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tert-butylbicyclophosphorothionate and flumazenil

tert-butylbicyclophosphorothionate has been researched along with flumazenil in 32 studies

Research

Studies (32)

TimeframeStudies, this research(%)All Research%
pre-19909 (28.13)18.7374
1990's21 (65.63)18.2507
2000's2 (6.25)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kukulka, KM; Mans, AM; McAvoy, KJ; Rokosz, NC1
Byrnes, JJ; Galpern, WR; Greenblatt, DJ; Miller, LG; Shader, RI1
Galpern, WR; Greenblatt, DJ; Lumpkin, M; Miller, LG; Shader, RI2
Blakeman, DP; Im, WB1
Basile, AS1
Kulkarni, SK; Ticku, MK1
Danielou, G; Lloyd, GK; Thuret, F1
Havoundjian, H; Skolnick, P; Trullas, R1
Greenblatt, DJ; Miller, LG; Roy, RB; Shader, RI; Summer, WR1
McIntyre, TD; Skolnick, P; Trullas, R1
Greenblatt, DJ; Lopez, F; Miller, LG; Roy, RB; Wecker, L1
Gaver, A; Greenblatt, DJ; Lopez, F; Miller, LG; Roy, RB; Shader, RI1
Engelstoft, M; Hansen, JB; Honoré, T; Jensen, LH; Schmiechen, R; Wätjen, F1
Haefely, W; Möhler, H; Richards, JG; Schoch, P1
Cohen, RM; Havoundjian, H; Paul, SM; Skolnick, P1
Ramanjaneyulu, R; Ticku, MK1
Carter, DB; Hamilton, BJ; Im, HK; Im, WB; Jacobsen, EJ; Pregenzer, JF1
Gruber, L; Maksay, G; Molnár, P1
Biggio, G; Concas, A; Cuccheddu, T; Maciocco, E; Santoro, G; Serra, M1
Chen, JS; Gee, KW; Johnson, D; Lan, NC1
Basile, AS; Drugan, RC; Ferland, RJ; Ha, JH1
Harris, RA; Klein, RL; McQuilkin, SJ; Sanna, E; Whiting, PJ1
Biggio, G; Cuccheddu, T; Floris, S; Ghiani, CA; Giusti, P; Motzo, C; Serra, M1
Hu, XJ; Ticku, MK1
Airaksinen, MM; Nieminen, SA; Railoma, O; Titievsky, AV1
Deutsch, SI; Hitri, A; Lukacs, LG; Park, CH1
Ai, J; Dekermendjian, K; Nielsen, M; Shan, R; Sterner, O; Witt, MR1
Hedblom, E; Kirkness, EF1
Gillardin, JM; Schlichter, R; Verleye, M1
Gillardin, J; Poisbeau, P; Rybalchenko, V; Schlichter, R; Verleye, M1
Atack, JR; Bromidge, F; Collinson, N; Dawson, GR; Hadingham, KL; Howell, O; Macaulay, A; McKernan, RM; Myers, J; Newman, R; O'Meara, G; Reynolds, DS; Rosahl, TW; Sur, C; Wafford, KA; Whiting, PJ1

Reviews

1 review(s) available for tert-butylbicyclophosphorothionate and flumazenil

ArticleYear
Benzodiazepine receptors resolved.
    Experientia, 1986, Feb-15, Volume: 42, Issue:2

    Topics: Animals; Antibodies, Monoclonal; Autoradiography; Benzodiazepines; Benzodiazepinones; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Chlorides; Clonazepam; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Histocytochemistry; Humans; Immunologic Techniques; Ionophores; Muscimol; Neurons; Radioisotopes; Radioligand Assay; Receptors, GABA-A; Spinal Cord; Synapses; Tissue Distribution

1986

Other Studies

31 other study(ies) available for tert-butylbicyclophosphorothionate and flumazenil

ArticleYear
Regional distribution and kinetics of three sites on the GABAA receptor: lack of effect of portacaval shunting.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1992, Volume: 12, Issue:2

    Topics: Animals; Autoradiography; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Flumazenil; Flunitrazepam; Image Processing, Computer-Assisted; Kinetics; Male; Muscimol; Portacaval Shunt, Surgical; Rats; Rats, Inbred Strains; Receptors, GABA-A; Tissue Distribution

1992
Chronic benzodiazepine administration. X. Concurrent administration of the peripheral-type benzodiazepine ligand PK11195 attenuates chronic effects of lorazepam.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:1

    Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Down-Regulation; Flumazenil; Isoquinolines; Ligands; Lorazepam; Male; Mice; Motor Activity; Receptors, GABA-A

1992
Chronic benzodiazepine administration. VII. Behavioral tolerance and withdrawal and receptor alterations associated with clonazepam administration.
    Psychopharmacology, 1991, Volume: 104, Issue:2

    Topics: Animals; Behavior, Animal; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Clonazepam; Convulsants; Drug Tolerance; Flumazenil; Male; Mice; Motor Activity; Muscimol; Receptors, GABA-A; Substance Withdrawal Syndrome

1991
Modification of gamma-aminobutyric acidA receptor binding and function by N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline in vitro and in vivo: effects of aging.
    Journal of neurochemistry, 1991, Volume: 56, Issue:4

    Topics: Aging; Animals; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Cerebral Cortex; Dose-Response Relationship, Drug; Flumazenil; gamma-Aminobutyric Acid; Kinetics; Lorazepam; Male; Mice; Mice, Inbred Strains; Quinolines; Receptors, GABA-A

1991
Correlation between gamma-aminobutyric acidA receptor ligand-induced changes in t-butylbicyclophosphoro[35S]thionate binding and 36Cl- uptake in rat cerebrocortical membranes.
    Molecular pharmacology, 1991, Volume: 39, Issue:3

    Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cerebral Cortex; Chloride Channels; Chlorides; Desoxycorticosterone; Diazepam; Ethanol; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Ligands; Membrane Proteins; Pentobarbital; Pregnanolone; Rats; Receptors, GABA-A; Synaptosomes

1991
The contribution of endogenous benzodiazepine receptor ligands to the pathogenesis of hepatic encephalopathy.
    Synapse (New York, N.Y.), 1991, Volume: 7, Issue:2

    Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chromatography, High Pressure Liquid; Diazepam; Flumazenil; Hepatic Encephalopathy; Kinetics; Ligands; Male; Mass Spectrometry; Muscimol; Peripheral Nerves; Rabbits; Radioligand Assay; Receptors, GABA-A; Sulfur Radioisotopes

1991
Chronic benzodiazepine antagonist treatment and its withdrawal upregulates components of GABA-benzodiazepine receptor ionophore complex in cerebral cortex of rat.
    Brain research, 1990, Jun-11, Volume: 519, Issue:1-2

    Topics: Affinity Labels; Animals; Azides; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Convulsants; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reference Values; Up-Regulation

1990
The activity of zolpidem and other hypnotics within the gamma-aminobutyric acid (GABAA) receptor supramolecular complex, as determined by 35S-t-butylbicyclophosphorothionate (35S-TBPS) binding to rat cerebral cortex membranes.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 255, Issue:2

    Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Hypnotics and Sedatives; In Vitro Techniques; Male; Pyridines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Zolpidem

1990
Stress-induced changes in t-[35S]butylbicyclophosphorothionate binding to gamma-aminobutyric acid-gated chloride channels are mimicked by in vitro occupation of benzodiazepine receptors.
    Journal of neurochemistry, 1987, Volume: 49, Issue:3

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cerebral Cortex; Chlorides; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Ion Channels; Kinetics; Male; Membranes; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological; Swimming

1987
Chronic benzodiazepine administration. II. Discontinuation syndrome is associated with upregulation of gamma-aminobutyric acidA receptor complex binding and function.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:1

    Topics: Animals; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Drug Tolerance; Flumazenil; Flunitrazepam; Ion Channels; Lorazepam; Male; Mice; Motor Activity; Muscimol; Receptors, GABA-A; Time Factors

1988
Asymmetrical activation of GABA-gated chloride channels in cerebral cortex.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 30, Issue:4

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Flumazenil; Functional Laterality; Ion Channels; Kinetics; Male; Organ Specificity; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
Dietary choline intake modulates benzodiazepine receptor binding and gamma-aminobutyric acidA receptor function in mouse brain.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:1

    Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; Choline; Diet; Flumazenil; Male; Membrane Proteins; Mice; Motor Activity; Receptors, GABA-A

1989
Chronic benzodiazepine administration. III. Upregulation of gamma-aminobutyric acidA receptor binding and function associated with chronic benzodiazepine antagonist administration.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:3

    Topics: Animals; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Chlorides; Flumazenil; Male; Membrane Proteins; Mice; Motor Activity; Receptors, GABA-A

1989
Oxadiazolylimidazobenzodiazepines, a new class of benzodiazepine receptor ligands.
    Advances in biochemical psychopharmacology, 1988, Volume: 45

    Topics: Animals; Avoidance Learning; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Conflict, Psychological; Convulsants; Flumazenil; Ligands; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
Differential sensitivity of "central" and "peripheral" type benzodiazepine receptors to phospholipase A2.
    Journal of neurochemistry, 1986, Volume: 46, Issue:3

    Topics: Animals; Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cerebral Cortex; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Kidney; Male; Myocardium; Pentobarbital; Phospholipases; Phospholipases A; Phospholipases A2; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A

1986
RO5-4864 inhibits the binding of [35S]t-butylbicyclophosphorothionate to rat brain membranes.
    Life sciences, 1984, Feb-13, Volume: 34, Issue:7

    Topics: Androstanes; Animals; Azasteroids; Benzodiazepinones; Bicuculline; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Cell Membrane; Cerebellum; Cerebral Cortex; Dose-Response Relationship, Drug; Flumazenil; Hippocampus; Male; Picrotoxin; Radioligand Assay; Rats

1984
Characterization of U-97775 as a GABAA receptor ligand of dual functionality in cloned rat GABAA receptor subtypes.
    British journal of pharmacology, 1995, Volume: 115, Issue:1

    Topics: Animals; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Chlorides; Electrophysiology; Flumazenil; Humans; Imidazoles; Ligands; Quinoxalines; Rats; Receptors, GABA-A; Recombinant Proteins

1995
Common modes of action of gamma-butyrolactones and pentylenetetrazol on the GABAA receptor-ionophore complex.
    European journal of pharmacology, 1994, Dec-15, Volume: 288, Issue:1

    Topics: 4-Butyrolactone; Androstanes; Animals; Azasteroids; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Cerebral Cortex; Convulsants; Electrophysiology; Flumazenil; GABA Antagonists; Ionophores; Male; Neurons; Patch-Clamp Techniques; Pentylenetetrazole; Prosencephalon; Rats; Rats, Wistar; Receptors, GABA-A; Stereoisomerism; Synaptosomes

1994
The effect of cyclopyrrolones on GABAA receptor function is different from that of benzodiazepines.
    Naunyn-Schmiedeberg's archives of pharmacology, 1994, Volume: 350, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Benzodiazepines; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Chlorine; Flumazenil; Hypnotics and Sedatives; Kinetics; Male; Mice; Mice, Inbred Strains; Muscimol; Naphthyridines; Piperazines; Radioisotopes; Receptors, GABA-A; Sulfur Compounds; Sulfur Radioisotopes; Tritium

1994
Differential effects of 4'-chlorodiazepam on expressed human GABAA receptors.
    Journal of neurochemistry, 1995, Volume: 64, Issue:2

    Topics: Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Clonazepam; Flumazenil; Humans; Quinolines; Receptors, GABA; Transfection

1995
The protective effects of stress control may be mediated by increased brain levels of benzodiazepine receptor agonists.
    Brain research, 1994, Oct-24, Volume: 661, Issue:1-2

    Topics: Analysis of Variance; Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Convulsants; Electroshock; Escape Reaction; Flumazenil; GABA-A Receptor Agonists; Hippocampus; Male; Picrotoxin; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Seizures; Sesterterpenes; Stress, Psychological; Strychnine; Sulfur Radioisotopes; Tritium

1994
Effects of 5-HT3 receptor antagonists on binding and function of mouse and human GABAA receptors.
    European journal of pharmacology, 1994, Jul-15, Volume: 268, Issue:2

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Flumazenil; Flunitrazepam; Humans; Indazoles; Indoles; Male; Mice; Mice, Inbred ICR; Receptors, GABA-A; Serotonin Antagonists; Tropanes; Tropisetron; Xenopus laevis

1994
Imidazenil, a new partial agonist of benzodiazepine receptors, reverses the inhibitory action of isoniazid and stress on gamma-aminobutyric acidA receptor function.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 269, Issue:1

    Topics: Animals; Benzodiazepines; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Flumazenil; GABA-A Receptor Antagonists; Imidazoles; Isoniazid; Male; Mice; Mice, Inbred Strains; Pentylenetetrazole; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Seizures; Stress, Physiological; Sulfur Radioisotopes; Tritium

1994
Chronic benzodiazepine agonist treatment produces functional uncoupling of the gamma-aminobutyric acid-benzodiazepine receptor ionophore complex in cortical neurons.
    Molecular pharmacology, 1994, Volume: 45, Issue:4

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Cerebral Cortex; Chloride Channels; Female; Flumazenil; Flurazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Ion Channel Gating; Macromolecular Substances; Male; Mice; Mice, Inbred C57BL; Nerve Tissue Proteins; Receptors, GABA; Receptors, GABA-A

1994
Influence of flumazenil on the learning-enhancing effect of ambocarb in rats.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 47, Issue:3

    Topics: Animals; Behavior, Animal; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Discrimination Learning; Discrimination, Psychological; Flumazenil; Flunitrazepam; Harmine; Learning; Ligands; Male; Muscimol; Rats; Rats, Wistar; Receptors, GABA-A

1994
Swim stress selectively alters the specific binding of a benzodiazepine antagonist in mice.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 45, Issue:2

    Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Flumazenil; Flurazepam; In Vitro Techniques; Kinetics; Male; Mice; Receptors, GABA-A; Stress, Physiological; Swimming; Tissue Distribution

1993
Characterisation of the furanocoumarin phellopterin as a rat brain benzodiazepine receptor partial agonist in vitro.
    Neuroscience letters, 1996, Nov-29, Volume: 219, Issue:3

    Topics: Animals; Binding Sites; Brain; Bridged Bicyclo Compounds, Heterocyclic; Coumarins; Diazepam; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; In Vitro Techniques; Male; Rats; Rats, Wistar; Receptors, GABA; Receptors, GABA-A

1996
A novel class of GABAA receptor subunit in tissues of the reproductive system.
    The Journal of biological chemistry, 1997, Jun-13, Volume: 272, Issue:24

    Topics: Amino Acid Sequence; Animals; Base Sequence; Binding Sites; Bridged Bicyclo Compounds, Heterocyclic; Cloning, Molecular; DNA, Complementary; Flumazenil; Humans; Molecular Sequence Data; Muscimol; Radioligand Assay; Rats; Receptors, GABA-A; RNA, Messenger

1997
Interactions of etifoxine with the chloride channel coupled to the GABA(A) receptor complex.
    Neuroreport, 1999, Oct-19, Volume: 10, Issue:15

    Topics: Animals; Anticonvulsants; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Cerebral Cortex; Chloride Channels; Convulsants; Flumazenil; GABA Modulators; Kinetics; Male; Mice; Oxazines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

1999
Modulation of GABAergic synaptic transmission by the non-benzodiazepine anxiolytic etifoxine.
    Neuropharmacology, 2000, Jul-10, Volume: 39, Issue:9

    Topics: Animals; Behavior, Animal; Bicuculline; Binding, Competitive; Brain; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Dose-Response Relationship, Drug; Drinking Behavior; Flumazenil; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hypothalamus; Isoquinolines; Male; Membrane Potentials; Membranes; Neurons; Oxazines; Patch-Clamp Techniques; Posterior Horn Cells; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, GABA-A; Sulfur Radioisotopes; Synaptic Transmission; Tetrodotoxin; Tranquilizing Agents

2000
Loss of the major GABA(A) receptor subtype in the brain is not lethal in mice.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2001, May-15, Volume: 21, Issue:10

    Topics: Animals; Autoradiography; Behavior, Animal; Binding, Competitive; Brain; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Electrophysiology; Flumazenil; Gait Disorders, Neurologic; Gene Expression; Homozygote; Ligands; Mice; Mice, Inbred Strains; Mice, Knockout; Motor Activity; Muscimol; Protein Subunits; Purkinje Cells; Radioligand Assay; Receptors, GABA-A; Survival Rate; Tissue Distribution

2001