Page last updated: 2024-09-05

tesaglitazar and methapyrilene

tesaglitazar has been researched along with methapyrilene in 1 studies

Compound Research Comparison

Studies
(tesaglitazar)
Trials
(tesaglitazar)
Recent Studies (post-2010)
(tesaglitazar)
Studies
(methapyrilene)
Trials
(methapyrilene)
Recent Studies (post-2010) (methapyrilene)
741325206325

Protein Interaction Comparison

ProteinTaxonomytesaglitazar (IC50)methapyrilene (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.744
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)1.391
Muscarinic acetylcholine receptor M2Homo sapiens (human)1.665
Muscarinic acetylcholine receptor M5Homo sapiens (human)3.265
Alpha-2A adrenergic receptorHomo sapiens (human)1.165
Cytochrome P450 2D6Homo sapiens (human)2.7564
Muscarinic acetylcholine receptor M1Homo sapiens (human)4.773
Alpha-2B adrenergic receptorHomo sapiens (human)3.318
Sodium-dependent noradrenaline transporter Homo sapiens (human)1.391
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.628
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.744
Sodium-dependent serotonin transporterHomo sapiens (human)0.2
Histamine H1 receptorHomo sapiens (human)0.016
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.843
5-hydroxytryptamine receptor 6Homo sapiens (human)3.091
Sodium-dependent dopamine transporter Homo sapiens (human)2.757

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1

Other Studies

1 other study(ies) available for tesaglitazar and methapyrilene

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
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