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tert-butylbicyclophosphorothionate and ro 5-4864

tert-butylbicyclophosphorothionate has been researched along with ro 5-4864 in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19907 (46.67)18.7374
1990's8 (53.33)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kokka, N; Longoni, B; Olsen, RW; Sapp, DW; Turner, DM; Witte, U1
Kokka, N; Olsen, RW; Sapp, DW; Witte, U1
Belelli, D; Gee, KW; McCauley, L1
Eshleman, AJ; Murray, TF1
Gee, KW; Lawrence, LJ; Yamamura, HI1
Devaud, LL; Murray, TF1
Culp, S; Liljequist, S; Tabakoff, B1
Brinton, RE; Gee, KW; McEwen, BS1
Cott, J; Skolnick, P; Weber, KH; Weissman, BA1
Gee, KW1
Ramanjaneyulu, R; Ticku, MK1
Deutsch, SI; Koetzner, L; Lukacs, LG; Mastropaolo, J; Morn, C; Park, CH1
Chen, JS; Gee, KW; Johnson, D; Lan, NC1
Friend, JM; Gee, KW; Xue, BG1
Saederup, E; Squires, RF1

Reviews

1 review(s) available for tert-butylbicyclophosphorothionate and ro 5-4864

ArticleYear
Interactions of pyrethroid insecticides with chloride ionophore-associated binding sites.
    Neurotoxicology, 1985,Summer, Volume: 6, Issue:2

    Topics: Animals; Benzodiazepinones; Brain; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Drug Interactions; Guinea Pigs; Ion Channels; Picrotoxin; Pyrethrins; Radioligand Assay; Rats; Receptors, GABA-A; Sesterterpenes

1985

Other Studies

14 other study(ies) available for tert-butylbicyclophosphorothionate and ro 5-4864

ArticleYear
Regional variation in steroid anesthetic modulation of [35S]TBPS binding to gamma-aminobutyric acidA receptors in rat brain.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:2

    Topics: Anesthetics; Animals; Benzodiazepinones; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Dose-Response Relationship, Drug; Pregnanediones; Rats; Receptors, GABA-A

1992
Sex differences in sensitivity to pentylenetetrazol but not in GABAA receptor binding.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 43, Issue:2

    Topics: Anesthetics; Animals; Anticonvulsants; Autoradiography; Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Diazepam; Electroshock; Ethanol; Female; Flunitrazepam; Male; Muscimol; Orchiectomy; Ovariectomy; Pentylenetetrazole; Pregnanediones; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Seizures; Sex Characteristics

1992
Heterotropic cooperativity between putative recognition sites for progesterone metabolites and the atypical benzodiazepine Ro 5-4864.
    Journal of neurochemistry, 1990, Volume: 55, Issue:1

    Topics: Animals; Benzodiazepinones; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Convulsants; gamma-Aminobutyric Acid; Male; Pregnanediol; Pregnanolone; Progesterone; Rats; Rats, Inbred Strains

1990
Dependence on gamma-aminobutyric acid of pyrethroid and 4'-chlorodiazepam modulation of the binding of t-[35S]butylbicyclophosphorothionate in piscine brain.
    Neuropharmacology, 1990, Volume: 29, Issue:7

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; gamma-Aminobutyric Acid; Kinetics; Nitriles; Pyrethrins; Receptors, GABA-A; Trout

1990
Involvement of peripheral-type benzodiazepine receptors in the proconvulsant actions of pyrethroid insecticides.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 247, Issue:1

    Topics: Animals; Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Dose-Response Relationship, Drug; In Vitro Techniques; Ion Channels; Isoquinolines; Male; Pyrethrins; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stereoisomerism

1988
The effect of ethanol on 35S-TBPS binding to mouse brain membranes in the presence of chloride.
    Pharmacology & toxicology, 1989, Volume: 65, Issue:5

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Benzodiazepinones; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Diazepam; Drug Tolerance; Ethanol; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred C57BL; Pentobarbital; Substance-Related Disorders; Sulfur Radioisotopes

1989
Regional distribution of a Ro5 4864 binding site that is functionally coupled to the gamma-aminobutyric acid/benzodiazepine receptor complex in rat brain.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:1

    Topics: Affinity Labels; Animals; Autoradiography; Azides; Benzodiazepines; Benzodiazepinones; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Clonazepam; Male; Photochemistry; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
Are "peripheral-type" binding sites for benzodiazepines in brain related to the convulsant actions of Ro 5-4864?
    Progress in clinical and biological research, 1985, Volume: 192

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Structure-Activity Relationship

1985
Phenylquinolines PK 8165 and PK 9084 allosterically modulate [35S]t-butylbicyclophosphorothionate binding to a chloride ionophore in rat brain via a novel Ro5 4864 binding site.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 240, Issue:3

    Topics: Animals; Anticonvulsants; Benzodiazepinones; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Convulsants; gamma-Aminobutyric Acid; Kinetics; Male; Quinolines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1987
RO5-4864 inhibits the binding of [35S]t-butylbicyclophosphorothionate to rat brain membranes.
    Life sciences, 1984, Feb-13, Volume: 34, Issue:7

    Topics: Androstanes; Animals; Azasteroids; Benzodiazepinones; Bicuculline; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Cell Membrane; Cerebellum; Cerebral Cortex; Dose-Response Relationship, Drug; Flumazenil; Hippocampus; Male; Picrotoxin; Radioligand Assay; Rats

1984
MK-801 alters the GABAA receptor complex and potentiates flurazepam's antiseizure efficacy.
    Pharmacology, biochemistry, and behavior, 1995, Volume: 51, Issue:4

    Topics: Animals; Anticonvulsants; Behavior, Animal; Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Convulsants; Dizocilpine Maleate; Drug Synergism; Electroshock; Flurazepam; Isoquinolines; Kinetics; Male; Mice; Receptors, GABA-A

1995
Differential effects of 4'-chlorodiazepam on expressed human GABAA receptors.
    Journal of neurochemistry, 1995, Volume: 64, Issue:2

    Topics: Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Clonazepam; Flumazenil; Humans; Quinolines; Receptors, GABA; Transfection

1995
Loreclezole modulates [35S]t-butylbicyclophosphorothionate and [3H]flunitrazepam binding via a distinct site on the GABAA receptor complex.
    European journal of pharmacology, 1996, Apr-04, Volume: 300, Issue:1-2

    Topics: Animals; Anticonvulsants; Benzodiazepinones; Binding Sites; Brain; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Drug Interactions; Flunitrazepam; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA; Triazoles

1996
Clozapine and some other antipsychotic drugs may preferentially block the same subset of GABA(A) receptors.
    Neurochemical research, 1997, Volume: 22, Issue:2

    Topics: Animals; Antidepressive Agents; Antipsychotic Agents; Benzodiazepines; Benzodiazepinones; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Clozapine; Drug Synergism; GABA Antagonists; gamma-Aminobutyric Acid; Naloxone; Prosencephalon; Rats; Receptors, GABA

1997