Page last updated: 2024-08-17

tetrabenazine and piperidines

tetrabenazine has been researched along with piperidines in 33 studies

Research

Studies (33)

TimeframeStudies, this research(%)All Research%
pre-199017 (51.52)18.7374
1990's6 (18.18)18.2507
2000's2 (6.06)29.6817
2010's7 (21.21)24.3611
2020's1 (3.03)2.80

Authors

AuthorsStudies
Henriksson, BG; Järbe, TU; Johansson, JO1
Crichlow, CA; Geyer, HM; Klioze, SS; Kruse, H; Martin, LL; Worm, M1
Bauer, VJ; Geyer, HM; Klioze, SS1
Alouf, JE; Buckle, M; Cesura, A; Da Prada, M; Geoffroy, C; Launay, JM; Mutel, V1
Bertocci, B; Cesura, AM; Da Prada, M1
Fuller, RW1
Gerhards, H; Kruse, H; Kunstmann, R; Leven, M; Paulus, EF; Schacht, U; Schmitt, K; Witte, PU1
Jurna, I; Regélhy, B1
Bachmann, T; Jurna, I; Theres, C1
Leonard, BE; Tonge, SR2
Leander, JD1
Feldtrauer, JJ; Paul, E; Stoecklin, K; Waldmeier, PC1
Burghard, H; Ellis, DB; Fortunato, J; Geyer, HM; Glamkowski, EJ; Ong, HH; Profitt, JA; Wilker, JC1
Allen, RC; Fortunato, JM; Geyer, HM; Glamkowski, EJ; Ong, HH; Wilker, JC1
Anderson, VB; Geyer, HM; Kruse, H; Ong, HH; Profitt, JA; Wilker, JC1
Erickson, JD; Varoqui, H1
Frey, KA; Kilbourn, MR; Wieland, DM1
Edwards, RH; Finn, JP; Merickel, A1
Chen, K; De Maeyer, E; Kung, MP; Meehan, WP; Ridd, MJ; Seif, I; Shih, JC1
An, H; Chervin, RD; Consens, FB; Gilman, S; Heumann, M; Junck, L; Koeppe, RA; Little, R2
BOFF, E; SCHECKEL, CL1
IWAMOTO, T; SATOH, T; TOKUMITSU, Y1
IWAMOTO, T; SATOH, T1
Klamer, D; Ponten, H; Waters, N; Waters, S1
Albin, RL; Bohnen, NI; Frey, KA; Koeppe, RA; Kotagal, V; Müller, ML; Petrou, M; Scott, PJ1
Czekaj, J; Kos, T; Popik, P; Skolnick, P1
Stevens, J1
Bonuccelli, U; Ceravolo, R; Mazzucchi, S; Palermo, G; Unti, E1
Bohnen, JLB; Bohnen, NI; Haugen, J; Müller, MLTM1
Bashir, H; Jankovic, J1
Depoortere, R; Jastrzębska-Więsek, M; Kołaczkowski, M; Newman-Tancredi, A; Varney, MA; Wesołowska, A1

Reviews

3 review(s) available for tetrabenazine and piperidines

ArticleYear
Biochemical pharmacology of the serotonin system.
    Advances in neurology, 1986, Volume: 43

    Topics: Alanine; Brain; Citalopram; Clomipramine; Fenfluramine; Fluoxetine; Fluvoxamine; Humans; Monoamine Oxidase Inhibitors; Neurons; Oximes; p-Chloroamphetamine; Paroxetine; Piperidines; Propylamines; Receptors, Serotonin; Reserpine; Serotonin; Serotonin Antagonists; Synapses; Tetrabenazine; Zimeldine

1986
Antipsychotic drugs in Huntington's disease.
    Expert review of neurotherapeutics, 2017, Volume: 17, Issue:3

    Topics: Antipsychotic Agents; Humans; Huntington Disease; Piperidines; Tetrabenazine

2017
Treatment options for chorea.
    Expert review of neurotherapeutics, 2018, Volume: 18, Issue:1

    Topics: Antipsychotic Agents; Chorea; Deep Brain Stimulation; Dopamine Antagonists; Humans; Piperidines; Tetrabenazine; Transcranial Magnetic Stimulation; Valine; Vesicular Monoamine Transport Proteins

2018

Trials

2 trial(s) available for tetrabenazine and piperidines

ArticleYear
REM sleep behavior disorder is related to striatal monoaminergic deficit in MSA.
    Neurology, 2003, Jul-08, Volume: 61, Issue:1

    Topics: Adult; Age Distribution; Aged; Binding, Competitive; Biogenic Monoamines; Carbon Radioisotopes; Corpus Striatum; Electromyography; Female; Humans; Iodine Radioisotopes; Male; Middle Aged; Multiple System Atrophy; Piperidines; Polysomnography; Predictive Value of Tests; Reference Values; REM Sleep Behavior Disorder; Sex Distribution; Tetrabenazine; Tetrahydronaphthalenes; Thalamus; Tomography, Emission-Computed; Tomography, Emission-Computed, Single-Photon

2003
Obstructive sleep apnea is related to a thalamic cholinergic deficit in MSA.
    Neurology, 2003, Jul-08, Volume: 61, Issue:1

    Topics: Adult; Age Distribution; Aged; Binding, Competitive; Carrier Proteins; Corpus Striatum; Female; Humans; Iodine Radioisotopes; Male; Membrane Glycoproteins; Membrane Transport Proteins; Middle Aged; Multiple System Atrophy; Neuropeptides; Pilot Projects; Piperidines; Pons; Receptors, Cholinergic; Reference Values; Regression Analysis; Sex Distribution; Sleep Apnea, Obstructive; Tetrabenazine; Tetrahydronaphthalenes; Thalamus; Tomography, Emission-Computed; Tomography, Emission-Computed, Single-Photon; Vesicular Acetylcholine Transport Proteins; Vesicular Biogenic Amine Transport Proteins; Vesicular Transport Proteins

2003

Other Studies

28 other study(ies) available for tetrabenazine and piperidines

ArticleYear
Drug discrimination in rats: the effects of phencyclidine and ditran.
    Psychopharmacologia, 1975, Apr-30, Volume: 42, Issue:1

    Topics: Animals; Cues; Cyclohexylamines; Discrimination Learning; Drug Combinations; Fenclonine; Glycolates; Imipramine; Ketamine; Male; Neostigmine; Phencyclidine; Physostigmine; Piperidines; Pyrrolidines; Rats; Tacrine; Tetrabenazine; Yohimbine

1975
Synthesis of spiro[isobenzofuran-1(3H),4'-piperidines] as potential central nervous system agents. 5. Conformationally mobile analogues derived by furan ring opening.
    Journal of medicinal chemistry, 1979, Volume: 22, Issue:11

    Topics: Animals; Antidepressive Agents; Benzofurans; Brain; In Vitro Techniques; Mice; Norepinephrine; Piperidines; Rats; Spiro Compounds; Structure-Activity Relationship; Synaptosomes; Tetrabenazine

1979
Synthesis of spiro[isobenzofuran-1(3H),4'-piperidines] as potential central nervous system agents. 2. Compounds containing a heteroatom attached to nitrogen.
    Journal of medicinal chemistry, 1977, Volume: 20, Issue:4

    Topics: Animals; Antidepressive Agents; Benzofurans; Blepharoptosis; Methods; Mice; Piperidines; Structure-Activity Relationship; Tetrabenazine

1977
One-step purification of the serotonin transporter located at the human platelet plasma membrane.
    The Journal of biological chemistry, 1992, Jun-05, Volume: 267, Issue:16

    Topics: Biological Transport; Blood Platelets; Blood Proteins; Carrier Proteins; Cell Membrane; Chromatography, Affinity; Electrophoresis, Gel, Two-Dimensional; Electrophoresis, Polyacrylamide Gel; Humans; Ouabain; Paroxetine; Piperidines; Serotonin; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins; Tetrabenazine

1992
Binding of [3H]dihydrotetrabenazine and [125I]azidoiodoketanserin photoaffinity labeling of the monoamine transporter of platelet 5-HT organelles.
    European journal of pharmacology, 1990, Sep-04, Volume: 186, Issue:1

    Topics: Affinity Labels; Animals; Azides; Biogenic Monoamines; Blood Platelets; Blood Proteins; Cell Membrane; Guinea Pigs; Humans; In Vitro Techniques; Iodine Radioisotopes; Ketanserin; Paroxetine; Photochemistry; Piperidines; Rabbits; Rats; Receptors, Serotonin; Subcellular Fractions; Tetrabenazine

1990
Resolution, absolute stereochemistry, and enantioselective activity of nomifensine and hexahydro-1H-indeno[1,2-b]pyridines.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:5

    Topics: Animals; Blepharoptosis; Brain; Chemical Phenomena; Chemistry; Dopamine; Drug Synergism; Indans; Indenes; Isomerism; Male; Mice; Molecular Conformation; Nomifensine; Norepinephrine; Piperidines; Rats; Serotonin; Structure-Activity Relationship; Synaptosomes; Tetrabenazine; Yohimbine

1987
The antagonism between reserpine and some antiparkinson drugs in electroseizure.
    Naunyn-Schmiedebergs Archiv fur experimentelle Pathologie und Pharmakologie, 1968, Volume: 259, Issue:5

    Topics: 1-Propanol; Animals; Atropine; Biperiden; Cyclohexanes; Dextroamphetamine; Dihydroxyphenylalanine; Electroshock; Methamphetamine; Parasympatholytics; Piperidines; Rats; Reserpine; Sympathomimetics; Tachyphylaxis; Tetrabenazine; Thiocarbamates; Tyrosine

1968
The effect of physostigmine and tetrabenazine on spinal motor control and its inhibition by drugs which influence reserpine rigidity.
    Naunyn-Schmiedebergs Archiv fur experimentelle Pathologie und Pharmakologie, 1969, Volume: 263, Issue:3

    Topics: 1-Propanol; Animals; Atropine; Biperiden; Dihydroxyphenylalanine; Electric Stimulation; Electromyography; Methamphetamine; Motor Neurons; Movement Disorders; Parasympatholytics; Phenytoin; Physostigmine; Piperidines; Rats; Reserpine; Spinal Cord; Spinal Nerves; Tetrabenazine; Trihexyphenidyl

1969
Interaction of phencyclidine with drugs affecting noradrenaline metabolism in the rat brain.
    Psychopharmacologia, 1972, Volume: 23, Issue:1

    Topics: Anesthetics; Animals; Brain; Brain Chemistry; Desipramine; Drug Antagonism; Drug Synergism; Norepinephrine; Normetanephrine; Phencyclidine; Piperidines; Rats; Tetrabenazine

1972
Partial antagonism of the behavioural and neurochemical effects of phencyclidine by drugs affecting monoamine metabolism.
    Psychopharmacologia, 1972, Volume: 24, Issue:4

    Topics: Anesthetics; Animals; Brain; Drug Antagonism; Hallucinogens; Hydroxyindoleacetic Acid; Imipramine; Injections, Intraperitoneal; Phencyclidine; Piperidines; Rats; Serotonin; Tetrabenazine

1972
Effects of tetrabenazine and phenylpiperidine analgesics during daily clorgyline treatment.
    Psychopharmacology, 1981, Volume: 74, Issue:3

    Topics: Analgesics; Analgesics, Opioid; Animals; Clorgyline; Columbidae; Conditioning, Operant; Drug Interactions; Male; Piperidines; Propylamines; Reinforcement Schedule; Tetrabenazine

1981
Reversibility of the interaction of CGP 11305 A with MAO A in vivo.
    European journal of pharmacology, 1983, Oct-14, Volume: 94, Issue:1-2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Brain; Clorgyline; Dopamine; Female; Homovanillic Acid; Hydroxyindoleacetic Acid; Liver; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Piperidines; Rats; Serotonin; Tetrabenazine

1983
Novel tetracyclic spiropiperidines. 3. 1-arylspiro[indoline-3,4'-piperidine]s as potential antidepressants.
    Journal of medicinal chemistry, 1983, Volume: 26, Issue:7

    Topics: 5-Hydroxytryptophan; Animals; Antidepressive Agents; Biological Assay; Blepharoptosis; Drug Synergism; Humans; Indicators and Reagents; Indoles; Piperidines; Stereotyped Behavior; Structure-Activity Relationship; Tetrabenazine

1983
Novel tetracyclic spiropiperidines. 4. Synthesis and pharmacological evaluation of spiro- and 6,7-dihydrospiro[benzo[b]pyrrolo[3,2,1-jk][1,4]benzodiazepine-2 (1H),4'-piperidine]s.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:1

    Topics: Animals; Antidepressive Agents; Benzodiazepines; Biological Assay; Blepharoptosis; Indicators and Reagents; Magnetic Resonance Spectroscopy; Piperidines; Rats; Spectrophotometry, Infrared; Spiro Compounds; Structure-Activity Relationship; Tetrabenazine

1984
Novel tetracyclic spiropiperidines. 1. 3-Aryl-1,3-dihydrospiro[benzo[c]thiophene-1,4'-piperidines] as potential antidepressants.
    Journal of medicinal chemistry, 1981, Volume: 24, Issue:1

    Topics: 5-Hydroxytryptophan; Animals; Antidepressive Agents, Tricyclic; Blepharoptosis; Chemical Phenomena; Chemistry; Drug Synergism; Male; Mice; Physostigmine; Piperidines; Spiro Compounds; Tetrabenazine

1981
Active transport of acetylcholine by the human vesicular acetylcholine transporter.
    The Journal of biological chemistry, 1996, Nov-01, Volume: 271, Issue:44

    Topics: Acetylcholine; Adrenal Gland Neoplasms; Animals; Biological Transport, Active; Carrier Proteins; Cytosol; Humans; Kinetics; Membrane Transport Proteins; Neuromuscular Depolarizing Agents; PC12 Cells; Pheochromocytoma; Piperidines; Rats; Recombinant Proteins; Substrate Specificity; Tetrabenazine; Transfection; Vesicular Acetylcholine Transport Proteins; Vesicular Transport Proteins

1996
Imaging of monoaminergic and cholinergic vesicular transporters in the brain.
    Advances in pharmacology (San Diego, Calif.), 1998, Volume: 42

    Topics: Acetylcholine; Alzheimer Disease; Brain; Carbon Radioisotopes; Carrier Proteins; Humans; Membrane Glycoproteins; Membrane Transport Proteins; Neuromuscular Depolarizing Agents; Neurons; Neuropeptides; Neurotransmitter Agents; Parkinson Disease; Piperidines; Tetrabenazine; Tomography, Emission-Computed; Tomography, Emission-Computed, Single-Photon; Tritium; Vesicular Acetylcholine Transport Proteins; Vesicular Biogenic Amine Transport Proteins; Vesicular Transport Proteins

1998
Analysis of neurotransmitter transport into secretory vesicles.
    Methods in enzymology, 1998, Volume: 296

    Topics: Acetylcholine; Animals; Carrier Proteins; Cell Membrane; CHO Cells; COS Cells; Cricetinae; Cytoplasmic Granules; Kinetics; Membrane Transport Proteins; Neurons; Neurotransmitter Agents; Piperidines; Recombinant Proteins; Tetrabenazine; Transfection; Vesicular Acetylcholine Transport Proteins; Vesicular Transport Proteins

1998
Ketanserin and tetrabenazine abolish aggression in mice lacking monoamine oxidase A.
    Brain research, 1999, Jul-24, Volume: 835, Issue:2

    Topics: Adrenergic Uptake Inhibitors; Aggression; Animals; Brain; Corpus Striatum; Drug Evaluation, Preclinical; Fluorobenzenes; Frontal Lobe; Ketanserin; Male; Mice; Mice, Knockout; Monoamine Oxidase; Neurotransmitter Agents; Piperidines; Radioligand Assay; Serotonin Antagonists; Tetrabenazine

1999
BEHAVIORAL EFFECTS OF INTERACTING IMIPRAMINE AND OTHER DRUGS WITH D-AMPHETAMINE, COCAINE, AND TETRABENAZINE.
    Psychopharmacologia, 1964, Feb-12, Volume: 5

    Topics: Amitriptyline; Atropine; Avoidance Learning; Chlorpromazine; Cocaine; Desipramine; Dextroamphetamine; Guanethidine; Imipramine; Iproniazid; Isocarboxazid; Methylphenidate; Parasympatholytics; Pharmacology; Piperidines; Promazine; Promethazine; Rats; Research; Scopolamine; Tetrabenazine; Trihexyphenidyl; Tyramine

1964
EFFECTS OF SOME TRANQUILLIZING AGENTS ON BRAIN NORADRENALINE AND DOPAMINE LEVELS OF SHOCKED RATS.
    Japanese journal of pharmacology, 1964, Volume: 14

    Topics: Blood-Brain Barrier; Brain; Chlordiazepoxide; Chlorpromazine; Cyproheptadine; Dopamine; Electricity; Fluorometry; Norepinephrine; Pharmacology; Piperidines; Rats; Research; Shock; Tetrabenazine; Thioridazine; Tranquilizing Agents

1964
EFFECTS OF CHLORPROMAZINE, TETRABENAZINE AND AZACYCLONOL ON BRAIN SEROTONIN LEVEL OF SHOCKED RATS.
    Japanese journal of pharmacology, 1964, Volume: 14

    Topics: Brain; Brain Chemistry; Chlorpromazine; Electricity; Electroshock; Pharmacology; Piperidines; Rats; Research; Serotonin; Shock; Tetrabenazine

1964
Co-administration of the Dopaminergic Stabilizer Pridopidine and Tetrabenazine in Rats.
    Journal of Huntington's disease, 2014, Volume: 3, Issue:3

    Topics: Animals; Behavior, Animal; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Drug Combinations; Drug Interactions; Locomotion; Male; Motor Activity; Piperidines; Rats; Rats, Sprague-Dawley; Tetrabenazine; Treatment Outcome

2014
Diabetes mellitus is independently associated with more severe cognitive impairment in Parkinson disease.
    Parkinsonism & related disorders, 2014, Volume: 20, Issue:12

    Topics: Aged; Butyrates; Carbon Isotopes; Cognition Disorders; Cross-Sectional Studies; Diabetes Complications; Diabetes Mellitus; Female; Humans; Male; Middle Aged; Neuroimaging; Neuropsychological Tests; Parkinson Disease; Piperidines; Positron-Emission Tomography; Severity of Illness Index; Tetrabenazine

2014
Effect of NMDAR antagonists in the tetrabenazine test for antidepressants: comparison with the tail suspension test.
    Acta neuropsychiatrica, 2015, Volume: 27, Issue:4

    Topics: Adrenergic Uptake Inhibitors; Animals; Antidepressive Agents; Blepharoptosis; Disease Models, Animal; Drug Evaluation, Preclinical; Excitatory Amino Acid Antagonists; Hindlimb Suspension; Ketamine; Male; Mice; Mice, Inbred C57BL; Motor Activity; Phenethylamines; Phenols; Piperidines; Pyridines; Pyrimidines; Receptors, N-Methyl-D-Aspartate; Tetrabenazine

2015
Market watch: Upcoming market catalysts in Q2 2016.
    Nature reviews. Drug discovery, 2016, Volume: 15, Issue:4

    Topics: Adrenergic Uptake Inhibitors; Antiparkinson Agents; Drug Approval; Drug Discovery; Humans; Piperidines; Tetrabenazine; United States; United States Food and Drug Administration; Urea

2016
Mentally stimulating activities associate with better cognitive performance in Parkinson disease.
    Journal of neural transmission (Vienna, Austria : 1996), 2017, Volume: 124, Issue:10

    Topics: Aged; Aged, 80 and over; Carbon Isotopes; Cognition Disorders; Cognitive Behavioral Therapy; Female; Humans; Magnetic Resonance Imaging; Male; Mental Status and Dementia Tests; Middle Aged; Neuropsychological Tests; Parkinson Disease; Phosphinic Acids; Piperidines; Positron-Emission Tomography; Regression Analysis; Tetrabenazine

2017
The selective 5-HT 1A receptor agonist, NLX-112, overcomes tetrabenazine-induced catalepsy and depression-like behavior in the rat.
    Behavioural pharmacology, 2022, 08-01, Volume: 33, Issue:5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antidepressive Agents; Buspirone; Catalepsy; Depression; Huntington Disease; Parkinsonian Disorders; Piperidines; Pyridines; Rats; Receptor, Serotonin, 5-HT1A; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin Receptor Agonists; Tetrabenazine

2022