger, D; Kubitz, R; Kühlkamp, T; Saha, N; vom Dahl, S; Wettstein, M | 1 |
Ding, L; Lang, W; Wang, H; Xiao, L | 1 |
Chen, JS; Exton, JH | 1 |
Ajioka, H; Akizawa, Y; Kanda, A; Kiniwa, M; Matsuura, N; Nakano, M; Nishihara, K; Nozawa, Y; Orimoto, N; Uji, T | 1 |
Chang, KC; Kang, YJ; Kim, HJ; Ko, YS; Lee, YS; Park, MK; Pyo, HS; Seo, HG; Yun-Choi, HS | 1 |
Eppig, JJ; O'brien, M; Viveiros, MM | 1 |
Cho, YW; Hahm, ET; Lee, JJ; Min, BI | 1 |
Jiménez, E; Montiel, M; Quesada, J | 1 |
Burrin, JM; Fowkes, RC; Grossman, AB; Khalaf, S; Korbonits, M; Mozid, AM; Nanzer, AM; Patel, MV | 1 |
Daosukho, C; Kiningham, KK; St Clair, DK | 1 |
Brodie, C; Cohen, A; Deutsch, E; Dovrat, S; Kazimirsky, G; Rubinfeld, H; Sarid, R | 1 |
Chen, PW; Kroog, GS | 1 |
Bristulf, J; Owman, C; Sabirsh, A | 1 |
Imamura, T; Ishisaki, A; Nakajima, K; Tsunobuchi, H | 1 |
Branchi, I; Capone, F; Costa, LG; Fattori, V; Giordano, G; Madia, F; Vitalone, A | 1 |
Closs, EI; Martiné, U; Rotmann, A; Strand, D | 1 |
Alviña, K; Boric, MP; Figueroa, XF; Garcés, G; Martínez, AD; Rosemblatt, M; Sáez, JC | 1 |
Leithe, E; Rivedal, E | 1 |
Gylfe, E; Rask, L; Sakwe, AM | 1 |
Madras, BK; Miller, GM; Yatin, SM | 1 |
Camden, JM; Camden, RE; Erb, L; González, FA; Schrader, AM; Seye, CI; Weisman, GA | 1 |
Kuan, YH; Lin, CN; Lin, RH; Tsao, LT; Wang, JP | 1 |
Cameron, P; Kanke, T; Macfarlane, SR; McKenzie, RC; Plevin, R; Sloss, CM | 1 |
Barnes-Davies, M; Bhattacharjee, A; Forsythe, ID; Hamann, M; Kaczmarek, LK; Oliver, DL; Song, P; Yang, Y | 1 |
Gerlo, S; Kooijman, R; Verdood, P | 1 |
Hu, N; Li, L; Sampat, K; Yuspa, SH; Zakari, J | 1 |
Clerk, A; Markou, T; Sugden, PH; Yong, CS | 1 |
Fujii, T; Fukushima, S; Kaneyuki, U; Kato, S; Kazanietz, MG; Maeda, M; Oshima, K; Shigemori, M | 1 |
Gosens, R; Grootte Bromhaar, MM; Maarsingh, H; Meurs, H; Nelemans, SA; ten Damme, A; Zaagsma, J | 1 |
Auersperg, N; Choi, KC; Kim, KY; Leung, PC | 1 |
Cho, NJ; Cho, TJ; Park, YS | 1 |
Akopian, A; Cristofanilli, M | 1 |
Doi, SQ; Glerum, S; Mendonça, MC; Sellitti, DF | 1 |
Linsdell, P; McDonald, TF; Missan, S | 1 |
Hayashi, H; Kondo, T; Suzuki, S; Takagi, K; Ueyama, J; Wakusawa, S | 1 |
Adrian, TE; Bell, RH; Ding, XZ; Flesche, JB; Robin, TP; Salabat, MR; Talamonti, MS; Ujiki, MB | 1 |
Aguilar, R; Bellido, C; Garrido-Gracia, JC; Sánchez-Criado, JE | 1 |
Fujino, H; Hirabayashi, T; Murayama, T; Nakamura, H; Shimizu, M; Taniguchi, T | 1 |
Di Jeso, B; Elia, MG; Marsigliante, S; Muscella, A; Storelli, C; Treglia, AS; Ulianich, L | 1 |
Chang, HC; Chen, IS; Cheng, HH; Chi, CC; Chu, ST; Ho, CM; Hsu, SS; Huang, CJ; Huang, JK; Jan, CR; Liu, SI; Lu, YC; Su, HH; Wang, JL | 1 |
Hara, A; Hirade, K; Hotta, K; Ito, H; Kato, K; Kozawa, O; Niwa, M | 1 |
Burek, CL; Sharma, RB; Traore, K; Trush, MA | 1 |
Bollinger, J; Cherny, VV; DeCoursey, TE; Finnegan, A; Gelb, MH; Morgan, D | 1 |
Abe, K; Nishiura, T | 1 |
Ding, WG; Horie, M; Ito, M; Matsuura, H; Toda, H; Toyoda, F; Yasuda, Y | 1 |
Cockerill, SL; Mitcheson, JS; Standen, NB; Tobin, AB; Torrecilla, I; Willars, GB | 1 |
Carlson, AE; Franceschi, RT; Gopalakrishnan, R; Suttamanatwong, S | 1 |
Chou, CC; Hsu, CY; Yung, BY | 1 |
Eggo, MC; Susarla, R; Watkinson, JC | 1 |
Bond, JA; Errington, R; Gescher, AJ; Lemoine, NR; Smith, PJ; Verschoyle, RD; Wiltshire, M; Wynford-Thomas, D | 1 |
Gergely, P; Kovács, I; Sipka, S; Szíjgyártó, Z; Szucs, K; Zákány, R | 1 |
D'Souza, T; Indig, FE; Morin, PJ | 1 |
Beltran, L; Digiovanni, J; Lu, J; Rho, O; Wilker, E | 1 |
Bocking, AD; Casciani, V; Challis, JR; Di Iorio, R; Marinoni, E; Moscarini, M | 1 |
Chen, P; Soo, J; Xue, R; Zhang, E | 1 |
Hanai, Y; Kozawa, O; Matsushima-Nishiwaki, R; Minamitani, C; Otsuka, T; Takai, S; Tokuda, H | 1 |
Aherne, SA; O'Brien, NM | 1 |
Arakawa, Y; Tomimatsu, N | 1 |
O'Sullivan, AW; Redmond, HP; Wang, JH | 1 |
Grichtchenko, II; Perry, C; Quissell, DO; Reyland, ME | 1 |
Pan, L; Song, K; Wu, X; Xu, J; Zhang, X | 1 |
Stricker, SA | 1 |
Chacko, S; Chang, S; Hypolite, JA; Mohanan, S; Wein, AJ; Zderic, SA | 1 |
Alrefai, WA; Annaba, F; Dwivedi, A; Gill, RK; Saksena, S; Sarwar, Z | 1 |
Ballim, RD; Mowla, S; Prince, S; Teng, H | 1 |
Boehm, S; Drobny, H; Kosenburger, K; Schicker, KW | 1 |
Bhamrah, M; Capasso, M; Cherny, VV; DeCoursey, TE; Dyer, MJ; Morgan, D; Musset, B | 1 |
Hu, T; Liu, Z; Shen, X | 1 |
Li, ZQ; Song, L; Yang, P; Yin, YQ | 1 |
Ali-Osman, F; Okamura, T; Singh, S | 1 |
Ceballos, NR; Volonteri, MC | 1 |
Hirata, K; Imamura, M; Ito, T; Kimura, Y; Kojima, T; Kyuno, D; Murata, M; Sawada, N; Takasawa, A; Tanaka, S; Yamaguchi, H | 1 |
Fukayama, M; Fukushima, N; Ishikawa, S; Kokudo, N; Shibahara, J; Shinozaki, A; Tanaka, M; Umeda, M | 1 |
Benjamin, A; Orogo-Wenn, M; Soukup, B; Walters, D | 1 |
Adachi, T; Hara, H; Kamiya, T; Makino, J | 1 |
Dai, Y; Kobayashi, K; Kogure, Y; Noguchi, K; Wan, Y; Wang, S; Yamanaka, H; Zhang, W; Zhu, W | 1 |
Jensen, RT; Nuche-Berenguer, B; Sancho, V | 1 |
Song, N; Wang, J; Wang, W; Xie, J; Zhang, H | 1 |
Chao, CY; Chen, HW; Li, CC; Lii, CK; Lin, LL; Liu, KL; Lu, CY | 1 |
Furue, MK; Hirata, M; Hirayama, N; Kawamura, S; Kinehara, M; Kohara, A; Matsumura, H; Mimura, S; Suga, M; Tateyama, D; Uchio-Yamada, K; Yanagihara, K | 1 |
Reetz, O; Strauss, U | 1 |
Chang, HT; Chen, FA; Cheng, HH; Cheng, JS; Chou, CT; Jan, CR; Kuo, CC; Kuo, DH; Liang, WZ; Shieh, P; Sun, TK; Tseng, HW | 1 |
Nazıroğlu, M | 1 |
Bhattacharya, S; Bible, PW; Cataisson, C; Gormley, AC; Kellett, MD; Morasso, MI; Palazzo, E; Sun, HW; Yuspa, SH | 1 |
Geng, Y; He, C; Li, L; Li, Y; Liang, X; Ma, Y; Shu, G; Song, X; Ye, G; Yin, L; Yin, Z; Yue, G; Zhang, R; Zhao, Y; Zou, Y | 1 |
294 other study(ies) available for tetradecanoylphorbol acetate and bisindolylmaleimide i
Article | Year |
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NF-kappa B-dependent induction of the NF-kappa B p50 subunit gene promoter underlies self-perpetuation of human immunodeficiency virus transcription in monocytic cells.
Topics: Base Sequence; Binding Sites; Cell Line; Cell Nucleus; Cytoplasm; Enhancer Elements, Genetic; HIV Long Terminal Repeat; HIV-1; Humans; Indoles; Isoenzymes; Macromolecular Substances; Maleimides; Molecular Sequence Data; Monocytes; NF-kappa B; Oligonucleotide Probes; Promoter Regions, Genetic; Protein Kinase C; Tetradecanoylphorbol Acetate; Transcription, Genetic; Virus Replication | 1992 |
Anti-inflammatory properties of Gö 6850: a selective inhibitor of protein kinase C.
Topics: Animals; Anti-Inflammatory Agents; Anti-Inflammatory Agents, Non-Steroidal; Arachidonic Acid; Dinoprostone; Enzyme Inhibitors; Female; Hypersensitivity, Delayed; Indoles; Macrophages, Peritoneal; Maleimides; Mice; Mice, Inbred BALB C; Neutrophils; Protein Kinase C; Superoxides; Tetradecanoylphorbol Acetate | 1995 |
Effects of Na+/H+ antiport and intracellular pH in the regulation of HL-60 cell apoptosis.
Topics: Amiloride; Apoptosis; DNA Damage; Enzyme Inhibitors; HL-60 Cells; Humans; Hydrogen-Ion Concentration; Indoles; Ionophores; Maleimides; Monensin; Protein Kinase C; Sodium-Hydrogen Exchangers; Tetradecanoylphorbol Acetate | 1995 |
Calcium mobilisation controls tyrosine protein phosphorylation independently of the activation of protein kinase C in human platelets.
Topics: Blood Platelets; Calcium; Edetic Acid; Enzyme Activation; Humans; Indoles; Maleimides; Phosphorylation; Phosphotyrosine; Platelet Activation; Platelet Aggregation; Protein Kinase C; Protein Kinases; Protein-Tyrosine Kinases; Signal Transduction; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin; Thrombin; Tyrosine | 1994 |
Insulin-like growth factor I, a unique calcium-dependent stimulator of 1,25-dihydroxyvitamin D3 production. Studies in cultured mouse kidney cells.
Topics: 25-Hydroxyvitamin D3 1-alpha-Hydroxylase; Animals; Binding, Competitive; Biological Transport; Calcitriol; Calcium; Calcium Channel Blockers; Cells, Cultured; Cycloheximide; Enzyme Inhibitors; Humans; Indoles; Insulin; Insulin-Like Growth Factor I; Kidney Tubules, Proximal; Male; Maleimides; Mice; Phosphates; Protein Kinase C; Protein Synthesis Inhibitors; Receptors, Calcitriol; Sodium; Tetradecanoylphorbol Acetate; Verapamil | 1995 |
Signal transduction pathway of acylation stimulating protein: involvement of protein kinase C.
Topics: Blood Proteins; Cells, Cultured; Complement C3a; Diglycerides; Enzyme Activation; Enzyme Inhibitors; Fibroblasts; Humans; Indoles; Maleimides; Naphthalenes; Protein Kinase C; Second Messenger Systems; Signal Transduction; Tetradecanoylphorbol Acetate; Triglycerides | 1995 |
Identification of the mechanism for the inhibition of Na+,K(+)-adenosine triphosphatase by hyperglycemia involving activation of protein kinase C and cytosolic phospholipase A2.
Topics: Animals; Arachidonic Acids; Biological Transport, Active; Cattle; Cells, Cultured; Cytosol; Enzyme Activation; Glucose; Humans; Hyperglycemia; Indoles; Maleimides; Muscle, Smooth, Vascular; Phospholipases A; Phospholipases A2; Phosphorylation; Protein Kinase C; Protein Processing, Post-Translational; Rats; Rats, Sprague-Dawley; Rubidium; Sodium-Potassium-Exchanging ATPase; Tetradecanoylphorbol Acetate | 1995 |
Amyloid precursor protein processing is stimulated by metabotropic glutamate receptors.
Topics: Alanine; Amyloid beta-Peptides; Amyloid beta-Protein Precursor; Animals; Cell Line; Chelating Agents; Cycloleucine; Embryo, Mammalian; Fetus; Glioma; Glutamic Acid; Hippocampus; Humans; Indoles; Kidney; Kinetics; Maleimides; N-Methylaspartate; Neuroblastoma; Neurons; Neurotoxins; PC12 Cells; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositol Phosphates; Protein Kinase C; Protein Processing, Post-Translational; Pyrimidines; Quinacrine; Quisqualic Acid; Rats; Receptors, Metabotropic Glutamate; Recombinant Proteins; Tetradecanoylphorbol Acetate; Transfection; Tumor Cells, Cultured | 1995 |
Protein kinase C mediates down-regulation of cystic fibrosis transmembrane conductance regulator levels in epithelial cells.
Topics: Adenocarcinoma; Colonic Neoplasms; Cycloheximide; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Dactinomycin; Epithelium; Gene Expression Regulation, Neoplastic; Humans; Indoles; Maleimides; Membrane Proteins; Pancreatic Neoplasms; Protein Biosynthesis; Protein Kinase C; RNA, Neoplasm; Tetradecanoylphorbol Acetate; Transcription, Genetic; Transfection; Tumor Cells, Cultured | 1993 |
Alpha 1-adrenoceptor activation increases ecto-5'-nucleotidase activity and adenosine release in rat cardiomyocytes by activating protein kinase C.
Topics: 5'-Nucleotidase; Adenosine; Adenosine Diphosphate; Adenosine Monophosphate; Animals; Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Activation; In Vitro Techniques; Indoles; Male; Maleimides; Methoxamine; Myocardium; Norepinephrine; Protein Kinase C; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Tetradecanoylphorbol Acetate | 1995 |
The protein kinase C inhibitor, bisindolylmaleimide, inhibits the TPA-induced but not the TNF-induced increase in LLC-PK1 transepithelial permeability.
Topics: Animals; Epithelium; In Vitro Techniques; Indoles; LLC-PK1 Cells; Maleimides; Permeability; Protein Kinase C; Swine; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha | 1995 |
Protein kinase C-independent activation of Raf-1 and mitogen-activated protein kinase by leukotriene B4 in guinea pig eosinophils.
Topics: Animals; Calcium-Calmodulin-Dependent Protein Kinases; Dose-Response Relationship, Drug; Enzyme Activation; Eosinophils; Glyceryl Ethers; Guinea Pigs; In Vitro Techniques; Indoles; Kinetics; Leukotriene B4; Male; Maleimides; Phenylpropionates; Protein Kinase C; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-raf; Receptors, Leukotriene B4; Tetradecanoylphorbol Acetate; Time Factors | 1995 |
Effects of protein kinase modulators on transferrin receptor expression in human leukaemic HL-60 cells.
Topics: Alkaloids; Bucladesine; Cell Division; Cell Line; Cyclic AMP-Dependent Protein Kinases; DNA, Neoplasm; Enzyme Activation; Gene Expression; Humans; Indoles; Isoquinolines; Leukemia, Promyelocytic, Acute; Maleimides; Protein Kinase C; Protein Kinases; Receptors, Transferrin; RNA, Messenger; Staurosporine; Sulfonamides; Tetradecanoylphorbol Acetate; Thymidine; Tumor Cells, Cultured | 1995 |
Preferential inhibition of phorbol ester-induced hydrolysis of phosphatidylethanolamine by N-acetylsphingosine in NIH 3T3 fibroblasts.
Topics: 3T3 Cells; Animals; Carbon Radioisotopes; Fibroblasts; Hydrolysis; Indoles; Kinetics; Maleimides; Mice; Palmitic Acid; Palmitic Acids; Phosphatidylethanolamines; Phospholipase D; Protein Kinase C; Radioisotope Dilution Technique; Rats; Sphingosine; Tetradecanoylphorbol Acetate | 1995 |
Thrombin and phorbol ester induce internalization of thrombin receptor of human mesangial cells through different pathways.
Topics: Alkaloids; Cell Membrane Permeability; Glomerular Mesangium; Humans; Indoles; Maleimides; Peptide Fragments; Protein Kinase C; Receptors, Thrombin; RNA, Messenger; Staurosporine; Tetradecanoylphorbol Acetate; Thrombin | 1995 |
The bisindolylmaleimide GF 109203X, a selective inhibitor of protein kinase C, does not inhibit the potentiating effect of phorbol ester on ethanol-induced phospholipase C-mediated hydrolysis of phosphatidylethanolamine.
Topics: 3T3 Cells; Animals; Ethanol; Ethanolamines; Indoles; Maleimides; Mice; Phosphatidylethanolamines; Protein Kinase C; Tetradecanoylphorbol Acetate; Type C Phospholipases | 1995 |
Differential modulation of human fibroblast and keratinocyte growth by the protein kinase C inhibitor GF 109203X.
Topics: Adolescent; Adult; Blotting, Northern; Casein Kinase II; Cell Differentiation; Cell Division; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Epidermal Growth Factor; Female; Fibroblasts; Gene Expression; Genes, fos; Genes, jun; Glyceraldehyde-3-Phosphate Dehydrogenases; Humans; Indoles; Keratinocytes; Maleimides; Middle Aged; Protein Binding; Protein Kinase C; Protein Serine-Threonine Kinases; RNA, Messenger; Tetradecanoylphorbol Acetate | 1994 |
Protein kinase C-dependent and -independent pathways of mitogen-activated protein kinase activation in macrophages by stimuli that activate phospholipase A2.
Topics: Animals; Arachidonic Acid; Calcimycin; Calcium-Calmodulin-Dependent Protein Kinases; Down-Regulation; Enzyme Activation; Ethers, Cyclic; Gene Expression Regulation, Enzymologic; Indoles; Isoenzymes; Macrophages, Peritoneal; Maleimides; Mice; Okadaic Acid; Phospholipases A; Phospholipases A2; Phosphoprotein Phosphatases; Phosphorylation; Protein Kinase C; Protein Kinase C-alpha; Signal Transduction; Tetradecanoylphorbol Acetate; Tyrosine; Zymosan | 1994 |
Increase of c-jun mRNA upon hypo-osmotic cell swelling of rat hepatoma cells.
Topics: Animals; Cell Size; Enzyme Activation; Indoles; Liver Neoplasms, Experimental; Maleimides; Osmolar Concentration; Protein Kinase C; Proto-Oncogene Proteins c-jun; Rats; RNA, Messenger; Signal Transduction; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1994 |
A protein kinase C-dependent activity modulates retinoic acid-induced transcription.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amino Acid Sequence; Animals; Cell Line; Cell Nucleus; Chlorocebus aethiops; DNA; Enzyme Induction; Humans; Indoles; Isoenzymes; Isoquinolines; Maleimides; Molecular Sequence Data; Phosphorylation; Piperazines; Promoter Regions, Genetic; Protein Binding; Protein Kinase C; Protein Processing, Post-Translational; Receptors, Retinoic Acid; Recombinant Fusion Proteins; Signal Transduction; Tetradecanoylphorbol Acetate; Transcription, Genetic; Tretinoin | 1993 |
PMA inhibits the growth of human fibroblasts after the induction of immediate-early genes.
Topics: Cell Cycle; Culture Media, Serum-Free; Fibroblasts; Gene Expression Regulation; Genes, fos; Genes, Immediate-Early; Genes, jun; Humans; Indoles; Maleimides; Protein Kinase C; RNA, Messenger; Tetradecanoylphorbol Acetate; Thrombin | 1994 |
Protein kinase C modulates the activity of a cloned gamma-aminobutyric acid transporter expressed in Xenopus oocytes via regulated subcellular redistribution of the transporter.
Topics: Animals; Biological Transport; Brain; Carrier Proteins; Cloning, Molecular; Cyclosporine; Cytoplasm; Female; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Gene Expression; Golgi Apparatus; Indoles; Kinetics; Maleimides; Membrane Proteins; Membrane Transport Proteins; Nerve Tissue Proteins; Oocytes; Organic Anion Transporters; Protein Kinase C; Rats; Serotonin; Subcellular Fractions; Tetradecanoylphorbol Acetate; Xenopus | 1994 |
N-protein kinase C isoenzymes may be involved in the regulation of various neutrophil functions.
Topics: Carbazoles; Enzyme Activation; Humans; In Vitro Techniques; Indoles; Isoenzymes; Maleimides; Muramidase; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Protein Kinase C; Respiratory Burst; Superoxides; Tetradecanoylphorbol Acetate | 1994 |
Calpain-induced downregulation of activated protein kinase C-alpha affects lung epithelial cell morphology.
Topics: Animals; Calpain; Cell Line; Cell Line, Transformed; Cytosol; Epithelial Cells; Epithelium; Indoles; Isoenzymes; Kinetics; Lung; Maleimides; Mice; Protein Kinase C; Tetradecanoylphorbol Acetate; Time Factors | 1994 |
Anti-CD3 and phorbol ester induce distinct phosphorylated sites in the SH2 domain of p56lck.
Topics: Amino Acid Sequence; Binding Sites; CD3 Complex; Cells, Cultured; Indoles; Lymphocyte Specific Protein Tyrosine Kinase p56(lck); Maleimides; Molecular Sequence Data; Peptide Mapping; Phosphorylation; Protein Kinase C; Protein-Tyrosine Kinases; Serine; Tetradecanoylphorbol Acetate; Trypsin | 1993 |
Anti-inflammatory properties of the protein kinase C inhibitor, 3-[1-[3-(dimethylamino)propyl]-1H-indol-3-yl]-4-(1H-indol-3-yl)-1H- pyrrole-2,5-dione monohydrochloride (GF109203X) in the PMA-mouse ear edema model.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Dinoprostone; Disease Models, Animal; Dose-Response Relationship, Drug; Ear; Edema; Eicosanoids; Female; Indoles; Inflammation; Maleimides; Mice; Neutrophils; Peroxidase; Protein Kinase C; Radioimmunoassay; Tetradecanoylphorbol Acetate | 1993 |
Muscarinic inhibition of ATP-sensitive K+ channels by protein kinase C in urinary bladder smooth muscle.
Topics: Adenosine Triphosphate; Animals; Benzopyrans; Carbachol; Cromakalim; Diglycerides; Glyburide; Guanosine Diphosphate; Guinea Pigs; In Vitro Techniques; Indoles; Maleimides; Membrane Potentials; Muscarinic Antagonists; Muscle, Smooth; Potassium Channels; Protein Kinase C; Pyrroles; Receptors, Muscarinic; Tetradecanoylphorbol Acetate; Thionucleotides; Urinary Bladder | 1993 |
The selective protein kinase C inhibitor GF 109203X inhibits phorbol ester-induced morphological and functional differentiation of SH-SY5Y human neuroblastoma cells.
Topics: Blotting, Northern; Cell Differentiation; Cell Line; Dose-Response Relationship, Drug; GAP-43 Protein; Gene Expression; Genes, fos; Humans; Indoles; Kinetics; Maleimides; Membrane Glycoproteins; Molecular Weight; Nerve Tissue Proteins; Neurites; Neuroblastoma; Neuropeptide Y; Phosphoproteins; Phosphorylation; Protein Kinase C; Proto-Oncogene Mas; Proto-Oncogene Proteins c-fos; RNA, Messenger; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1993 |
Distinct mechanisms of phospholipase D activation and attenuation utilized by different mitogens in NIH-3T3 fibroblasts.
Topics: 3T3 Cells; Alkaloids; Animals; Dinoprost; Dose-Response Relationship, Drug; Enzyme Activation; Hydrolysis; Indoles; Maleimides; Mice; Mitogens; Phosphatidic Acids; Phospholipase D; Phospholipids; Platelet-Derived Growth Factor; Staurosporine; Tetradecanoylphorbol Acetate | 1993 |
Overexpression of protein kinase C-delta and -epsilon in NIH 3T3 cells induces opposite effects on growth, morphology, anchorage dependence, and tumorigenicity.
Topics: 3T3 Cells; Animals; Biological Transport; Blotting, Northern; Blotting, Western; Brain; Cell Adhesion; Cell Division; Cell Transformation, Neoplastic; Cloning, Molecular; Enzyme Activation; Enzyme Stability; Indoles; Isoenzymes; Kinetics; Maleimides; Mice; Mice, Inbred C57BL; Mice, Nude; Neoplasms, Experimental; Protein Kinase C; Tetradecanoylphorbol Acetate | 1993 |
Overexpression of epsilon-protein kinase C enhances nerve growth factor-induced phosphorylation of mitogen-activated protein kinases and neurite outgrowth.
Topics: Amino Acid Sequence; Analysis of Variance; Animals; Blotting, Western; Calcium-Calmodulin-Dependent Protein Kinases; Cell Differentiation; Enzyme Inhibitors; Ethanol; Fluorescent Antibody Technique; Gene Expression; Indoles; Isoenzymes; Maleimides; Microscopy, Fluorescence; Molecular Sequence Data; Nerve Growth Factors; Neurites; PC12 Cells; Peptides; Phosphorylation; Protein Kinase C; Rats; Recombinant Proteins; Substrate Specificity; Tetradecanoylphorbol Acetate; Transfection | 1995 |
Inhibition of protein kinase C suppresses megakaryocytic differentiation and stimulates erythroid differentiation in HEL cells.
Topics: Aphidicolin; Biomarkers; Blood Proteins; Cell Cycle; Cell Differentiation; Enzyme Inhibitors; Erythroid Precursor Cells; Gene Expression Regulation, Leukemic; Globins; Glycophorins; Hematopoietic Stem Cells; Hemin; Humans; Indoles; Leukemia, Erythroblastic, Acute; Maleimides; Megakaryocytes; Neoplasm Proteins; Phorbol 12,13-Dibutyrate; Phosphoproteins; Phosphorylation; Platelet Membrane Glycoproteins; Protein Kinase C; Protein Processing, Post-Translational; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1996 |
Protein kinase C regulates tyrosine phosphorylation of pp125FAK in platelets adherent to fibrinogen.
Topics: Adenosine Diphosphate; Apyrase; Blood Platelets; Calcium; Cell Adhesion Molecules; Cell Size; Egtazic Acid; Enzyme Inhibitors; Fibrinogen; Focal Adhesion Kinase 1; Focal Adhesion Protein-Tyrosine Kinases; Humans; Indoles; Maleimides; Phosphoproteins; Phosphorylation; Platelet Adhesiveness; Platelet Glycoprotein GPIIb-IIIa Complex; Protein Kinase C; Protein Processing, Post-Translational; Protein-Tyrosine Kinases; Signal Transduction; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin; Tyrosine | 1996 |
1,25-dihydroxyvitamin D3 primes acute promyelocytic cells for TPA-induced monocytic differentiation through both PKC and tyrosine phosphorylation cascades.
Topics: Alkaloids; Calcitriol; Cell Differentiation; Enzyme Inhibitors; Genistein; Humans; Indoles; Isoflavones; Leukemia, Promyelocytic, Acute; Maleimides; Monocytes; Phagocytosis; Phosphorylation; Protein Kinase C; Protein Tyrosine Phosphatases; Protein-Tyrosine Kinases; Signal Transduction; Staurosporine; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Tyrosine; Vanadates | 1996 |
Phorbol ester-stimulated phosphorylation of PU.1: association with leukemic cell growth inhibition.
Topics: Base Sequence; Bryostatins; Cell Differentiation; Cell Division; DNA, Neoplasm; Enhancer Elements, Genetic; Enzyme Inhibitors; Gene Expression Regulation, Leukemic; Humans; Indoles; Lactones; Lymphoma, Large B-Cell, Diffuse; Macrolides; Maleimides; Molecular Sequence Data; Neoplasm Proteins; Phosphorylation; Protein Binding; Protein Kinase C; Protein Processing, Post-Translational; Proto-Oncogene Proteins; Proto-Oncogenes; RNA, Messenger; RNA, Neoplasm; Tetradecanoylphorbol Acetate; Trans-Activators; Transcription Factors; Transcription, Genetic; Tumor Cells, Cultured | 1996 |
Mechanism of apoptosis suppression by phorbol ester in IL-6-starved murine plasmacytomas: role of PKC modulation and cell cycle.
Topics: Alkaloids; Animals; Apoptosis; Benzophenanthridines; Cell Cycle; Cell Line; Cytosol; Enzyme Activation; Enzyme Inhibitors; Indoles; Interleukin-6; Isoenzymes; Lactams; Maleimides; Mice; Phenanthridines; Phorbol Esters; Plasmacytoma; Protein Kinase C; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1996 |
Modulation of keratinocyte growth factor (KGF) mRNA expression in human dermal fibroblasts grown in monolayer or within a collagen matrix.
Topics: Adolescent; Adult; Breast; Cell Division; Cells, Cultured; Cholera Toxin; Culture Media, Conditioned; Enzyme Inhibitors; Epidermal Growth Factor; Female; Fibroblast Growth Factor 10; Fibroblast Growth Factor 7; Fibroblast Growth Factors; Fibroblasts; Growth Substances; Humans; Indoles; Keratinocytes; Maleimides; Middle Aged; Protein Kinase C; RNA, Messenger; Signal Transduction; Skin; Surgery, Plastic; Tetradecanoylphorbol Acetate; Transcription, Genetic | 1996 |
Inhibition of T lymphocyte activation by cAMP is associated with down-regulation of two parallel mitogen-activated protein kinase pathways, the extracellular signal-related kinase and c-Jun N-terminal kinase.
Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Bucladesine; Calcium-Calmodulin-Dependent Protein Kinases; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Inhibitors; ErbB Receptors; Humans; Indoles; Isoenzymes; JNK Mitogen-Activated Protein Kinases; Leukemia-Lymphoma, Adult T-Cell; Lymphocyte Activation; Lymphocyte Specific Protein Tyrosine Kinase p56(lck); Lymphoma, T-Cell; Maleimides; Mice; Mitogen-Activated Protein Kinases; Mitogens; Molecular Sequence Data; Muromonab-CD3; Nerve Tissue Proteins; Peptide Fragments; Phosphorylation; Protein Kinase C; Protein Processing, Post-Translational; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-jun; Signal Transduction; T-Lymphocytes; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1996 |
Protein kinase C-epsilon is implicated in neurite outgrowth in differentiating human neuroblastoma cells.
Topics: Cell Differentiation; Down-Regulation; Enzyme Inhibitors; Growth Substances; Humans; Indoles; Isoenzymes; Maleimides; Neurites; Neuroblastoma; Neurons; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-epsilon; Tetradecanoylphorbol Acetate; Transcription, Genetic | 1996 |
The kinase inhibitor iso-H7 stimulates rat satellite cell differentiation through a non-protein kinase C pathway by increasing myogenin expression level.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Blotting, Northern; Cell Differentiation; Creatine Kinase; Enzyme Inhibitors; Indoles; Isoquinolines; Maleimides; Muscle, Skeletal; Myogenin; Myosin Light Chains; Protein Kinase C; Rats; Rats, Wistar; RNA, Messenger; Sulfonamides; Tetradecanoylphorbol Acetate | 1996 |
Transcriptional control of the heme oxygenase gene in mouse M1 cells during their TPA-induced differentiation into macrophages.
Topics: Acetylcysteine; Animals; Binding Sites; Carcinogens; Cell Differentiation; Electrophoresis; Enzyme Inhibitors; Free Radical Scavengers; Gene Expression Regulation, Neoplastic; Genes, fos; Genes, jun; Heme Oxygenase (Decyclizing); Hydrogen Peroxide; Indoles; Leukemia, Myeloid; Macrophages; Maleimides; Mice; NF-kappa B; Nuclear Proteins; Protein Kinase C; Signal Transduction; Tetradecanoylphorbol Acetate; Transcription Factor AP-1; Transcription, Genetic; Tumor Cells, Cultured | 1996 |
Direct proof that phorbol ester accelerates the use of choline phosphate for phosphatidylcholine synthesis in intact cells.
Topics: 3T3 Cells; Animals; Carbon Radioisotopes; Choline; Choline-Phosphate Cytidylyltransferase; Enzyme Inhibitors; Indoles; Kinetics; Maleimides; Mice; Nucleotidyltransferases; Phosphatidylcholines; Phosphorylcholine; Protein Kinase C; Radioisotope Dilution Technique; Tetradecanoylphorbol Acetate | 1996 |
Protein kinase C activity and phosphoprotein pattern in stimulated alveolar macrophages.
Topics: Animals; Cattle; Cytosol; Electrophoresis, Gel, Two-Dimensional; In Vitro Techniques; Indoles; Macrophage Activation; Macrophages, Alveolar; Maleimides; Phosphoproteins; Protein Kinase C; Rats; Spectrometry, Fluorescence; Staurosporine; Tetradecanoylphorbol Acetate | 1996 |
Activation of G-proteins with AIF-4 induces LFA-1-mediated adhesion of T-cell hybridoma cells to ICAM-1 by signal pathways that differ from phorbol ester- and manganese-induced adhesion.
Topics: Aluminum Compounds; Androstadienes; Animals; Cell Adhesion; Enzyme Activation; Enzyme Inhibitors; Estrenes; Fluorides; Genistein; GTP-Binding Proteins; Humans; Hybridomas; Indoles; Intercellular Adhesion Molecule-1; Isoflavones; Lymphocyte Function-Associated Antigen-1; Maleimides; Manganese; Mice; Neoplasm Invasiveness; Neoplasm Proteins; Phosphatidylinositol 3-Kinases; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositol Diacylglycerol-Lyase; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Phosphotransferases (Alcohol Group Acceptor); Protein Kinase C; Protein-Tyrosine Kinases; Pyrrolidinones; Signal Transduction; T-Lymphocytes; Tetradecanoylphorbol Acetate; Wortmannin | 1997 |
Inhibition of cytosolic phospholipase A2 by annexin V in differentiated permeabilized HL-60 cells. Evidence of crucial importance of domain I type II Ca2+-binding site in the mechanism of inhibition.
Topics: Annexin A5; Arachidonic Acid; Bacterial Proteins; Binding Sites; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Cell Differentiation; Cell Membrane Permeability; Cytosol; Enzyme Inhibitors; Female; Guanosine 5'-O-(3-Thiotriphosphate); HL-60 Cells; Humans; Indoles; Kinetics; Maleimides; N-Formylmethionine Leucyl-Phenylalanine; Phospholipases A; Phospholipases A2; Placenta; Pregnancy; Protein Kinase C; Recombinant Proteins; Streptolysins; Tetradecanoylphorbol Acetate | 1997 |
Prostaglandin F2alpha stimulates tyrosine phosphorylation and mitogen-activated protein kinase in osteoblastic MC3T3-E1 cells via protein kinase C activation.
Topics: Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Dinoprost; Enzyme Activation; Enzyme Inhibitors; Immunosorbent Techniques; Indoles; Maleimides; Osteoblasts; Phosphorylation; Phosphotyrosine; Protein Kinase C; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-raf; Tetradecanoylphorbol Acetate | 1997 |
Activation of ecto-5'-nucleotidase by protein kinase C and its role in ischaemic tolerance in the canine heart.
Topics: 5'-Nucleotidase; Animals; Dogs; Enzyme Activation; Female; Hemodynamics; Indoles; Ischemic Preconditioning; Male; Maleimides; Myocardial Infarction; Myocardial Ischemia; Phosphorylation; Protein Kinase C; Tetradecanoylphorbol Acetate | 1997 |
CSF-1-induced and constitutive Il6 gene expression in mouse macrophages: evidence for PKC-dependent and -independent pathways.
Topics: Animals; Drug Synergism; Enzyme Inhibitors; Gene Expression Regulation; Indoles; Interleukin-6; Macrophage Colony-Stimulating Factor; Macrophages, Peritoneal; Male; Maleimides; Mice; Mice, Inbred C57BL; Mice, SCID; Protein Kinase C; Signal Transduction; Staurosporine; Tetradecanoylphorbol Acetate | 1997 |
Expression of CD44 isoforms in neuroblastoma cells is regulated by PI 3-kinase and protein kinase C.
Topics: Carcinogens; Cell Adhesion; Enzyme Inhibitors; Humans; Hyaluronan Receptors; Hyaluronic Acid; Indoles; Insulin-Like Growth Factor I; Maleimides; Models, Molecular; Neuroblastoma; Phosphatidylinositol 3-Kinases; Phosphotransferases (Alcohol Group Acceptor); Platelet-Derived Growth Factor; Protein Kinase C; Signal Transduction; Surface Properties; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Up-Regulation | 1997 |
Phosphorylation of the respiratory burst oxidase subunit p67(phox) during human neutrophil activation. Regulation by protein kinase C-dependent and independent pathways.
Topics: Enzyme Activation; Enzyme Inhibitors; Humans; Indoles; Lymphocyte Activation; Maleimides; N-Formylmethionine Leucyl-Phenylalanine; NADH, NADPH Oxidoreductases; NADPH Oxidases; Neutrophils; Peptide Mapping; Phosphoproteins; Phosphorylation; Protein Kinase C; Serine; Tetradecanoylphorbol Acetate | 1997 |
N-6 and n-3 polyunsaturated fatty acids stimulate translocation of protein kinase Calpha, -betaI, -betaII and -epsilon and enhance agonist-induced NADPH oxidase in macrophages.
Topics: Calcimycin; Docosahexaenoic Acids; Enzyme Inhibitors; Fatty Acids, Unsaturated; Histones; HL-60 Cells; Humans; Indoles; Ionophores; Isoenzymes; Luminescent Measurements; Macrophages; Maleimides; Monocytes; N-Formylmethionine Leucyl-Phenylalanine; NADPH Oxidases; Phosphorylation; Protein Kinase C; Tetradecanoylphorbol Acetate | 1997 |
Activation of mitogen-activated protein kinase by the nociceptin receptor expressed in Chinese hamster ovary cells.
Topics: Androstadienes; Animals; Calcium-Calmodulin-Dependent Protein Kinases; CHO Cells; Chromones; Cricetinae; Cricetulus; Down-Regulation; Enzyme Activation; Enzyme Inhibitors; Indoles; Maleimides; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Morpholines; Nociceptin Receptor; Phosphatidylinositol 3-Kinases; Phosphotransferases (Alcohol Group Acceptor); Protein Binding; Protein Kinase C; Protein-Tyrosine Kinases; Receptors, Opioid; Recombinant Proteins; Tetradecanoylphorbol Acetate; Wortmannin | 1997 |
Down-regulation of gap junctional intercellular communication between osteoblastic MC3T3-E1 cells by basic fibroblast growth factor and a phorbol ester (12-O-tetradecanoylphorbol-13-acetate).
Topics: 3T3 Cells; Animals; Blotting, Northern; Blotting, Western; Carcinogens; Cell Communication; DNA; Dose-Response Relationship, Drug; Down-Regulation; Fibroblast Growth Factor 2; Gap Junctions; Humans; Indoles; Maleimides; Mice; Osteoblasts; Protein Kinase C; Recombinant Proteins; Tetradecanoylphorbol Acetate | 1997 |
Cellular relocalisation of protein kinase C-theta caused by staurosporine and some of its analogues.
Topics: Alkaloids; Antineoplastic Agents; Blotting, Western; Cell Membrane; Cell Nucleus; Cytosol; Enzyme Inhibitors; Fluorescent Antibody Technique, Indirect; Humans; Indoles; Isoenzymes; Maleimides; Microscopy, Confocal; Models, Chemical; Protein Kinase C; Protein Kinase C-theta; Staurosporine; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Zinc Fingers | 1997 |
Upregulation of CD9 expression during TPA treatment of K562 cells.
Topics: Antigens, CD; Cell Differentiation; Flow Cytometry; Gene Expression Regulation, Neoplastic; Humans; Indoles; Integrin alpha1beta1; Integrins; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Maleimides; Megakaryocytes; Membrane Glycoproteins; Platelet Glycoprotein GPIIb-IIIa Complex; Promoter Regions, Genetic; RNA, Messenger; Tetradecanoylphorbol Acetate; Tetraspanin 29; Time Factors; Tumor Cells, Cultured; Up-Regulation | 1997 |
Role of protein kinases in the in vitro differentiation of human epidermal HaCaT cells.
Topics: Adenine; Cell Differentiation; Cell Line; Enzyme Inhibitors; Epidermal Cells; Epidermis; Genistein; Humans; Indoles; Isoenzymes; Isoflavones; Keratinocytes; Maleimides; Okadaic Acid; Phosphoprotein Phosphatases; Protein Kinase C; Protein Kinases; Protein-Tyrosine Kinases; Staurosporine; Tetradecanoylphorbol Acetate | 1997 |
Priming of mouse macrophages with the macrophage colony-stimulating factor (CSF-1) induces a variety of pathways that regulate expression of the interleukin 6 (Il6) and granulocyte-macrophage colony-stimulating factor (Csfgm) genes.
Topics: Animals; Cells, Cultured; Down-Regulation; Enzyme Inhibitors; Flow Cytometry; Granulocyte-Macrophage Colony-Stimulating Factor; Indoles; Interleukin-6; Kinetics; Macrophage Colony-Stimulating Factor; Macrophages, Peritoneal; Male; Maleimides; Mice; Mice, Inbred C57BL; Polymerase Chain Reaction; Protein Kinase Inhibitors; Protein Kinases; Receptor, Macrophage Colony-Stimulating Factor; RNA, Messenger; Staurosporine; Tetradecanoylphorbol Acetate; Transcription, Genetic | 1997 |
Roles for protein kinase C and mitogen-activated protein kinase in nicotine-induced secretion from bovine adrenal chromaffin cells.
Topics: Adrenal Medulla; Animals; Calcimycin; Calcium-Calmodulin-Dependent Protein Kinases; Cattle; Cells, Cultured; Chromaffin Cells; Enzyme Activation; Enzyme Inhibitors; Exocytosis; Flavonoids; Indoles; Kinetics; Maleimides; Nicotine; Norepinephrine; Potassium Chloride; Protein Kinase C; Signal Transduction; Tetradecanoylphorbol Acetate | 1997 |
Effect of the protein kinase C inhibitor GF 109 203X on elastase release and respiratory burst of human neutrophils.
Topics: Calcimycin; Calcium; Enzyme Inhibitors; Exocytosis; Humans; In Vitro Techniques; Indoles; L-Lactate Dehydrogenase; Leukocyte Elastase; Maleimides; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Protein Kinase C; Respiratory Burst; Superoxides; Tetradecanoylphorbol Acetate | 1996 |
Serine phosphorylation-regulated ubiquitination and degradation of beta-catenin.
Topics: Amino Acid Sequence; beta Catenin; Consensus Sequence; Cytoskeletal Proteins; DNA-Binding Proteins; Enzyme Inhibitors; Humans; I-kappa B Proteins; Indoles; Maleimides; Molecular Sequence Data; Mutagenesis, Site-Directed; Naphthalenes; NF-kappa B; NF-KappaB Inhibitor alpha; Phosphorylation; Phosphoserine; Point Mutation; Protein Kinase C; Protein Processing, Post-Translational; Sequence Alignment; Serine; Substrate Specificity; Tetradecanoylphorbol Acetate; Trans-Activators; Ubiquitins | 1997 |
Mitogen-activated protein kinases mediate the stimulation of bile acid secretion by tauroursodeoxycholate in rat liver.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Bucladesine; Calcium-Calmodulin-Dependent Protein Kinases; Cells, Cultured; Colforsin; Enzyme Activation; Enzyme Inhibitors; Flavonoids; GTP-Binding Proteins; Indoles; Isomerism; Isoproterenol; Kinetics; Liver; Male; Maleimides; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Models, Biological; Protein Kinase C; Protein-Tyrosine Kinases; Rats; Rats, Wistar; Signal Transduction; Taurochenodeoxycholic Acid; Taurocholic Acid; Tetradecanoylphorbol Acetate | 1997 |
Inactivation of melatonin receptors by protein kinase C in human prostate epithelial cells.
Topics: Aged; Aged, 80 and over; Animals; Calcium Chloride; Carcinogens; Cells, Cultured; Cyclic GMP; Enzyme Inhibitors; Epithelial Cells; Epithelium; Humans; Indoles; Iodine Radioisotopes; Male; Maleimides; Melatonin; Middle Aged; Prostate; Protein Kinase C; Rats; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Tetradecanoylphorbol Acetate; Thymidine; Tritium | 1997 |
Role of protein kinase C-alpha in activation of ecto-5'-nucleotidase in the preconditioned canine myocardium.
Topics: Adenosine Triphosphatases; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Biological Transport; Blood Pressure; Cell Membrane; Dogs; Enzyme Activation; Enzyme Inhibitors; Heart Rate; Indoles; Ischemic Preconditioning, Myocardial; Isoenzymes; Maleimides; Methoxamine; Myocardium; Okadaic Acid; Prazosin; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-delta; Protein Kinase C-epsilon; Tetradecanoylphorbol Acetate | 1997 |
Both the catalytic and regulatory domains of protein kinase C chimeras modulate the proliferative properties of NIH 3T3 cells.
Topics: 3T3 Cells; Animals; Binding Sites; Catalysis; Cell Division; Enzyme Inhibitors; Indoles; Isoenzymes; Maleimides; Mice; Platelet-Derived Growth Factor; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-delta; Protein Kinase C-epsilon; Recombinant Fusion Proteins; Tetradecanoylphorbol Acetate; Transfection | 1997 |
Molecular mechanisms for the growth factor action of gastrin.
Topics: Animals; Benzodiazepinones; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Devazepide; DNA-Binding Proteins; Enzyme Inhibitors; ets-Domain Protein Elk-1; Flavonoids; Gastrins; Genes, fos; Hormone Antagonists; Humans; Indoles; Luciferases; Maleimides; Mitogen-Activated Protein Kinase 1; Pancreas; Pertussis Toxin; Promoter Regions, Genetic; Protein Kinase C; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-fos; Rats; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Recombinant Proteins; Tetradecanoylphorbol Acetate; Transcription Factors; Transcription, Genetic; Transfection; Virulence Factors, Bordetella | 1997 |
Cholecystokinin-stimulated tyrosine phosphorylation of p125FAK and paxillin is mediated by phospholipase C-dependent and -independent mechanisms and requires the integrity of the actin cytoskeleton and participation of p21rho.
Topics: Actins; Animals; Calcimycin; Calcium; Cell Adhesion Molecules; Cytoskeletal Proteins; Cytoskeleton; Enzyme Inhibitors; Focal Adhesion Kinase 1; Focal Adhesion Protein-Tyrosine Kinases; GTP-Binding Proteins; Indoles; Inositol Phosphates; Kinetics; Male; Maleimides; Models, Biological; Pancreas; Paxillin; Phospholipases; Phosphoproteins; Phosphorylation; Protein Kinase C; Protein-Tyrosine Kinases; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; rho GTP-Binding Proteins; Sincalide; Tetradecanoylphorbol Acetate; Tyrosine | 1997 |
Neuromedin B receptor activation causes tyrosine phosphorylation of p125FAK by a phospholipase C independent mechanism which requires p21rho and integrity of the actin cytoskeleton.
Topics: Actin Cytoskeleton; Actins; ADP Ribose Transferases; Animals; Botulinum Toxins; Calcimycin; Calcium; Cell Adhesion Molecules; Colchicine; Cytochalasin D; Enzyme Inhibitors; Focal Adhesion Kinase 1; Focal Adhesion Protein-Tyrosine Kinases; Gastrin-Releasing Peptide; GTP-Binding Proteins; Indoles; Maleimides; Mice; Neurokinin B; Nitriles; Phosphorylation; Phosphotyrosine; Protein-Tyrosine Kinases; Rats; Receptors, Bombesin; rho GTP-Binding Proteins; Tetradecanoylphorbol Acetate; Thapsigargin; Transfection; Tumor Cells, Cultured; Type C Phospholipases; Tyrphostins | 1997 |
Acetylcholine agonists stimulate mitogen-activated protein kinase in oligodendrocyte progenitors by muscarinic receptors.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Animals, Newborn; Atropine; Brain; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Cells, Cultured; Cholinergic Agents; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Indoles; Maleimides; Mitogen-Activated Protein Kinase 1; Oligodendroglia; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Signal Transduction; Stem Cells; Tetradecanoylphorbol Acetate | 1997 |
P2U purinergic receptor inhibits apical IsK/KvLQT1 channel via protein kinase C in vestibular dark cells.
Topics: Adenosine Triphosphate; Amino Acid Sequence; Animals; Base Sequence; Calcium Channels; Cloning, Molecular; DNA Primers; Enzyme Activation; Enzyme Inhibitors; Epithelial Cells; Estrenes; Gerbillinae; Humans; In Vitro Techniques; Indoles; KCNQ Potassium Channels; KCNQ1 Potassium Channel; Maleimides; Membrane Potentials; Molecular Sequence Data; Polymerase Chain Reaction; Potassium Channels; Potassium Channels, Voltage-Gated; Protein Kinase C; Pyrrolidinones; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2Y2; Sequence Alignment; Tetradecanoylphorbol Acetate; Type C Phospholipases; Vestibule, Labyrinth | 1997 |
Induction of 12-lipoxygenase expression by phorbol 12-myristate 13-acetate in human epidermoid carcinoma A431 cells.
Topics: Arachidonate 12-Lipoxygenase; Base Sequence; Blotting, Western; Carcinoma, Squamous Cell; DNA-Binding Proteins; Enzyme Induction; Genes, Reporter; Humans; Indoles; Luciferases; Maleimides; Microsomes; Molecular Sequence Data; Mutagenesis, Site-Directed; Nuclear Proteins; Promoter Regions, Genetic; RNA, Messenger; Sp1 Transcription Factor; Tetradecanoylphorbol Acetate; Transfection; Tumor Cells, Cultured | 1998 |
The microbial alkaloid toxin staurosporine blocks the phorbol ester-induced increase in beta-amyloid precursor protein in PC12 cells.
Topics: Alkaloids; Amyloid beta-Protein Precursor; Animals; Dose-Response Relationship, Drug; Down-Regulation; Enzyme Inhibitors; Indoles; Isomerism; Maleimides; PC12 Cells; Protein Kinase C; Rats; Staurosporine; Tetradecanoylphorbol Acetate; Time Factors | 1997 |
Extracellular signal-regulated kinase (ERK) activity is required for TPA-mediated inhibition of drug-induced apoptosis.
Topics: Anisomycin; Apoptosis; Calcium-Calmodulin-Dependent Protein Kinases; DNA Fragmentation; Enzyme Activation; Enzyme Inhibitors; Flavonoids; HL-60 Cells; Humans; Indoles; JNK Mitogen-Activated Protein Kinases; Maleimides; Mitogen-Activated Protein Kinases; Naphthalenes; Protein Kinase C; Tetradecanoylphorbol Acetate | 1998 |
Induction of apoptosis by hepatocyte growth factor/scatter factor and its augmentation by phorbol esters in Meth A cells.
Topics: Animals; Apoptosis; Benzimidazoles; Cell Cycle; Cell Survival; DNA Fragmentation; DNA Replication; Flow Cytometry; Fluorescent Dyes; Hepatocyte Growth Factor; Indoles; Maleimides; Mice; Protein Kinase C; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1998 |
Cross-talk between protein kinase C-alpha (PKC-alpha) and -delta (PKC-delta): PKC-alpha elevates the PKC-delta protein level, altering its mRNA transcription and degradation.
Topics: Animals; Enzyme Activation; Enzyme Stability; Indoles; Isoenzymes; Leukemia, Promyelocytic, Acute; Lymphoma, B-Cell; Maleimides; Mice; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-delta; RNA, Messenger; Tetradecanoylphorbol Acetate; Transcription, Genetic; Tumor Cells, Cultured; Up-Regulation | 1998 |
Osmotic swelling-induced activation of the extracellular-signal-regulated protein kinases Erk-1 and Erk-2 in intestine 407 cells involves the Ras/Raf-signalling pathway.
Topics: ADP Ribose Transferases; Androstadienes; Botulinum Toxins; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Cell Size; Enzyme Activation; Epidermal Growth Factor; Flavonoids; Humans; Hypotonic Solutions; Indoles; Intestines; Iodine Radioisotopes; Maleimides; Osmotic Pressure; Phosphorylation; ras Proteins; Rubidium Radioisotopes; Signal Transduction; Tetradecanoylphorbol Acetate; Wortmannin | 1998 |
Transforming G protein-coupled receptors block insulin and ras-induced adipocytic differentiation in 3T3-L1 cells: evidence for a PKC and MAP kinase independent pathway.
Topics: 3T3 Cells; Adaptor Proteins, Signal Transducing; Adaptor Proteins, Vesicular Transport; Adipocytes; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Cell Differentiation; GRB2 Adaptor Protein; GTP-Binding Proteins; Histocytochemistry; Indoles; Insulin; Insulin Receptor Substrate Proteins; Maleimides; Mice; Phosphoproteins; Phosphorylation; Protein Kinase C; Proteins; ras Proteins; Receptors, Muscarinic; Shc Signaling Adaptor Proteins; Signal Transduction; Src Homology 2 Domain-Containing, Transforming Protein 1; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha | 1998 |
Protein kinase C-alpha activity inversely modulates invasion and growth of intestinal cells.
Topics: Animals; Cadherins; Carbazoles; Cell Adhesion; Cell Movement; Cell Size; Gene Expression Regulation, Neoplastic; Humans; Indoles; Maleimides; Mice; Mice, Nude; Mutagenesis, Site-Directed; Neoplasm Invasiveness; Neoplasms, Experimental; Protein Kinase C; Tetradecanoylphorbol Acetate; Transfection; Transplantation, Heterologous; Tumor Cells, Cultured; Urokinase-Type Plasminogen Activator | 1998 |
Desmosomes are regulated by protein kinase C in primary rat epithelial cells.
Topics: Animals; Cell Adhesion; Cells, Cultured; Cytoplasm; Desmosomes; Enzyme Inhibitors; Epithelial Cells; Indoles; Keratinocytes; Macromolecular Substances; Maleimides; Microscopy, Electron; Microscopy, Fluorescence; Morphogenesis; Phosphorylation; Protein Kinase C; Protein Processing, Post-Translational; Rats; Rats, Sprague-Dawley; Tetradecanoylphorbol Acetate; Tongue | 1998 |
Simultaneous cross-linking of CD6 and CD28 induces cell proliferation in resting T cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adult; Antibodies, Monoclonal; Antigens, CD; Carcinogens; CD28 Antigens; CD3 Complex; Cell Division; Cyclosporine; Dose-Response Relationship, Drug; Enzyme Inhibitors; Humans; Immunosuppressive Agents; Indoles; Interleukin-2; Lymphocyte Activation; Maleimides; Protein Kinase C; RNA, Messenger; T-Lymphocytes; Tetradecanoylphorbol Acetate | 1998 |
Induction of cell death by stimulation of protein kinase C in human epithelial cells expressing a mutant ras oncogene: a potential therapeutic target.
Topics: Apoptosis; Blotting, Western; Cell Death; Cell Line; Down-Regulation; Electrophoresis, Agar Gel; Epithelial Cells; Genes, ras; Humans; Indoles; Maleimides; Microscopy, Electron; Mutation; Protein Kinase C; ras Proteins; Tetradecanoylphorbol Acetate; Thyroid Gland | 1998 |
The role of protein kinase C signaling in activated DRA transcription.
Topics: B-Lymphocytes; Burkitt Lymphoma; Cell Membrane; Cytosol; Enzyme Activation; Enzyme Inhibitors; Gene Expression Regulation; HLA-DR alpha-Chains; HLA-DR Antigens; Humans; Indoles; Isoenzymes; Maleimides; Microscopy, Fluorescence; Promoter Regions, Genetic; Protein Kinase C; Second Messenger Systems; Tetradecanoylphorbol Acetate; Transcription Factor AP-1; Transfection | 1998 |
Interleukin-1alpha and tumor necrosis factor alpha synergistically stimulate prostaglandin E2-dependent production of interleukin-11 in rheumatoid synovial fibroblasts.
Topics: Arthritis, Rheumatoid; Carcinogens; Cells, Cultured; Dinoprostone; Drug Synergism; Enzyme Inhibitors; Fibroblasts; Gene Expression Regulation, Enzymologic; Humans; Indoles; Interleukin-1; Interleukin-11; Isoquinolines; Maleimides; Protein Kinase C; Signal Transduction; Sulfonamides; Synovial Membrane; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha | 1998 |
The role of protein kinase C alpha and epsilon isozymes in DNA synthesis induced by muscarinic receptors in a glial cell line.
Topics: Astrocytoma; Atropine; Carbachol; Carcinogens; DNA; Dose-Response Relationship, Drug; Down-Regulation; Drug Synergism; Enzyme Inhibitors; Humans; Indoles; Isoenzymes; Maleimides; Muscarinic Agonists; Muscarinic Antagonists; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-epsilon; Radioligand Assay; Receptors, Muscarinic; Staurosporine; Tetradecanoylphorbol Acetate; Time Factors; Tumor Cells, Cultured | 1998 |
Role of p38 MAP kinase in myocardial stress.
Topics: Adenosine; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Cell Survival; Cells, Cultured; Enzyme Inhibitors; Flavonoids; Imidazoles; Indoles; Ischemic Preconditioning, Myocardial; Maleimides; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinases; Myocardial Ischemia; Myocardium; p38 Mitogen-Activated Protein Kinases; Protein Kinase C; Pyridines; Rats; Tetradecanoylphorbol Acetate | 1998 |
Pervanadate activates NADPH oxidase via protein kinase C-independent phosphorylation of p47-phox.
Topics: Amino Acid Sequence; Animals; Binding Sites; Biological Transport; Enzyme Activation; Guinea Pigs; Indoles; Maleimides; Mice; Molecular Sequence Data; NADPH Dehydrogenase; NADPH Oxidases; Neutrophils; Phosphoproteins; Phosphorylation; Protein Kinase C; Protein Kinases; Protein Tyrosine Phosphatases; Superoxides; Tetradecanoylphorbol Acetate; Vanadates | 1999 |
Transcriptional activation of gonadotropin-releasing hormone (GnRH) receptor gene by GnRH: involvement of multiple signal transduction pathways.
Topics: Animals; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Genes, Reporter; Gonadotropin-Releasing Hormone; Indoles; Maleimides; Mice; Pituitary Gland; Promoter Regions, Genetic; Protein Kinase C; Proto-Oncogene Proteins c-raf; Rats; Receptors, LHRH; Signal Transduction; Tetradecanoylphorbol Acetate; Transcriptional Activation; Transfection | 1999 |
Intracellular signaling mechanisms of interleukin-1beta in synovial fibroblasts.
Topics: Animals; Calcimycin; Calcium Channel Blockers; Cell Line; Enzyme Inhibitors; Fibroblasts; Indoles; Interleukin-1; Intracellular Membranes; Ionophores; Maleimides; Nifedipine; Rabbits; Signal Transduction; Synovial Membrane; Tetradecanoylphorbol Acetate; Verapamil | 1999 |
Specific signaling pathways in the regulation of TNF-alpha mRNA synthesis and TNF-alpha secretion in RBL-2H3 mast cells stimulated through the high affinity IgE receptor.
Topics: Androstadienes; Animals; beta-N-Acetylhexosaminidases; Egtazic Acid; Enzyme Inhibitors; Gene Expression; Indoles; Leukemia, Basophilic, Acute; Maleimides; Mast Cells; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase C; Rats; Receptors, IgE; Reverse Transcriptase Polymerase Chain Reaction; Ribonucleases; RNA, Messenger; Signal Transduction; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha; Wortmannin | 1998 |
Bradykinin stimulates interleukin-8 production by human lung fibroblasts.
Topics: Blotting, Northern; Bradykinin; Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Inhibitors; Fibroblasts; Gene Expression; Humans; Indoles; Interleukin-1; Interleukin-8; Lung; Maleimides; Protein Kinase C; Receptors, Interleukin-1; Recombinant Proteins; Stimulation, Chemical; Tetradecanoylphorbol Acetate; Time Factors | 1998 |
Resistance to TNF-alpha cytotoxicity can be achieved through different signaling pathways in rat mesangial cells.
Topics: Animals; Apoptosis; Calcium-Calmodulin-Dependent Protein Kinases; Cell Cycle Proteins; Cells, Cultured; Cycloheximide; Drug Resistance; Dual Specificity Phosphatase 1; Enzyme Activation; Enzyme Inhibitors; Glomerular Mesangium; Immediate-Early Proteins; Indoles; JNK Mitogen-Activated Protein Kinases; Male; Maleimides; Mitogen-Activated Protein Kinases; Phosphoprotein Phosphatases; Protein Kinase C; Protein Phosphatase 1; Protein Tyrosine Phosphatases; Rats; Rats, Sprague-Dawley; Signal Transduction; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha | 1999 |
Sp1 is involved in a protein kinase C-independent activation of human T cell leukemia virus type I long terminal repeat by 12-O-tetradecanoylphorbol-13-acetate.
Topics: Anti-Inflammatory Agents; Base Sequence; Enzyme Inhibitors; Gene Products, tax; HIV Long Terminal Repeat; Human T-lymphotropic virus 1; Humans; Indoles; Jurkat Cells; Maleimides; Molecular Sequence Data; Protein Kinase C; Protein Processing, Post-Translational; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-ets; Restriction Mapping; Sp1 Transcription Factor; Terminal Repeat Sequences; Tetradecanoylphorbol Acetate; Transcription Factors; Transcriptional Activation | 1999 |
Involvement of p21 in the PKC-induced regulation of the G2/M cell cycle transition.
Topics: Aphidicolin; CDC2 Protein Kinase; Cyclin B; Cyclin-Dependent Kinase Inhibitor p21; Cyclins; DNA; Dose-Response Relationship, Drug; Enzyme Activation; Flow Cytometry; G2 Phase; Humans; Indoles; Maleimides; Mitosis; Phosphorylation; Precipitin Tests; Protein Kinase C; Signal Transduction; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Up-Regulation | 1999 |
Phosphatidylinositol 3-kinase and protein kinase C are required for the inhibition of caspase activity by epidermal growth factor.
Topics: Alkaloids; Androstadienes; Apoptosis; Benzophenanthridines; Blotting, Western; Caspase 3; Caspase Inhibitors; Caspases; Chromatin; Chromones; DNA Fragmentation; Enzyme Precursors; Epidermal Growth Factor; Flow Cytometry; Humans; Indoles; Maleimides; Molecular Weight; Morpholines; Phenanthridines; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Poly(ADP-ribose) Polymerases; Protein Kinase C; Staurosporine; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Wortmannin | 1999 |
Protein kinase C mediates experimental colitis in the rat.
Topics: Animals; Colitis; Colon; Enzyme Inhibitors; Ethanol; Indoles; Intestinal Mucosa; Isoenzymes; Male; Maleimides; Neutropenia; Peroxidase; Protein Kinase C; Rats; Rats, Sprague-Dawley; Staurosporine; Tetradecanoylphorbol Acetate; Trinitrobenzenesulfonic Acid | 1999 |
The essential role of phorbol ester-sensitive protein kinase C isoforms in activation-induced cell death of Th1 cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Apoptosis; Cells, Cultured; Enzyme Activation; Enzyme Inhibitors; Fas Ligand Protein; fas Receptor; Indoles; Isoenzymes; Maleimides; Membrane Glycoproteins; Mice; Mice, Transgenic; Mitogens; Protein Kinase C; Tetradecanoylphorbol Acetate; Th1 Cells; Th2 Cells | 1999 |
1,25-dihydroxyvitamin D3 and TPA activate phospholipase D in Caco-2 cells: role of PKC-alpha.
Topics: Caco-2 Cells; Calcitriol; Calcium; Carbazoles; Enzyme Activation; Enzyme Inhibitors; Humans; Indoles; Ionomycin; Isoenzymes; Kinetics; Maleimides; Phospholipase D; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-alpha; Protein Kinase C-delta; Tetradecanoylphorbol Acetate | 1999 |
Regulation of actin cytoskeleton in lymphocytes: PKC-delta disrupts IL-3-induced membrane ruffles downstream of Rac1.
Topics: Actins; Animals; B-Lymphocytes; Cell Line; Cell Membrane; Cell Size; Cytochalasin D; Cytoskeleton; GTP-Binding Proteins; Indoles; Interleukin-3; Isoenzymes; Maleimides; Mice; Phenotype; Protein Kinase C; Protein Kinase C-delta; rac GTP-Binding Proteins; Tetradecanoylphorbol Acetate; Tubulin | 1999 |
The role of protein kinases A and C pathways in the regulation of mitogen-activated protein kinase activation in response to gonadotropin-releasing hormone receptor activation.
Topics: Animals; Bucladesine; Buserelin; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Inhibitors; Epidermal Growth Factor; ErbB Receptors; Indoles; Kinetics; Maleimides; Protein Kinase C; Rats; Receptors, LHRH; Signal Transduction; Tetradecanoylphorbol Acetate; Transfection | 1999 |
VEGF activates protein kinase C-dependent, but Ras-independent Raf-MEK-MAP kinase pathway for DNA synthesis in primary endothelial cells.
Topics: 3T3 Cells; Adenoviridae; Androstadienes; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Carbazoles; Chromones; DNA Replication; Endothelial Growth Factors; Endothelium, Vascular; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Genes, ras; Genetic Vectors; Indoles; Lymphokines; Maleimides; MAP Kinase Kinase Kinase 1; Mice; Morpholines; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Isoforms; Protein Kinase C; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins c-raf; Proto-Oncogene Proteins p21(ras); Rats; Receptor Protein-Tyrosine Kinases; Receptors, Growth Factor; Receptors, Vascular Endothelial Growth Factor; Signal Transduction; Tetradecanoylphorbol Acetate; Transfection; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors; Wortmannin | 1999 |
Hyperglycemia in vitro attenuates insulin-stimulated chemokinesis in normal human neutrophils. Role of protein kinase C activation.
Topics: Adult; Cell Movement; Cell Size; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Humans; Hyperglycemia; Indoles; Insulin; Maleimides; Neutrophils; Protein Kinase C; Tetradecanoylphorbol Acetate | 1999 |
Activated Ki-Ras suppresses 12-O-tetradecanoylphorbol-13-acetate-induced activation of the c-Jun NH2-terminal kinase pathway in human colon cancer cells.
Topics: Alleles; Amino Acid Substitution; Calcium-Calmodulin-Dependent Protein Kinases; Chromones; Colonic Neoplasms; Culture Media, Serum-Free; Depression, Chemical; Enzyme Activation; Enzyme Inhibitors; Gene Expression Regulation, Neoplastic; Genes, Immediate-Early; Genes, ras; Humans; Indoles; Isoenzymes; JNK Mitogen-Activated Protein Kinases; Maleimides; MAP Kinase Kinase 1; MAP Kinase Kinase 2; MAP Kinase Kinase 4; MAP Kinase Kinase Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Morpholines; Mutation, Missense; Neoplasm Proteins; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Protein Isoforms; Protein Kinase C; Protein Kinases; Protein Processing, Post-Translational; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Proto-Oncogene Proteins p21(ras); Signal Transduction; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1999 |
Phosphoinositide 3-kinase-dependent and -independent activation of the small GTPase Rac2 in human neutrophils.
Topics: Androstadienes; Chromones; Enzyme Activation; GTP-Binding Proteins; Guanosine Triphosphate; Humans; Indoles; Leukotriene B4; Maleimides; Morpholines; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Pertussis Toxin; Phosphatidylinositol 3-Kinases; Protein Binding; Protein Serine-Threonine Kinases; rac GTP-Binding Proteins; Signal Transduction; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella; Wortmannin | 1999 |
Involvement of group VI Ca2+-independent phospholipase A2 in protein kinase C-dependent arachidonic acid liberation in zymosan-stimulated macrophage-like P388D1 cells.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Calcium; Diglycerides; Egtazic Acid; Group VI Phospholipases A2; Indoles; Leukemia P388; Maleimides; Mice; Naphthalenes; Oligonucleotides, Antisense; Organophosphonates; Phospholipases A; Phospholipases A2; Protein Kinase C; Pyrones; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Zymosan | 1999 |
Role of diacylglycerol (DAG) in hormonal induction of S phase in hepatocytes: the DAG-dependent protein kinase C pathway is not activated by epidermal growth factor (EGF), but is involved in mediating the enhancement of responsiveness to EGF by vasopressi
Topics: Angiotensin II; Animals; Bacterial Proteins; Calcium-Calmodulin-Dependent Protein Kinases; Carcinogens; Cells, Cultured; Diglycerides; DNA; Enzyme Activation; Enzyme Inhibitors; Epidermal Growth Factor; G1 Phase; GTP-Binding Proteins; Indoles; Liver; Male; Maleimides; Neuropeptides; Norepinephrine; Phospholipase D; Protein Kinase C; Rats; Rats, Wistar; S Phase; Tetradecanoylphorbol Acetate; Vasopressins | 1999 |
PAR1 activation initiates integrin engagement and outside-in signalling in megakaryoblastic CHRF-288 cells.
Topics: Blood Platelets; Calcium; Cell Adhesion; Cell Cycle Proteins; Cell Line; Fibrinogen; Humans; Indoles; Maleimides; Peptide Fragments; Phosphatidylinositol 3-Kinases; Phosphorylation; Platelet Glycoprotein GPIIb-IIIa Complex; Protein Binding; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-vav; Receptor, PAR-1; Receptors, Thrombin; Signal Transduction; Tetradecanoylphorbol Acetate; Thrombin | 1999 |
Sphingosine and phorbol ester modulate protein kinase C activity and modify ATP-evoked calcium mobilization in glioma C6 cells.
Topics: Adenosine Triphosphate; Animals; Calcium; Calcium Signaling; Endoplasmic Reticulum; Enzyme Activation; Glioma; Indoles; Maleimides; Protein Kinase C; Rats; Sphingosine; Tetradecanoylphorbol Acetate; Thapsigargin; Time Factors; Tumor Cells, Cultured; Type C Phospholipases | 1999 |
Evidence on the participation of protein kinase C alpha in the proliferation of cultured myoblasts.
Topics: Animals; Cell Differentiation; Cell Division; Chick Embryo; DNA Replication; Indoles; Isoenzymes; Maleimides; Muscle, Skeletal; Naphthalenes; Protein Kinase C; Protein Kinase C-alpha; Tetradecanoylphorbol Acetate | 1999 |
Opposite effects of Ras or PKC activation on the expression of the SPRR2A keratinocyte terminal differentiation marker.
Topics: Calcium; Cell Differentiation; Cells, Cultured; Cornified Envelope Proline-Rich Proteins; Enzyme Activation; Epidermal Growth Factor; Gene Expression Regulation; Genes, fos; Humans; Indoles; Keratinocytes; Maleimides; Membrane Proteins; Mutation; Oncogene Protein p21(ras); Promoter Regions, Genetic; Protein Kinase C; Protein Precursors; Proto-Oncogene Proteins c-jun; RNA, Messenger; Signal Transduction; Tetradecanoylphorbol Acetate; Transcription, Genetic | 1999 |
Involvement of desmoplakin phosphorylation in the regulation of desmosomes by protein kinase C, in HeLa cells.
Topics: Animals; Cytoskeletal Proteins; Desmogleins; Desmoplakins; Desmosomes; Enzyme Inhibitors; gamma Catenin; HeLa Cells; Humans; Indoles; Maleimides; Mice; Phosphorylation; Protein Kinase C; Solubility; Tetradecanoylphorbol Acetate | 1999 |
Thioredoxin reductase is the major selenoprotein expressed in human umbilical-vein endothelial cells and is regulated by protein kinase C.
Topics: Blotting, Western; Calcimycin; Calcium; Cells, Cultured; Endothelium, Vascular; Gene Expression Regulation, Enzymologic; Humans; Indoles; Maleimides; Molecular Weight; Organ Specificity; Protein Kinase C; Proteins; Selenoproteins; Sodium Selenite; Tetradecanoylphorbol Acetate; Thioredoxin-Disulfide Reductase; Thyroid Gland; Time Factors; Tumor Cells, Cultured; Umbilical Veins | 1999 |
Role of protein kinase C in facilitation of luteinizing hormone (LH)-releasing hormone-induced LH surges by neuropeptide Y.
Topics: Animals; Enzyme Activation; Enzyme Inhibitors; Female; Follicle Stimulating Hormone; Gonadotropin-Releasing Hormone; In Vitro Techniques; Indoles; Kinetics; Luteinizing Hormone; Maleimides; Neuropeptide Y; Pituitary Gland, Anterior; Proestrus; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, LHRH; Tetradecanoylphorbol Acetate; Time Factors | 1999 |
A role of protein kinase C in the regulation of cytosolic phospholipase A(2) in bradykinin-induced PGI(2) synthesis by human vascular endothelial cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Base Sequence; Bradykinin; Calcium; Cells, Cultured; Cytosol; DNA Primers; Endothelium, Vascular; Enzyme Inhibitors; Epoprostenol; Humans; Indoles; Inositol 1,4,5-Trisphosphate; Kinetics; Maleimides; Mutagenesis, Site-Directed; Phospholipases A; Protein Kinase C; RNA, Messenger; Tetradecanoylphorbol Acetate | 1999 |
Distinct protein kinase C isozymes signal mitogenesis and apoptosis in human colon cancer cells.
Topics: Acetamides; Antineoplastic Agents; Apoptosis; Biological Transport; Colonic Neoplasms; Colorectal Neoplasms; Down-Regulation; Enzyme Inhibitors; Ethers, Cyclic; Humans; Indoles; Isoenzymes; Maleimides; Mitosis; Osmolar Concentration; Protein Kinase C; Pyrans; Signal Transduction; Spiro Compounds; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1999 |
Bradykinin induces interleukin-6 expression in astrocytes through activation of nuclear factor-kappaB.
Topics: Animals; Animals, Newborn; Astrocytes; Benzylamines; Bradykinin; Brain; Calcium-Calmodulin-Dependent Protein Kinases; Cells, Cultured; Enzyme Inhibitors; Gene Expression Regulation; Humans; Indoles; Interleukin-6; Kinetics; Luciferases; Maleimides; Mice; NF-kappa B; Promoter Regions, Genetic; Protein Kinase C; Recombinant Fusion Proteins; Sulfonamides; Tetradecanoylphorbol Acetate; Thapsigargin; Transcription, Genetic; Transfection | 1999 |
Cholecystokinin activates PYK2/CAKbeta by a phospholipase C-dependent mechanism and its association with the mitogen-activated protein kinase signaling pathway in pancreatic acinar cells.
Topics: Adaptor Proteins, Signal Transducing; Animals; Biological Transport; Calcimycin; Calcium; Cell Adhesion Molecules; Cholecystokinin; Colchicine; Cytochalasin D; Focal Adhesion Kinase 1; Focal Adhesion Kinase 2; Focal Adhesion Protein-Tyrosine Kinases; GRB2 Adaptor Protein; In Vitro Techniques; Indoles; Male; Maleimides; MAP Kinase Signaling System; Models, Biological; Pancreas; Phosphorylation; Protein-Tyrosine Kinases; Proteins; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-crk; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Sincalide; Tetradecanoylphorbol Acetate; Thapsigargin; Type C Phospholipases | 1999 |
Gq/11-coupled receptors and protein synthesis in rat cardiomyocytes: role of Gi-proteins and protein kinase C-isozymes.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-Agonists; Animals; Animals, Newborn; Bridged Bicyclo Compounds, Heterocyclic; Carbachol; Dose-Response Relationship, Drug; Endothelin-1; Enzyme Inhibitors; Fatty Acids, Unsaturated; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Proteins; Heart Ventricles; Hydrazines; Indoles; Inositol Phosphates; Isoenzymes; Maleimides; Norepinephrine; Pertussis Toxin; Phenylalanine; Protein Biosynthesis; Protein Kinase C; Proteins; Rats; Receptors, Cell Surface; Tetradecanoylphorbol Acetate; Tritium; Virulence Factors, Bordetella | 1999 |
Stimulation of A(2A) adenosine receptor phosphorylation by protein kinase C activation: evidence for regulation by multiple protein kinase C isoforms.
Topics: Acetophenones; Animals; Benzopyrans; Carbazoles; CHO Cells; Consensus Sequence; Cricetinae; Cyclic AMP; Dogs; Endothelin-1; Enzyme Activation; Enzyme Inhibitors; Glioma; Indoles; Isoenzymes; Maleimides; Mutagenesis, Site-Directed; Phosphorylation; Protein Kinase C; Rats; Receptor, Adenosine A2A; Receptors, Purinergic P1; Signal Transduction; Tetradecanoylphorbol Acetate; Triazines; Triazoles; Tumor Cells, Cultured | 1999 |
'Outside-in' signalling mechanisms underlying CD11b/CD18-mediated NADPH oxidase activation in human adherent blood eosinophils.
Topics: Androstadienes; Carbazoles; CD18 Antigens; Cell Adhesion; Cell Count; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Eosinophils; Humans; Imidazoles; Indoles; Isoenzymes; Macrophage-1 Antigen; Maleimides; Mitogen-Activated Protein Kinases; N-Formylmethionine Leucyl-Phenylalanine; NADPH Oxidases; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase C; Pyrazoles; Pyridines; Pyrimidines; Signal Transduction; src-Family Kinases; Superoxides; Tetradecanoylphorbol Acetate; Wortmannin | 1999 |
The involvement of protein kinase C in nitric oxide-induced damage to rat isolated colonic mucosal cells.
Topics: Animals; Azoles; Cell Survival; Colon; Cyclic N-Oxides; Dose-Response Relationship, Drug; Enzyme Activation; Imidazoles; Indoles; Intestinal Mucosa; Isoenzymes; Isoindoles; Male; Maleimides; Nitric Oxide; Nitric Oxide Donors; Organoselenium Compounds; Penicillamine; Protein Kinase C; Rats; Rats, Sprague-Dawley; Staurosporine; Tetradecanoylphorbol Acetate | 1999 |
Prevention of neuronal apoptosis by phorbol ester-induced activation of protein kinase C: blockade of p38 mitogen-activated protein kinase.
Topics: Amyloid beta-Peptides; Animals; Brain-Derived Neurotrophic Factor; Cell Hypoxia; Cells, Cultured; Cerebral Cortex; Coculture Techniques; Culture Media, Serum-Free; Cycloheximide; Enzyme Inhibitors; Flavonoids; Imidazoles; Indoles; JNK Mitogen-Activated Protein Kinases; Kinetics; Maleimides; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinases; Neurons; p38 Mitogen-Activated Protein Kinases; Peptide Fragments; Phorbol Esters; Protein Kinase C; Pyridines; Staurosporine; Tetradecanoylphorbol Acetate | 1999 |
Mechanisms involved in desensitization of particulate guanylyl cyclase in human airway smooth muscle: the role of protein kinase C.
Topics: 1-Methyl-3-isobutylxanthine; Atrial Natriuretic Factor; Cells, Cultured; Cyclic GMP; Dose-Response Relationship, Drug; Enzyme Activation; Guanylate Cyclase; Humans; Indoles; Maleimides; Muscle, Smooth; Phorbols; Phosphodiesterase Inhibitors; Protein Kinase C; Respiratory System; Solubility; Tetradecanoylphorbol Acetate; Time Factors | 1999 |
Activation of protein kinase C is required for the stable attachment of adherent platelets to collagen but is not needed for the initial rapid adhesion under flow conditions.
Topics: Animals; Antibodies; Blood Flow Velocity; Blood Platelets; Blood Proteins; Carbazoles; Carcinogens; Cell Adhesion Molecules; Collagen; Enzyme Inhibitors; Enzyme Precursors; Focal Adhesion Kinase 1; Focal Adhesion Protein-Tyrosine Kinases; Humans; Indoles; Integrins; Intracellular Signaling Peptides and Proteins; Maleimides; Phosphoproteins; Phosphorylation; Platelet Adhesiveness; Protein Conformation; Protein Kinase C; Protein-Tyrosine Kinases; Rats; Receptors, Collagen; Skin; Stimulation, Chemical; Syk Kinase; Tetradecanoylphorbol Acetate; Tyrosine | 1999 |
Rapid signalling by androgen receptor in prostate cancer cells.
Topics: Adenocarcinoma; Androgen Antagonists; Cell Nucleus; Cytoplasm; Dihydrotestosterone; DNA-Binding Proteins; Enzyme Activation; Enzyme Inhibitors; ets-Domain Protein Elk-1; Flavonoids; Gene Expression Regulation, Neoplastic; Humans; Indoles; Ligands; Male; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Neoplasm Proteins; Neoplasms, Hormone-Dependent; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Prostatic Neoplasms; Protein Kinase C; Protein Processing, Post-Translational; Proto-Oncogene Proteins; Receptors, Androgen; Recombinant Fusion Proteins; Testosterone; Tetradecanoylphorbol Acetate; Transcription Factors; Transfection; Tumor Cells, Cultured | 1999 |
PKC-epsilon regulates basolateral endocytosis in human T84 intestinal epithelia: role of F-actin and MARCKS.
Topics: Acetophenones; Acetylcholine; Actin Cytoskeleton; Actins; Amino Acid Sequence; Benzopyrans; Biological Transport; Carbachol; Carbazoles; Carcinogens; Cell Membrane; Cell Polarity; Cells, Cultured; Cholinergic Agonists; Cross-Linking Reagents; Cytochalasin D; Diglycerides; Endocytosis; Enzyme Inhibitors; Epithelial Cells; Humans; Indoles; Intestines; Intracellular Signaling Peptides and Proteins; Isoenzymes; Maleimides; Membrane Proteins; Molecular Sequence Data; Myristoylated Alanine-Rich C Kinase Substrate; Nucleic Acid Synthesis Inhibitors; Pinocytosis; Protein Kinase C; Protein Kinase C-epsilon; Proteins; Tetradecanoylphorbol Acetate | 1999 |
Effect of contraction on mitogen-activated protein kinase signal transduction in skeletal muscle. Involvement Of the mitogen- and stress-activated protein kinase 1.
Topics: 3-O-Methylglucose; Amino Acid Sequence; Animals; Biological Transport; Electric Stimulation; Enzyme Inhibitors; Flavonoids; Glycogen; Imidazoles; In Vitro Techniques; Indoles; Insulin; Male; Maleimides; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Muscle Contraction; Muscle, Skeletal; p38 Mitogen-Activated Protein Kinases; Phosphopeptides; Phosphorylation; Pyridines; Rats; Rats, Wistar; Signal Transduction; Tetradecanoylphorbol Acetate | 2000 |
Exposure to 60-Hz magnetic fields and proliferation of human astrocytoma cells in vitro.
Topics: Animals; Astrocytoma; Brain Neoplasms; Carbachol; Carcinogens; Cell Division; Cerebral Cortex; Cholinergic Agents; Cold Temperature; DNA Replication; DNA, Neoplasm; Drug Synergism; Electromagnetic Fields; Enzyme Inhibitors; Humans; Indoles; Maleimides; Protein Kinase C; Rats; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 2000 |
Interleukin-1beta regulates CFTR expression in human intestinal T84 cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenocarcinoma; Benzoquinones; Cell Line; Colon; Colonic Neoplasms; Cycloheximide; Cystic Fibrosis Transmembrane Conductance Regulator; Enzyme Inhibitors; Genistein; Humans; Indoles; Interleukin-1; Lactams, Macrocyclic; Maleimides; Neoplasm Proteins; Phosphorylation; Protein Kinase C; Protein Processing, Post-Translational; Protein Synthesis Inhibitors; Quinones; Rifabutin; RNA, Messenger; RNA, Neoplasm; Signal Transduction; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Up-Regulation | 2000 |
Inhibition of bradykinin-induced phosphoinositide hydrolysis and Ca2+ mobilisation by phorbol ester in rat cultured vascular smooth muscle cells.
Topics: Animals; Biological Transport; Bradykinin; Calcium Signaling; Cells, Cultured; Enzyme Activation; Enzyme Inhibitors; Indoles; Inositol 1,4,5-Trisphosphate; Isoenzymes; Kinetics; Maleimides; Muscle, Smooth, Vascular; Phosphatidylinositols; Protein Kinase C; Rats; Rats, Sprague-Dawley; Staurosporine; Tetradecanoylphorbol Acetate | 1999 |
CCK stimulates mob-1 expression and NF-kappaB activation via protein kinase C and intracellular Ca(2+).
Topics: Animals; Biological Transport; Calcium; Carcinogens; Cell Nucleus; Chelating Agents; Chemokine CXCL10; Chemokines, CXC; Cholecystokinin; Cytokines; DNA-Binding Proteins; Egtazic Acid; Enzyme Inhibitors; Gene Expression; In Vitro Techniques; Indoles; Ionomycin; Ionophores; Male; Maleimides; NF-kappa B; Pancreas; Phosphorylation; Protein Kinase C; Rats; Rats, Wistar; RNA, Messenger; Tetradecanoylphorbol Acetate | 2000 |
A protein kinase C-independent pathway leading to c-Jun-dependent expression of 100-kDa Ras GTPase-activating protein in JEG-3 human choriocarcinoma cells.
Topics: Cell Differentiation; Choriocarcinoma; Enzyme Activation; Enzyme Inhibitors; Female; Gene Expression Regulation, Neoplastic; Genes, fos; Genes, jun; Humans; Indoles; JNK Mitogen-Activated Protein Kinases; Maleimides; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinases; Molecular Weight; Neoplasm Proteins; Okadaic Acid; Oligonucleotides, Antisense; Protein Isoforms; Protein Kinase C; Proto-Oncogene Proteins c-fos; Proto-Oncogene Proteins c-jun; ras GTPase-Activating Proteins; RNA, Messenger; RNA, Neoplasm; Signal Transduction; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Uterine Neoplasms | 2000 |
Induction of cell cornification and enhanced squamous-cell marker SPRR1 gene expression by phorbol ester are regulated by different signaling pathways in human conducting airway epithelial cells.
Topics: Biomarkers; Cell Size; Cornified Envelope Proline-Rich Proteins; Enzyme Activation; Enzyme Inhibitors; Epithelial Cells; Flavonoids; Gene Expression Regulation; Humans; Indoles; Lactams; Maleimides; Membrane Proteins; Microscopy, Phase-Contrast; Mitogen-Activated Protein Kinases; Protein Kinase C; Proteins; RNA, Messenger; Signal Transduction; Tetradecanoylphorbol Acetate; Time Factors; Trachea; Transcriptional Activation | 2000 |
The m3 muscarinic acetylcholine receptor is coupled to mitogen-activated protein kinase via protein kinase C and epidermal growth factor receptor kinase.
Topics: Carbachol; Cell Line; Enzyme Activation; Enzyme Inhibitors; Epidermal Growth Factor; ErbB Receptors; Humans; Indoles; Maleimides; Mitogen-Activated Protein Kinases; Protein Kinase C; Receptor, Muscarinic M3; Receptors, Muscarinic; Recombinant Proteins; Tetradecanoylphorbol Acetate; Transfection | 2000 |
Differential effects of protein kinase C on the levels of epithelial Na+ channel subunit proteins.
Topics: Aldosterone; Animals; Biological Transport; Blotting, Western; Cell Line; Dose-Response Relationship, Drug; Electrophysiology; Enzyme Activation; Enzyme Inhibitors; Epithelial Sodium Channels; Indoles; Kinetics; Maleimides; Naphthalenes; Protein Kinase C; Protein Structure, Tertiary; RNA, Messenger; Sodium; Sodium Channels; Tetradecanoylphorbol Acetate; Time Factors; Xenopus | 2000 |
Dexamethasone inhibits the induction of NAD(+)-dependent 15-hydroxyprostaglandin dehydrogenase by phorbol ester in human promonocytic U937 cells.
Topics: Anti-Inflammatory Agents; Dexamethasone; Dose-Response Relationship, Drug; Enzyme Induction; Humans; Hydroxyprostaglandin Dehydrogenases; Indoles; Maleimides; Mifepristone; Phorbol Esters; Staurosporine; Tetradecanoylphorbol Acetate; Time Factors; U937 Cells | 2000 |
Inhibition and stimulation of growth of Entamoeba histolytica in culture: association with PKC activity and protein phosphorylation.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Culture Media; Down-Regulation; Entamoeba histolytica; Enzyme Inhibitors; Indoles; Maleimides; Marine Toxins; Okadaic Acid; Oxazoles; Phosphorylation; Protein Kinase C; Tetradecanoylphorbol Acetate; Threonine | 2000 |
4-Hydroxynonenal-induced MEL cell differentiation involves PKC activity translocation.
Topics: Aldehydes; Animals; Biological Transport, Active; Cell Differentiation; Cell Division; Dimethyl Sulfoxide; Enzyme Inhibitors; Hemoglobins; Indoles; Leukemia, Erythroblastic, Acute; Maleimides; Mice; Protein Kinase C; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 2000 |
Protein kinase C activity modulates dendritic differentiation of rat Purkinje cells in cerebellar slice cultures.
Topics: Animals; Carcinogens; Cell Differentiation; Cell Size; Dendrites; Enzyme Inhibitors; Indoles; Isoenzymes; Maleimides; Organ Culture Techniques; Protein Kinase C; Purkinje Cells; Rats; Rats, Sprague-Dawley; Tetradecanoylphorbol Acetate; Tetrodotoxin | 2000 |
Modulation of neutrophil migration and superoxide anion release by metoprolol.
Topics: Adrenergic beta-Antagonists; Cells, Cultured; Chemotaxis, Leukocyte; Enzyme Inhibitors; Humans; Indoles; Isoenzymes; Maleimides; Metoprolol; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-alpha; Respiratory Burst; Staurosporine; Superoxides; Tetradecanoylphorbol Acetate; Time Factors | 2000 |
Different regulation of phospholipase D activity in glioma C6 cells by sphingosine, propranolol, imipramine and phorbol ester.
Topics: Animals; Brain Neoplasms; Cell Compartmentation; Drug Interactions; Enzyme Activation; Enzyme Inhibitors; Glioma; Imipramine; Indoles; Isoenzymes; Maleimides; Neoplasm Proteins; Phospholipase D; Propranolol; Protein Kinase C; Rats; Sphingosine; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 2000 |
The effect of rapamycin on single ENaC channel activity and phosphorylation in A6 cells.
Topics: Drug Interactions; Enzyme Inhibitors; Epithelial Sodium Channels; Immunophilins; Immunosuppressive Agents; Indoles; Maleimides; Patch-Clamp Techniques; Phosphorylation; Protein Kinase C; Sirolimus; Sodium Channels; Tacrolimus; Tacrolimus Binding Proteins; Tetradecanoylphorbol Acetate | 2000 |
Changes in activity and regulation of the cardiac Ca2+ channel (L-type) by protein kinase C in chronic alcohol-exposed rats.
Topics: Alcoholism; Animals; Calcium Channels, L-Type; Electric Stimulation; Enzyme Inhibitors; Ethanol; Indoles; Isoenzymes; Maleimides; Manganese; Myocardium; Protein Kinase C; Rats; Rats, Sprague-Dawley; Tetradecanoylphorbol Acetate | 2000 |
Protein kinase C theta and epsilon promote T-cell survival by a rsk-dependent phosphorylation and inactivation of BAD.
Topics: bcl-Associated Death Protein; Carrier Proteins; Cell Line; Cell Survival; Humans; Indoles; Isoenzymes; Maleimides; Phosphorylation; Protein Kinase C; Protein Kinase C-theta; Protein Kinases; Ribosomal Protein S6 Kinases; T-Lymphocytes; Tetradecanoylphorbol Acetate | 2000 |
Phorbor myristate acetate induces NADPH oxidase activity of cytochalasin B-primed neutrophils through the protein kinase C-independent pathway.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adult; Androstadienes; Cytochalasin B; Ethanol; Granulocyte Colony-Stimulating Factor; Humans; Indoles; Maleimides; NADPH Oxidases; Neutrophils; Phosphatidylinositol 3-Kinases; Phospholipase D; Protein Kinase C; Superoxides; Tetradecanoylphorbol Acetate; Wortmannin | 2000 |
Role of protein kinase C in alpha(1)-adrenergic regulation of a(Na)(i) in guinea pig ventricular myocytes.
Topics: Adrenergic alpha-Agonists; Animals; Enzyme Inhibitors; Extracellular Space; Guinea Pigs; Heart Ventricles; Indoles; Intracellular Membranes; Maleimides; Myocardium; Phenylephrine; Potassium; Protein Kinase C; Receptors, Adrenergic, alpha; Sodium; Staurosporine; Strophanthidin; Tetradecanoylphorbol Acetate; Tetrodotoxin | 2000 |
Permissive role of protein kinase C alpha but not protein kinase C delta in sphingosine 1-phosphate-induced Rho A activation in C2C12 myoblasts.
Topics: Acetophenones; Animals; Benzopyrans; Carbazoles; Cell Fractionation; Cell Line; Cell Membrane; Endoplasmic Reticulum; Endosomes; Enzyme Inhibitors; Golgi Apparatus; Indoles; Isoenzymes; Lysophospholipids; Maleimides; Mice; Muscle, Skeletal; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-delta; Protein Transport; rhoA GTP-Binding Protein; Sphingosine; Tetradecanoylphorbol Acetate | 2000 |
Differential localization of protein kinase C isotypes in equine eosinophils and neutrophils.
Topics: Animals; Brain; Cell Membrane; Cell Nucleus; Cytoplasmic Granules; Enzyme Activation; Enzyme Inhibitors; Eosinophils; Horses; Indoles; Intracellular Membranes; Isoenzymes; Maleimides; Neutrophils; Organ Specificity; Protein Kinase C; Rats; Respiratory Burst; Staurosporine; Subcellular Fractions; Superoxides; Tetradecanoylphorbol Acetate | 2000 |
AP-1 proteins mediate hyperglycemia-induced activation of the human TGF-beta1 promoter in mesangial cells.
Topics: Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Gene Expression Regulation; Glomerular Mesangium; Glucose; Humans; Hyperglycemia; Imidazoles; Indoles; Maleimides; Mitogen-Activated Protein Kinases; Nuclear Proteins; p38 Mitogen-Activated Protein Kinases; Podophyllin; Podophyllotoxin; Promoter Regions, Genetic; Pyridines; RNA, Messenger; Sp1 Transcription Factor; Tetradecanoylphorbol Acetate; Tissue Distribution; Transcription Factor AP-1; Transforming Growth Factor beta; Transforming Growth Factor beta1 | 2000 |
High glucose level and free fatty acid stimulate reactive oxygen species production through protein kinase C--dependent activation of NAD(P)H oxidase in cultured vascular cells.
Topics: Animals; Aorta; Blood Vessels; Cattle; Cells, Cultured; Electron Spin Resonance Spectroscopy; Endothelium, Vascular; Enzyme Activation; Enzyme Inhibitors; Fatty Acids, Nonesterified; Glucose; Indoles; Maleimides; Muscle, Smooth, Vascular; NADPH Oxidases; Onium Compounds; Palmitic Acid; Protein Kinase C; Reactive Oxygen Species; Tetradecanoylphorbol Acetate | 2000 |
Agonist-induced long-term desensitization of the human prostacyclin receptor.
Topics: beta-Adrenergic Receptor Kinases; Cell Line; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Fibroblasts; G-Protein-Coupled Receptor Kinase 5; Humans; Iloprost; Indoles; Kinetics; Maleimides; Phosphorylation; Polymerase Chain Reaction; Protein Kinase C; Protein Serine-Threonine Kinases; Receptors, Epoprostenol; Receptors, Prostaglandin; Recombinant Fusion Proteins; Tetradecanoylphorbol Acetate; Transfection | 2000 |
Stimulation of extracellular signal-regulated kinases and proliferation in rat osteoblastic cells by parathyroid hormone is protein kinase C-dependent.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Blotting, Western; Cell Division; Cell Line; Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Epidermal Growth Factor; Flavonoids; Indoles; Maleimides; Mitogen-Activated Protein Kinases; Osteoblasts; Parathyroid Hormone; Peptides; Phosphorylation; Plasmids; Protein Kinase C; Proto-Oncogene Proteins p21(ras); Rats; Signal Transduction; Tetradecanoylphorbol Acetate; Time Factors; Transfection | 2001 |
Serotonin transporter phosphorylation modulated by tetanus toxin.
Topics: Animals; Biological Transport; Brain; Carrier Proteins; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Indoles; Isoenzymes; Isotope Labeling; Maleimides; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Phospholipase C gamma; Phosphorylation; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-alpha; Rats; Rats, Sprague-Dawley; Serine; Serotonin; Serotonin Plasma Membrane Transport Proteins; Synaptosomes; Tetanus Toxin; Tetradecanoylphorbol Acetate; Tritium; Type C Phospholipases; Tyrosine | 2000 |
Protein kinase C activation modulates pro- and anti-apoptotic signaling pathways.
Topics: Antineoplastic Agents; Apoptosis; Apoptotic Protease-Activating Factor 1; Blotting, Western; Bryostatins; Calcitriol; Caspases; Cell Cycle; Cell Differentiation; Enzyme Activation; Enzyme Inhibitors; Fas Ligand Protein; fas Receptor; Flow Cytometry; Humans; Indoles; Isoenzymes; Lactones; Macrolides; Maleimides; Membrane Glycoproteins; Protein Kinase C; Proteins; Proto-Oncogene Proteins c-bcl-2; Receptors, Tumor Necrosis Factor; Signal Transduction; Tetradecanoylphorbol Acetate; Tretinoin; Tumor Necrosis Factor-alpha; U937 Cells | 2000 |
Protein kinase C-alpha is an upstream activator of the IkappaB kinase complex in the TPA signal transduction pathway to NF-kappaB in U2OS cells.
Topics: Butadienes; DNA-Binding Proteins; Enzyme Activation; Genes, Dominant; Humans; I-kappa B Kinase; I-kappa B Proteins; Indoles; Isoenzymes; Kinetics; Maleimides; MAP Kinase Kinase 1; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Multienzyme Complexes; Mutation; NF-kappa B; NF-KappaB Inhibitor alpha; Nitriles; Protein Kinase C; Protein Kinase C-alpha; Protein Processing, Post-Translational; Protein Serine-Threonine Kinases; Ribosomal Protein S6 Kinases; Signal Transduction; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha | 2000 |
p53-independent elevation of p21 expression by PMA results from PKC-mediated mRNA stabilization.
Topics: Cyclin-Dependent Kinase Inhibitor p21; Cyclins; Dactinomycin; Enzyme Activation; Enzyme Inhibitors; Gene Expression Regulation; Genes, Reporter; Humans; Indoles; Kinetics; Luciferases; Maleimides; Okadaic Acid; Promoter Regions, Genetic; Protein Kinase C; RNA, Messenger; Signal Transduction; Tetradecanoylphorbol Acetate; Transfection; Tumor Suppressor Protein p53; U937 Cells | 2001 |
Modulation of cyclin D1 and its signaling components by the phorbol ester TPA and the tyrosine phosphatase inhibitor vanadate.
Topics: Animals; Cell Division; Cell Line; Cell Membrane; Cyclin D1; Cytosol; Enzyme Activation; Enzyme Inhibitors; Epidermal Growth Factor; Fibroblasts; Flavonoids; Indoles; Isoenzymes; Kinetics; Maleimides; MAP Kinase Signaling System; Mice; Mitogen-Activated Protein Kinases; Platelet-Derived Growth Factor; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-epsilon; Protein Tyrosine Phosphatases; Signal Transduction; Tetradecanoylphorbol Acetate; Vanadates | 2001 |
Characterization of the 5'-flanking region of the rat TIS11 gene.
Topics: Animals; Cell Line; DNA-Binding Proteins; Enzyme Inhibitors; Flavonoids; Gene Expression Regulation; Genes, Immediate-Early; Genes, Reporter; Immediate-Early Proteins; Indoles; Luciferases; Maleimides; Mitogen-Activated Protein Kinase Kinases; PC12 Cells; Promoter Regions, Genetic; Protein Kinase C; Rats; Sequence Deletion; Tetradecanoylphorbol Acetate; Tristetraprolin | 2000 |
The stimulation of MAP kinase by 1,25(OH)(2)-vitamin D(3) in skeletal muscle cells is mediated by protein kinase C and calcium.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcimycin; Calcitriol; Calcium; Calmodulin; Chick Embryo; Egtazic Acid; Enzyme Activation; Fluphenazine; Indoles; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Muscle, Skeletal; Naphthalenes; Neomycin; Phosphorylation; Protein Kinase C; Tetradecanoylphorbol Acetate; Thapsigargin; Type C Phospholipases; Verapamil | 2001 |
Oxidized-LDL enhances coronary vasoconstriction by increasing the activity of protein kinase C isoforms alpha and epsilon.
Topics: Animals; Blotting, Western; Calcium; Calcium Channel Blockers; Carbazoles; Coronary Vessels; Enzyme Activation; Enzyme Inhibitors; Fura-2; In Vitro Techniques; Indoles; Isoenzymes; Isometric Contraction; Lipoproteins, LDL; Male; Maleimides; Muscle, Smooth, Vascular; Potassium Chloride; Protein Kinase C; Serotonin; Subcellular Fractions; Swine; Tetradecanoylphorbol Acetate; Vasoconstriction; Verapamil | 2001 |
Glycated serum albumin-induced vascular smooth muscle cell proliferation through activation of the mitogen-activated protein kinase/extracellular signal-regulated kinase pathway by protein kinase C.
Topics: Animals; Cell Division; Cell Line; DNA; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Glycated Serum Albumin; Glycation End Products, Advanced; Humans; Indoles; Isoenzymes; Luciferases; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Muscle, Smooth, Vascular; Protein Kinase C; Rats; Recombinant Fusion Proteins; Serum Albumin; Tetradecanoylphorbol Acetate; Transcriptional Activation | 2001 |
Synergistic induction of apoptosis in human leukemia cells (U937) exposed to bryostatin 1 and the proteasome inhibitor lactacystin involves dysregulation of the PKC/MAPK cascade.
Topics: Acetylcysteine; Amanitins; Aminoacetonitrile; Apoptosis; Benzoquinones; Bryostatins; Butadienes; Curcumin; Cysteine Endopeptidases; Dactinomycin; Diterpenes; Drug Synergism; Enzyme Activation; Flavonoids; Humans; Imidazoles; Indoles; JNK Mitogen-Activated Protein Kinases; Lactams, Macrocyclic; Lactones; Macrolides; Maleimides; MAP Kinase Kinase 4; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Multienzyme Complexes; Neoplasm Proteins; Nitriles; Nucleic Acid Synthesis Inhibitors; p38 Mitogen-Activated Protein Kinases; Protease Inhibitors; Proteasome Endopeptidase Complex; Protein Kinase C; Protein Synthesis Inhibitors; Proto-Oncogene Proteins c-raf; Pyridines; Quinones; Terpenes; Tetradecanoylphorbol Acetate; Transcription Factor AP-1; Type C Phospholipases; U937 Cells; Ubiquitins | 2001 |
Modulation of rat erg1, erg2, erg3 and HERG K+ currents by thyrotropin-releasing hormone in anterior pituitary cells via the native signal cascade.
Topics: Animals; Arachidonic Acid; Cation Transport Proteins; Cells, Cultured; Cholecystokinin; Colforsin; DNA-Binding Proteins; Enzyme Inhibitors; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Flavonoids; Humans; Indoles; Isoquinolines; Kinetics; Maleimides; Membrane Potentials; Membrane Transport Proteins; Patch-Clamp Techniques; Pituitary Gland, Anterior; Potassium Channels; Potassium Channels, Voltage-Gated; Protein Kinase Inhibitors; Protein Kinases; Rats; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Thyrotropin-Releasing Hormone; Trans-Activators; Transcriptional Regulator ERG; Tyrphostins; Vasoactive Intestinal Peptide | 2001 |
Differential effects of growth hormone and insulin-like growth factor I on human endothelial cell migration.
Topics: Cell Line; Cell Movement; Endothelin-1; Endothelium, Vascular; Enzyme Inhibitors; Epidermal Growth Factor; Human Growth Hormone; Humans; Indoles; Insulin-Like Growth Factor I; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Protein Kinase C; Recombinant Proteins; Signal Transduction; Tetradecanoylphorbol Acetate | 2001 |
Altered expression of glutamate transporters under hypoxic conditions in vitro.
Topics: Amino Acid Transport System X-AG; Animals; Aspartic Acid; Carrier Proteins; Cell Death; Cell Hypoxia; Excitatory Amino Acid Transporter 2; Excitatory Amino Acid Transporter 3; Gene Expression Regulation; Glioma; Glutamate Plasma Membrane Transport Proteins; Glutamic Acid; Hypothalamic Neoplasms; Indoles; Maleimides; Mice; Mitochondria; Nerve Tissue Proteins; Neuroglia; Neurons; Protein Kinase C; Rats; Receptors, Neurotransmitter; Recombinant Fusion Proteins; RNA, Messenger; Symporters; Tetradecanoylphorbol Acetate; Transfection; Tumor Cells, Cultured | 2001 |
Key role of PKC and Ca2+ in EGF protection of microtubules and intestinal barrier against oxidants.
Topics: Calcimycin; Calcium; Calcium-Transporting ATPases; Cell Membrane; Cell Membrane Permeability; Cytosol; Enzyme Activation; Enzyme Inhibitors; Epidermal Growth Factor; Humans; Hydrogen Peroxide; Hypochlorous Acid; Indoles; Intestinal Mucosa; Isoenzymes; Maleimides; Microtubules; Models, Biological; Oxidants; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-alpha; Signal Transduction; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 2001 |
Upregulation of p21(WAF1/CIP1) leads to morphologic changes and esterase activity in TPA-mediated differentiation of human prostate cancer cell line TSU-Pr1.
Topics: Adenoviridae; Blotting, Northern; Blotting, Western; Carcinogens; Cell Differentiation; Cyclin-Dependent Kinase Inhibitor p21; Cyclins; DNA Primers; Enzyme Inhibitors; Flavonoids; Humans; Indoles; Male; Maleimides; Mitogen-Activated Protein Kinases; Naphthol AS D Esterase; Prostatic Neoplasms; Protein Kinase C; Recombinant Proteins; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Up-Regulation | 2001 |
Leukotriene D(4) affects localisation of vinculin in intestinal epithelial cells via distinct tyrosine kinase and protein kinase C controlled events.
Topics: Actins; alpha Catenin; Cadherins; Carcinogens; Cell Adhesion; Cell Line; Cytoskeletal Proteins; Enzyme Inhibitors; Focal Adhesions; Humans; Indoles; Integrin beta1; Intestinal Mucosa; Leukotriene D4; Maleimides; Phosphorylation; Protein Kinase C; Protein-Tyrosine Kinases; Pyrazoles; Pyrimidines; Tetradecanoylphorbol Acetate; Tyrosine; Vinculin | 2001 |
Extracellular ATP stimulates an inhibitory pathway towards growth factor-induced cRaf-1 and MEKK activation in astrocyte cultures.
Topics: Adenosine Triphosphate; Animals; Animals, Newborn; Astrocytes; Cells, Cultured; Cerebral Cortex; Enzyme Inhibitors; Fibroblast Growth Factor 2; Indoles; Kinetics; Maleimides; MAP Kinase Kinase 1; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Models, Biological; Norepinephrine; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins c-raf; Rats; Serotonin; Tetradecanoylphorbol Acetate | 2001 |
TSH-induced differentiated functions correlate with enhancement of phosphotyrosine phosphatase activity in thyroid cells. Effect of phorbol 12-myristate 13-acetate.
Topics: Adenylyl Cyclases; Animals; Cell Culture Techniques; Cell Differentiation; Cyclic AMP; Enzyme Inhibitors; Indoles; Iodine; Maleimides; Protein Kinase C; Protein Tyrosine Phosphatases; Swine; Tetradecanoylphorbol Acetate; Thyroid Gland; Thyrotropin | 2001 |
Saturated non-esterified fatty acids stimulate de novo diacylglycerol synthesis and protein kinase c activity in cultured aortic smooth muscle cells.
Topics: Animals; Aorta; Arachidonic Acid; Cattle; Cells, Cultured; Coenzyme A Ligases; Diglycerides; Enzyme Inhibitors; Fatty Acids, Nonesterified; Indoles; Kinetics; Maleimides; Mitogen-Activated Protein Kinases; Muscle, Smooth, Vascular; Oleic Acid; Palmitic Acid; Protein Kinase C; Stearic Acids; Tetradecanoylphorbol Acetate; Triazenes | 2001 |
Thrombin activates p38 mitogen-activated protein kinase in vascular smooth muscle cells.
Topics: Animals; Aorta, Thoracic; Cell Division; Cells, Cultured; DNA; Enzyme Activation; Enzyme Inhibitors; Heterotrimeric GTP-Binding Proteins; Imidazoles; Indoles; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Muscle, Smooth, Vascular; p38 Mitogen-Activated Protein Kinases; Protein Kinase C; Protein-Tyrosine Kinases; Pyridines; Rats; Tetradecanoylphorbol Acetate; Thrombin | 2001 |
Down-modulation of L-selectin by lipopolysaccharide is not required for lipopolysaccharide-induced expression of CD14 in mouse bone marrow granulocytes.
Topics: Animals; Bone Marrow Cells; Cells, Cultured; Down-Regulation; Enzyme Inhibitors; Granulocytes; Indoles; L-Selectin; Ligands; Lipopolysaccharide Receptors; Lipopolysaccharides; Maleimides; Mice; Mice, Inbred C3H; Mice, Inbred C57BL; Mice, Knockout; Protein Binding; Protein Kinase C; Tetradecanoylphorbol Acetate | 2001 |
Bradykinin induces protein kinase C-dependent activation of phospholipase D in A-431 cells.
Topics: Acetophenones; Benzopyrans; Bradykinin; Carbazoles; Enzyme Activation; Enzyme Inhibitors; Epidermal Growth Factor; Humans; Immunoblotting; Indoles; Isoenzymes; Kinetics; Maleimides; Phospholipase D; Phospholipids; Protein Kinase C; Staurosporine; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 2001 |
Insulin- and glucose-induced phosphorylation of the Na(+),K(+)-adenosine triphosphatase alpha-subunits in rat skeletal muscle.
Topics: Animals; Cell Membrane; Enzyme Inhibitors; Extracellular Space; Glucose; Indoles; Insulin; Male; Maleimides; Muscle, Skeletal; Phosphoamino Acids; Phosphorylation; Rats; Rats, Wistar; Sodium-Potassium-Exchanging ATPase; Tetradecanoylphorbol Acetate; Tissue Distribution; Tyrosine | 2001 |
Serotonin activation of the ERK pathway in Hermissenda: contribution of calcium-dependent protein kinase C.
Topics: Animals; Calcium; Carbazoles; Chelating Agents; Conditioning, Classical; Egtazic Acid; Enzyme Inhibitors; Indoles; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Mollusca; Phosphorylation; Serotonin; Tetradecanoylphorbol Acetate | 2001 |
Pharmacological evidence for system-dependent involvement of protein kinase C isoenzymes in phorbol ester-suppressed gap junctional communication.
Topics: Carbazoles; Cell Communication; Cells, Cultured; Connexin 43; Dose-Response Relationship, Drug; Gap Junctions; Indoles; Isoenzymes; Maleimides; Protein Kinase C; Protein Kinase C-delta; Protein Kinase C-epsilon; Tetradecanoylphorbol Acetate | 2001 |
Inorganic lead stimulates DNA synthesis in human astrocytoma cells: role of protein kinase Calpha.
Topics: Astrocytes; Astrocytoma; Carbachol; Carcinogens; Cell Cycle; Cell Division; Cholinergic Agonists; Culture Media, Serum-Free; DNA; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flow Cytometry; Humans; Immunoblotting; Indoles; Isoenzymes; Maleimides; Organometallic Compounds; Protein Kinase C; Protein Kinase C-alpha; Staurosporine; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 2001 |
Regulation of MDR1 promoter activity in human breast carcinoma cells by protein kinase C isozymes alpha and theta.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; Breast Neoplasms; Catalysis; Chloramphenicol O-Acetyltransferase; Drug Resistance, Neoplasm; Enzyme Inhibitors; Gene Deletion; Gene Expression Regulation, Enzymologic; Genes, Reporter; Humans; Indoles; Isoenzymes; Maleimides; Phenotype; Promoter Regions, Genetic; Protein Isoforms; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-theta; Tetradecanoylphorbol Acetate; Transcription, Genetic; Transfection; Tumor Cells, Cultured | 2001 |
Protein kinase epsilon dampens the secretory response of model intestinal epithelia during ischemia.
Topics: Biological Transport; Bryostatins; Carcinogens; Cell Hypoxia; Cell Line; Chlorides; Enzyme Activation; Enzyme Inhibitors; Humans; Indoles; Intestinal Mucosa; Ischemia; Isoenzymes; Lactones; Macrolides; Maleimides; Mitogens; Protein Kinase C; Protein Kinase C-epsilon; Tetradecanoylphorbol Acetate | 2001 |
Identification of protein kinase Calpha as an essential, but not sufficient, cytosolic factor for Ca2+-induced alpha- and dense-core granule secretion in platelets.
Topics: Adenosine Triphosphate; Animals; Blood Platelets; Blotting, Western; Brain; Calcium; Chromatography, Gel; Cytosol; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; HeLa Cells; Humans; Indoles; Isoenzymes; Jurkat Cells; Maleimides; Protein Binding; Protein Kinase C; Protein Kinase C-alpha; Rats; Tetradecanoylphorbol Acetate | 2001 |
Protein kinase C regulates the phosphorylation and cellular localization of occludin.
Topics: Alkaline Phosphatase; Animals; Binding Sites; Calcium; Carcinogens; Cell Line; Cells, Cultured; Cytoplasm; Detergents; Diglycerides; Dogs; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Indoles; Maleimides; Membrane Proteins; Mice; Microscopy, Fluorescence; Occludin; Octoxynol; Phosphorylation; Precipitin Tests; Protein Kinase C; Protein Structure, Tertiary; Recombinant Proteins; Serine; Spectrometry, Mass, Electrospray Ionization; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization; Tetradecanoylphorbol Acetate; Tight Junctions; Time Factors | 2001 |
Mechanisms in fluoride-induced interleukin-8 synthesis in human lung epithelial cells.
Topics: Androstadienes; Benzylamines; Cell Line; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Egtazic Acid; Epithelial Cells; Flavonoids; Genistein; Humans; Indoles; Interleukin-8; Isoquinolines; Lung; Maleimides; Okadaic Acid; Pertussis Toxin; Protein Kinase C; Signal Transduction; Sodium Fluoride; Sulfonamides; Tetradecanoylphorbol Acetate; Vanadates; Virulence Factors, Bordetella; Wortmannin | 2001 |
Docosahexaenoic acid modulates phorbol ester-induced activation of extracellular signal-regulated kinases 1 and 2 in NIH/3T3 cells.
Topics: 3T3 Cells; Animals; Cell Division; Docosahexaenoic Acids; Enzyme Activation; Enzyme Inhibitors; Indoles; Maleimides; MAP Kinase Kinase Kinase 1; MAP Kinase Signaling System; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase C; Protein Serine-Threonine Kinases; Tetradecanoylphorbol Acetate; Transforming Growth Factor alpha | 2001 |
Coupling strength between localized Ca(2+) transients and K(+) channels is regulated by protein kinase C.
Topics: Animals; Calcium Channel Blockers; Calcium Channels; Colon; Enzyme Inhibitors; Imidazoles; In Vitro Techniques; Indoles; Inositol 1,4,5-Trisphosphate; Maleimides; Mice; Mice, Inbred BALB C; Microscopy, Confocal; Muscle, Smooth; Potassium Channels; Protein Kinase C; Second Messenger Systems; Tetradecanoylphorbol Acetate | 2001 |
Protein kinase C modulates telomerase activity in human cervical cancer cells.
Topics: Alternative Splicing; Carbazoles; Catalytic Domain; Enzyme Inhibitors; Female; HeLa Cells; Humans; Indoles; Maleimides; Protein Kinase C; RNA, Messenger; Telomerase; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Uterine Cervical Neoplasms | 2001 |
TNF-alpha enhances intracellular glucocorticoid availability.
Topics: 11-beta-Hydroxysteroid Dehydrogenase Type 2; Animals; Cells, Cultured; Colforsin; Corticosterone; Cyclic AMP-Dependent Protein Kinases; Down-Regulation; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Glucocorticoids; Glucose; Hydroxysteroid Dehydrogenases; Imidazoles; Indoles; Maleimides; Mitogen-Activated Protein Kinases; Pyridines; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha | 2001 |
Enhancement of phospholipase D activity by overexpression of amyloid precursor protein in P19 mouse embryonic carcinoma cells.
Topics: Amyloid beta-Protein Precursor; Animals; Cell Differentiation; Enzyme Activation; Enzyme Inhibitors; Indoles; Maleimides; Mice; Neurons; Peptide Fragments; Phospholipase D; Protein Kinase C; Reference Values; Tetradecanoylphorbol Acetate; Transfection; Tretinoin; Tumor Cells, Cultured | 2001 |
Phosphorylation-dependent regulation of phospholipase D2 by protein kinase C delta in rat Pheochromocytoma PC12 cells.
Topics: Acetophenones; Adenoviridae; Animals; Benzopyrans; Bradykinin; Cell Membrane; Cytosol; Dose-Response Relationship, Drug; Enzyme Inhibitors; Immunoblotting; Immunohistochemistry; Indoles; Isoenzymes; Maleimides; Microscopy, Fluorescence; Mutation; PC12 Cells; Peptide Mapping; Phospholipase D; Phosphorylation; Precipitin Tests; Protein Binding; Protein Isoforms; Protein Kinase C; Protein Kinase C-delta; Protein Transport; Rats; Tetradecanoylphorbol Acetate; Time Factors; Up-Regulation | 2002 |
The P2X(7) receptor-mediated phospholipase D activation is regulated by both PKC-dependent and PKC-independent pathways in a rat brain-derived Type-2 astrocyte cell line, RBA-2.
Topics: Adenosine Triphosphate; Animals; Astrocytes; Brain; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Drug Synergism; Enzyme Activation; Enzyme Inhibitors; Indoles; Kinetics; Maleimides; Phospholipase D; Protein Kinase C; Protein-Tyrosine Kinases; Purinergic P2 Receptor Agonists; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2X7; RNA, Messenger; Signal Transduction; Tetradecanoylphorbol Acetate; Type C Phospholipases | 2002 |
Protein Kinase C is a mediator of the synthesis and secretion of osteoprotegerin in osteoblast-like cells.
Topics: Animals; Antibodies; Blotting, Northern; Blotting, Western; Cell Line; Cell Survival; Cells, Cultured; Dose-Response Relationship, Drug; Electrophoresis, Polyacrylamide Gel; Enzyme Inhibitors; Glycoproteins; Humans; Indoles; Maleimides; Osteoblasts; Osteoprotegerin; Promoter Regions, Genetic; Protein Kinase C; Rats; Receptors, Cytoplasmic and Nuclear; Receptors, Tumor Necrosis Factor; Recombinant Proteins; RNA, Messenger; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 2002 |
Activation of Erk1/Erk2 and transiently increased p53 levels together may account for p21 expression associated with phorbol ester-induced transient growth inhibition in HepG2 cells.
Topics: Cell Division; Cyclin-Dependent Kinase Inhibitor p21; Cyclins; Enzyme Activation; Enzyme Inhibitors; Humans; Indoles; Kinetics; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Protein Kinase C; Proto-Oncogene Proteins c-raf; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Tumor Suppressor Protein p53 | 2002 |
Protein kinase C-dependent, CCAAT/enhancer-binding protein beta-mediated expression of insulin-like growth factor I gene.
Topics: Base Sequence; Binding Sites; CCAAT-Enhancer-Binding Protein-alpha; CCAAT-Enhancer-Binding Protein-beta; Enzyme Inhibitors; Gene Expression Regulation; Humans; Indoles; Insulin-Like Growth Factor I; Maleimides; Promoter Regions, Genetic; Protein Kinase C; Protein Processing, Post-Translational; Recombinant Fusion Proteins; RNA, Messenger; Serine; Tetradecanoylphorbol Acetate; Transcription, Genetic; Tumor Cells, Cultured | 2002 |
Effect of wortmannin and phorbol ester on Paramecium fluid-phase uptake in the presence of transferrin.
Topics: Androstadienes; Animals; Biomarkers; Endocytosis; Endosomes; Enzyme Activation; Indoles; Isoquinolines; Maleimides; Paramecium; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase C; Tetradecanoylphorbol Acetate; Transferrin; Wortmannin | 2001 |
FGF-2 and TPA induce matrix metalloproteinase-9 secretion in MCF-7 cells through PKC activation of the Ras/ERK pathway.
Topics: Acetophenones; Benzopyrans; Carbazoles; Collagenases; Enzyme Inhibitors; Fibroblast Growth Factor 2; Genes, Dominant; Humans; Indoles; Maleimides; MAP Kinase Kinase 1; MAP Kinase Kinase 2; Matrix Metalloproteinase 9; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Models, Biological; Phosphorylation; Protein Kinase C; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-raf; ras Proteins; Signal Transduction; Tetradecanoylphorbol Acetate; Transfection; Tumor Cells, Cultured | 2002 |
Blocking NF-kappaB activation in Jurkat leukemic T cells converts the survival agent and tumor promoter PMA into an apoptotic effector.
Topics: Apoptosis; Carbazoles; Caspase 8; Caspase 9; Caspases; DNA-Binding Proteins; Enzyme Activation; Enzyme Inhibitors; Fas Ligand Protein; fas Receptor; Gene Expression Regulation, Leukemic; Humans; I-kappa B Proteins; Indoles; Isoenzymes; Jurkat Cells; Maleimides; Membrane Glycoproteins; Neoplasm Proteins; NF-kappa B; NF-KappaB Inhibitor alpha; Protein Kinase C; Recombinant Fusion Proteins; Sequence Deletion; Tetradecanoylphorbol Acetate | 2002 |
Phorbol myristate acetate induces ruffling of the acrosome of human sperm.
Topics: Acrosome; Acrosome Reaction; Actins; Cells, Cultured; Cytochalasin B; Cytochalasin D; Enzyme Inhibitors; Female; Humans; Indoles; Male; Maleimides; Microscopy, Electron; Microscopy, Electron, Scanning; Oocytes; Polymers; Protein Kinase C; Pyrimidine Nucleosides; Tetradecanoylphorbol Acetate; Zona Pellucida | 2002 |
Protein kinase C regulates endocytosis and recycling of E-cadherin.
Topics: Actins; Adherens Junctions; Animals; Cadherins; Cell Adhesion; Cell Line; Cell Membrane; Dogs; Endocytosis; Endosomes; Enzyme Inhibitors; Indoles; Maleimides; Polymers; Protein Kinase C; Tetradecanoylphorbol Acetate | 2002 |
Excitation of smooth muscles isolated from the guinea-pig gastric antrum in response to depolarization.
Topics: Acetylcholine; Alkaloids; Animals; Benzophenanthridines; Boron Compounds; Calcium; Calcium Signaling; Carbonyl Cyanide m-Chlorophenyl Hydrazone; Carcinogens; Electric Stimulation; Enzyme Inhibitors; Evoked Potentials; Guinea Pigs; Indoles; Ionophores; Lanthanum; Male; Maleimides; Muscle, Smooth; Phenanthridines; Protein Kinase C; Pyloric Antrum; Tetradecanoylphorbol Acetate; Thapsigargin | 2002 |
Phosphospecific site tyrosine phosphorylation of p125FAK and proline-rich kinase 2 is differentially regulated by cholecystokinin receptor type A activation in pancreatic acini.
Topics: Animals; Binding Sites; Calcium; Cholecystokinin; Diglycerides; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Focal Adhesion Kinase 1; Focal Adhesion Kinase 2; Focal Adhesion Protein-Tyrosine Kinases; Hydrolysis; Indoles; Inositol Phosphates; Kinetics; Male; Maleimides; Pancreas; Phosphatidylinositol 4,5-Diphosphate; Phosphorylation; Phosphotyrosine; Protein Kinase C; Protein-Tyrosine Kinases; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Sincalide; Tetradecanoylphorbol Acetate; Thapsigargin; Type C Phospholipases | 2003 |
BCR targets cyclin D2 via Btk and the p85alpha subunit of PI3-K to induce cell cycle progression in primary mouse B cells.
Topics: Adaptor Proteins, Signal Transducing; Agammaglobulinaemia Tyrosine Kinase; Amides; Animals; Antibodies, Anti-Idiotypic; Apoptosis; B-Lymphocytes; Calcium Signaling; Carrier Proteins; Cell Cycle; Chromones; Class Ib Phosphatidylinositol 3-Kinase; Crosses, Genetic; Cyclin D2; Cyclins; Enzyme Inhibitors; Female; Imidazoles; Immunologic Deficiency Syndromes; Indoles; Ionomycin; Isoenzymes; Macromolecular Substances; Male; Maleimides; Mice; Mice, Inbred C57BL; Mice, Inbred CBA; Mice, Knockout; Mice, Mutant Strains; Models, Immunological; Morpholines; Nitriles; Phenotype; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phospholipase C gamma; Phosphoproteins; Phosphorylation; Protein Interaction Mapping; Protein Processing, Post-Translational; Protein Subunits; Protein-Tyrosine Kinases; Receptors, Antigen, B-Cell; Signal Transduction; src-Family Kinases; Tetradecanoylphorbol Acetate; Type C Phospholipases | 2003 |
Effect of protein kinase C activation and inhibition on rat hepatic stellate cell activation.
Topics: Actins; Alkaloids; Animals; Benzophenanthridines; Cell Division; Cells, Cultured; Enzyme Activation; Enzyme Activators; Enzyme Inhibitors; In Vitro Techniques; Indoles; Liver; Male; Maleimides; Phenanthridines; Phorbol Esters; Protein Kinase C; Rats; Rats, Sprague-Dawley; Signal Transduction; Staurosporine; Tetradecanoylphorbol Acetate | 2003 |
Modification of intracellular free calcium in cultured A10 vascular smooth muscle cells by exogenous phosphatidic acid.
Topics: Animals; Boron Compounds; Calcium; Carbamates; Cells, Cultured; Diltiazem; Drug Interactions; Egtazic Acid; Indoles; Macrocyclic Compounds; Maleimides; Muscle, Smooth, Vascular; Oxazoles; Pertussis Toxin; Phenylcarbamates; Phosphatidic Acids; Rats; Tetradecanoylphorbol Acetate; Thapsigargin; Verapamil | 2003 |
Fatty acid and phorbol ester-mediated interference of mitogenic signaling via novel protein kinase C isoforms in pancreatic beta-cells (INS-1).
Topics: Acetophenones; Benzopyrans; Cell Line; Enzyme Activation; Enzyme Inhibitors; Fatty Acids, Nonesterified; Humans; Indoles; Insulin-Like Growth Factor I; Islets of Langerhans; Isoenzymes; Maleimides; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Mitogens; Phosphorylation; Protein Kinase C; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Tetradecanoylphorbol Acetate | 2003 |
Recovery of gap junctional intercellular communication after phorbol ester treatment requires proteasomal degradation of protein kinase C.
Topics: Animals; Blotting, Western; Cell Communication; Cells, Cultured; Connexin 43; Cysteine Endopeptidases; Cysteine Proteinase Inhibitors; Down-Regulation; Enzyme Inhibitors; Epithelial Cells; Gap Junctions; Indoles; Isoenzymes; Leupeptins; Liver; Maleimides; Multienzyme Complexes; Peptide Hydrolases; Proteasome Endopeptidase Complex; Protein Kinase C; Rats; Tetradecanoylphorbol Acetate | 2003 |
Protein kinase C modulates tumor necrosis factor-related apoptosis-inducing ligand-induced apoptosis by targeting the apical events of death receptor signaling.
Topics: Adaptor Proteins, Signal Transducing; Apoptosis; Apoptosis Regulatory Proteins; BH3 Interacting Domain Death Agonist Protein; Carrier Proteins; Caspase 3; Caspase 8; Caspase 9; Caspases; Cytochromes c; Enzyme Activation; Enzyme Inhibitors; Fas-Associated Death Domain Protein; HeLa Cells; Humans; I-kappa B Proteins; Indoles; Maleimides; Membrane Glycoproteins; Mitochondria; NF-kappa B; NF-KappaB Inhibitor alpha; Phosphatidylserines; Phosphorylation; Protein Kinase C; Receptors, TNF-Related Apoptosis-Inducing Ligand; Receptors, Tumor Necrosis Factor; Signal Transduction; Tetradecanoylphorbol Acetate; TNF-Related Apoptosis-Inducing Ligand; Tumor Necrosis Factor-alpha | 2003 |
Staurosporine induces rapid homotypic intercellular adhesion of U937 cells via multiple kinase activation.
Topics: Acetophenones; Adenosine Triphosphate; Benzopyrans; Calcium-Calmodulin-Dependent Protein Kinases; Carbazoles; CD18 Antigens; Cell Aggregation; Cycloheximide; Cytoskeleton; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Genistein; Humans; Imidazoles; Indoles; Integrin beta1; Isoenzymes; Maleimides; Mitogen-Activated Protein Kinases; Naphthalenes; Phosphorylation; Phosphotransferases; Protein Kinase C; Protein-Tyrosine Kinases; Pyridines; Staurosporine; Temperature; Tetradecanoylphorbol Acetate; Time Factors; Tyrosine; U937 Cells | 2003 |
15-Deoxy-Delta12,14-prostaglandin J2 regulates endogenous Cot MAPK kinase kinase 1 activity induced by lipopolysaccharide.
Topics: Animals; Antineoplastic Agents, Phytogenic; Blotting, Western; Carcinogens; Cell Division; Cell Line; Enzyme Activation; Enzyme Inhibitors; Fibrinolytic Agents; Gene Expression Regulation, Enzymologic; Indoles; Ligands; Lipopolysaccharides; Macrophages; Maleimides; MAP Kinase Kinase Kinases; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Paclitaxel; Phosphorylation; Precipitin Tests; Prostaglandin D2; Protein Isoforms; Protein-Tyrosine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-raf; RNA, Messenger; Rosiglitazone; Tetradecanoylphorbol Acetate; Thiazolidinediones; Time Factors | 2003 |
Activation of P2X7 purinoceptor-stimulated TGF-beta 1 mRNA expression involves PKC/MAPK signalling pathway in a rat brain-derived type-2 astrocyte cell line, RBA-2.
Topics: Adenosine; Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphate; Animals; Astrocytes; Blotting, Northern; Blotting, Western; Brain; Carbazoles; Cell Line; Dose-Response Relationship, Drug; Flavonoids; Gene Expression; Indoles; Kinetics; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase C; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2X4; Receptors, Purinergic P2X7; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetradecanoylphorbol Acetate; Transforming Growth Factor beta; Transforming Growth Factor beta1 | 2003 |
Diacylglycerols containing Omega 3 and Omega 6 fatty acids bind to RasGRP and modulate MAP kinase activation.
Topics: Animals; Binding, Competitive; Brain; Diglycerides; DNA-Binding Proteins; DNA, Complementary; Docosahexaenoic Acids; Dose-Response Relationship, Drug; Eicosapentaenoic Acid; Enzyme Activation; Enzyme Inhibitors; Escherichia coli; Fatty Acids; Fatty Acids, Omega-3; Fatty Acids, Omega-6; Guanine Nucleotide Exchange Factors; Humans; Immunoblotting; Indoles; Inhibitory Concentration 50; Jurkat Cells; Kinetics; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Plasmids; Protein Binding; Rats; Tetradecanoylphorbol Acetate; Time Factors; Transfection | 2004 |
Ca2+-dependent protein kinase C isoforms induce cholestasis in rat liver.
Topics: Animals; Bacterial Proteins; Bile; Biological Transport; Blotting, Western; Calcium; Carbazoles; Cell Line; Cell Membrane; Cells, Cultured; Cholestasis; Cloning, Molecular; Densitometry; Detergents; Dose-Response Relationship, Drug; Enzyme Activation; Hepatocytes; Humans; Indoles; Liver; Luminescent Proteins; Male; Maleimides; Microscopy, Confocal; Models, Biological; Perfusion; Phorbol Esters; Polymerase Chain Reaction; Protein Isoforms; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-epsilon; Protein Transport; Rats; Rats, Wistar; Signal Transduction; Taurocholic Acid; Tetradecanoylphorbol Acetate; Time Factors; Transfection | 2004 |
Cooperation between PKC-alpha and PKC-epsilon in the regulation of JNK activation in human lung cancer cells.
Topics: Animals; Carbazoles; Carcinoma, Non-Small-Cell Lung; Carcinoma, Small Cell; Cell Membrane; Cytoplasm; Humans; Indoles; Isoenzymes; JNK Mitogen-Activated Protein Kinases; Lung Neoplasms; Maleimides; Mice; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-epsilon; rac1 GTP-Binding Protein; Signal Transduction; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 2004 |
Regulation of phospholipase D2 activity by protein kinase C alpha.
Topics: Animals; COS Cells; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Gene Expression Regulation, Enzymologic; Genetic Vectors; Indoles; Maleimides; Phospholipase D; Phosphorylation; Precipitin Tests; Protein Binding; Protein Kinase C; Protein Kinase C-alpha; Serine; Subcellular Fractions; Tetradecanoylphorbol Acetate; Threonine; Time Factors; Transfection | 2004 |
Protein kinase C activation by Helicobacter pylori in human gastric epithelial cells limits interleukin-8 production through suppression of extracellular signal-regulated kinase.
Topics: Animals; Calcium-Calmodulin-Dependent Protein Kinases; Cell Adhesion Molecules; Cell Survival; Dose-Response Relationship, Drug; Down-Regulation; Epithelial Cells; Extracellular Signal-Regulated MAP Kinases; Gastric Mucosa; Helicobacter pylori; Humans; I-kappa B Kinase; Indoles; Interleukin-8; Maleimides; Methods; Naphthalenes; Protein Kinase C; Protein Serine-Threonine Kinases; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 2004 |
Induction of manganese-superoxide dismutase by YS 51, a synthetic 1-(beta-naphtylmethyl)6,7-dihydroxy- 1,2,3,4-tetrahydroisoquinoline alkaloid: implication for anti-inflammatory actions.
Topics: Animals; Blotting, Northern; Curcumin; Cycloheximide; Dactinomycin; Dose-Response Relationship, Drug; Drug Synergism; Drug Therapy, Combination; Endothelial Cells; Endothelium, Vascular; Enzyme Induction; Flavonoids; Gene Expression Regulation, Enzymologic; HeLa Cells; Humans; Imidazoles; Indoles; JNK Mitogen-Activated Protein Kinases; Maleimides; Mitogen-Activated Protein Kinase 3; p38 Mitogen-Activated Protein Kinases; Phorbol Esters; Phosphorylation; Pulmonary Artery; Pyridines; RNA, Messenger; Sheep; Superoxide Dismutase; Tetradecanoylphorbol Acetate; Tetrahydroisoquinolines; Tumor Necrosis Factor-alpha | 2004 |
Protein kinase C activity regulates the onset of anaphase I in mouse oocytes.
Topics: Anaphase; Animals; Dose-Response Relationship, Drug; Embryonic Development; Enzyme Activation; Enzyme Inhibitors; Female; Fertilization in Vitro; Indoles; Maleimides; Metaphase; Mice; Mice, Inbred Strains; Oocytes; Protein Kinase C; Tetradecanoylphorbol Acetate | 2004 |
Activation of protein kinase C antagonizes the opioid inhibition of calcium current in rat spinal dorsal horn neurons.
Topics: Analgesics, Opioid; Animals; Animals, Newborn; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Colforsin; Drug Interactions; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enzyme Activation; Enzyme Inhibitors; Female; Indoles; Isoquinolines; Male; Maleimides; Membrane Potentials; Narcotics; Patch-Clamp Techniques; Posterior Horn Cells; Potassium Channel Blockers; Protein Kinase C; Rats; Rats, Sprague-Dawley; Sulfonamides; Tetradecanoylphorbol Acetate; Tetraethylammonium; Tetrodotoxin | 2004 |
Activation of second messenger-dependent protein kinases induces muscarinic acetylcholine receptor desensitization in rat thyroid epithelial cells.
Topics: Animals; Arsenicals; Calcium; Calcium Channels; Carbachol; Colforsin; Cyclic AMP-Dependent Protein Kinases; Endocytosis; Epithelial Cells; Indoles; Maleimides; Muscarinic Agonists; Protein Kinase C; Rats; Rats, Inbred F344; Receptors, Muscarinic; Second Messenger Systems; Sucrose; Tetradecanoylphorbol Acetate; Thyroid Gland | 2004 |
Ghrelin exerts a proliferative effect on a rat pituitary somatotroph cell line via the mitogen-activated protein kinase pathway.
Topics: Androstadienes; Animals; Butadienes; Carcinogens; Cell Division; Cell Line, Tumor; Dose-Response Relationship, Drug; Enzyme Inhibitors; Ghrelin; Indoles; Maleimides; MAP Kinase Signaling System; Nitriles; Peptide Hormones; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Pituitary Gland; Pituitary Neoplasms; Rats; RNA, Messenger; Tetradecanoylphorbol Acetate; Tyrphostins; Wortmannin | 2004 |
IkappaBalpha (inhibitory kappaBalpha) identified as labile repressor of MnSOD (manganese superoxide dismutase) expression.
Topics: Cell Line; Cycloheximide; DNA; Down-Regulation; Enhancer Elements, Genetic; Gene Expression Regulation, Enzymologic; Humans; I-kappa B Proteins; Indoles; Introns; Isoenzymes; Maleimides; NF-kappa B; NF-KappaB Inhibitor alpha; Protein Binding; Protein Biosynthesis; Protein Kinase C; Protein Processing, Post-Translational; Protein Transport; Repressor Proteins; RNA, Messenger; Superoxide Dismutase; Tetradecanoylphorbol Acetate; Time Factors; Transcription Factor AP-1 | 2004 |
Role of protein kinase C delta in reactivation of Kaposi's sarcoma-associated herpesvirus.
Topics: Acetophenones; Benzopyrans; Cell Line; Enzyme Inhibitors; Herpesvirus 8, Human; Humans; Indoles; Maleimides; Protein Kinase C; Protein Kinase C-delta; Tetradecanoylphorbol Acetate; Virus Activation; Virus Latency | 2004 |
Alterations in receptor expression or agonist concentration change the pathways gastrin-releasing peptide receptor uses to regulate extracellular signal-regulated kinase.
Topics: 3T3 Cells; Animals; Bombesin; Cell Line; Enzyme Activation; Enzyme Inhibitors; Extracellular Signal-Regulated MAP Kinases; Gene Expression Regulation; Humans; Indoles; Maleimides; Mice; Microscopy, Confocal; Protein Transport; Receptors, Bombesin; Tetradecanoylphorbol Acetate | 2004 |
Exploring the pharmacology of the leukotriene B4 receptor BLT1, without the confounding effects of BLT2.
Topics: Boron Compounds; Calcium; Calcium Channel Blockers; Cytosol; Dantrolene; Dose-Response Relationship, Drug; Estrenes; Fatty Alcohols; Glycols; HeLa Cells; Humans; Imidazoles; Indoles; Intracellular Space; Maleimides; Nickel; Nifedipine; Plasmids; Propranolol; Protein Kinase Inhibitors; Pyrrolidinones; Receptors, Leukotriene B4; Staurosporine; Tetradecanoylphorbol Acetate; Thapsigargin; Transfection | 2004 |
Possible involvement of protein kinase C activation in differentiation of human umbilical vein endothelium-derived cell into smooth muscle-like cell.
Topics: Carbazoles; Carcinogens; Cell Differentiation; Cells, Cultured; Endothelium, Vascular; Enzyme Activation; Enzyme Inhibitors; Humans; Indoles; Maleimides; Myocytes, Smooth Muscle; Protein Kinase C; Signal Transduction; Tetradecanoylphorbol Acetate; Umbilical Veins | 2004 |
Differential in vitro neurotoxicity of the flame retardant PBDE-99 and of the PCB Aroclor 1254 in human astrocytoma cells.
Topics: Apoptosis; Astrocytes; Astrocytoma; Cell Line, Tumor; Cell Survival; Chlorodiphenyl (54% Chlorine); Dose-Response Relationship, Drug; Down-Regulation; Enzyme Inhibitors; Flame Retardants; Formazans; Halogenated Diphenyl Ethers; Humans; Indoles; Isoenzymes; L-Lactate Dehydrogenase; Maleimides; Phenyl Ethers; Protein Kinase C; Tetradecanoylphorbol Acetate; Tetrazolium Salts; Trypan Blue; Tumor Suppressor Protein p53 | 2004 |
Protein kinase C activation promotes the internalization of the human cationic amino acid transporter hCAT-1. A new regulatory mechanism for hCAT-1 activity.
Topics: Animals; Biotinylation; Cationic Amino Acid Transporter 1; Enzyme Activation; Enzyme Inhibitors; Gene Expression; Glioblastoma; Green Fluorescent Proteins; Homeostasis; Humans; Indoles; Maleimides; Microscopy, Fluorescence; Mutagenesis, Site-Directed; Oocytes; Phosphorylation; Protein Kinase C; Recombinant Fusion Proteins; Tetradecanoylphorbol Acetate; Transfection; Tumor Cells, Cultured; Xenopus laevis | 2004 |
Histamine reduces gap junctional communication of human tonsil high endothelial cells in culture.
Topics: Cells, Cultured; Chlorpheniramine; Coloring Agents; Connexin 43; Cyclic AMP; Cyclooxygenase Inhibitors; Cytoskeleton; Dose-Response Relationship, Drug; Endothelial Cells; Enzyme Inhibitors; Gap Junctions; Histamine; Humans; Immunoblotting; Indoles; Indomethacin; Inflammation; Ionophores; Maleimides; Microscopy, Fluorescence; Palatine Tonsil; Phalloidine; Phosphorylation; Protein Kinase C; Tetradecanoylphorbol Acetate; Time Factors | 2004 |
Connexin43 synthesis, phosphorylation, and degradation in regulation of transient inhibition of gap junction intercellular communication by the phorbol ester TPA in rat liver epithelial cells.
Topics: Animals; Blotting, Western; Carcinogens; Cell Communication; Cell Line; Cell Line, Tumor; Connexin 43; Cycloheximide; Dactinomycin; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Epithelial Cells; Flavonoids; Fluorescent Dyes; Gap Junctions; Image Processing, Computer-Assisted; Indoles; Isoquinolines; Liver; Maleimides; MAP Kinase Signaling System; Phosphorylation; Protein Kinase C; Protein Synthesis Inhibitors; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Time Factors | 2005 |
Protein kinase C modulates agonist-sensitive release of Ca2+ from internal stores in HEK293 cells overexpressing the calcium sensing receptor.
Topics: Calcium; Carbazoles; Cations; Cell Line; Culture Media, Serum-Free; Down-Regulation; Enzyme Activation; Enzyme Inhibitors; Humans; Immunoblotting; Indoles; Maleimides; Neomycin; Protein Isoforms; Protein Kinase C; Protein Kinase C-epsilon; Receptors, Calcium-Sensing; Signal Transduction; Subcellular Fractions; Tetradecanoylphorbol Acetate; Time Factors | 2005 |
Dopamine and norepinephrine transporter-dependent c-Fos production in vitro: relevance to neuroadaptation.
Topics: Adaptation, Physiological; Brain Chemistry; Cell Line; Dopamine; Dopamine Agonists; Dopamine Plasma Membrane Transport Proteins; Enzyme Inhibitors; Gene Expression Regulation; Humans; Indoles; Maleimides; Membrane Glycoproteins; Membrane Transport Modulators; Membrane Transport Proteins; Nerve Tissue Proteins; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Phosphorylation; Protein Kinase C; Proto-Oncogene Proteins c-fos; Symporters; Tetradecanoylphorbol Acetate | 2005 |
P2Y2 nucleotide receptors enhance alpha-secretase-dependent amyloid precursor protein processing.
Topics: ADAM Proteins; ADAM17 Protein; Amino Acid Chloromethyl Ketones; Amyloid beta-Protein Precursor; Amyloid Precursor Protein Secretases; Aspartic Acid Endopeptidases; Blotting, Western; Butadienes; Calcium; Cell Line, Tumor; Central Nervous System; Chelating Agents; Dose-Response Relationship, Drug; Down-Regulation; Egtazic Acid; Endopeptidases; Furin; Humans; Indoles; Maleimides; MAP Kinase Signaling System; Metalloendopeptidases; Nitriles; Phorbol Esters; Protein Kinase C; Protein Structure, Tertiary; Receptors, Purinergic P2; Receptors, Purinergic P2Y2; RNA, Small Interfering; Tetradecanoylphorbol Acetate; Time Factors; Transfection; Uridine Triphosphate | 2005 |
Artocarpol A stimulation of superoxide anion generation in neutrophils involved the activation of PLC, PKC and p38 mitogen-activated PK signaling pathways.
Topics: Animals; Butadienes; Calcium; Cell-Free System; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Estrenes; Flavonoids; Heterocyclic Compounds, 4 or More Rings; Imidazoles; Immunoblotting; Indoles; Maleimides; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Nitriles; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase C; Pyridines; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Signal Transduction; Superoxides; Tetradecanoylphorbol Acetate; Type C Phospholipases | 2005 |
The role of intracellular Ca2+ in the regulation of proteinase-activated receptor-2 mediated nuclear factor kappa B signalling in keratinocytes.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Calcium; Cell Line; Chelating Agents; Egtazic Acid; Enzyme Inhibitors; Estrenes; Humans; I-kappa B Kinase; Indoles; Keratinocytes; Maleimides; Mitogen-Activated Protein Kinases; NF-kappa B; Oligonucleotides; Phosphodiesterase Inhibitors; Protein Binding; Protein Kinase C; Protein Serine-Threonine Kinases; Pyrrolidinones; Receptor, PAR-2; Signal Transduction; Tacrolimus; Tetradecanoylphorbol Acetate; Trypsin; Type C Phospholipases | 2005 |
Effect of protein kinase C activation on intracellular Ca2+ signaling and integrity of intestinal epithelial cells.
Topics: Acetophenones; Animals; Benzopyrans; Calcium; Calcium Channel Blockers; Calcium Signaling; Carbazoles; Cell Line; Cell Survival; Chelating Agents; Dose-Response Relationship, Drug; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; Epithelial Cells; Indoles; Intestinal Mucosa; Intracellular Space; Maleimides; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-delta; Protein Kinase C-epsilon; Tetradecanoylphorbol Acetate; Verapamil | 2005 |
Acoustic environment determines phosphorylation state of the Kv3.1 potassium channel in auditory neurons.
Topics: Acoustic Stimulation; Action Potentials; Animals; Animals, Newborn; Brain Stem; CHO Cells; Cricetinae; Cricetulus; Dose-Response Relationship, Radiation; Electric Stimulation; Enzyme Inhibitors; Functional Laterality; Gene Expression Regulation; Immunohistochemistry; In Vitro Techniques; Indoles; Maleimides; Neurons; Patch-Clamp Techniques; Phosphorylation; Protein Kinase C; Rats; Rats, Sprague-Dawley; Tetradecanoylphorbol Acetate | 2005 |
Tumor necrosis factor-alpha activates the extrapituitary PRL promoter in myeloid leukemic cells.
Topics: Analysis of Variance; Cell Line; Drug Interactions; Electrophoretic Mobility Shift Assay; Enzyme Activation; Enzyme Inhibitors; Gene Expression Regulation; Humans; Indoles; Leukemia, Myeloid; Maleimides; Mutagenesis; Prolactin; Promoter Regions, Genetic; Tetradecanoylphorbol Acetate; Transfection; Tumor Necrosis Factor-alpha | 2006 |
Protein kinase C negatively regulates Akt activity and modifies UVC-induced apoptosis in mouse keratinocytes.
Topics: Adenoviridae; Animals; Apoptosis; Cells, Cultured; Immunoblotting; Immunoprecipitation; Indoles; Insulin-Like Growth Factor I; Keratinocytes; Maleimides; Mice; Phosphoprotein Phosphatases; Phosphorylation; Protein Isoforms; Protein Kinase C; Protein Kinase C-delta; Protein Kinase C-epsilon; Protein Phosphatase 2; Protein Transport; Proto-Oncogene Proteins c-akt; Serine; Signal Transduction; Skin; Tetradecanoylphorbol Acetate; Time Factors; Ultraviolet Rays | 2006 |
Regulation of protein kinase C delta by phorbol ester, endothelin-1, and platelet-derived growth factor in cardiac myocytes.
Topics: Animals; Animals, Newborn; Cell Culture Techniques; Cell Extracts; Cells, Cultured; Chromatography, Gel; Chromones; Endothelin-1; Enzyme Inhibitors; Gene Expression Regulation, Enzymologic; Immunoblotting; Indoles; Maleimides; Morpholines; Myocytes, Cardiac; Phosphorylation; Platelet-Derived Growth Factor; Precipitin Tests; Protein Kinase C-delta; Pyrimidines; Rats; Rats, Sprague-Dawley; Solubility; Tetradecanoylphorbol Acetate; Time Factors | 2006 |
Regulation of vascular smooth muscle proliferation and migration by beta2-chimaerin, a non-protein kinase C phorbol ester receptor.
Topics: Animals; Blotting, Western; Cell Line; Cell Line, Tumor; Cell Movement; Cell Proliferation; Cells, Cultured; Gene Expression; GTPase-Activating Proteins; Humans; Immunohistochemistry; Indoles; Infant, Newborn; Maleimides; Mitogens; Muscle, Smooth, Vascular; Neoplasm Proteins; Platelet-Derived Growth Factor; Protein Kinase C; Rats; Reverse Transcriptase Polymerase Chain Reaction; Tetradecanoylphorbol Acetate | 2006 |
Bradykinin augments EGF-induced airway smooth muscle proliferation by activation of conventional protein kinase C isoenzymes.
Topics: Animals; Bradykinin; Carbazoles; Cattle; Cell Proliferation; Cells, Cultured; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Activation; Enzyme Inhibitors; Epidermal Growth Factor; Indoles; Isoenzymes; Maleimides; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Myocytes, Smooth Muscle; Protein Kinase C; Receptor, Bradykinin B2; Tetradecanoylphorbol Acetate; Thymidine; Trachea; Tritium | 2006 |
Mechanism of gonadotropin-releasing hormone (GnRH)-I and -II-induced cell growth inhibition in ovarian cancer cells: role of the GnRH-I receptor and protein kinase C pathway.
Topics: Adenocarcinoma; Cell Proliferation; Enzyme Activation; Enzyme Inhibitors; Female; Gonadotropin-Releasing Hormone; Humans; Indoles; Maleimides; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Oligopeptides; Ovarian Neoplasms; Protein Kinase C; Receptors, LHRH; RNA, Small Interfering; Signal Transduction; Tetradecanoylphorbol Acetate; Transfection; Tumor Cells, Cultured | 2006 |
Stimulation of cyclic AMP production by the Caenorhabditis elegans muscarinic acetylcholine receptor GAR-3 in Chinese hamster ovary cells.
Topics: Animals; Caenorhabditis elegans; Caenorhabditis elegans Proteins; Calcium; Carbachol; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; GTP-Binding Protein alpha Subunits, Gi-Go; Indoles; Maleimides; Muscarinic Agonists; Muscarinic Antagonists; Pertussis Toxin; Protein Isoforms; Protein Kinase C; Receptors, Muscarinic; Tetradecanoylphorbol Acetate | 2006 |
Calcium channel and glutamate receptor activities regulate actin organization in salamander retinal neurons.
Topics: Actins; Alkaloids; Animals; Benzophenanthridines; Calcium; Calcium Channels, L-Type; Carcinogens; Cell Survival; Electrophysiology; Enzyme Inhibitors; Glutamic Acid; Indoles; Maleimides; Neurons, Afferent; Phenanthridines; Potassium; Protein Kinase C; Receptors, Glutamate; Retinal Ganglion Cells; Tetradecanoylphorbol Acetate; Urodela | 2006 |
Increase of C-type natriuretic peptide expression by serum and platelet-derived growth factor-BB in human aortic smooth muscle cells is dependent on protein kinase C activation.
Topics: Animals; Aorta; Becaplermin; Blood; Cells, Cultured; Culture Media; Endothelial Cells; Enzyme Activation; Gene Expression; Genistein; Humans; Indoles; Maleimides; Muscle, Smooth, Vascular; Natriuretic Peptide, C-Type; Platelet-Derived Growth Factor; Protein Kinase C; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-sis; Rats; Receptors, Atrial Natriuretic Factor; RNA, Messenger; Species Specificity; Tetradecanoylphorbol Acetate; Tyrphostins | 2006 |
Role of kinases and G-proteins in the hyposmotic stimulation of cardiac IKs.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Cell Line; Chromans; Colforsin; Cricetinae; Cyclic AMP-Dependent Protein Kinases; Cytochalasin D; Cytoskeleton; GTP-Binding Proteins; Guinea Pigs; Indoles; Isoquinolines; KCNQ1 Potassium Channel; Maleimides; Mitogen-Activated Protein Kinases; Myocytes, Cardiac; Osmotic Pressure; Phosphatidylinositol 3-Kinases; Potassium Channels; Protein Kinase C; Protein-Tyrosine Kinases; Sulfonamides; Tetradecanoylphorbol Acetate; Tyrphostins | 2006 |
Protein kinase Cbeta isoform down-regulates the expression of MDR3 P-glycoprotein in human Chang liver cells.
Topics: ATP Binding Cassette Transporter, Subfamily B; ATP-Binding Cassette Transporters; Carbazoles; Cells, Cultured; Down-Regulation; Humans; Indoles; Isoenzymes; Liver; Maleimides; Protein Kinase C; Protein Kinase C beta; Tetradecanoylphorbol Acetate | 2006 |
On the mechanisms of 12-O-tetradecanoylphorbol-13-acetate-induced growth arrest in pancreatic cancer cells.
Topics: Cell Division; Cell Line, Tumor; Cell Proliferation; Cyclin A; Cyclin B; Cyclin B1; Cyclin E; Cyclin-Dependent Kinase Inhibitor p21; Flavonoids; G2 Phase; Gene Expression Regulation, Neoplastic; Humans; Indoles; Maleimides; MAP Kinase Kinase Kinases; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Pancreatic Neoplasms; Phosphorylation; Protein Kinase C; Protein Kinase Inhibitors; RNA, Messenger; Tetradecanoylphorbol Acetate | 2006 |
Protein kinase C cross-talk with gonadotrope progesterone receptor is involved in GnRH-induced LH secretion.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Bodily Secretions; Cells, Cultured; Chelating Agents; Colforsin; Egtazic Acid; Enzyme Inhibitors; Female; Gonadotropin-Releasing Hormone; Imines; Indoles; Ionomycin; Luteinizing Hormone; Maleimides; Mifepristone; Nifedipine; Pituitary Gland, Anterior; Protein Kinase C; Rats; Rats, Wistar; Receptors, Progesterone; Signal Transduction; Tetradecanoylphorbol Acetate | 2006 |
Hydrogen peroxide-induced arachidonic acid release in L929 cells; roles of Src, protein kinase C and cytosolic phospholipase A2alpha.
Topics: Animals; Arachidonic Acid; Calcimycin; Calcium; Cell Line, Tumor; Cytosol; Dose-Response Relationship, Drug; Enzyme Inhibitors; Fibroblasts; Group IV Phospholipases A2; Humans; Hydrogen Peroxide; Indoles; Ionophores; Maleimides; Mice; Phospholipases A; Protein Kinase C; Protein Kinase C-alpha; Protein Transport; Pyrimidines; Pyrrolidines; Signal Transduction; src-Family Kinases; Tetradecanoylphorbol Acetate; Transfection | 2006 |
The sarcoplasmic-endoplasmic reticulum Ca2+ ATPase 2b regulates the Ca2+ transients elicited by P2Y2 activation in PC Cl3 thyroid cells.
Topics: Adenosine Triphosphate; Animals; Barium; Biological Transport, Active; Calcium; Carbazoles; Cell Line; Enzyme Activation; Indoles; Maleimides; Manganese; Microscopy, Fluorescence; Protein Kinase C; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2Y2; Sarcoplasmic Reticulum; Sarcoplasmic Reticulum Calcium-Transporting ATPases; Tetradecanoylphorbol Acetate; Thapsigargin; Thyroid Gland; Uridine Triphosphate | 2006 |
Phospholipase A2-independent Ca2+ entry and subsequent apoptosis induced by melittin in human MG63 osteosarcoma cells.
Topics: Apoptosis; Calcium; Calcium Channels, L-Type; Cell Line, Tumor; Cell Survival; Egtazic Acid; Enzyme Inhibitors; Fluorescent Dyes; Fura-2; Humans; Indoles; Maleimides; Melitten; Osteoblasts; Osteosarcoma; Phospholipases A; Phospholipases A2; Tetradecanoylphorbol Acetate | 2007 |
TNF-alpha decreases hsp 27 in human blood mononuclear cells: involvement of protein kinase c.
Topics: Carcinogens; Cells, Cultured; Enzyme Activation; Enzyme Inhibitors; Heat-Shock Proteins; HSP70 Heat-Shock Proteins; Humans; Indoles; Leukocytes, Mononuclear; Maleimides; Phosphorylation; Protein Kinase C; Protein Processing, Post-Translational; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha | 2006 |
Role of ROS and MAPK in TPA-induced ICAM-1 expression in the myeloid ML-1 cell line.
Topics: Blotting, Western; Butadienes; Cell Line, Tumor; Extracellular Signal-Regulated MAP Kinases; Flavonoids; Flow Cytometry; Gene Expression Regulation, Neoplastic; Humans; Indoles; Intercellular Adhesion Molecule-1; Leukemia, Myeloid; Maleimides; Mitogen-Activated Protein Kinases; Models, Biological; NF-kappa B; Nitriles; Oligonucleotide Array Sequence Analysis; Protein Kinase C; Reactive Oxygen Species; Signal Transduction; Sulfones; Tetradecanoylphorbol Acetate | 2007 |
Sustained activation of proton channels and NADPH oxidase in human eosinophils and murine granulocytes requires PKC but not cPLA2 alpha activity.
Topics: Animals; Arachidonic Acids; Carcinogens; Enzyme Activation; Enzyme Inhibitors; Eosinophils; Granulocytes; Group IV Phospholipases A2; Humans; Indoles; Ion Channels; Maleimides; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, SCID; N-Formylmethionine Leucyl-Phenylalanine; NADPH Oxidases; Okadaic Acid; Phospholipases A; Protein Kinase C; Protons; Signal Transduction; Tetradecanoylphorbol Acetate | 2007 |
Alpha1-adrenergic receptor stimulation induces the expression of receptor activator of nuclear factor kappaB ligand gene via protein kinase C and extracellular signal-regulated kinase pathways in MC3T3-E1 osteoblast-like cells.
Topics: 3T3 Cells; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blotting, Western; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Extracellular Signal-Regulated MAP Kinases; Flavonoids; Indoles; Maleimides; Mice; Osteoblasts; Phenylephrine; Prazosin; Propranolol; Protein Kinase C; Receptor Activator of Nuclear Factor-kappa B; Receptors, Adrenergic, alpha-1; Reverse Transcriptase Polymerase Chain Reaction; Tetradecanoylphorbol Acetate; Yohimbine | 2007 |
Stimulatory action of protein kinase C(epsilon) isoform on the slow component of delayed rectifier K+ current in guinea-pig atrial myocytes.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Delayed Rectifier Potassium Channels; Dose-Response Relationship, Drug; Enzyme Activation; Guinea Pigs; Heart Atria; In Vitro Techniques; Indoles; Isoenzymes; Maleimides; Membrane Potentials; Myocytes, Cardiac; Patch-Clamp Techniques; Peptide Fragments; Phenylephrine; Prazosin; Protein Kinase C-epsilon; Protein Kinase Inhibitors; Receptors, Adrenergic, alpha-1; Tetradecanoylphorbol Acetate; Time Factors | 2007 |
Modulation of hERG potassium currents in HEK-293 cells by protein kinase C. Evidence for direct phosphorylation of pore forming subunits.
Topics: Calcium; Cell Line; Diglycerides; Enzyme Activators; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Humans; Indoles; Ion Channel Gating; Ionomycin; Ionophores; Maleimides; Membrane Potentials; Methacholine Chloride; Muscarinic Agonists; Mutation; Phosphorylation; Potassium; Protein Kinase C; Protein Kinase Inhibitors; Receptor, Muscarinic M3; Signal Transduction; Tetradecanoylphorbol Acetate; Transfection | 2007 |
Regulation of matrix Gla protein by parathyroid hormone in MC3T3-E1 osteoblast-like cells involves protein kinase A and extracellular signal-regulated kinase pathways.
Topics: 3T3 Cells; Animals; Butadienes; Calcium-Binding Proteins; Colforsin; Cyclic AMP-Dependent Protein Kinases; Extracellular Matrix Proteins; Extracellular Signal-Regulated MAP Kinases; Gene Expression Regulation; Indoles; Isoquinolines; Maleimides; Matrix Gla Protein; Mice; Nitriles; Osteoblasts; Parathyroid Hormone; Promoter Regions, Genetic; Protein Kinase C; Recombinant Proteins; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate | 2007 |
Involvement of nPKC-MAPK pathway in the decrease of nucleophosmin/B23 during megakaryocytic differentiation of human myelogenous leukemia K562 cells.
Topics: Carbazoles; Cell Differentiation; Cell Line, Tumor; Humans; Indoles; K562 Cells; Leukemia, Myeloid; Maleimides; Megakaryocytes; Mitogen-Activated Protein Kinases; Nuclear Proteins; Nucleolin; Nucleophosmin; Phosphoproteins; Proteasome Endopeptidase Complex; Proteasome Inhibitors; Protein Kinase C; RNA-Binding Proteins; Tetradecanoylphorbol Acetate | 2007 |
Regulation of plasminogen activators in human thyroid follicular cells and their relationship to differentiated function.
Topics: Adenylyl Cyclases; Aprotinin; Cell Differentiation; Cells, Cultured; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Activators; Epidermal Growth Factor; Fibroblast Growth Factors; Flavonoids; Humans; Indoles; Insulin; Iodine; Iodine Radioisotopes; Maleimides; Mesylates; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Plasminogen Inactivators; Protein Kinase C; Protein Kinase C beta; Protein Kinase Inhibitors; Pyrroles; RNA, Messenger; Serine Proteinase Inhibitors; Signal Transduction; Tetradecanoylphorbol Acetate; Thyroid Gland; Thyrotropin; Time Factors; Tissue Plasminogen Activator; Urokinase-Type Plasminogen Activator | 2007 |
Cytotoxic action of phorbol esters on human pancreatic cancer cells.
Topics: Animals; Apoptosis; Cell Line, Tumor; Cell Proliferation; Cell Survival; Dose-Response Relationship, Drug; Enzyme Inhibitors; Humans; Indoles; Inhibitory Concentration 50; Intracellular Signaling Peptides and Proteins; Maleimides; Membrane Proteins; Mice; Myristoylated Alanine-Rich C Kinase Substrate; Pancreatic Neoplasms; Phorbol 12,13-Dibutyrate; Phorbol Esters; Phosphorylation; Protein Kinase C; Tetradecanoylphorbol Acetate; Xenograft Model Antitumor Assays | 2007 |
The role of protein kinase C isoenzymes in the regulation of calcineurin activity in human peripheral blood mononuclear cells.
Topics: Adaptor Proteins, Signal Transducing; Base Sequence; Calcimycin; Calcineurin; Calcineurin Inhibitors; Carbazoles; DNA Primers; Enzyme Activation; Humans; In Vitro Techniques; Indoles; Ionophores; Isoenzymes; Leukocytes, Mononuclear; Maleimides; Phosphorylation; Protein Kinase C; Protein Kinase Inhibitors; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; Tetradecanoylphorbol Acetate | 2007 |
Phosphorylation of claudin-4 by PKCepsilon regulates tight junction barrier function in ovarian cancer cells.
Topics: Cell Line, Tumor; Claudin-4; Female; Humans; Indoles; Maleimides; Membrane Proteins; Mutation; Ovarian Neoplasms; Phosphorylation; Protein Isoforms; Protein Kinase C-epsilon; Signal Transduction; Tetradecanoylphorbol Acetate; Tight Junctions | 2007 |
Activation of epidermal akt by diverse mouse skin tumor promoters.
Topics: Animals; Anthracenes; Anticoagulants; Carcinogens; Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Epidermis; ErbB Receptors; Female; Heparin; Indoles; Keratinocytes; Maleimides; Mice; Mice, Inbred ICR; Okadaic Acid; Phosphorylation; Protein Kinase C; Proto-Oncogene Proteins c-akt; Skin Neoplasms; Tetradecanoylphorbol Acetate | 2007 |
Opposite effect of phorbol ester PMA on PTGS2 and PGDH mRNA expression in human chorion trophoblast cells.
Topics: Calcium; Carcinogens; Cells, Cultured; Chorion; Cyclooxygenase 2; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Gene Expression Regulation, Enzymologic; Humans; Hydroxyprostaglandin Dehydrogenases; Imidazoles; Indoles; Maleimides; MAP Kinase Kinase 1; MAP Kinase Kinase 2; MAP Kinase Kinase 4; MAP Kinase Signaling System; p38 Mitogen-Activated Protein Kinases; Pregnancy; Protein Kinase C; Pyridines; RNA, Messenger; Tetradecanoylphorbol Acetate; Trophoblasts | 2008 |
Effects of phorbol ester on vesicle dynamics as revealed by total internal reflection fluorescence microscopy.
Topics: Animals; Cytoplasmic Vesicles; Diglycerides; Electrophysiology; Enzyme Inhibitors; Exocytosis; Green Fluorescent Proteins; Indoles; Maleimides; Microscopy, Fluorescence; Movement; Neuropeptide Y; PC12 Cells; Protein Kinase C; Rats; Tetradecanoylphorbol Acetate | 2008 |
P70 S6 kinase negatively regulates fibroblast growth factor 2-stimulated interleukin-6 synthesis in osteoblasts: function at a point downstream from protein kinase C.
Topics: Animals; Carbazoles; Cells, Cultured; Fibroblast Growth Factor 2; Indoles; Interleukin-6; Maleimides; Mice; Osteoblasts; Phosphorylation; Protein Kinase C; Ribosomal Protein S6 Kinases, 70-kDa; Sirolimus; Tetradecanoylphorbol Acetate | 2008 |
Modulation of cytokine production by plant sterols in stimulated human Jurkat T cells.
Topics: Cell Division; Cell Survival; Cholesterol; Concanavalin A; Cytokines; Enzyme Inhibitors; Humans; Immunologic Factors; Immunosuppressive Agents; Indoles; Interleukin-2; Jurkat Cells; Lymphocyte Activation; Maleimides; Phytosterols; Protein Kinase C; Sitosterols; T-Lymphocytes; Tacrolimus; Tetradecanoylphorbol Acetate | 2008 |
Protein kinase C-mediated protection of motoneurons from excitotoxicity.
Topics: Animals; Cell Survival; Dose-Response Relationship, Drug; Drug Interactions; Embryo, Mammalian; Enzyme Inhibitors; Excitatory Amino Acids; Glutamic Acid; Indoles; Maleimides; Motor Neurons; Neuroprotective Agents; Protein Kinase C; Rats; Spinal Cord; Tetradecanoylphorbol Acetate | 2008 |
The role of P38 MAPK and PKC in BLP induced TNF-alpha release, apoptosis, and NFkappaB activation in THP-1 monocyte cells.
Topics: Apoptosis; Bacterial Proteins; Cell Line; Dose-Response Relationship, Drug; Enzyme Inhibitors; Humans; Imidazoles; Indoles; Inflammation; Lipopolysaccharides; Lipoproteins; Maleimides; Monocytes; NF-kappa B; p38 Mitogen-Activated Protein Kinases; Protein Kinase C; Pyridines; Signal Transduction; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha | 2009 |
Electrogenic NBCe1 (SLC4A4), but not electroneutral NBCn1 (SLC4A7), cotransporter undergoes cholinergic-stimulated endocytosis in salivary ParC5 cells.
Topics: Animals; Bicarbonates; Biotinylation; Calmodulin; Carbachol; Cell Line; Cell Membrane; Cell Polarity; Cholinergic Agonists; Endocytosis; Endosomes; Gene Transfer Techniques; Hydrogen-Ion Concentration; Indoles; Maleimides; Microscopy, Confocal; Monensin; Parotid Gland; Protein Kinase C; Protein Kinase Inhibitors; Protein Transport; Rats; Receptors, Muscarinic; Sodium-Bicarbonate Symporters; Sulfonamides; Tetradecanoylphorbol Acetate; Time Factors; Xenopus laevis | 2008 |
Exogenous nitric oxide-induced release of calcium from intracellular IP3 receptor-sensitive stores via S-nitrosylation in respiratory burst-dependent neutrophils.
Topics: Calcium; Cells, Cultured; Humans; Indoles; Inositol 1,4,5-Trisphosphate Receptors; Maleimides; Neutrophils; Nitric Oxide; Nitric Oxide Donors; Nitroprusside; Protein Kinase C; Protein Kinase Inhibitors; Respiratory Burst; Tetradecanoylphorbol Acetate | 2008 |
Roles of protein kinase C isotypes during seawater-versus cAMP-induced oocyte maturation in a marine worm.
Topics: Animals; Bridged-Ring Compounds; Diglycerides; Dose-Response Relationship, Drug; Enzyme Inhibitors; Immunoblotting; Indoles; Invertebrates; Isoenzymes; Maleimides; Neomycin; Norbornanes; Oocytes; Protein Kinase C; Seawater; Signal Transduction; Tetradecanoylphorbol Acetate; Thiocarbamates; Thiones | 2009 |
Alteration of the PKC-mediated signaling pathway for smooth muscle contraction in obstruction-induced hypertrophy of the urinary bladder.
Topics: Animals; Disease Models, Animal; Humans; Hypertrophy; In Vitro Techniques; Indoles; Male; Maleimides; Muscle Contraction; Muscle Proteins; Muscle, Smooth; Phosphoproteins; Phosphorylation; Potassium Chloride; Protein Kinase C; Rabbits; Signal Transduction; Tetradecanoylphorbol Acetate; Urinary Bladder; Urinary Bladder Neck Obstruction | 2009 |
Modulation of ileal apical Na+-dependent bile acid transporter ASBT by protein kinase C.
Topics: Bile Acids and Salts; Caco-2 Cells; Calcium; Cell Membrane; Chelating Agents; Chromones; Egtazic Acid; Enzyme Activators; Humans; Ileum; Indoles; Intestinal Mucosa; Kinetics; Maleimides; Morpholines; Organic Anion Transporters, Sodium-Dependent; Peptides; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase C; Protein Kinase Inhibitors; Protein Processing, Post-Translational; Symporters; Tetradecanoylphorbol Acetate; Transfection | 2009 |
Phosphorylation of histone H3 by protein kinase C signaling plays a critical role in the regulation of the developmentally important TBX2 gene.
Topics: Binding Sites; Blotting, Western; Cell Line; Chromatin Immunoprecipitation; Enzyme Inhibitors; Fibroblasts; Flavonoids; Gene Expression; Histones; Humans; Imidazoles; Indoles; Maleimides; Mitogen-Activated Protein Kinases; Phosphorylation; Promoter Regions, Genetic; Protein Binding; Protein Kinase C; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; Ribosomal Protein S6 Kinases, 90-kDa; RNA Interference; Serine; Signal Transduction; Sp1 Transcription Factor; T-Box Domain Proteins; Tetradecanoylphorbol Acetate | 2009 |
Differential fading of inhibitory and excitatory B2 bradykinin receptor responses in rat sympathetic neurons: a role for protein kinase C.
Topics: Adrenergic beta-Antagonists; Animals; Animals, Newborn; Bradykinin; Calcium; Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Inhibitors; Indoles; Maleimides; Membrane Potentials; Neural Inhibition; Neurons; Norepinephrine; Patch-Clamp Techniques; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B2; Sodium Channel Blockers; Statistics, Nonparametric; Superior Cervical Ganglion; Tetradecanoylphorbol Acetate; Tetrodotoxin; Time Factors; Tritium | 2009 |
Identification of Thr29 as a critical phosphorylation site that activates the human proton channel Hvcn1 in leukocytes.
Topics: Amino Acid Substitution; Carcinogens; Cell Line; Enzyme Inhibitors; Humans; Indoles; Ion Channel Gating; Ion Channels; Leukocytes; Maleimides; Mutation, Missense; NADPH Oxidases; Phosphorylation; Protein Kinase C-delta; Respiratory Burst; Tetradecanoylphorbol Acetate; Threonine | 2010 |
Roles of phospholipase D in phorbol myristate acetate-stimulated neutrophil respiratory burst.
Topics: 1-Butanol; Calcium; Cells, Cultured; Diglycerides; Enzyme Inhibitors; Estrenes; Humans; Indoles; Maleimides; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Phosphatidic Acids; Phosphodiesterase Inhibitors; Phospholipase D; Protein Kinase C; Protein Transport; Pyrrolidinones; Respiratory Burst; Tetradecanoylphorbol Acetate | 2011 |
Protein kinase C regulates neurite outgrowth in spinal cord neurons.
Topics: Animals; Cells, Cultured; Dose-Response Relationship, Drug; Embryo, Mammalian; Enzyme Activators; Enzyme Inhibitors; Indoles; Maleimides; Neurites; Neurons; Protein Kinase C; Rats; Rats, Sprague-Dawley; Spinal Cord; Tetradecanoylphorbol Acetate; Time Factors | 2010 |
Serine phosphorylation of glutathione S-transferase P1 (GSTP1) by PKCα enhances GSTP1-dependent cisplatin metabolism and resistance in human glioma cells.
Topics: Antineoplastic Agents; bcl-2-Associated X Protein; Cell Line, Tumor; Cisplatin; Drug Resistance, Neoplasm; Glioma; Glutathione S-Transferase pi; Humans; Indoles; Maleimides; Phosphorylation; Protein Kinase C-alpha; Protein Transport; RNA, Small Interfering; Serine; Tetradecanoylphorbol Acetate | 2010 |
Mechanism of hCG-induced spermiation in the toad Rhinella arenarum (Amphibia, Anura).
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Amiloride; Animals; Bufo arenarum; Chorionic Gonadotropin; Cyclic AMP-Dependent Protein Kinases; Indoles; Isoquinolines; Male; Maleimides; Ouabain; Protein Kinase C; Sertoli Cells; Sodium-Potassium-Exchanging ATPase; Spermatozoa; Staurosporine; Sulfonamides; Tetradecanoylphorbol Acetate | 2010 |
Transcriptional regulation of claudin-18 via specific protein kinase C signaling pathways and modification of DNA methylation in human pancreatic cancer cells.
Topics: Carcinoma, Pancreatic Ductal; Cell Line, Tumor; Claudins; DNA Methylation; Enzyme Activation; Gene Expression Regulation, Neoplastic; Humans; Indoles; Isoenzymes; Maleimides; Membrane Proteins; Pancreatic Ducts; Phosphorylation; Promoter Regions, Genetic; Protein Kinase C; Signal Transduction; Tetradecanoylphorbol Acetate; Tight Junctions; Up-Regulation | 2011 |
Claudin-18 is an early-stage marker of pancreatic carcinogenesis.
Topics: Adenocarcinoma, Mucinous; Biomarkers, Tumor; Carcinoma, Pancreatic Ductal; Carcinoma, Papillary; Cell Transformation, Neoplastic; Claudins; Enzyme Inhibitors; Humans; Indoles; Maleimides; Membrane Proteins; Pancreas; Pancreatic Neoplasms; Pancreatitis, Chronic; Protein Kinase C; Retrospective Studies; Stomach Neoplasms; Tetradecanoylphorbol Acetate | 2011 |
Physiological effect of protein kinase C on ENaC-mediated lung liquid regulation in the adult rat lung.
Topics: Amiloride; Animals; Benzophenanthridines; Biological Transport; Cells, Cultured; Electric Impedance; Enzyme Inhibitors; Epithelial Cells; Epithelial Sodium Channels; Indoles; Ionomycin; Isotonic Solutions; Lung; Male; Maleimides; Protein Kinase C; Rats; Rats, Wistar; Ringer's Solution; Signal Transduction; Sodium Channel Blockers; Terbutaline; Tetradecanoylphorbol Acetate | 2012 |
TPA induces the expression of EC-SOD in human monocytic THP-1 cells: involvement of PKC, MEK/ERK and NOX-derived ROS.
Topics: Butadienes; Cell Differentiation; Cell Line, Tumor; Extracellular Signal-Regulated MAP Kinases; Flavonoids; Humans; Indoles; Macrophages; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Monocytes; NADPH Oxidases; Nitriles; Protein Kinase C; Reactive Oxygen Species; Superoxide Dismutase; Tetradecanoylphorbol Acetate | 2012 |
Potentiation of the P2X3 ATP receptor by PAR-2 in rat dorsal root ganglia neurons, through protein kinase-dependent mechanisms, contributes to inflammatory pain.
Topics: Adenosine Triphosphate; Animals; Carbazoles; Colforsin; Cyclic AMP-Dependent Protein Kinases; Ganglia, Spinal; Indoles; Inflammation; Male; Maleimides; MAP Kinase Signaling System; Membrane Potentials; Neurons; Pain; Phosphorylation; Protein Kinase C; Protein Transport; Purinergic P2X Receptor Agonists; Purinergic P2X Receptor Antagonists; Pyrroles; Rats, Sprague-Dawley; Receptor, PAR-2; Receptors, Purinergic P2X3; Tetradecanoylphorbol Acetate | 2012 |
The Src kinase Yes is activated in pancreatic acinar cells by gastrointestinal hormones/neurotransmitters, but not pancreatic growth factors, which stimulate its association with numerous other signaling molecules.
Topics: Acinar Cells; Animals; Bombesin; Calcimycin; Calcium Ionophores; Calcium Signaling; Carbachol; Cholecystokinin; Enzyme Activation; Focal Adhesion Kinase 1; Focal Adhesion Kinase 2; Gastrointestinal Hormones; Indoles; Intercellular Signaling Peptides and Proteins; Male; Maleimides; Neurotransmitter Agents; Pancreas; Peptide Fragments; Phosphorylation; Protein Kinase C; Protein Processing, Post-Translational; Proto-Oncogene Proteins c-yes; Rats; Rats, Sprague-Dawley; Tetradecanoylphorbol Acetate; Thapsigargin | 2012 |
6-Hydroxydopamine upregulates iron regulatory protein 1 by activating certain protein kinase C isoforms in the dopaminergic MES23.5 cell line.
Topics: Cation Transport Proteins; Cell Line; Dopaminergic Neurons; Enzyme Activation; Indoles; Iron; Iron Regulatory Protein 1; Isoenzymes; Maleimides; Oxidopamine; Protein Kinase C; Tetradecanoylphorbol Acetate; Up-Regulation | 2012 |
Inhibition of matrix metalloproteinase-9 expression by docosahexaenoic acid mediated by heme oxygenase 1 in 12-O-tetradecanoylphorbol-13-acetate-induced MCF-7 human breast cancer cells.
Topics: Adenocarcinoma; Androstadienes; Antineoplastic Agents; Breast Neoplasms; Carcinogens; Cell Movement; Cell Survival; Docosahexaenoic Acids; Dose-Response Relationship, Drug; Drug Antagonism; Enzyme Activation; Female; Flavonoids; Gene Expression Regulation, Neoplastic; Gene Silencing; Heme Oxygenase-1; Humans; Indoles; Maleimides; Matrix Metalloproteinase 9; MCF-7 Cells; Neoplasm Invasiveness; Tetradecanoylphorbol Acetate; Time Factors; Wortmannin | 2013 |
Protein kinase C regulates human pluripotent stem cell self-renewal.
Topics: Activins; Alkaline Phosphatase; Blotting, Western; Carbazoles; Cell Line; Cell Proliferation; Chromones; Extracellular Signal-Regulated MAP Kinases; Fibroblast Growth Factor 2; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Immunohistochemistry; Indoles; Maleimides; Morpholines; Phosphatidylinositol 3-Kinases; Phosphorylation; Pluripotent Stem Cells; Protein Kinase C; Protein Kinase C-delta; Protein Kinase C-epsilon; Proto-Oncogene Proteins c-akt; RNA Interference; Signal Transduction; Tetradecanoylphorbol Acetate | 2013 |
Protein kinase C activation inhibits rat and human hyperpolarization activated cyclic nucleotide gated channel (HCN)1--mediated current in mammalian cells.
Topics: Animals; Cell Line; HEK293 Cells; Humans; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Indoles; Maleimides; Membrane Potentials; Mice; Patch-Clamp Techniques; Protein Kinase C; Protein Kinase Inhibitors; Rats; Tetradecanoylphorbol Acetate | 2013 |
Naproxen-induced Ca2+ movement and death in MDCK canine renal tubular cells.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Calcium; Calcium Channel Blockers; Cell Death; Dogs; Imidazoles; Indoles; Madin Darby Canine Kidney Cells; Maleimides; Naproxen; Nifedipine; Protein Kinase C; Protein Kinase Inhibitors; Tetradecanoylphorbol Acetate | 2015 |
Activation of TRPM2 and TRPV1 Channels in Dorsal Root Ganglion by NADPH Oxidase and Protein Kinase C Molecular Pathways: a Patch Clamp Study.
Topics: Acetophenones; Action Potentials; Animals; Calcium Signaling; Capsaicin; Cells, Cultured; Cinnamates; Ganglia, Spinal; Indoles; Male; Maleimides; NADPH Oxidases; Neurons; ortho-Aminobenzoates; Oxidative Stress; Protein Kinase C; Rats; Rats, Wistar; Tetradecanoylphorbol Acetate; TRPM Cation Channels; TRPV Cation Channels | 2017 |
A novel DLX3-PKC integrated signaling network drives keratinocyte differentiation.
Topics: Animals; Antimicrobial Cationic Peptides; Calcium; Cell Adhesion; Cell Differentiation; Cell Proliferation; Cells, Cultured; Chemokines; Cytokines; Epidermis; Homeodomain Proteins; Humans; Hyperplasia; Indoles; Keratinocytes; Leukocytes; Maleimides; Mice; Mice, Transgenic; Protein Kinase C-alpha; Signal Transduction; Tetradecanoylphorbol Acetate; Transcription Factors | 2017 |
α-Cyperone Inhibits PMA-Induced EPCR Shedding through PKC Pathway.
Topics: ADAM17 Protein; Cell Survival; Endothelial Protein C Receptor; Human Umbilical Vein Endothelial Cells; Humans; Indoles; JNK Mitogen-Activated Protein Kinases; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Naphthalenes; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase C; Tetradecanoylphorbol Acetate | 2017 |