Page last updated: 2024-09-05

tesaglitazar and pioglitazone

tesaglitazar has been researched along with pioglitazone in 6 studies

Compound Research Comparison

Studies
(tesaglitazar)
Trials
(tesaglitazar)
Recent Studies (post-2010)
(tesaglitazar)
Studies
(pioglitazone)
Trials
(pioglitazone)
Recent Studies (post-2010) (pioglitazone)
7413254,3388242,277

Protein Interaction Comparison

ProteinTaxonomytesaglitazar (IC50)pioglitazone (IC50)
CDGSH iron-sulfur domain-containing protein 1Rattus norvegicus (Norway rat)1
Bile salt export pumpRattus norvegicus (Norway rat)2
Peroxisome proliferator-activated receptor gammaRattus norvegicus (Norway rat)0.7
Bile salt export pumpHomo sapiens (human)0.337
Carbonic anhydrase 2Homo sapiens (human)0.114
Steryl-sulfataseHomo sapiens (human)0.8
Peroxisome proliferator-activated receptor alphaMus musculus (house mouse)1.15
Amine oxidase [flavin-containing] BHomo sapiens (human)0.298
Peroxisome proliferator-activated receptor gammaHomo sapiens (human)3.0379
Peroxisome proliferator-activated receptor gammaMus musculus (house mouse)0.7
CDGSH iron-sulfur domain-containing protein 2Homo sapiens (human)4.8
CDGSH iron-sulfur domain-containing protein 1Homo sapiens (human)8.65

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (50.00)29.6817
2010's3 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Deussen, HJ; Ebdrup, S; Fleckner, J; Frost Jensen, A; Mortensen, SB; Nygaard, L; Pettersson, I; Pridal, L; Rasmussen, HB; Sauerberg, P1
Lindberg, MB; Ohman, KP; Ose, L; Retterstøl, K; Svensson, M; Tonstad, S1
Bays, H; Bryzinski, BS; McElhattan, J1
Hamrén, B; Karlsson, MO; Ohman, KP; Svensson, MK1
Blander, G; Bobadilla, M; Catlett, NL; Deehan, R; Edgar, A; Elliston, KO; Haefliger, C; Ladd, W; Maerz-Weiss, P; Mizrahi, J; Steiner, G; Wong, B; Wright, MB1
Benavidez, JM; Black, M; Blednov, YA; Edenberg, HJ; Ferguson, LB; Foroud, T; Goate, AM; Harris, RA; Hesselbrock, V; Schoenhard, GL; Wetherill, L1

Trials

3 trial(s) available for tesaglitazar and pioglitazone

ArticleYear
The dual peroxisome proliferator-activated receptor alpha/gamma agonist tesaglitazar further improves the lipid profile in dyslipidemic subjects treated with atorvastatin.
    Metabolism: clinical and experimental, 2007, Volume: 56, Issue:9

    Topics: Adult; Alkanesulfonates; Anticholesteremic Agents; Atorvastatin; Chemotherapy, Adjuvant; Cross-Over Studies; Drug Combinations; Drug Synergism; Dyslipidemias; Female; Heptanoic Acids; Humans; Hypoglycemic Agents; Lipids; Male; Middle Aged; Phenylpropionates; Pioglitazone; Placebos; PPAR alpha; PPAR gamma; Pyrroles; Thiazolidinediones

2007
A double-blind, randomised trial of tesaglitazar versus pioglitazone in patients with type 2 diabetes mellitus.
    Diabetes & vascular disease research, 2007, Volume: 4, Issue:3

    Topics: Adult; Aged; Aged, 80 and over; Alkanesulfonates; Blood Glucose; Cholesterol, HDL; Cholesterol, LDL; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Double-Blind Method; Female; Glycated Hemoglobin; Humans; Hypoglycemic Agents; Male; Middle Aged; Phenylpropionates; Pioglitazone; Thiazolidinediones; Time Factors

2007
Pharmacokinetic-pharmacodynamic assessment of the interrelationships between tesaglitazar exposure and renal function in patients with type 2 diabetes mellitus.
    Journal of clinical pharmacology, 2012, Volume: 52, Issue:9

    Topics: Aged; Alkanesulfonates; Creatinine; Diabetes Mellitus, Type 2; Female; Glomerular Filtration Rate; Humans; Hypoglycemic Agents; Kidney; Male; Middle Aged; Models, Biological; Phenylpropionates; Pioglitazone; Thiazolidinediones

2012

Other Studies

3 other study(ies) available for tesaglitazar and pioglitazone

ArticleYear
Synthesis and biological and structural characterization of the dual-acting peroxisome proliferator-activated receptor alpha/gamma agonist ragaglitazar.
    Journal of medicinal chemistry, 2003, Apr-10, Volume: 46, Issue:8

    Topics: Binding Sites; Crystallography, X-Ray; Hypoglycemic Agents; Ligands; Models, Molecular; Oxazines; Phenylpropionates; Radioligand Assay; Receptors, Cytoplasmic and Nuclear; Stereoisomerism; Transcription Factors

2003
Comparative transcriptional network modeling of three PPAR-α/γ co-agonists reveals distinct metabolic gene signatures in primary human hepatocytes.
    PloS one, 2012, Volume: 7, Issue:4

    Topics: Alkanesulfonates; Cells, Cultured; Fenofibrate; Hepatocytes; Humans; Oxazoles; Phenylpropionates; Pioglitazone; PPAR alpha; PPAR gamma; Thiazolidinediones; Thiophenes

2012
Peroxisome proliferator-activated receptors α and γ are linked with alcohol consumption in mice and withdrawal and dependence in humans.
    Alcoholism, clinical and experimental research, 2015, Volume: 39, Issue:1

    Topics: Adult; Alcohol Drinking; Alcoholism; Alkanesulfonates; Animals; Bezafibrate; Brain; Female; Fenofibrate; Genome-Wide Association Study; Humans; Liver; Male; Mice; Phenylpropionates; Pioglitazone; Polymorphism, Single Nucleotide; PPAR alpha; PPAR gamma; Thiazoles; Thiazolidinediones

2015