Page last updated: 2024-08-23

tertatolol and pindolol

tertatolol has been researched along with pindolol in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19902 (20.00)18.7374
1990's6 (60.00)18.2507
2000's2 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Carrupt, PA; el Tayar, N; Testa, B; Van de Waterbeemd, H1
Carrupt, PA; Gaillard, P; Schambel, P; Testa, B1
Kompa, AR; Molenaar, P; Pak, HS; Roberts, SJ; Summers, RJ1
Ferrari, MD; Heiligers, JP; Saxena, PR; Villalón, CM1
De Blasi, A; Fratelli, M; Marasco, O1
Assie, MB; Koek, W1
Clifford, EM; Cowen, PJ; Gartside, SE; Sharp, T1
Fornal, CA; Jacobs, BL; Martin, FJ; Metzler, CW1
Castro, ME; Harrison, PJ; Pazos, A; Sharp, T1
Bench, CJ; Castro, ME; Cowen, PJ; Grasby, PM; Gunn, RN; Harrison, PJ; Koepp, MJ; Meyer, JH; Pazos, A; Rabiner, EA; Sargent, PA; Sharp, T1

Reviews

1 review(s) available for tertatolol and pindolol

ArticleYear
Modeling of beta-adrenoceptors based on molecular electrostatic potential studies of agonists and antagonists.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:11

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Models, Molecular; Receptors, Adrenergic, beta; Structure-Activity Relationship

1988

Trials

1 trial(s) available for tertatolol and pindolol

ArticleYear
beta-blocker binding to human 5-HT(1A) receptors in vivo and in vitro: implications for antidepressant therapy.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2000, Volume: 23, Issue:3

    Topics: Adrenergic beta-Antagonists; Adult; Aged; Antidepressive Agents; Autoradiography; Autoreceptors; Brain Chemistry; Female; Humans; In Vitro Techniques; Male; Middle Aged; Penbutolol; Pindolol; Piperazines; Propanolamines; Pyridines; Receptors, Neurotransmitter; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Thiophenes; Tomography, Emission-Computed

2000

Other Studies

8 other study(ies) available for tertatolol and pindolol

ArticleYear
Binding of arylpiperazines, (aryloxy)propanolamines, and tetrahydropyridylindoles to the 5-HT1A receptor: contribution of the molecular lipophilicity potential to three-dimensional quantitative structure-affinity relationship models.
    Journal of medicinal chemistry, 1996, Jan-05, Volume: 39, Issue:1

    Topics: Indoles; Ligands; Models, Molecular; Molecular Conformation; Molecular Structure; Piperazines; Propanolamines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Structure-Activity Relationship; Tetrahydronaphthalenes

1996
Localization of (-)-[125I]cyanopindolol binding in guinea-pig heart: characteristics of non-beta-adrenoceptor related binding in cardiac pacemaker and conducting regions.
    Neuroscience letters, 1992, Feb-17, Volume: 136, Issue:1

    Topics: Alprenolol; Animals; Ascorbic Acid; Binding Sites; Ethanolamines; Female; Guinea Pigs; Haloperidol; Heart Conduction System; Isoproterenol; Male; Myocardium; Peroxidase; Phentolamine; Pindolol; Propanolamines; Propranolol; Protein Binding; Receptors, Adrenergic, beta; Serotonin; Thiophenes; Trachea

1992
Effects of tertatolol, a beta-adrenoceptor antagonist with agonist affinity at 5-HT1A receptors, in an animal model of migraine: comparison with propranolol and pindolol.
    European journal of pharmacology, 1992, Sep-10, Volume: 220, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Carotid Arteries; Disease Models, Animal; Hemodynamics; Injections, Intravenous; Migraine Disorders; Pindolol; Propanolamines; Propranolol; Receptors, Serotonin; Swine; Thiophenes

1992
Certain beta-blockers can decrease beta-adrenergic receptor number: I. Acute reduction in receptor number by tertatolol and bopindolol.
    Circulation research, 1988, Volume: 63, Issue:2

    Topics: Adrenergic beta-Antagonists; Binding, Competitive; Humans; Leukocytes, Mononuclear; Lymphoma; Male; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Stereoisomerism; Sympathomimetics; Thiophenes; Tumor Cells, Cultured

1988
(-)-pindolol and (+/-)-tertatolol affect rat hippocampal 5-HT levels through mechanisms involving not only 5-HT1A, but also 5-HT1B receptors.
    Neuropharmacology, 1996, Volume: 35, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Betaxolol; Hippocampus; Male; Microdialysis; Pindolol; Propanolamines; Rats; Receptors, Serotonin; Serotonin; Thiophenes

1996
Effects of (-)-tertatolol, (-)-penbutolol and (+/-)-pindolol in combination with paroxetine on presynaptic 5-HT function: an in vivo microdialysis and electrophysiological study.
    British journal of pharmacology, 1999, Volume: 127, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Antidepressive Agents; Drug Synergism; Electrophysiology; In Vitro Techniques; Male; Membrane Potentials; Microdialysis; Paroxetine; Patch-Clamp Techniques; Penbutolol; Pindolol; Propanolamines; Prosencephalon; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Presynaptic; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Thiophenes

1999
Pindolol suppresses serotonergic neuronal activity and does not block the inhibition of serotonergic neurons produced by 8-hydroxy-2-(di-n-propylamino)tetralin in awake cats.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 291, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Cats; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Neurons; Pindolol; Propanolamines; Raphe Nuclei; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Thiophenes

1999
Affinity of (+/-)-pindolol, (-)-penbutolol, and (-)-tertatolol for pre- and postsynaptic serotonin 5-HT(1A) receptors in human and rat brain.
    Journal of neurochemistry, 2000, Volume: 75, Issue:2

    Topics: Aged; Animals; Anti-Arrhythmia Agents; Autoradiography; Brain; Dentate Gyrus; Female; Hippocampus; Humans; Male; Penbutolol; Pindolol; Piperazines; Propanolamines; Pyridines; Radioligand Assay; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Presynaptic; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Synapses; Thiophenes; Tritium

2000