Page last updated: 2024-08-16

tetracaine and torpedo

tetracaine has been researched along with torpedo in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19903 (17.65)18.7374
1990's8 (47.06)18.2507
2000's5 (29.41)29.6817
2010's1 (5.88)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
McCarthy, MP; Stroud, RM1
Bigelow, J; Michel, L; Oswald, RE1
Haring, R; Kloog, Y1
McCarthy, MP; Moore, MA1
Baenziger, JE; McCarthy, MP; Méthot, N1
Baenziger, JE; Demers, CN; Méthot, N1
Eterović, VA; Ferchmin, PA; Hann, RM; Lee, YH; Li, L; McNamee, MG; Rodriguez, AD1
Chen, CH; Roth, LG; Zuklie, BM1
Baenziger, JE; Ryan, SE1
Cohen, JB; Middleton, RE; Strnad, NP1
Cohen, JB; Gallagher, MJ1
Chiara, DC; Cohen, JB; Gallagher, MJ1
Arias, HR; Bayer, EZ; Blanton, MP; Gallagher, MJ; McCardy, EA1
Arias, HR; Barrantes, FJ; Horváth, LI; Mantipragada, SB; Marsh, D; Sandhoff, K; Schwarzmann, G1
Arias, HR; Bhumireddy, P; Bouzat, C; Spitzmaul, G; Trudell, JR1
Baenziger, JE; daCosta, CJ; Goodreid, MM; Ryan, SE; Sturgeon, RM; Vuong, NQ1
Bruzik, KS; Chiara, DC; Cohen, JB; Savechenkov, PY; Yu, Z1

Other Studies

17 other study(ies) available for tetracaine and torpedo

ArticleYear
Conformational states of the nicotinic acetylcholine receptor from Torpedo californica induced by the binding of agonists, antagonists, and local anesthetics. Equilibrium measurements using tritium-hydrogen exchange.
    Biochemistry, 1989, Jan-10, Volume: 28, Issue:1

    Topics: Animals; Binding, Competitive; Bungarotoxins; Carbachol; Electric Organ; Hydrogen; In Vitro Techniques; Procaine; Protein Conformation; Receptors, Nicotinic; Tetracaine; Torpedo; Tritium

1989
Mechanism of binding of a benzomorphan opiate to the acetylcholine receptor from Torpedo electroplaque.
    Molecular pharmacology, 1986, Volume: 29, Issue:2

    Topics: Affinity Labels; Animals; Binding Sites; Bungarotoxins; Carbachol; Decamethonium Compounds; In Vitro Techniques; Kinetics; Phenazocine; Phencyclidine; Receptors, Cholinergic; Structure-Activity Relationship; Tetracaine; Torpedo; Tritium; Tubocurarine

1986
Multiple binding sites for phencyclidine on the nicotinic acetylcholine receptor from Torpedo ocellata electric organ.
    Life sciences, 1984, Mar-12, Volume: 34, Issue:11

    Topics: Acetylcholine; Animals; Binding Sites; Bungarotoxins; Carbachol; Dibucaine; Electric Organ; Kinetics; Phencyclidine; Receptors, Cholinergic; Tetracaine; Torpedo; Tubocurarine

1984
The effects of drugs on the incorporation of a conformationally-sensitive, hydrophobic probe into the ion channel of the nicotinic acetylcholine receptor.
    Biochimica et biophysica acta, 1994, Mar-23, Volume: 1190, Issue:2

    Topics: Anesthetics, Local; Animals; Azirines; Binding Sites; Bungarotoxins; Chlorpromazine; Dibucaine; Iodine Radioisotopes; Ion Channels; Molecular Conformation; Receptors, Nicotinic; Tetracaine; Torpedo; Ultraviolet Rays

1994
Secondary structure of the nicotinic acetylcholine receptor: implications for structural models of a ligand-gated ion channel.
    Biochemistry, 1994, Jun-21, Volume: 33, Issue:24

    Topics: Animals; Carbachol; Electric Organ; Ion Channel Gating; Ion Channels; Models, Molecular; Protein Conformation; Protein Structure, Secondary; Receptors, Nicotinic; Spectrometry, Fluorescence; Spectrophotometry, Infrared; Spectroscopy, Fourier Transform Infrared; Tetracaine; Torpedo

1994
Structure of both the ligand- and lipid-dependent channel-inactive states of the nicotinic acetylcholine receptor probed by FTIR spectroscopy and hydrogen exchange.
    Biochemistry, 1995, Nov-21, Volume: 34, Issue:46

    Topics: Animals; Carbachol; Cholesterol; Deuterium; Hydrogen; Hydrogen Bonding; Ion Channels; Lipid Bilayers; Membrane Lipids; Phosphatidic Acids; Phosphatidylcholines; Protein Structure, Secondary; Receptors, Nicotinic; Spectrophotometry; Spectroscopy, Fourier Transform Infrared; Tetracaine; Torpedo

1995
The ion channel of muscle and electric organ acetylcholine receptors: differing affinities for noncompetitive inhibitors.
    Cellular and molecular neurobiology, 1993, Volume: 13, Issue:2

    Topics: Amino Acid Sequence; Animals; Cell Line; Diterpenes; Electric Organ; Ion Channel Gating; Magnesium; Membrane Potentials; Mice; Molecular Sequence Data; Muscle Proteins; Nerve Tissue Proteins; Nicotinic Antagonists; Oocytes; Organ Specificity; Phencyclidine; Recombinant Proteins; Sequence Homology, Amino Acid; Sodium Channels; Tetracaine; Torpedo; Xenopus laevis

1993
Elucidation of biphasic alterations on acetylcholinesterase (AChE) activity and membrane fluidity in the structure-functional effects of tetracaine on AChE-associated membrane vesicles.
    Archives of biochemistry and biophysics, 1998, Mar-01, Volume: 351, Issue:1

    Topics: 1-Propanol; Acetylcholinesterase; Anesthetics, Local; Animals; Calorimetry, Differential Scanning; Cell Membrane; Electric Organ; Ethanol; Fluorescence Polarization; Lipid Bilayers; Liposomes; Membrane Fluidity; Membrane Lipids; Membrane Proteins; Temperature; Tetracaine; Thermodynamics; Torpedo

1998
A structure-based approach to nicotinic receptor pharmacology.
    Molecular pharmacology, 1999, Volume: 55, Issue:2

    Topics: Anesthetics, Local; Animals; Binding Sites; Binding, Competitive; Carbachol; Dibucaine; Lidocaine; Neurotransmitter Agents; Prilocaine; Protein Conformation; Receptors, Nicotinic; Spectroscopy, Fourier Transform Infrared; Tetracaine; Torpedo

1999
Photoaffinity labeling the torpedo nicotinic acetylcholine receptor with [(3)H]tetracaine, a nondesensitizing noncompetitive antagonist.
    Molecular pharmacology, 1999, Volume: 56, Issue:2

    Topics: Animals; Binding Sites; Cell Membrane; Ligands; Nicotinic Antagonists; Photoaffinity Labels; Radioligand Assay; Receptors, Nicotinic; Serine Endopeptidases; Tetracaine; Torpedo; Tritium

1999
Identification of amino acids of the torpedo nicotinic acetylcholine receptor contributing to the binding site for the noncompetitive antagonist [(3)H]tetracaine.
    Molecular pharmacology, 1999, Volume: 56, Issue:2

    Topics: Amino Acids; Animals; Binding Sites; Nicotinic Antagonists; Photoaffinity Labels; Protein Structure, Secondary; Receptors, Nicotinic; Sequence Analysis; Tetracaine; Torpedo; Tritium

1999
Interactions between 3-(Trifluoromethyl)-3-(m-[(125)I]iodophenyl)diazirine and tetracaine, phencyclidine, or histrionicotoxin in the Torpedo series nicotinic acetylcholine receptor ion channel.
    Molecular pharmacology, 2001, Volume: 59, Issue:6

    Topics: Affinity Labels; Amphibian Venoms; Anesthetics, Local; Animals; Azirines; Ceramides; Drug Interactions; Excitatory Amino Acid Antagonists; Iodine Radioisotopes; Membrane Proteins; Phencyclidine; Receptors, Nicotinic; Tetracaine; Torpedo

2001
Allosterically linked noncompetitive antagonist binding sites in the resting nicotinic acetylcholine receptor ion channel.
    Archives of biochemistry and biophysics, 2002, Jul-01, Volume: 403, Issue:1

    Topics: Allosteric Site; Amobarbital; Anesthetics, Local; Animals; Binding Sites; Binding, Competitive; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Modulators; Inhibitory Concentration 50; Ions; Ketamine; Kinetics; Light; Models, Molecular; Phencyclidine; Protein Binding; Protein Conformation; Receptors, Nicotinic; Tetracaine; Torpedo

2002
Lipid-protein interactions and effect of local anesthetics in acetylcholine receptor-rich membranes from Torpedo marmorata electric organ.
    Biochemistry, 2003, Aug-05, Volume: 42, Issue:30

    Topics: Anesthetics, Local; Animals; Benzocaine; Binding, Competitive; Electric Organ; Electron Spin Resonance Spectroscopy; Gangliosides; Hydrophobic and Hydrophilic Interactions; Membrane Proteins; Models, Chemical; Phosphatidylinositols; Phospholipids; Procaine; Receptors, Nicotinic; Spectrometry, Fluorescence; Spin Labels; Stearic Acids; Synaptic Membranes; Tetracaine; Torpedo

2003
Molecular mechanisms and binding site location for the noncompetitive antagonist crystal violet on nicotinic acetylcholine receptors.
    Biochemistry, 2006, Feb-21, Volume: 45, Issue:7

    Topics: Allosteric Regulation; Amobarbital; Animals; Binding Sites; Fluorescent Dyes; Gentian Violet; Ion Channels; Models, Molecular; Nicotinic Agonists; Nicotinic Antagonists; Pentobarbital; Phencyclidine; Protein Binding; Protein Conformation; Quaternary Ammonium Compounds; Receptors, Nicotinic; Temperature; Tetracaine; Thiophenes; Torpedo; Tritium

2006
Lipid composition alters drug action at the nicotinic acetylcholine receptor.
    Molecular pharmacology, 2008, Volume: 73, Issue:3

    Topics: Anesthetics, Local; Animals; Cholesterol; Dose-Response Relationship, Drug; Inhibitory Concentration 50; Kinetics; Lipid Bilayers; Lipids; Phosphatidic Acids; Phosphatidylcholines; Protein Conformation; Receptors, Nicotinic; Spectroscopy, Fourier Transform Infrared; Tetracaine; Torpedo

2008
A photoreactive analog of allopregnanolone enables identification of steroid-binding sites in a nicotinic acetylcholine receptor.
    The Journal of biological chemistry, 2019, 05-10, Volume: 294, Issue:19

    Topics: Animals; Binding Sites; Fish Proteins; Molecular Docking Simulation; Pregnanolone; Receptors, Nicotinic; Steroids; Tetracaine; Torpedo

2019