tetracaine has been researched along with dibucaine in 197 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 150 (76.14) | 18.7374 |
1990's | 24 (12.18) | 18.2507 |
2000's | 13 (6.60) | 29.6817 |
2010's | 10 (5.08) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET | 1 |
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J | 1 |
Carrupt, PA; Guillarme, D; Henchoz, Y; Rudaz, S; Veuthey, JL | 1 |
Batts, TW; Brown, ML; Jones, PJ; Landry, V; Patel, MK; Wang, Y | 1 |
Gozalbes, R; Pineda-Lucena, A | 1 |
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ | 1 |
Brouillette, WJ; Brown, GB; Zha, C | 1 |
Hendrickson, HS | 1 |
Hendrickson, HS; van Dam-Mieras, MC | 1 |
Hellmann, G; Scharinger, B; Suko, J; Winkler, F | 1 |
Jacobson, K; Papahadjopoulos, D; Poste, G; Vail, WJ | 2 |
Büchi, J; Merki, F; Perlia, X | 2 |
Cascella, PJ; DeFrancisco, M; Feldman, S | 1 |
Blanchard, SG; Dunn, SM; Elliott, J; Raftery, MA | 1 |
Kono, T; Suzuki, K | 1 |
Koblin, DD; Lester, HA | 1 |
Dawson, AP; Fulton, DV; Selwyn, MJ | 1 |
Feinstein, MG; Fiekers, J; Fraser, C | 1 |
Nicolson, GL | 1 |
DeStefano, MJ; Rabinovitch, M | 1 |
Landmesser, CM | 1 |
Feinstein, MB; Makriyannis, A; Perrie, S; Sha'afi, RI; Volpi, M | 1 |
Kunze, H; Nahas, N; Traynor, JR; Wurl, M | 1 |
Lee, AG | 1 |
Kunze, H; Traynor, JR | 1 |
Corkedale, S; Katz, AM; Repke, DI; Schwarz, J | 1 |
Nicolson, GL; Poste, G; Smith, JR | 1 |
de Meis, L; Pacheco, AG; Wolosker, H | 1 |
Bridal, TR; Busath, D | 1 |
Fujiwara, Y; Kuroda, Y; Nakagawa, T; Wakita, M | 1 |
Hishinuma, S; Uchida, MK | 2 |
García-Martín, E; González-Cabanillas, S; Gutiérrez-Merino, C | 1 |
Cragoe, EJ; Hayakawa, M; Hori, T; Ito, F; Nango, M; Oku, N; Shibamoto, S | 1 |
Crăcium, C; Tarba, C | 1 |
Filion, PR; Khazen, T; Lavoie, PA | 1 |
Diez, A; Escudero, B; Gutiérrez-Merino, C; Laynez, J; Molina, A | 1 |
Harada, S; Yanagi, K | 1 |
Enyeart, JJ; Hinkle, PM; Phillips, WJ | 1 |
Kamaya, H; Kaminoh, Y; Ueda, I | 1 |
Hansen, J; Kreilgård, B | 1 |
Ivanov, II; Semin, BK; Tshudinovskich, MN | 1 |
Fischer, T; Hansen, J; Kreilgård, B | 1 |
Bevers, EM; Comfurius, P; Verhallen, PF; Zwaal, RF | 2 |
Balgavý, P; Ondrias, K; Stasko, A | 1 |
Béderová, E; Pisková, L; Racanský, V | 1 |
Nozawa, Y; Umeki, S | 1 |
Attwood, D; Fletcher, P | 1 |
Lavoie, PA; Mekhail-Ishak, K; Sharkawi, M | 1 |
Garcia-Martin, E; Gutiérrez-Merino, C | 1 |
Adade, AB; O'Brien, KL; Vanderkooi, G | 1 |
Abe, K; Mashimo, T; Yoshiya, I | 1 |
Fujita, I; Irita, K; Minakami, S; Takeshige, K; Yoshitake, J | 1 |
Deuticke, B; Haest, CW; Plasa, G; Schneider, E | 1 |
Abdelaziz, AA; el-Nakeeb, MA | 1 |
Beck, MH; Holden, A | 1 |
Ferrell, JE; Huestis, WH; Mitchell, KT | 1 |
Escudero, B; Gutiérrez-Merino, C | 1 |
Fujiwara, Y; Kuroda, Y | 1 |
Kontani, H; Koshiura, R | 1 |
Akerman, SB | 1 |
Feinstein, MB; Paimre, M | 1 |
Aledort, LM; Niemetz, J | 1 |
Mertens, W; Steinbach, H; Zipf, HF | 1 |
Dereymaeker, A; Sorel, L | 1 |
Libelius, R; Sonesson, B; Stamenović, BA; Thesleff, S | 1 |
Cerbón, J | 1 |
Bohn, E; Kunze, H; Vogt, W | 1 |
Gotterer, GS | 1 |
Swamy, VC; Triggle, DJ | 1 |
Daly, JW; Huang, M; Shimizu, H; Takenoshita, M | 1 |
Camu, F | 1 |
Beaudoin, AR; Dunnigan, J; Marois, C; Morisset, J | 1 |
Farhadieh, B; Hall, NA; Hammarlund, ER | 1 |
Fisher, PA; Luduena, FP | 1 |
Fink, BR; Kenny, GE; Simpson, WE | 2 |
Moran, JF; Swamy, VC; Triggle, DJ | 1 |
Eichberg, J; Hauser, G | 1 |
Papahadjopoulos, D | 2 |
Foldes, FF; Smith, JC | 1 |
Corssen, G | 1 |
Black, RG; Bonica, JJ | 1 |
Singer, MA | 1 |
Becker, CE | 1 |
Changeux, JP; Weber, M | 1 |
Belobrov, VM; Komissarov, IV; Makarova, LE; Rudenko, NZ; Titov, EV | 1 |
Dure-Smith, P; Freundlich, IM | 1 |
Foster, B; Young, TM | 1 |
Defalque, RJ | 1 |
Johnson, EM; Ludlum, DB | 1 |
Montoya, RG | 1 |
Oki, S | 1 |
Komissarov, IV; Makarova, LE; Rudenko, NZ | 1 |
Bickers, WM | 1 |
Standaert, F; Usubiaga, JE | 1 |
Andersen, NB | 1 |
Fuchs, F; Wilcox, WD | 1 |
Beck, IT; Dinda, PK | 1 |
Iwata, Y; Kimura, F; Nakamura, T; Takamura, M; Tsunoo, M | 1 |
Bangham, AD; Miller, N; Standish, MM | 1 |
Blaustein, MP; Goldman, DE | 1 |
Bridenbaugh, LD; Moore, DC | 1 |
Daniel, EE; Wolowyk, M | 1 |
Ishikawa, F; Kitahara, T | 1 |
Hersh, L | 1 |
Bond, GH; Hudgins, PM | 1 |
Nyquist-Battie, C; Sidek, HM; Vanderkooi, G | 1 |
Lavoie, PA | 1 |
Chazotte, B; Chignell, D; Vanderkooi, G | 1 |
Coller, BS | 1 |
Allison, WS; Goldenberg, TM; Laikind, PK | 1 |
Adade, AB; Chignell, D; Vanderkooi, G | 1 |
Bussereau, F; Genty, N | 1 |
Brodal, B; Røed, A | 1 |
Hidaka, H; Tanaka, T | 1 |
Chazotte, B; Vanderkooi, G | 1 |
Ito, S; Pastan, I; Richert, N | 1 |
Balgavý, P; Horváth, LI; Ondrias, K; Stolc, S | 1 |
Chang, HH; Galton, N; Lampe, RA; Magruder, CD; Michaelis, EK; Michaelis, ML | 1 |
Fazly Bazaz, BS; Salt, WG | 3 |
Bradford, P; Marinetti, GV | 1 |
Harris, EJ; Jackson, MJ; Jones, DA | 1 |
Ohki, S | 1 |
Ieiri, M; Oura, K; Shinohara, M | 1 |
Haring, R; Kloog, Y | 1 |
Maloney, MS | 1 |
Covino, BG; Feldman, HS | 1 |
Berg, T; Holte, K; Tolleshaug, H | 1 |
Canellakis, ES; Chen, KY; Kyriakidis, DA | 1 |
Leyko, W; Surewicz, WK | 1 |
Glass, F; Kadowitz, PJ; Lippton, H | 1 |
Concepcion, MA; Covino, BG; Francis, DM; Rocco, AG; Wark, JA | 1 |
Mori, T | 1 |
Cullis, PR; Hornby, AP | 1 |
Bell, FP | 1 |
Minakuchi, R; Mori, T; Nishizuka, Y; Takai, Y; Yu, B | 1 |
Coffe, G; Genna, JM; Pudles, J | 1 |
Stadler, JK; Vaughan, VL | 1 |
Jain, MK; Singer, MA | 1 |
McCarthy, MP; Moore, MA | 1 |
Jones, EW; Manning, R | 1 |
Muteki, T; Sugiyama, K | 1 |
Clark, DT; Lewis, DA; Pankhurst, CL | 1 |
Andoh, K; Haga, S; Hashimoto, Y; Koga, Y; Momose, K; Shima, T | 1 |
Masuda, R; Yokoyama, K | 1 |
Andriamainty, F; Balgavý, P; Filípek, J; Kovács, P | 1 |
Anteneodo, C; Louro, SR; Wajnberg, E | 1 |
Bircher, AJ; Messmer, SL; Rufli, T; Surber, C | 1 |
Agafonov, AV; Opanasenko, VK; Semenova, GA | 1 |
Borgo, M; Luzzati, V; Márquez, G; Mateu, L; Morán, O; Padrón, R; Vonasek, E | 1 |
Turner, T; Weightman, W | 1 |
Baenziger, JE; Ryan, SE | 1 |
Inoue, T; Masuda, R; Yokoyama, K | 1 |
Irita, K; Kansha, M; Nagata, T; Takahashi, S | 1 |
Mutlu, Z; Tulga, F | 1 |
Abadir, AR; Gintautas, J; Yaman, M | 1 |
Hino, Y; Ikeda, N; Kudo, K; Tsuji, A | 1 |
Benoit, E; Charpentier, G; Kado, R; Luzzati, V; Mateu, L; Vachette, P | 1 |
Hino, Y; Ikeda, N; Inoue, H; Kudo, K; Takahashi, S | 1 |
Amador Kane, S; Floyd, SD | 1 |
Chakrabarti, A; Mondal, M | 1 |
BABICHEV, VA | 3 |
BARTELS, E; HIGMAN, HB; ROSENBERG, P | 1 |
ZAKHAREVSKII, AS | 1 |
ADRIANI, J; ZEPERNICK, R | 2 |
EARLE, RW | 1 |
ADRIANI, J | 1 |
KOMROWER, GM | 1 |
WENDL, HK | 1 |
ANDERSEN, NB; GRAVENSTEIN, JS | 1 |
Chattopadhyay, A; Kalipatnapu, S | 1 |
Hidaka, N; Ibusuki, S; Katsuki, H; Takasaki, M; Tateyama, S; Yano, T | 1 |
Ball, C; Westhorpe, R | 1 |
Boonme, P; Junyaprasert, VB; Krauel, K; Rades, T; Songkro, S | 1 |
Boonme, P; Junyaprasert, VB; Rades, T; Wurster, DE | 1 |
ADRIANI, J; BRAY, KE; KATZ, S | 1 |
EDGE, ND; SOMERS, GF | 1 |
Bach, D; Miller, IR; Sela, B | 1 |
HILL, EF | 1 |
Brinca, A; Cabral, R; Gonçalo, M | 1 |
Huster, D; Scheidt, HA; Weizenmann, N | 1 |
Avranas, A; Horovitz, O; Mocanu, A; Pasca, RD; Tomoaia, G; Tomoaia-Cotisel, M | 1 |
Chakrabarti, A; Patra, M | 1 |
Schmutz, JL | 1 |
Saito, S; Tobe, M | 1 |
Brás, S; Lobo, L; Matos-Pires, E; Pina-Trincão, D | 1 |
3 review(s) available for tetracaine and dibucaine
Article | Year |
---|---|
Studies on the mechanism of action of local anesthetics with phospholipid model membranes.
Topics: Anesthetics, Local; Calcium; Cocaine; Dibucaine; Diffusion; Electric Conductivity; Lidocaine; Macromolecular Substances; Magnetic Resonance Spectroscopy; Membrane Potentials; Membranes, Artificial; Models, Biological; Permeability; Phospholipids; Procaine; Sodium; Surface Properties; Tetracaine | 1972 |
Allergic contact dermatitis from lignocaine: report of 29 cases and review of the literature.
Topics: Adolescent; Adult; Aged; Aged, 80 and over; Anesthetics, Local; Bupivacaine; Carticaine; Child; Child, Preschool; Cross Reactions; Dermatitis, Allergic Contact; Diagnosis, Differential; Dibucaine; Female; Humans; Lidocaine; Male; Mepivacaine; Middle Aged; Patch Tests; Prilocaine; Tetracaine | 1998 |
History of T-cain: a local anesthetic developed and manufactured in Japan.
Topics: Administration, Topical; Anesthesia, Local; Anesthesia, Spinal; Anesthetics, Local; Dibucaine; Humans; Japan; Neurotoxicity Syndromes; Tetracaine | 2015 |
2 trial(s) available for tetracaine and dibucaine
Article | Year |
---|---|
A clinical double-blind study of dibucaine and tetracaine in spinal anesthesia.
Topics: Adult; Aged; Anesthesia, Spinal; Dibucaine; Double-Blind Method; Humans; Hypotension; Middle Aged; Random Allocation; Tetracaine; Time Factors | 1982 |
Prophylactic application of an intra-alveolar socket medicament to reduce postextraction complications in HIV-seropositive patients.
Topics: Acquired Immunodeficiency Syndrome; Adult; Anesthetics, Local; Aspirin; Chlortetracycline; Dental Care for Chronically Ill; Dibucaine; Drug Combinations; Dry Socket; Female; HIV Infections; HIV Seropositivity; Humans; Male; Middle Aged; Occlusive Dressings; Surgical Wound Infection; Tetracaine; Tooth Extraction; Wound Healing | 1994 |
192 other study(ies) available for tetracaine and dibucaine
Article | Year |
---|---|
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium | 1985 |
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase | 2008 |
High-throughput log P determination by ultraperformance liquid chromatography: a convenient tool for medicinal chemists.
Topics: Chemical Phenomena; Chemistry, Pharmaceutical; Chemistry, Physical; Chromatography, Liquid; Mathematics; Pharmaceutical Preparations; Software | 2008 |
Ligand-based design and synthesis of novel sodium channel blockers from a combined phenytoin-lidocaine pharmacophore.
Topics: Drug Design; Expert Systems; Inhibitory Concentration 50; Lidocaine; Ligands; Models, Molecular; Phenytoin; Sodium Channel Blockers; Structure-Activity Relationship | 2009 |
QSAR-based solubility model for drug-like compounds.
Topics: Databases, Factual; Models, Molecular; Pharmaceutical Preparations; Quantitative Structure-Activity Relationship; Solubility; Water | 2010 |
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship | 2012 |
A highly predictive 3D-QSAR model for binding to the voltage-gated sodium channel: design of potent new ligands.
Topics: Ligands; Models, Molecular; Quantitative Structure-Activity Relationship; Voltage-Gated Sodium Channels | 2014 |
The penetration of local anesthetics into phosphatidylcholine monolayers.
Topics: 4-Aminobenzoic Acid; Anesthetics, Local; Biological Transport; Dibucaine; Kinetics; Lidocaine; Membranes, Artificial; Models, Biological; Permeability; Phosphatidylcholines; Procaine; Structure-Activity Relationship; Tetracaine; Triglycerides | 1976 |
Local anesthetic inhibition of pancreatic phospholipase A2 action on lecithin monolayers.
Topics: 4-Aminobenzoic Acid; Anesthetics, Local; Calcium; Dibucaine; Kinetics; Lidocaine; Membranes, Artificial; Models, Biological; Pancreas; Phosphatidylcholines; Phospholipases; Procaine; Spectrophotometry, Ultraviolet; Surface Properties; Tetracaine | 1976 |
Aspects of the mechanism of action of local anesthetics on the sarcoplasmic reticulum of skeletal muscle.
Topics: Adenosine Diphosphate; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Calcium; Dibucaine; Dose-Response Relationship, Drug; Enzyme Activation; In Vitro Techniques; Kinetics; Lidocaine; Muscles; Phosphoproteins; Procaine; Rabbits; Sarcoplasmic Reticulum; Tetracaine | 1976 |
Effects of local anesthetics on membrane properties. II. Enhancement of the susceptibility of mammalian cells to agglutination by plant lectins.
Topics: Agglutination; Anesthetics, Local; Animals; Binding Sites, Antibody; Cell Line; Cell Membrane; Cell Transformation, Neoplastic; Cells, Cultured; Colchicine; Concanavalin A; Cricetinae; Cytochalasin B; Dibucaine; Dose-Response Relationship, Drug; Freeze Fracturing; Lectins; Mice; Mice, Inbred BALB C; Polarography; Polyomavirus; Procaine; Proteins; Simian virus 40; Temperature; Tetracaine | 1975 |
[Relationship between the physico-chemical properties, the chemical reactivity and the local anesthetic effect. 32. 2: The binding capacity of structural protein (wool) for local anesthetics].
Topics: Adsorption; Anesthetics, Local; Animals; Benzoates; Dibucaine; Hydrogen-Ion Concentration; Keratins; Procaine; Protein Binding; Proteins; Structure-Activity Relationship; Tetracaine; Wool | 1975 |
Activity of local anesthetic agents in goldfish.
Topics: Anesthetics, Local; Animals; Cyprinidae; Dibucaine; Goldfish; Hydrogen-Ion Concentration; Kinetics; Lidocaine; Procaine; Solubility; Structure-Activity Relationship; Tetracaine | 1975 |
Specific binding of perhydrohistrionicotoxin to Torpedo acetylcholine receptor.
Topics: Acetylcholine; Amphibian Venoms; Animals; Binding, Competitive; Dibucaine; Electric Organ; Fishes; Kinetics; Parasympatholytics; Receptors, Cholinergic; Tetracaine | 1979 |
Internalization and degradation of fat cell-bound insulin. Separation and partial characterization of subcellular vesicles associated with iodoinsulin.
Topics: Adipose Tissue; Animals; Chloroquine; Dibucaine; Immunoassay; Insulin; Iodine Radioisotopes; Kinetics; Lidocaine; Lysosomes; Male; Procaine; Rats; Receptor, Insulin; Subcellular Fractions; Tetracaine | 1979 |
Voltage-dependent and voltage-independent blockade of acetylcholine receptors by local anesthetics in Electrophorus electroplaques.
Topics: Acetylcholine; Anesthetics, Local; Animals; Benzocaine; Chlorpromazine; Dibucaine; Electric Conductivity; Electric Organ; Electrophorus; In Vitro Techniques; Kinetics; Lidocaine; Membrane Potentials; Procaine; Receptors, Cholinergic; Receptors, Nicotinic; Tetracaine | 1979 |
Inhibition of Ca2+ efflux from mitochondria by nupercaine and tetracaine.
Topics: Animals; Biological Transport, Active; Brain; Calcium; Cell-Free System; Dibucaine; Mitochondria; Mitochondria, Liver; Rats; Ruthenium Red; Tetracaine | 1979 |
An analysis of the mechanism of local anesthetic inhibition of platelet aggregation and secretion.
Topics: Adenosine Diphosphate; Animals; Blood Platelets; Calcimycin; Calcium; Calcium Radioisotopes; Collagen; Depression, Chemical; Dibucaine; In Vitro Techniques; Platelet Aggregation; Serotonin; Tetracaine; Thrombin | 1976 |
Cell shape changes and transmembrane receptor uncoupling induced by tertiary amine local anesthetic.
Topics: Agglutination; Anesthetics, Local; Calcimycin; Calcium; Cell Line; Cell Membrane; Cells, Cultured; Concanavalin A; Dibucaine; Lasalocid; Microtubules; Procaine; Receptors, Concanavalin A; Receptors, Drug; Tetracaine | 1976 |
Cell shape changes induced by cationic anesthetics.
Topics: Anesthetics, Local; Animals; Benzocaine; Cell Adhesion; Cell Fusion; Cell Membrane; Cell Movement; Chlorpromazine; Culture Media; Dibucaine; Edetic Acid; Egtazic Acid; Female; HEPES; Lidocaine; Macrophages; Mice; Prilocaine; Pseudopodia; Structure-Activity Relationship; Tetracaine; Tetrodotoxin; Tromethamine | 1976 |
More on baricity.
Topics: Anesthesia, Spinal; Densitometry; Dibucaine; Humans; Tetracaine | 1977 |
Mechanisms of local anesthetic action on the permeability of erythrocytes, leukocytes, and liposomes containing the erythrocyte anion channel protein.
Topics: Alcohols; Anesthetics, Local; Animals; Blood Proteins; Cell Membrane Permeability; Dibucaine; Erythrocytes; Female; Humans; In Vitro Techniques; Liposomes; Male; Neutrophils; Rabbits; Sulfates; Tetracaine | 1977 |
Effects of local anaesthetics on phospholipases.
Topics: Anesthetics, Local; Calcium; Chlorpromazine; Cocaine; Dibucaine; Humans; Kinetics; Lidocaine; Male; Phospholipases; Procaine; Semen; Snake Venoms; Tetracaine | 1976 |
Interactions between anaesthetics and lipid mixtures. Amines.
Topics: Anesthetics, Local; Benzocaine; Binding Sites; Calcium; Chlorophyll; Dibucaine; Lipids; Membranes, Artificial; Myristic Acids; Neural Conduction; Palmitic Acids; Procaine; Sodium; Temperature; Tetracaine | 1976 |
Local anaesthetics increase susceptibility of untransformed cells to agglutination by concanavalin A.
Topics: Agglutination; Anesthetics, Local; Animals; Binding Sites; Calcium; Cell Line; Cell Transformation, Neoplastic; Concanavalin A; Dibucaine; Fibroblasts; Mice; Mice, Inbred BALB C; Microscopy, Electron; Procaine; Tetracaine | 1975 |
[Relations between the physico-chemical properties, the chemical reactivity and the local anesthetic activity. 32. (Part 1): Binding capacity of a structural protein (wool) to local anesthetics].
Topics: Albumins; Anesthetics, Local; Animals; Binding Sites; Dibucaine; Kinetics; Lipoproteins; Nerve Tissue Proteins; Protein Binding; Protein Conformation; Proteins; Ranvier's Nodes; Receptors, Drug; Structure-Activity Relationship; Tetracaine; Wool | 1975 |
Inhibition of rat liver cholesterol esterase by local anaesthetics.
Topics: Anesthetics, Local; Animals; Carboxylic Ester Hydrolases; Chlorpromazine; Cholesterol; Deoxycholic Acid; Dibucaine; Dose-Response Relationship, Drug; Female; Kinetics; Liver; Oleic Acids; Polyethylene Glycols; Rats; Sterol Esterase; Taurocholic Acid; Tetracaine | 1975 |
Effects of local anaesthetics on calcium transport by canine cardiac microsomes (fragmented sarcoplasmic reticulum).
Topics: Anesthetics, Local; Animals; Biological Transport, Active; Calcium; Dibucaine; Dogs; Heart; In Vitro Techniques; Lidocaine; Microsomes; Myocardium; Oxalates; Procainamide; Sarcoplasmic Reticulum; Tetracaine | 1975 |
Effects of local anesthetics on cell morphology and membrane-associated cytoskeletal organization in BALB/3T3 cells.
Topics: Cell Line; Cell Membrane; Cells, Cultured; Dibucaine; Dose-Response Relationship, Drug; Microtubules; Procaine; Tetracaine | 1976 |
Local anesthetics induce fast Ca2+ efflux through a nonenergized state of the sarcoplasmic reticulum Ca(2+)-ATPase.
Topics: Anesthetics, Local; Animals; Benzocaine; Calcium; Calcium-Transporting ATPases; Dibucaine; Dose-Response Relationship, Drug; Heparin; Kinetics; Muscles; Polyamines; Proadifen; Procaine; Rabbits; Ruthenium Red; Sarcoplasmic Reticulum; Tetracaine | 1992 |
Inhibition of gramicidin channel activity by local anesthetics.
Topics: 4-Aminobenzoic Acid; Anesthetics, Local; Dibucaine; Electric Conductivity; Gramicidin; Ion Channels; Kinetics; Tetracaine | 1992 |
Conformations of dibucaine and tetracaine in small unilamellar phosphatidylcholine vesicles as studied by nuclear Overhauser effects in 1H nuclear magnetic resonance spectroscopy.
Topics: Dibucaine; Lipid Bilayers; Magnetic Resonance Spectroscopy; Molecular Conformation; Molecular Structure; Phosphatidylcholines; Tetracaine | 1992 |
Blockade by the local anaesthetic, tetracaine, of desensitization of Ca-induced Ca release after muscarinic stimulation in smooth muscle.
Topics: Animals; Caffeine; Calcium; Carbachol; Dibucaine; Female; Guinea Pigs; Histamine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Parasympathomimetics; Potassium; Receptors, Histamine H1; Tetracaine | 1991 |
Modulation of calcium fluxes across synaptosomal plasma membrane by local anesthetics.
Topics: Adenosine Triphosphate; Adsorption; Anesthetics, Local; Animals; Ca(2+) Mg(2+)-ATPase; Calcium; Calcium Channels; Carrier Proteins; Cell Membrane; Cell Membrane Permeability; Dibucaine; Kinetics; Lidocaine; Osmotic Pressure; Procaine; Rats; Rats, Inbred Strains; Sodium-Calcium Exchanger; Synaptosomes; Tetracaine | 1990 |
Inhibitory effect of local anesthetics on Na+/H+ antiporter in brush border membrane-reconstituted vesicles.
Topics: Anesthetics, Local; Animals; Antiporters; Carrier Proteins; Dibucaine; In Vitro Techniques; Kidney; Lidocaine; Microvilli; Protons; Rats; Sodium; Tetracaine | 1990 |
A comparative study of the effects of procaine, lidocaine, tetracaine and dibucaine on the functions and ultrastructure of isolated rat liver mitochondria.
Topics: Animals; Dibucaine; Female; Intracellular Membranes; Kinetics; Lidocaine; Membrane Potentials; Microscopy, Electron; Mitochondria, Liver; Oxidative Phosphorylation; Oxygen Consumption; Procaine; Rats; Rats, Inbred Strains; Submitochondrial Particles; Tetracaine | 1990 |
Mechanisms of the inhibition of fast axonal transport by local anesthetics.
Topics: Adenosine Triphosphate; Anesthetics, Local; Animals; Axonal Transport; Dibucaine; Ganglia, Spinal; In Vitro Techniques; Lidocaine; Phosphocreatine; Rana catesbeiana; Reference Values; Sciatic Nerve; Spinal Nerves; Tetracaine | 1989 |
Interaction of the local anesthetics dibucaine and tetracaine with sarcoplasmic reticulum membranes. Differential scanning calorimetry and fluorescence studies.
Topics: Animals; Binding Sites; Ca(2+) Mg(2+)-ATPase; Calcium-Transporting ATPases; Calorimetry, Differential Scanning; Dibucaine; In Vitro Techniques; Intracellular Membranes; Protein Denaturation; Rabbits; Sarcoplasmic Reticulum; Spectrometry, Fluorescence; Temperature; Tetracaine | 1989 |
Destabilization of herpes simplex virus type 1 virions by local anesthetics, alkaline pH, and calcium depletion.
Topics: Anesthetics, Local; Calcium; Capsid; Centrifugation, Density Gradient; Dibucaine; Hydrogen-Ion Concentration; Lidocaine; Magnesium; Simplexvirus; Tetracaine; Virion; Virus Activation | 1989 |
Pituitary thyrotropin-releasing hormone receptors: local anesthetic effects on binding and responses.
Topics: Anesthetics, Local; Animals; Benzocaine; Chlordiazepoxide; Chlorpromazine; Dibucaine; Hydrogen-Ion Concentration; Imipramine; Lidocaine; Pituitary Gland; Procaine; Prolactin; Propranolol; Rats; Receptors, Neurotransmitter; Receptors, Thyrotropin-Releasing Hormone; Tetracaine; Thyrotropin-Releasing Hormone; Trifluoperazine; Verapamil | 1989 |
Differential affinity of charged local anesthetics to solid-gel and liquid-crystalline states of dimyristoylphosphatidic acid vesicle membranes.
Topics: Anesthetics, Local; Chemical Phenomena; Chemistry, Physical; Dibucaine; Glycerophospholipids; Lidocaine; Liposomes; Mathematics; Phosphatidic Acids; Procaine; Temperature; Tetracaine; Thermodynamics | 1989 |
Aspects of pharmaceutical and chemical standardization of patch test materials.
Topics: Acrolein; Acyclic Monoterpenes; Allergens; Benzocaine; Cellulose; Dermatitis, Contact; Dibucaine; Eugenol; Humans; Patch Tests; Pharmaceutical Vehicles; Povidone; Propanols; Quality Control; Skin Tests; Terpenes; Tetracaine; Thiazoles | 1989 |
Local anesthetics-induced inhibition of chloroplast electron transport.
Topics: Anesthetics, Local; Benzocaine; Chlorophyll; Chloroplasts; Dibucaine; Electron Transport; Hydrogen-Ion Concentration; Light; Light-Harvesting Protein Complexes; Mitochondria; Osmolar Concentration; Photosynthesis; Photosynthetic Reaction Center Complex Proteins; Plant Proteins; Tetracaine; Trimecaine | 1989 |
Chemical, pharmaceutical and clinical standardization of the TRUE Test caine mix.
Topics: Adult; Aged; Benzocaine; Cellulose; Chromatography, High Pressure Liquid; Dibucaine; Drug Hypersensitivity; Female; Humans; Male; Middle Aged; Patch Tests; Pharmaceutical Vehicles; Povidone; Reference Standards; Skin Tests; Tetracaine | 1989 |
Correlation between calpain-mediated cytoskeletal degradation and expression of platelet procoagulant activity. A role for the platelet membrane-skeleton in the regulation of membrane lipid asymmetry?
Topics: Blood Coagulation; Blood Platelets; Calcimycin; Calcium; Calpain; Collagen; Contractile Proteins; Cytoskeletal Proteins; Cytoskeleton; Dibucaine; Enzyme Activation; Filamins; Humans; Kinetics; Membrane Lipids; Microfilament Proteins; Myosins; Talin; Tetracaine; Thrombin; Thromboplastin | 1987 |
Spin label study of the perturbation effect of the local anaesthetics tetracaine and dibucaine on synaptosomes at pharmacological concentrations.
Topics: Anesthetics, Local; Animals; Brain; Dibucaine; Electron Spin Resonance Spectroscopy; In Vitro Techniques; Magnetic Resonance Spectroscopy; Membrane Lipids; Rats; Spin Labels; Stearic Acids; Synaptosomes; Temperature; Tetracaine | 1987 |
The influence of local anesthetics on the gel-liquid crystal phase transition in model dipalmitoylphosphatidylcholine membranes.
Topics: 1,2-Dipalmitoylphosphatidylcholine; Anesthetics, Local; Cocaine; Dibucaine; Electron Spin Resonance Spectroscopy; Gels; Lidocaine; Lipid Bilayers; Microscopy, Polarization; Physical Phenomena; Physics; Piperidines; Tetracaine | 1988 |
Effect of local anesthetics on stearoyl-CoA desaturase of Tetrahymena microsomes.
Topics: Anesthetics, Local; Animals; Dibucaine; Fatty Acid Desaturases; Kinetics; Lidocaine; Microsomes; NADPH-Ferrihemoprotein Reductase; Procaine; Propranolol; Stearoyl-CoA Desaturase; Structure-Activity Relationship; Tetracaine; Tetrahymena pyriformis | 1986 |
Self-association of local anaesthetic drugs in aqueous solution.
Topics: Anesthetics, Local; Chemistry, Pharmaceutical; Dibucaine; Light; Micelles; Osmolar Concentration; Radiation; Scattering, Radiation; Solutions; Tetracaine | 1986 |
Biphasic effect of local anesthetics on the adenosine triphosphate-dependent calcium uptake by lysed brain synaptosomes.
Topics: Anesthetics, Local; Animals; Biological Transport, Active; Calcium; Calcium-Transporting ATPases; Cerebral Cortex; Dibucaine; Kinetics; Lidocaine; Male; Rats; Rats, Inbred Strains; Synaptosomes; Tetracaine | 1986 |
Local anesthetics inhibit the Ca2+, Mg2+-ATPase activity of rat brain synaptosomes.
Topics: Anesthetics, Local; Animals; Brain; Ca(2+) Mg(2+)-ATPase; Calcium-Transporting ATPases; Dibucaine; Kinetics; Lidocaine; Procaine; Quinacrine; Rats; Rats, Inbred Strains; Synaptosomes; Tetracaine | 1986 |
Temperature dependence and mechanism of local anesthetic effects on mitochondrial adenosinetriphosphatase.
Topics: Adenosine Triphosphatases; Anesthetics, Local; Animals; Cattle; Chloroform; Chlorpromazine; Dibucaine; Dithionitrobenzoic Acid; Kinetics; Mitochondria, Heart; Tetracaine; Thermodynamics | 1987 |
Dual effect of local anesthetics on the function of excitable rod outer segment disk membrane.
Topics: Anesthetics, Local; Animals; Benzocaine; Bupivacaine; Calcium; Cattle; Dibucaine; Dose-Response Relationship, Drug; Hydrogen-Ion Concentration; In Vitro Techniques; Lidocaine; Light; Photoreceptor Cells; Protons; Rhodopsin; Rod Cell Outer Segment; Tetracaine | 1986 |
Cinchocaine and amethocaine inhibit activation and activity of superoxide production in human neutrophils.
Topics: Blood Proteins; Calcium; Depression, Chemical; Dibucaine; Humans; In Vitro Techniques; NADH, NADPH Oxidoreductases; NADPH Oxidases; Neutrophils; Phosphorylation; Superoxides; Tetracaine | 1986 |
On the regulatory role of the cytoskeleton in the expression of platelet procoagulant activity.
Topics: Blood Coagulation Factors; Blood Platelets; Calcimycin; Calpain; Cytoskeleton; Dibucaine; Dose-Response Relationship, Drug; Electrophoresis, Polyacrylamide Gel; Enzyme Activation; Humans; Phosphatidylserines; Platelet Aggregation; Stimulation, Chemical; Tetracaine | 1986 |
Bacterial cytotoxins, amphotericin B and local anesthetics enhance transbilayer mobility of phospholipids in erythrocyte membranes. Consequences for phospholipid asymmetry.
Topics: Amphotericin B; Anesthetics, Local; Animals; Cytotoxins; Dibucaine; Erythrocyte Membrane; Membrane Lipids; Phosphatidylethanolamines; Phosphatidylserines; Phospholipases A; Phospholipases A2; Phospholipids; Pseudomonas aeruginosa; Rabbits; Rats; Staphylococcus aureus; Tetracaine; Type C Phospholipases | 1986 |
Sporicidal activity of local anaesthetics and their binary combinations with preservatives.
Topics: Anesthetics, Local; Anti-Infective Agents, Local; Aspergillus niger; Bacillus subtilis; Cetrimonium; Cetrimonium Compounds; Chlorhexidine; Cresols; Dibucaine; Ethylene Glycols; Lidocaine; Pharmaceutic Aids; Phenylmercury Compounds; Preservatives, Pharmaceutical; Procaine; Spores, Bacterial; Spores, Fungal; Temperature; Tetracaine | 1987 |
Benzocaine--an unsatisfactory indicator of topical local anaesthetic sensitization for the U.K.
Topics: Benzocaine; Dibucaine; Drug Hypersensitivity; Humans; Patch Tests; Retrospective Studies; Tetracaine | 1988 |
Membrane bilayer balance and platelet shape: morphological and biochemical responses to amphipathic compounds.
Topics: Adult; Anions; Blood Platelets; Cations; Cell Membrane; Chlorpromazine; Dibucaine; Dimyristoylphosphatidylcholine; Erythrocytes; Humans; Lipid Bilayers; Membrane Lipids; Membrane Proteins; Phosphatidic Acids; Phosphatidylcholines; Phosphatidylserines; Phosphorylation; Platelet Activating Factor; Tetracaine; Thrombin | 1988 |
Effects of local anaesthetics on short-term desensitization of guinea-pig taenia caecum to histamine.
Topics: Anesthetics, Local; Animals; Calcium; Cecum; Dibucaine; Female; Guinea Pigs; Histamine; Histamine Antagonists; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Tetracaine | 1987 |
Effects of local anesthetics on the passive permeability of sarcoplasmic reticulum vesicles to Ca2+ and Mg2+.
Topics: Anesthetics, Local; Animals; Calcium; Dibucaine; In Vitro Techniques; Lidocaine; Light; Magnesium; Permeability; Procaine; Rabbits; Sarcoplasmic Reticulum; Scattering, Radiation; Sucrose; Tetracaine | 1987 |
Locations and dynamical perturbations for lipids of cationic forms of procaine, tetracaine, and dibucaine in small unilamellar phosphatidylcholine vesicles as studied by nuclear Overhauser effects in 1H nuclear magnetic resonance spectroscopy.
Topics: Cations; Chemical Phenomena; Chemistry; Dibucaine; Lipid Bilayers; Liposomes; Magnetic Resonance Spectroscopy; Membrane Fluidity; Membrane Lipids; Phosphatidylcholines; Procaine; Structure-Activity Relationship; Tetracaine | 1987 |
The effects of tetrodotoxin, papaverine and verapamil on the increase in the rate of spontaneous afferent discharges induced by local anesthetics from the pulmonary mechanoreceptors of the bullfrog.
Topics: Aconitine; Action Potentials; Anesthetics, Local; Animals; Dibucaine; In Vitro Techniques; Lung; Mechanoreceptors; Neurons, Afferent; Papaverine; Procaine; Rana catesbeiana; Tetracaine; Tetrodotoxin; Verapamil | 1985 |
A methodological study of spinal (subarachnoid) anaesthesia in the rat and the mouse.
Topics: Anesthesia, Spinal; Animals; Bupivacaine; Dibucaine; Dose-Response Relationship, Drug; Lidocaine; Male; Mepivacaine; Mice; Models, Biological; Motor Neurons; Nerve Block; Rats; Rats, Inbred Strains; Tetracaine; Time Factors | 1985 |
Specific reaction of local anesthetics with phosphodiester groups.
Topics: 4-Aminobenzoic Acid; Anesthetics, Local; Chemical Phenomena; Chemistry; Cocaine; Dibucaine; Electrophoresis; Hydrogen-Ion Concentration; Phosphates; Phospholipids; Procaine; Proteins; RNA; Tetracaine | 1966 |
Dissociation of platelet aggregation from clot retraction, potassium loss, and adenosine triphosphatase activity.
Topics: 4-Aminobenzoic Acid; Adenosine Triphosphatases; Anesthetics, Local; Blood Coagulation; Blood Platelets; Cocaine; Dibucaine; Lidocaine; Potassium; Procaine; Tetracaine; Thrombin | 1968 |
[Influence of lipid composition on the binding of local anesthetics to "cephalin"-cholesterol membranes].
Topics: Cholesterol; Dibucaine; Electrochemistry; Electrodes; Membranes, Artificial; Phosphatidylethanolamines; Procaine; Surface Properties; Tetracaine | 1968 |
Lack of depression of the cortical neurons activity by topical anesthetics in the rabbit.
Topics: 4-Aminobenzoic Acid; Anesthetics, Local; Animals; Cerebral Cortex; Cortical Spreading Depression; Dibucaine; Electroencephalography; Lidocaine; Propoxycaine; Rabbits; Seizures; Tetracaine | 1969 |
Denervation-like changes in skeletal muscle after treatment with a local anaesthetic (Marchaine).
Topics: Adenosine Triphosphatases; Anesthetics, Local; Anilides; Animals; Denervation; Dibucaine; Male; Muscular Atrophy; Myofibrils; Pipecolic Acids; Rats; Succinate Dehydrogenase; Tetracaine | 1970 |
NMR evidence for the hydrophobic interaction of local anaesthetics. Possible relation to their potency.
Topics: 4-Aminobenzoic Acid; Anesthetics, Local; Animals; Brain; Calcium; Cattle; Dibucaine; Lysophosphatidylcholines; Magnetic Resonance Spectroscopy; Membranes, Artificial; Molecular Conformation; Phosphatidylcholines; Phosphatidylethanolamines; Phospholipids; Procaine; Structure-Activity Relationship; Surface Properties; Tetracaine; Time Factors; Vibration | 1972 |
Effects of local anaesthetics on prostaglandin biosynthesis in vitro.
Topics: 4-Aminobenzoic Acid; Anesthetics, Local; Animals; Benzocaine; Calcium; Carbon Radioisotopes; Cattle; Chlorpromazine; Chromatography, Thin Layer; Cocaine; Dibucaine; Edetic Acid; Kinetics; Lidocaine; Linoleic Acids; Male; Mepivacaine; Oleic Acids; Phosphatidylethanolamines; Phospholipases; Procaine; Prostaglandins; Seminal Vesicles; Sheep; Snakes; Species Specificity; Tetracaine; Triglycerides | 1974 |
Rat liver D-beta-hydroxybutyrate dehydrogenase. 3. Inhibition by topical anesthetics.
Topics: Acetoacetates; Alcohols; Anesthetics, Local; Animals; Dibucaine; Hydroxybutyrate Dehydrogenase; Kinetics; Lipids; Liver; Mitochondria, Liver; NAD; Phosphatidylcholines; Propranolol; Quinine; Rats; Solubility; Tetracaine | 1969 |
2-Halogenoethylamines and the role of Ca 2+ in adrenergic -receptor activation in the rat vas deferens.
Topics: Animals; Binding Sites; Bromine; Calcium; Diazoxide; Dibucaine; Drug Antagonism; Drug Interactions; Ethylamines; In Vitro Techniques; Male; Methylamines; Muscle Contraction; Naphthalenes; Norepinephrine; Phenethylamines; Phenoxybenzamine; Proadifen; Rats; Receptors, Adrenergic; Receptors, Drug; Synaptic Transmission; Tetracaine; Vas Deferens | 1972 |
Accumulation of adenosine 3',5'-monophosphate in brain slices: interaction of local anaesthetics and depolarizing agents.
Topics: Adenosine; Anesthetics, Local; Animals; Brain; Carbon Isotopes; Cocaine; Cyclic AMP; Dibucaine; Drug Interactions; Guinea Pigs; Histamine; In Vitro Techniques; Lidocaine; Neuromuscular Depolarizing Agents; Norepinephrine; Ouabain; Potassium Chloride; Procaine; Tetracaine | 1973 |
Effects of local anesthetics on glucose-stimulated insulin secretion from rat pancreas in vitro.
Topics: Anesthetics, Local; Animals; Antigens; Bupivacaine; Caffeine; Calcium; Cyclic AMP; Dibucaine; Glucose; In Vitro Techniques; Insulin; Insulin Antibodies; Insulin Secretion; Lidocaine; Mepivacaine; Neutralization Tests; Pancreas; Potassium; Prilocaine; Procaine; Rats; Stimulation, Chemical; Tetracaine | 1973 |
Biochemical reactions involved in pancreatic enzyme secretion. I. Activation of the adenylate cyclase complex.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Amylases; Animals; Bethanechol Compounds; Bucladesine; Cholecystokinin; Dibucaine; Enzyme Activation; Male; Oxygen Consumption; Pancreas; Procaine; Tetracaine | 1974 |
Aggregation of certain medicinal amines in aqueous solutions of their salts.
Topics: Dibucaine; Diphenhydramine; Histamine H1 Antagonists; Osmosis; Potassium Chloride; Procaine; Solutions; Tetracaine; Tripelennamine; Water | 1967 |
Effects of various drugs on the bronchoconstriction produced by transmural stimulation of the perfused guinea pig lung.
Topics: Acetylcholine; Aminobenzoates; Animals; Atropine; Biphenyl Compounds; Bronchi; Cocaine; Cyproheptadine; Dibucaine; Drug Antagonism; Drug Synergism; Electric Stimulation; Ganglionic Blockers; Guinea Pigs; Hexamethonium Compounds; Histamine; Isoproterenol; Lung; Nicotine; Perfusion; Physostigmine; Pilocarpine; Serotonin; Tetracaine; Tremorine | 1967 |
Anesthetic potency compared with intensity of effect on oxygen consumption in monolayer cultures.
Topics: Amobarbital; Anesthetics; Anesthetics, Local; Animals; Barbiturates; Chloroform; Culture Techniques; Dibucaine; Ethers; Ethyl Ethers; Halothane; Lidocaine; Methohexital; Methoxyflurane; Mice; Oxygen Consumption; Phenobarbital; Prilocaine; Procaine; Secobarbital; Tetracaine; Thiamylal; Thiopental | 1968 |
Irreversible antagonism at the adrenergic alpha-receptor: the role of calcium.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Calcium; Calcium Isotopes; Diazoxide; Dibenzylchlorethamine; Dibucaine; In Vitro Techniques; Indomethacin; Male; Naphthalenes; Norepinephrine; Phenethylamines; Phenoxybenzamine; Rats; Sympatholytics; Tetracaine; Vas Deferens | 1970 |
Stimulation by local anesthetics of the metabolism of acidic phospholipids in the rat pineal gland.
Topics: Anesthetics, Local; Animals; Chromatography, Thin Layer; Cocaine; Cytidine; Dibucaine; Dose-Response Relationship, Drug; Lidocaine; Phosphatidic Acids; Phosphatidylinositols; Phospholipids; Phosphorus Radioisotopes; Pineal Gland; Procaine; Propranolol; Rats; Tetracaine; Tritium | 1974 |
The recognition of atypical plasma cholinesterase by relative substrate hydrolysis rate.
Topics: Acetylcholine; Benzoates; Choline; Cholinesterases; Dibucaine; Drug Resistance; Gene Frequency; Genetic Code; Genotype; Heterozygote; Homozygote; Humans; Hydrolysis; Procaine; Tetracaine | 1972 |
Toxic effects of local anaesthetics on human respiratory epithelium.
Topics: Anesthetics, Local; Bronchi; Cilia; Cocaine; Dibucaine; Epithelium; Humans; In Vitro Techniques; Lidocaine; Procaine; Respiratory System; Tetracaine; Time Factors; Trachea | 1973 |
Analgesic blocks.
Topics: Analgesia; Anesthesia, Conduction; Anesthesia, Local; Anesthetics, Local; Autonomic Nerve Block; Bupivacaine; Cranial Nerves; Dibucaine; Ethanol; Ganglia, Autonomic; Humans; Methods; Pain; Pain Management; Phenols; Prognosis; Spinal Nerves; Splanchnic Nerves; Stellate Ganglion; Tetracaine | 1973 |
Interaction of local anesthetics and salicylate with phospholipid membranes.
Topics: Anesthetics, Local; Calcium Chloride; Dibucaine; Electrophoresis; Liposomes; Membranes, Artificial; Phosphatidylcholines; Phospholipids; Salicylates; Sodium Isotopes; Surface Properties; Tetracaine | 1973 |
Cholinesterase genotype and hydrolysis of choline esters, procaine and tetracaine.
Topics: Acetylcholine; Benzoates; Butyrates; Choline; Cholinesterases; Dibucaine; Female; Fluorides; Genetic Variation; Genotype; Humans; Kinetics; Male; Pedigree; Procaine; Spectrophotometry, Ultraviolet; Tetracaine | 1973 |
Binding of Naja nigricollis (3H)alpha-toxin to membrane fragments from Electrophorus and Torpedo electric organs. 3. Effects of local anaesthetics on the binding of the tritiated alpha-neurotoxin.
Topics: Anesthetics, Local; Animals; Antitoxins; Binding Sites; Dibucaine; Electric Organ; Electrophorus; Fishes; In Vitro Techniques; Isoquinolines; Kinetics; Membranes; Parasympatholytics; Prilocaine; Procaine; Protein Binding; Receptors, Cholinergic; Snakes; Tetracaine; Toxins, Biological; Tritium | 1974 |
[Role of carbonyl in the anesthetic effect of local anesthetics].
Topics: Anesthetics, Local; Dibucaine; Lidocaine; Procaine; Spectrum Analysis; Structure-Activity Relationship; Tetracaine | 1972 |
Bronchography: the rational use of premedication and local anesthesia.
Topics: Anesthetics, Local; Atropine; Body Weight; Bronchography; Bronchoscopy; Cocaine; Codeine; Cough; Dibucaine; Humans; Lidocaine; Methods; Pentobarbital; Phosphates; Premedication; Propiophenones; Tetracaine; Vasoconstrictor Agents | 1971 |
Equipment for spinal anaesthesia.
Topics: Anesthesia, Spinal; Dibucaine; Humans; Sterilization; Tetracaine | 1969 |
Retrobulbar block for oculocardiac reflex: duration of protection by common local anesthetics.
Topics: Anesthesia, General; Anesthetics, Local; Animals; Cornea; Dibucaine; Dogs; Eye; Heart; Injections; Lidocaine; Mepivacaine; Miotics; Prilocaine; Procaine; Propoxycaine; Pupil; Reflex; Secobarbital; Tetracaine; Time Factors | 1969 |
Aggregation of local anesthetics in solution.
Topics: Anesthetics, Local; Chemical Phenomena; Chemistry; Colloids; Dibucaine; Hydrochloric Acid; Light; Macromolecular Substances; Polymers; Procaine; Scattering, Radiation; Sodium Chloride; Solutions; Tetracaine; Water | 1969 |
Combined effects of some local anesthetics with sodium benzoate.
Topics: Anesthetics, Local; Animals; Benzoates; Cocaine; Cornea; Dental Pulp; Dibucaine; Drug Synergism; Hydrogen-Ion Concentration; Lidocaine; Procaine; Rabbits; Sodium; Tetracaine | 1970 |
Phospholipid model membranes. 3. Antagonistic effects of Ca2+ and local anesthetics on the permeability of phosphatidylserine vesicles.
Topics: Anesthetics, Local; Calcium; Cocaine; Dibucaine; Electrophoresis; Hydrogen-Ion Concentration; Lidocaine; Membranes, Artificial; Permeability; Phosphatidylethanolamines; Procaine; Sodium Isotopes; Tetracaine | 1970 |
Effect of local anesthetics on phospholipid bilayers.
Topics: Anesthetics, Local; Animals; Anura; Calcium; Cocaine; Dibucaine; Electricity; Electrophysiology; In Vitro Techniques; Membranes, Artificial; Phosphatidylcholines; Phosphatidylethanolamines; Phospholipids; Procaine; Sciatic Nerve; Tetracaine | 1970 |
[Local anesthetizing activity and electron donating properties of anesthetic molecules].
Topics: Anesthetics, Local; Animals; Benzoates; Chelating Agents; Chemistry, Pharmaceutical; Densitometry; Dibucaine; Electrons; Glycerophosphates; Guinea Pigs; Lidocaine; Procaine; Spectrophotometry; Sulfhydryl Compounds; Tetracaine | 1970 |
Epidural analgesia in obstetrics.
Topics: Absorption; Anesthesia, Epidural; Anesthesia, Obstetrical; Cesarean Section; Delivery, Obstetric; Dibucaine; Diffusion; Dura Mater; Episiotomy; Female; Humans; Injections, Spinal; Labor, Obstetric; Lidocaine; Methods; Obstetric Labor Complications; Oxytocin; Pregnancy; Procaine; Tetracaine | 1970 |
The effects of local anesthetics on motor nerve terminals.
Topics: Anesthetics, Local; Animals; Cats; Depression, Chemical; Dibucaine; Leg; Lidocaine; Muscle Contraction; Peripheral Nerves; Procaine; Tetanus; Tetracaine | 1968 |
The effect of local anesthetic and pH on sodium and potassium flux in human red cells.
Topics: Biological Transport, Active; Cell Membrane Permeability; Cocaine; Depression, Chemical; Dibucaine; Erythrocytes; Hematocrit; Hemolysis; Humans; Hydrogen-Ion Concentration; Lidocaine; Potassium; Potassium Isotopes; Procaine; Sodium; Sodium Isotopes; Tetracaine | 1968 |
Depression of oxygen uptake in cell culture by volatile, barbiturate and local anesthetics.
Topics: Anesthesia, Inhalation; Anesthetics; Anesthetics, Local; Animals; Barbiturates; Chloroform; Culture Media; Culture Techniques; Depression, Chemical; Dibucaine; Ethyl Ethers; Halothane; Lidocaine; Methoxyflurane; Mice; Oxygen Consumption; Partial Pressure; Prilocaine; Procaine; Tetracaine | 1969 |
Spinal analgesia.
Topics: Anesthesia, Spinal; Dibucaine; Drug and Narcotic Control; Economics; Humans; Lidocaine; Procaine; Tetracaine | 1969 |
The effect of some local anesthetic compounds on sarcotubular calcium transport.
Topics: Animals; Biological Transport; Calcium; Dibucaine; Lidocaine; Muscle Contraction; Muscles; Procaine; Rabbits; Tetracaine | 1969 |
The effect of local anesthetics on the transmural potential difference of the small intestine of the rat.
Topics: Anesthetics, Local; Animals; Biological Transport; Dibucaine; Electrophysiology; Female; Glucose; Intestinal Absorption; Intestine, Small; Mannitol; Osmolar Concentration; Procaine; Rats; Sodium; Tetracaine | 1969 |
[Mast-cell disruptive effect of local anesthetics and its prevention, with special reference to the effect of aliphatic anesthetics].
Topics: Anesthetics, Local; Animals; Chloral Hydrate; Dibucaine; Ethyl Ethers; Female; Male; Mast Cells; Procaine; Rats; Tetracaine | 1969 |
Cation permeability of phospholipid model membranes: effect of narcotics.
Topics: Alcohols; Cell Membrane Permeability; Chloroform; Cocaine; Dibucaine; Ethyl Ethers; Models, Theoretical; Phosphatidylcholines; Procaine; Tetracaine | 1965 |
Action of anionic and cationic nerve-blocking agents: experiment and interpretation.
Topics: Anesthetics, Local; Calcium; Chemical Phenomena; Chemistry; Detergents; Dibucaine; Lidocaine; Mepivacaine; Phosphatidylethanolamines; Procaine; Tetracaine; Thiopental | 1966 |
Spinal (subarachnoid) block. A review of 11,574 cases.
Topics: Anesthesia, Spinal; Dibucaine; Epinephrine; Humans; Phenylephrine; Procaine; Subarachnoid Space; Tetracaine | 1966 |
The contractile response of the uterus to cocaine.
Topics: Acetylcholine; Animals; Atropine; Calcium; Catecholamines; Cocaine; Dibucaine; Diethylstilbestrol; Epinephrine; Estrogens; Female; Glycerol; Hemolysis; Histamine; In Vitro Techniques; Lidocaine; Muscle Contraction; Norepinephrine; Oxytocin; Phenoxybenzamine; Procaine; Progesterone; Rabbits; Sensory Receptor Cells; Serotonin; Strontium; Tetracaine; Uterus | 1966 |
On the control of spinal anesthetic levels.
Topics: Abdomen; Anesthesia, Spinal; Anesthetics, Local; Dibucaine; Humans; Iodine Radioisotopes; Solutions; Tetracaine | 1967 |
The interaction of local anesthetics with lecithin monolayers.
Topics: Anesthetics, Local; Dibucaine; Ephedrine; Phosphatidylcholines; Procaine; Quinine; Surface Tension; Tetracaine | 1967 |
Inhibition of dog kidney Na+, K+-ATPase activity by procaine, tetracaine and dibucaine.
Topics: 4-Nitrophenylphosphatase; Adenosine Triphosphatases; Animals; Cation Transport Proteins; Dibucaine; Dogs; Kidney; Kinetics; Potassium; Procaine; Sodium; Sodium-Potassium-Exchanging ATPase; Tetracaine | 1984 |
Inhibition of synaptosomal enzymes by local anesthetics.
Topics: Adenosine Triphosphatases; Anesthetics, Local; Animals; Ca(2+) Mg(2+)-ATPase; Cerebral Cortex; Cholinesterase Inhibitors; Dibucaine; Kinetics; Lidocaine; Procaine; Rats; Sodium-Potassium-Exchanging ATPase; Synaptosomes; Tetracaine | 1984 |
Block of fast axonal transport in vitro by the local anesthetics dibucaine and etidocaine.
Topics: Acetanilides; Animals; Axonal Transport; Dibucaine; Etidocaine; Ganglia, Spinal; In Vitro Techniques; Rana catesbeiana; Spinal Nerve Roots; Spinal Nerves; Tetracaine | 1982 |
Further studies on F1-ATPase inhibition by local anesthetics.
Topics: Adenosine Triphosphatases; Anesthetics, Local; Animals; Cattle; Chlorpromazine; Dibucaine; Kinetics; Lidocaine; Mitochondria; Mitochondria, Heart; Oxidative Phosphorylation Coupling Factors; Procainamide; Procaine; Propranolol; Proton-Translocating ATPases; Submitochondrial Particles; Tetracaine | 1982 |
Effects of tertiary amine local anesthetics on von Willebrand factor-dependent platelet function: alteration of membrane reactivity and degradation of GPIb by a calcium-dependent protease(s).
Topics: Anesthetics, Local; Animals; Aspirin; Blood Coagulation Factors; Cattle; Cell Membrane; Depression, Chemical; Dibucaine; Dose-Response Relationship, Drug; Epoprostenol; Glycoproteins; Humans; Lidocaine; Membrane Proteins; Peptide Hydrolases; Platelet Aggregation; Platelet Membrane Glycoproteins; Tetracaine; von Willebrand Factor | 1982 |
On the mechanism of inhibition of the bovine heart F1-ATPase by local anesthetics.
Topics: Anesthetics, Local; Animals; Cattle; Chlorpromazine; Dibucaine; Dicyclohexylcarbodiimide; Kinetics; Mitochondria, Heart; Proton-Translocating ATPases; Structure-Activity Relationship; Tetracaine | 1982 |
Local anesthetics: a new class of partial inhibitors of mitochondrial ATPase.
Topics: Anesthetics, Local; Animals; Cattle; Chlorpromazine; Dibucaine; Dose-Response Relationship, Drug; Hydrogen-Ion Concentration; Kinetics; Lidocaine; Magnesium; Mitochondria, Heart; Proton-Translocating ATPases; Tetracaine | 1984 |
Is cytoskeleton involved in vesicular stomatitis virus reproduction?
Topics: Animals; Cell Line; Colchicine; Cytochalasin B; Cytoskeleton; Dibucaine; Microtubules; Procaine; Tetracaine; Vacuoles; Vesicular stomatitis Indiana virus | 1980 |
Inhibition of sarcolemma ATPases by some membrane-stabilizing drugs.
Topics: Animals; Calcium-Transporting ATPases; Chlorpromazine; Dibucaine; Dose-Response Relationship, Drug; Ouabain; Procaine; Propranolol; Rats; Sarcolemma; Sodium-Potassium-Exchanging ATPase; Tetracaine | 1981 |
Interaction of local anesthetics with calmodulin.
Topics: 2',3'-Cyclic-Nucleotide Phosphodiesterases; Animals; Calcium; Calcium-Binding Proteins; Calmodulin; Cattle; Chickens; Dibucaine; Gizzard, Avian; Kinetics; Lidocaine; Myocardium; Myosin-Light-Chain Kinase; Phosphoric Diester Hydrolases; Protein Kinases; Tetracaine | 1981 |
Cytochrome c oxidase inhibition by anesthetics: thermodynamic analysis.
Topics: Butanols; Dibucaine; Electron Transport Complex IV; Mitochondria, Liver; Protein Conformation; Temperature; Tetracaine; Thermodynamics | 1982 |
Vinculin phosphorylation by the src kinase: inhibition by chlorpromazine, imipramine and local anesthetics.
Topics: Anesthetics, Local; Animals; Caseins; Chlorpromazine; Dibucaine; Imipramine; Muscle Proteins; Phosphatidylglycerols; Phosphorylation; Phosphotransferases; Rats; Tetracaine; Vinculin | 1982 |
A spin label study of the perturbation effect of tertiary amine anesthetics on brain lipid liposomes and synaptosomes.
Topics: Anesthetics, Local; Animals; Cerebral Cortex; Dibucaine; Electron Spin Resonance Spectroscopy; Intracellular Membranes; Lidocaine; Liposomes; Membrane Lipids; Piperidines; Rats; Spin Labels; Synaptosomes; Tetracaine | 1983 |
Effects of amphipathic drugs on L'[3H]glutamate binding to synaptic membranes and the purified binding protein.
Topics: Anesthetics, Local; Animals; Chlorpromazine; Dibucaine; Glutamates; Kinetics; Male; Quinacrine; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Glutamate; Synaptic Membranes; Tetracaine | 1984 |
Local anaesthetic induced turbidity increases: implications of interactions with intact bacterial cells and with subcellular fractions.
Topics: Anesthetics, Local; Cell Membrane; Cytoplasm; Dibucaine; Escherichia coli; Lidocaine; Lipids; Nephelometry and Turbidimetry; Procaine; Spectrophotometry; Subcellular Fractions; Tetracaine | 1983 |
Local anaesthetics as antibacterial agents: effects on cellular respiration and the leakage of cytoplasmic constituents.
Topics: Anesthetics, Local; Cytoplasm; Dibucaine; Escherichia coli; Lidocaine; Oxidoreductases; Oxygen Consumption; Pentoses; Phosphates; Procaine; Tetracaine | 1983 |
Local anaesthetics as antimicrobial agents: structure-action considerations.
Topics: Anesthetics, Local; Anti-Bacterial Agents; Bacillus megaterium; Dibucaine; Escherichia coli; Klebsiella pneumoniae; Lidocaine; Procaine; Pseudomonas aeruginosa; Structure-Activity Relationship; Tetracaine | 1983 |
Trinitrobenzenesulfonic acid and fluorodinitrobenzene: probes to study local anesthetic effects in cell membranes.
Topics: 4-Aminobenzoic Acid; Anesthetics, Local; Dibucaine; Dinitrofluorobenzene; Erythrocyte Membrane; Erythrocytes; Humans; Kinetics; Nitrobenzenes; Phosphatidylethanolamines; Phosphatidylserines; Temperature; Tetracaine; Trinitrobenzenesulfonic Acid | 1981 |
Inhibition of lipid peroxidation in muscle homogenates by phospholipase A2 inhibitors.
Topics: Animals; Chloroquine; Chlorpromazine; Dibucaine; Female; Free Radicals; In Vitro Techniques; Iron; Lipid Peroxides; Mice; Muscles; Phospholipases; Phospholipases A; Phospholipases A2; Procaine; Quinacrine; Tetracaine | 1984 |
Adsorption of local anesthetics on phospholipid membranes.
Topics: Adsorption; Anesthetics, Local; Dibucaine; Electrophoresis; Liposomes; Phosphatidylcholines; Phosphatidylserines; Procaine; Tetracaine | 1984 |
[Acute toxicity tests on prones-pasta].
Topics: Anesthesia, Dental; Anesthetics, Local; Animals; Dibucaine; Ethanolamines; Female; Male; Mice; Tetracaine | 1983 |
Multiple binding sites for phencyclidine on the nicotinic acetylcholine receptor from Torpedo ocellata electric organ.
Topics: Acetylcholine; Animals; Binding Sites; Bungarotoxins; Carbachol; Dibucaine; Electric Organ; Kinetics; Phencyclidine; Receptors, Cholinergic; Tetracaine; Torpedo; Tubocurarine | 1984 |
Pharmacological evidence for cell surface control of oral regeneration in Stentor coeruleus.
Topics: Animals; Calcium; Ciliophora; Dibucaine; Dose-Response Relationship, Drug; Mouth; Phytohemagglutinins; Procaine; Regeneration; Tetracaine; Time Factors | 1980 |
A chronic model for investigation of experimental spinal anesthesia in the dog.
Topics: Anesthesia, Spinal; Anesthetics, Local; Animals; Bupivacaine; Catheters, Indwelling; Dibucaine; Dogs; Female; Half-Life; Injections, Spinal; Lidocaine; Male; Mepivacaine; Methods; Models, Biological; Procaine; Subarachnoid Space; Tetracaine | 1981 |
Effects of local anesthetics and related compounds on the endocytosis and catabolism of asialo-glycoproteins in isolated hepatocytes.
Topics: Anesthetics, Local; Animals; Antineoplastic Agents; Asialoglycoproteins; Cadaverine; Dibucaine; Endocytosis; Glycoproteins; In Vitro Techniques; Kinetics; Liver; Procaine; Rats; Tetracaine | 1982 |
The inhibition of the serum-stimulated increase of ornithine decarboxylase by ionophores and local anesthetics.
Topics: Anesthetics, Local; Animals; Blood; Carboxy-Lyases; Cell Line; Culture Media; Dibucaine; Dose-Response Relationship, Drug; Ionophores; Leukemia, Experimental; Mice; Neuroblastoma; Ornithine Decarboxylase Inhibitors; Tetracaine; Valinomycin | 1982 |
The effect of local anaesthetics on the osmotic fragility of liposomes.
Topics: Anesthetics, Local; Chemical Phenomena; Chemistry; Dibucaine; Liposomes; Membrane Lipids; Osmotic Fragility; Procaine; Tetracaine | 1982 |
Differential effects of local anesthetics and propranolol on arachidonic acid and adenosine 5'-diphosphate-induced aggregation in rabbit platelets.
Topics: Adenosine Diphosphate; Anesthetics, Local; Animals; Arachidonic Acids; Dibucaine; Humans; Lidocaine; Platelet Aggregation; Procaine; Propranolol; Rabbits; Tetracaine | 1980 |
Effects of various membrane phospholipid-interacting drugs on three species of multifunctional protein kinases.
Topics: Animals; Cattle; Chlorpromazine; Dibucaine; Phospholipids; Protein Kinase Inhibitors; Protein Kinases; Rats; Tetracaine | 1981 |
Influence of local and neutral anaesthetics on the polymorphic phase preferences of egg yolk phosphatidylethanolamine.
Topics: Anesthetics; Butanols; Chemical Phenomena; Chemistry; Chlorpromazine; Dibucaine; Ethanol; Lipid Bilayers; Phosphatidylethanolamines; Procaine; Structure-Activity Relationship; Temperature; Tetracaine | 1981 |
Cholesterol esterification by rat adrenal gland. Inhibition by local anesthetics in vitro.
Topics: Acyl Coenzyme A; Acyltransferases; Adrenal Glands; Anesthetics, Local; Animals; Benzocaine; Cholesterol Esters; Dibucaine; Lidocaine; Male; Oleic Acids; Rats; Sterol O-Acyltransferase; Tetracaine | 1981 |
Inhibitory action of chlorpromazine, dibucaine, and other phospholipid-interacting drugs on calcium-activated, phospholipid-dependent protein kinase.
Topics: Animals; Brain; Calcium; Chlorpromazine; Cytosol; Dibucaine; Enzyme Activation; Imipramine; Kinetics; Phentolamine; Phospholipids; Protein Kinases; Rats; Tetracaine; Verapamil | 1980 |
Effects of tertiary amine local anesthetics on the assembly and disassembly of brain microtubules in vitro.
Topics: Animals; Brain; Calcium; Dibucaine; Kinetics; Macromolecular Substances; Microscopy, Electron; Microtubules; Procaine; Rats; Swine; Temperature; Tetracaine; Tubulin | 1980 |
Isolation and genetic characterization of dibucaine-resistant variants of a mouse lymphocytic cell line.
Topics: Animals; Benzocaine; Cell Division; Cell Line; Dibucaine; Dose-Response Relationship, Drug; Drug Resistance; Ethyl Methanesulfonate; Hybrid Cells; Leukemia L5178; Lymphocytes; Mice; Mutation; Procaine; Tetracaine | 1980 |
Interaction of four local anesthetics with phospholipid bilayer membranes: permeability effects and possible mechanisms.
Topics: Anesthetics, Local; Benzocaine; Chemical Phenomena; Chemistry; Dibucaine; Kinetics; Lipid Bilayers; Phosphatidylcholines; Procaine; Sodium; Structure-Activity Relationship; Temperature; Tetracaine | 1980 |
The effects of drugs on the incorporation of a conformationally-sensitive, hydrophobic probe into the ion channel of the nicotinic acetylcholine receptor.
Topics: Anesthetics, Local; Animals; Azirines; Binding Sites; Bungarotoxins; Chlorpromazine; Dibucaine; Iodine Radioisotopes; Ion Channels; Molecular Conformation; Receptors, Nicotinic; Tetracaine; Torpedo; Ultraviolet Rays | 1994 |
Cytotoxic effects of membrane-active agents in human leukaemia cell lines.
Topics: Antineoplastic Agents; Cell Division; Cell Line; Cell Survival; Culture Media, Serum-Free; Dibucaine; Humans; Leukemia, Erythroblastic, Acute; Leukemia, Promyelocytic, Acute; Phospholipid Ethers; Tetracaine; Thymidine; Tumor Cells, Cultured | 1995 |
Local anesthetics depress the calcium current of rat sensory neurons in culture.
Topics: Animals; Bupivacaine; Calcium; Dibucaine; Ganglia, Spinal; Lidocaine; Membrane Potentials; Procaine; Rats; Rats, Sprague-Dawley; Tetracaine | 1994 |
[Combined spinal and epidural analgesia for caesarean section].
Topics: Anesthesia, Epidural; Anesthesia, Obstetrical; Anesthesia, Spinal; Cesarean Section; Dibucaine; Female; Humans; Lidocaine; Pregnancy; Tetracaine | 1993 |
[Density, specific gravity and baricity of various spinal anesthetics and those of normal human cerebrospinal fluid in Japanese].
Topics: Anesthesia, Spinal; Anesthetics, Local; Asian People; Bupivacaine; Cerebrospinal Fluid; Dibucaine; Glucose; Humans; Japan; Lidocaine; Solutions; Specific Gravity; Tetracaine | 1995 |
Effect of local anesthetic [2-(alkyloxy)phenyl]-2-(1-piperidinyl)ethyl esters of carbamic acid on the activity of purified sarcoplasmic reticulum (Ca-Mg)ATPase.
Topics: Anesthetics, Local; Animals; Ca(2+) Mg(2+)-ATPase; Carbamates; Dibucaine; Female; In Vitro Techniques; Piperidines; Rabbits; Sarcoplasmic Reticulum; Structure-Activity Relationship; Tetracaine | 1996 |
Interaction of alkanols and local anesthetics with spin-labeled Ca(2+)-ATPase of sarcoplasmic reticulum vesicles.
Topics: 1-Butanol; Anesthetics, Local; Animals; Butanols; Calcium-Transporting ATPases; Dibucaine; Electron Spin Resonance Spectroscopy; Hydrogen-Ion Concentration; Maleimides; Muscle, Skeletal; Rabbits; Sarcoplasmic Reticulum; Spin Labels; Tetracaine | 1996 |
Delayed-type hypersensitivity to subcutaneous lidocaine with tolerance to articaine: confirmation by in vivo and in vitro tests.
Topics: Adult; Anesthetics, Local; Benzocaine; Bupivacaine; Carticaine; Cross Reactions; Dermatitis, Allergic Contact; Dibucaine; Drug Eruptions; Drug Tolerance; Eczema; Edema; Female; Humans; Hypersensitivity, Delayed; Injections, Subcutaneous; Lidocaine; Lymphocyte Activation; Mepivacaine; Parabens; Patch Tests; Preservatives, Pharmaceutical; Prilocaine; Procaine; Quinolines; Recurrence; Skin Tests; Sulfites; Tetracaine | 1996 |
Light-induced reversible local fusions of thylakoid membranes in the presence of dibucaine or tetracaine.
Topics: Anesthetics, Local; Chloroplasts; Dibucaine; Hydrogen-Ion Concentration; Intracellular Membranes; Light; Membrane Fusion; Microscopy, Electron; Pisum sativum; Tetracaine | 1996 |
The action of local anesthetics on myelin structure and nerve conduction in toad sciatic nerve.
Topics: Action Potentials; Anesthetics, Local; Animals; Biophysical Phenomena; Biophysics; Bufo marinus; Crystallography, X-Ray; Dibucaine; In Vitro Techniques; Lidocaine; Molecular Structure; Myelin Sheath; Neural Conduction; Procaine; Scattering, Radiation; Sciatic Nerve; Tetracaine; X-Rays | 1997 |
A structure-based approach to nicotinic receptor pharmacology.
Topics: Anesthetics, Local; Animals; Binding Sites; Binding, Competitive; Carbachol; Dibucaine; Lidocaine; Neurotransmitter Agents; Prilocaine; Protein Conformation; Receptors, Nicotinic; Spectroscopy, Fourier Transform Infrared; Tetracaine; Torpedo | 1999 |
[Spread of spinal anesthesia with 3 different hyperbaric solutions used in Japan].
Topics: Adult; Aged; Anesthesia, Spinal; Anesthetics, Local; Dibucaine; Female; Glucose; Humans; Injections, Spinal; Male; Middle Aged; Sodium Chloride; Solutions; Specific Gravity; Tetracaine | 1998 |
Dibucaine and tetracaine inhibit the activation of mitogen-activated protein kinase mediated by L-type calcium channels in PC12 cells.
Topics: Anesthetics, Local; Animals; Blotting, Western; Calcium Channels, L-Type; Dibucaine; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Ionomycin; Mitogen-Activated Protein Kinases; PC12 Cells; Phosphorylation; Potassium Chloride; Proto-Oncogene Proteins c-fos; Rats; Tetracaine | 1999 |
Four types of topical anaesthetic agents: evaluation of clinical effectiveness.
Topics: Administration, Topical; Adolescent; Anesthesia, Dental; Anesthetics, Local; Benzocaine; Child; Dibucaine; Evaluation Studies as Topic; Facial Pain; Female; Gels; Humans; Injections; Lidocaine; Lidocaine, Prilocaine Drug Combination; Male; Pain Measurement; Prilocaine; Tetracaine | 1999 |
Modulation of phospholipid metabolism, leukotrienes and prostaglandin synthesis by local anesthetic agents.
Topics: Anesthetics, Local; Animals; Cattle; Chromatography, Thin Layer; Dibucaine; In Vitro Techniques; Leukotrienes; Lysophosphatidylcholines; Microsomes; Phosphatidylcholine-Sterol O-Acyltransferase; Phospholipids; Prostaglandins; Tetracaine | 1999 |
Sensitive and selective determination of tetracaine and its metabolite in human samples by gas chromatography-mass spectrometry.
Topics: 4-Aminobenzoic Acid; Adipose Tissue; Anesthetics, Local; Brain Chemistry; Dibucaine; Gas Chromatography-Mass Spectrometry; Humans; Liver; Muscle, Skeletal; para-Aminobenzoates; Reproducibility of Results; Sensitivity and Specificity; Tetracaine | 2000 |
Physical structure of the excitable membrane of unmyelinated axons: X-ray scattering study and electrophysiological properties of pike olfactory nerve.
Topics: Anesthetics, Local; Animals; Axons; Cell Membrane; Cytoplasm; Dibucaine; Electrophysiology; Esocidae; Microtubules; Molecular Conformation; Myelin Sheath; Olfactory Nerve; Potassium Chloride; Statistics as Topic; Synchrotrons; Temperature; Tetracaine; Tetrodotoxin; Veratridine; X-Ray Diffraction | 2000 |
Blood concentrations of tetracaine and its metabolite following spinal anesthesia.
Topics: 4-Aminobenzoic Acid; Adult; Aged; Anesthesia, Spinal; Anesthetics, Local; Cause of Death; Dibucaine; Forensic Medicine; Gas Chromatography-Mass Spectrometry; Humans; Mepivacaine; Middle Aged; para-Aminobenzoates; Tetracaine | 2001 |
Interaction of local anesthetics with phospholipids in Langmuir monolayers.
Topics: 1,2-Dipalmitoylphosphatidylcholine; Anesthetics, Local; Biophysical Phenomena; Biophysics; Dibucaine; In Vitro Techniques; Membranes, Artificial; Microscopy, Fluorescence; Phospholipids; Tetracaine | 2000 |
The tertiary amine local anesthetic dibucaine binds to the membrane skeletal protein spectrin.
Topics: Amines; Anesthetics, Local; Animals; Circular Dichroism; Dibucaine; Dose-Response Relationship, Drug; Erythrocyte Membrane; Goats; Hot Temperature; Ions; Kinetics; Lidocaine; Procaine; Protein Binding; Protein Structure, Tertiary; Spectrin; Spectrometry, Fluorescence; Temperature; Tetracaine; Thermodynamics; Tryptophan; Ultraviolet Rays | 2002 |
[Comparative effects of novocaine, dicaine, and sovcaine on blood circulation and respiration in cats and rabbits].
Topics: Anesthetics; Anesthetics, Local; Animals; Blood Pressure; Blood Pressure Determination; Cats; Dibucaine; Plethysmography; Procaine; Rabbits; Respiration; Tetracaine | 1956 |
[Comparative characteristics of the terminal stage of anesthesia with certain local anesthetics; novocaine, cocaine, dicaine, and sovcaine].
Topics: Anesthesia; Anesthetics; Anesthetics, Local; Cardiovascular Agents; Cocaine; Dibucaine; Humans; Procaine; Tetracaine | 1956 |
[Effect of novocaine, dicaine and sovcaine on the system; comparative experimental research].
Topics: Anesthetics; Anesthetics, Local; Dibucaine; Procaine; Tetracaine | 1956 |
The active structure of local anesthetics. Effects on electrical and cholinesterase activity.
Topics: Acetylcholinesterase; Anesthetics; Anesthetics, Local; Cocaine; Dibucaine; Electricity; Tetracaine | 1963 |
[Effect of serotonin and some indole derivatives on the local anesthetic activity of cocaine, novocain, dicaine and sovcaine].
Topics: Analgesia; Anesthesia; Anesthesia and Analgesia; Anesthesia, Local; Anesthetics; Anesthetics, Local; Cocaine; Dibucaine; Procaine; Serotonin; Tetracaine | 1962 |
SOME RECENT STUDIES ON THE CLINICAL PHARMACOLOGY OF LOCAL ANESTHETICS OF PRACTICAL SIGNIFICANCE.
Topics: Adjuvants, Anesthesia; Anesthetics; Anesthetics, Local; Cocaine; Dibucaine; Humans; Lidocaine; Metabolism; Pharmacology; Procaine; Tetracaine | 1963 |
FACTORS INVOLVED IN SELECTION OF A LOCAL ANESTHETIC.
Topics: Anesthesia, Local; Anesthetics; Anesthetics, Local; Cats; Cocaine; Dibucaine; Guinea Pigs; Mice; Procaine; Research; Tetracaine; Toxicology | 1963 |
CLINICAL EFFECTIVENESS OF DRUGS USED FOR TOPICAL ANESTHESIA.
Topics: Anesthesia, Local; Anesthetics; Anesthetics, Local; Benzocaine; Cocaine; Dibucaine; Electric Stimulation; Humans; Lidocaine; Lip; Mepivacaine; Mucous Membrane; Palate; Pharmacology; Procaine; Sympathomimetics; Tetracaine; Tongue; Treatment Outcome; Tripelennamine | 1964 |
SOME ASPECTS OF THE PHARMACOLOGY OF LOCAL ANESTHETICS OF CLINICAL IMPORTANCE.
Topics: Anesthetics; Anesthetics, Local; Cardiovascular Agents; Dibucaine; Lidocaine; Mepivacaine; Pharmacology; Procaine; Tetracaine; Toxicology | 1964 |
TO-DAY'S DRUGS. LOCAL ANALGESICS.
Topics: Analgesia; Analgesics; Dibucaine; Lidocaine; Pain; Pharmacology; Procaine; Tetracaine; Toxicology | 1964 |
PERIDURAL ANESTHESIA TECHNIQUES AND LOCAL ANESTHETIC AGENTS.
Topics: Anesthesia, Epidural; Anesthesia, Local; Anesthesia, Spinal; Anesthetics; Anesthetics, Local; Dibucaine; Humans; Lidocaine; Procaine; Tetracaine | 1964 |
EFFECTS OF LOCAL ANESTHETICS ON SODIUM AND POTASSIUM IN HUMAN RED CELLS.
Topics: Anesthetics, Local; Cocaine; Computers, Analog; Dibucaine; Electronic Data Processing; Erythrocytes; Hemolysis; Humans; Ions; Lidocaine; Metabolism; Pharmacology; Potassium; Procaine; Research; Sodium; Tetracaine | 1965 |
Interaction of serotonin1A receptors from bovine hippocampus with tertiary amine local anesthetics.
Topics: Amines; Anesthetics, Local; Animals; Binding Sites; Binding, Competitive; Cattle; Cell Membrane; Cholesterol; Dibucaine; Dose-Response Relationship, Drug; Hippocampus; Lidocaine; Ligands; Membrane Fluidity; Membrane Lipids; Molecular Structure; Neurons; Procaine; Receptor, Serotonin, 5-HT1A; Serotonin Antagonists; Serotonin Receptor Agonists; Subcellular Fractions; Tetracaine | 2004 |
[Glucose attenuating local anesthetic-induced hemolysis].
Topics: Anesthetics, Local; Dibucaine; Dose-Response Relationship, Drug; Erythrocyte Membrane; Glucose; Hemolysis; Humans; In Vitro Techniques; Lidocaine; Neurotoxicity Syndromes; Tetracaine | 2004 |
Local anaesthetics--Nupercaine and Amethcaine.
Topics: Anesthesia, Spinal; Anesthetics, Local; Dibucaine; History, 20th Century; Humans; Tetracaine | 2004 |
Transdermal delivery of hydrophobic and hydrophilic local anesthetics from o/w and w/o Brij 97-based microemulsions.
Topics: 1-Butanol; Administration, Cutaneous; Anesthetics, Local; Calorimetry, Differential Scanning; Dibucaine; Electric Conductivity; Emulsions; Epidermis; Humans; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; In Vitro Techniques; Lidocaine; Molecular Weight; Palmitates; Permeability; Plant Oils; Polyethylene Glycols; Skin Absorption; Tetracaine; Viscosity; Water | 2007 |
Aerosol OT microemulsions as carriers for transdermal delivery of hydrophobic and hydrophilic local anesthetics.
Topics: 1-Butanol; Administration, Cutaneous; Anesthetics, Local; Calorimetry, Differential Scanning; Chromatography, High Pressure Liquid; Dibucaine; Dioctyl Sulfosuccinic Acid; Drug Carriers; Electric Conductivity; Emulsions; Epidermis; Humans; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; In Vitro Techniques; Lidocaine; Palmitates; Permeability; Refractometry; Skin Absorption; Surface-Active Agents; Tetracaine; Viscosity | 2008 |
The effect of epinephrine, ephedrine and neosynephrine on the duration of spinal anesthesia with nupercaine and pontocaine; preliminary report.
Topics: Adrenal Cortex Hormones; Anesthesia, Spinal; Dibucaine; Ephedrine; Epinephrine; Phenylephrine; Tetracaine | 1948 |
Comparative activities of amethocaine, cinchocaine and procaine.
Topics: Anesthesia; Anesthesiology; Anesthetics, Local; Dibucaine; Humans; Procaine; Tetracaine | 1947 |
Thermotropic properties of brain lipids in the presence and absence of local anesthetics.
Topics: Anesthetics, Local; Animals; Brain Chemistry; Calorimetry, Differential Scanning; Cattle; Chemical Phenomena; Chemistry, Physical; Dibucaine; Hot Temperature; Lipids; Tetracaine; Time Factors | 1980 |
Amethocaine or nupercaine.
Topics: Anesthesia; Anesthesiology; Dibucaine; Tetracaine | 1947 |
Contact allergy to local anaesthetics-value of patch testing with a caine mix in the baseline series.
Topics: Adult; Anesthetics, Local; Benzocaine; Cross Reactions; Dermatitis, Allergic Contact; Dibucaine; Female; Humans; Male; Middle Aged; Patch Tests; Tetracaine; Young Adult | 2013 |
Interaction of local anesthetics with lipid bilayers investigated by ¹H MAS NMR spectroscopy.
Topics: Anesthetics, Local; Cell Membrane; Dibucaine; Hydrophobic and Hydrophilic Interactions; Lidocaine; Lipid Bilayers; Magnetic Resonance Spectroscopy; Procaine; Tetracaine | 2012 |
Selective effect of procaine, tetracaine and dibucaine on gold nanoparticles.
Topics: Anesthetics, Local; Dibucaine; Gold; Metal Nanoparticles; Microscopy, Electron, Transmission; Procaine; Static Electricity; Tetracaine | 2012 |
Differential interactions of two local anesthetics with phospholipid membrane and nonerythroid spectrin: Localization in presence of cholesterol and ganglioside, GM1.
Topics: Algorithms; Anesthetics, Local; Animals; Brain; Cell Membrane; Cholesterol; Circular Dichroism; Dibucaine; G(M1) Ganglioside; Kinetics; Membrane Lipids; Models, Chemical; Models, Molecular; Phospholipids; Protein Binding; Sheep; Spectrin; Spectrometry, Fluorescence; Tetracaine; Thermodynamics | 2015 |
[Generalised contact eczema: Care is needed in selecting a lubricant for digital rectal examination].
Topics: Aged, 80 and over; Anesthetics, Local; Benzocaine; Conjunctivitis; Dermatitis, Allergic Contact; Dibucaine; Digital Rectal Examination; Eczema; Humans; Lubricants; Male; Ophthalmic Solutions; Patch Tests; Recurrence; Tetracaine | 2015 |
Baboon syndrome caused by anti-haemorrhoidal ointment.
Topics: Anesthetics, Local; Buttocks; Dermatitis, Allergic Contact; Dibucaine; Erythema; Hemorrhoids; Humans; Male; Middle Aged; Ointments; Syndrome; Tetracaine | 2018 |