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tertatolol and 8-hydroxy-2-(di-n-propylamino)tetralin

tertatolol has been researched along with 8-hydroxy-2-(di-n-propylamino)tetralin in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's13 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Carrupt, PA; Gaillard, P; Schambel, P; Testa, B1
Bizot-Espiard, J; Costentin, J; Guardiola, B; Schiavi, P; Simon, P1
Laubie, M; Mennecier, P; Verbeuren, TJ1
Adrien, J; Fattaccini, CM; Gozlan, H; Guardiola-Lemaitre, B; Haj-Dahmane, S; Hamon, M; Jolas, T; Kidd, EJ; Lanfumey, L1
Andrews, N; File, SE; Gonzalez, LE; Hogg, S1
Emerit, MB; Hamon, M; Riad, M1
Artigas, F; Celada, P; Romero, L1
Cagnotto, A; De Blasi, A; Esposito, E; Mennini, T; Prisco, S; Talone, D1
Bietti, G; Borsini, F; Ceci, A; Donetti, A1
File, SE; Gonzalez, LE1
Assie, MB; Koek, W1
Andrews, N; File, SE; Gonzalez, LE1
Fornal, CA; Jacobs, BL; Martin, FJ; Metzler, CW1

Other Studies

13 other study(ies) available for tertatolol and 8-hydroxy-2-(di-n-propylamino)tetralin

ArticleYear
Binding of arylpiperazines, (aryloxy)propanolamines, and tetrahydropyridylindoles to the 5-HT1A receptor: contribution of the molecular lipophilicity potential to three-dimensional quantitative structure-affinity relationship models.
    Journal of medicinal chemistry, 1996, Jan-05, Volume: 39, Issue:1

    Topics: Indoles; Ligands; Models, Molecular; Molecular Conformation; Molecular Structure; Piperazines; Propanolamines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Structure-Activity Relationship; Tetrahydronaphthalenes

1996
5-HT1A receptor agonists prevent in rats the yawning and penile erections induced by direct dopamine agonists.
    Psychopharmacology, 1992, Volume: 108, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Aminoquinolines; Animals; Body Temperature; Buspirone; Chromans; Dopamine Agents; Male; Mice; Penile Erection; Propanolamines; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Serotonin; Spiro Compounds; Thiophenes; Yawning

1992
5-Hydroxytryptamine-induced vasodilatation in the isolated perfused rat kidney: are endothelial 5-HT1A receptors involved?
    European journal of pharmacology, 1991, Aug-16, Volume: 201, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Angiotensin II; Animals; Atrial Natriuretic Factor; Endothelium, Vascular; Kidney; Male; Nitroglycerin; Papaverine; Piperazines; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes; Thiophenes; Vasodilation

1991
(-)Tertatolol is a potent antagonist at pre- and postsynaptic serotonin 5-HT1A receptors in the rat brain.
    Naunyn-Schmiedeberg's archives of pharmacology, 1993, Volume: 347, Issue:5

    Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Brain; Electrophysiology; Hydroxyindoleacetic Acid; Isomerism; Male; Neurons; Propanolamines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Thiophenes

1993
5-HT1A receptors in the median raphe nucleus and dorsal hippocampus may mediate anxiolytic and anxiogenic behaviours respectively.
    European journal of pharmacology, 1994, Nov-03, Volume: 264, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Anxiety; Autoreceptors; Dendrites; Grooming; Hippocampus; Male; Motor Activity; Propanolamines; Raphe Nuclei; Rats; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Social Behavior; Thiophenes

1994
Neurotrophic effects of ipsapirone and other 5-HT1A receptor agonists on septal cholinergic neurons in culture.
    Brain research. Developmental brain research, 1994, Oct-14, Volume: 82, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Autoradiography; Brain; Cell Division; Cells, Cultured; Choline O-Acetyltransferase; Dose-Response Relationship, Drug; Female; Fetus; Immunohistochemistry; Nerve Growth Factors; Neurons; Piperazines; Pregnancy; Propanolamines; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiophenes; Tritium

1994
Reduction of in vivo striatal 5-hydroxytryptamine release by 8-OH-DPAT after inactivation of Gi/G(o) proteins in dorsal raphe nucleus.
    European journal of pharmacology, 1994, Nov-14, Volume: 265, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Autoreceptors; Citalopram; Corpus Striatum; GTP-Binding Proteins; Male; Pertussis Toxin; Potassium Channels; Propanolamines; Raphe Nuclei; Rats; Rats, Wistar; Serotonin; Thiophenes; Virulence Factors, Bordetella

1994
Tertatolol, a new beta-blocker, is a serotonin (5-hydroxytryptamine1A) receptor antagonist in rat brain.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain; Electrophysiology; Male; Membranes; Neurons; Propanolamines; Radioligand Assay; Raphe Nuclei; Rats; Serotonin Antagonists; Thiophenes

1993
BIMT 17, a 5-HT1A receptor agonist/5-HT2A receptor antagonist, directly activates postsynaptic 5-HT inhibitory responses in the rat cerebral cortex.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Antidepressive Agents; Benzimidazoles; Binding, Competitive; Buspirone; Cerebral Cortex; Dose-Response Relationship, Drug; In Vitro Techniques; Iontophoresis; Male; Microelectrodes; Neurons; Piperazines; Prazosin; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiophenes

1995
Anxiolytic effects in the plus-maze of 5-HT1A-receptor ligands in dorsal raphé and ventral hippocampus.
    Pharmacology, biochemistry, and behavior, 1996, Volume: 54, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Anti-Anxiety Agents; Anxiety; Hippocampus; Ligands; Male; Propanolamines; Raphe Nuclei; Rats; Receptors, Serotonin; Serotonin Receptor Agonists; Stereotaxic Techniques; Thiophenes

1996
(-)-pindolol and (+/-)-tertatolol affect rat hippocampal 5-HT levels through mechanisms involving not only 5-HT1A, but also 5-HT1B receptors.
    Neuropharmacology, 1996, Volume: 35, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Betaxolol; Hippocampus; Male; Microdialysis; Pindolol; Propanolamines; Rats; Receptors, Serotonin; Serotonin; Thiophenes

1996
5-HT1A and benzodiazepine receptors in the basolateral amygdala modulate anxiety in the social interaction test, but not in the elevated plus-maze.
    Brain research, 1996, Sep-02, Volume: 732, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholinesterase; Adrenergic beta-Antagonists; Amygdala; Analysis of Variance; Animals; Anxiety; GABA Modulators; Infusions, Parenteral; Male; Maze Learning; Midazolam; Motor Activity; Neurons; Propanolamines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists; Social Behavior; Thiophenes

1996
Pindolol suppresses serotonergic neuronal activity and does not block the inhibition of serotonergic neurons produced by 8-hydroxy-2-(di-n-propylamino)tetralin in awake cats.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 291, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Cats; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Neurons; Pindolol; Propanolamines; Raphe Nuclei; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Thiophenes

1999