Page last updated: 2024-08-17

tetrabenazine and lobeline

tetrabenazine has been researched along with lobeline in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19901 (10.00)18.7374
1990's1 (10.00)18.2507
2000's3 (30.00)29.6817
2010's5 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chagkutip, J; Crooks, PA; Dwoskin, LP; Nickell, JR; Vartak, AP1
Crooks, PA; Deaciuc, AG; Dwoskin, LP; Grinevich, VP; Hojahmat, M; Horton, DB; Miller, DK; Norrholm, SD1
Zetler, G1
Crooks, PA; Dwoskin, LP; Teng, L1
Crooks, PA; Dwoskin, LP; Grinevich, VP; Miller, DK; Norrholm, SD; Zheng, G1
Crooks, PA; Deaciuc, AG; Dwoskin, LP; Zhan, CG; Zheng, F; Zheng, G1
Bardo, MT; Beckmann, JS; Crooks, PA; Denehy, ED; Dwoskin, LP; Horton, DB; Nickell, JR; Siripurapu, KB; Vartak, A1
Crooks, PA; Deaciuc, AG; Dwoskin, LP; Nickell, JR; Penthala, NR; Ponugoti, PR1
Crooks, PA; Dwoskin, LP; Horton, DB; Nickell, JR; Zheng, G1
Crooks, PA; Ding, D; Dwoskin, LP; Nickell, JR1

Other Studies

10 other study(ies) available for tetrabenazine and lobeline

ArticleYear
Pyrrolidine analogues of lobelane: relationship of affinity for the dihydrotetrabenazine binding site with function of the vesicular monoamine transporter 2 (VMAT2).
    Journal of medicinal chemistry, 2009, Dec-10, Volume: 52, Issue:23

    Topics: Binding Sites; Lobeline; Protein Binding; Pyrrolidines; Structure-Activity Relationship; Tetrabenazine; Vesicular Monoamine Transport Proteins

2009
Lobeline esters as novel ligands for neuronal nicotinic acetylcholine receptors and neurotransmitter transporters.
    Bioorganic & medicinal chemistry, 2010, Jan-15, Volume: 18, Issue:2

    Topics: Animals; Esters; Ligands; Lobeline; Male; Molecular Structure; Neurons; Neurotransmitter Transport Proteins; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Stereoisomerism; Structure-Activity Relationship

2010
Drug-induced catalepsy as influenced by convulsant and anticonvulsant drugs.
    Neuropharmacology, 1973, Volume: 12, Issue:8

    Topics: Animals; Anticonvulsants; Arecoline; Bemegride; Caffeine; Catalepsy; Central Nervous System Stimulants; Drug Synergism; Ethosuximide; Haloperidol; Humans; Lobeline; Male; Mice; Mice, Inbred Strains; Nicotine; Nikethamide; Paraoxon; Pentylenetetrazole; Pilocarpine; Tetrabenazine; Tremorine; Trifluoperazine

1973
Lobeline displaces [3H]dihydrotetrabenazine binding and releases [3H]dopamine from rat striatal synaptic vesicles: comparison with d-amphetamine.
    Journal of neurochemistry, 1998, Volume: 71, Issue:1

    Topics: Animals; Binding, Competitive; Biological Transport; Corpus Striatum; Dextroamphetamine; Dopamine; Dopamine Agents; Lobeline; Male; Membrane Glycoproteins; Membrane Transport Proteins; Neuropeptides; Neurotransmitter Agents; Nicotinic Agonists; Rats; Rats, Sprague-Dawley; Synaptic Vesicles; Tetrabenazine; Tritium; Vesicular Biogenic Amine Transport Proteins; Vesicular Monoamine Transport Proteins

1998
Lobeline analogs with enhanced affinity and selectivity for plasmalemma and vesicular monoamine transporters.
    The Journal of pharmacology and experimental therapeutics, 2004, Volume: 310, Issue:3

    Topics: Aconitine; Animals; Biological Transport; Carrier Proteins; Cells, Cultured; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Ganglionic Stimulants; Humans; Iodine Radioisotopes; Kinetics; Lobeline; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Neuropeptides; Nicotine; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Rats; Rats, Sprague-Dawley; Rubidium; Serotonin; Serotonin Plasma Membrane Transport Proteins; Symporters; Tetrabenazine; Tritium; Vesicular Biogenic Amine Transport Proteins; Vesicular Monoamine Transport Proteins

2004
Computational neural network analysis of the affinity of lobeline and tetrabenazine analogs for the vesicular monoamine transporter-2.
    Bioorganic & medicinal chemistry, 2007, Apr-15, Volume: 15, Issue:8

    Topics: Artificial Intelligence; Crystallography, X-Ray; Least-Squares Analysis; Ligands; Lobeline; Neural Networks, Computer; Nicotinic Agonists; Nonlinear Dynamics; Structure-Activity Relationship; Tetrabenazine; Vesicular Monoamine Transport Proteins

2007
The novel pyrrolidine nor-lobelane analog UKCP-110 [cis-2,5-di-(2-phenethyl)-pyrrolidine hydrochloride] inhibits VMAT2 function, methamphetamine-evoked dopamine release, and methamphetamine self-administration in rats.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 335, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Aconitine; Amphetamine-Related Disorders; Animals; Behavior, Animal; Cell Membrane; Conditioning, Operant; Corpus Striatum; Dopamine; Drug Tolerance; Lobeline; Male; Methamphetamine; Nicotine; Protein Binding; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Reinforcement, Psychology; Self Administration; Synaptic Vesicles; Tetrabenazine; Vesicular Monoamine Transport Proteins

2010
Pyrrolidine analogs of GZ-793A: synthesis and evaluation as inhibitors of the vesicular monoamine transporter-2 (VMAT2).
    Bioorganic & medicinal chemistry letters, 2013, Jun-01, Volume: 23, Issue:11

    Topics: Animals; Binding Sites; Dopamine; Lobeline; Protein Binding; Pyrrolidines; Rats; Synaptic Vesicles; Tetrabenazine; Vesicular Monoamine Transport Proteins

2013
GZ-793A, a lobelane analog, interacts with the vesicular monoamine transporter-2 to inhibit the effect of methamphetamine.
    Journal of neurochemistry, 2013, Volume: 127, Issue:2

    Topics: Adrenergic Uptake Inhibitors; Animals; Data Interpretation, Statistical; Dopamine; Dopamine Uptake Inhibitors; Lobeline; Male; Methamphetamine; Neostriatum; Rats; Rats, Sprague-Dawley; Reserpine; Synaptic Vesicles; Tetrabenazine; Vesicular Monoamine Transport Proteins

2013
Quinolyl analogues of norlobelane: novel potent inhibitors of [(3)H]dihydrotetrabenazine binding and [(3)H]dopamine uptake at the vesicular monoamine transporter-2.
    Bioorganic & medicinal chemistry letters, 2015, Jul-01, Volume: 25, Issue:13

    Topics: Amphetamine-Related Disorders; Animals; Binding Sites; Dopamine; Humans; In Vitro Techniques; Kinetics; Lobeline; Methamphetamine; Rats; Structure-Activity Relationship; Synaptic Vesicles; Tetrabenazine; Vesicular Monoamine Transport Proteins

2015