tert-butylbicyclophosphorothionate has been researched along with diazepam in 47 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 18 (38.30) | 18.7374 |
| 1990's | 26 (55.32) | 18.2507 |
| 2000's | 3 (6.38) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Kokka, N; Olsen, RW; Sapp, DW; Witte, U | 1 |
| Maksay, G; Simonyi, M; Tegyey, Z | 1 |
| Biggio, G; Concas, A; Mascia, MP; Sanna, E; Santoro, G; Serra, M | 1 |
| Gee, KW; Lan, NC | 1 |
| Biggio, G; Concas, A; Sanna, E; Serra, M | 1 |
| Biggio, G; Concas, A; Sanna, E; Santoro, G; Serra, M | 1 |
| Biggio, G; Concas, A; Foddi, C; Sanna, E; Serra, M | 1 |
| Niles, L | 1 |
| Blakeman, DP; Im, WB | 1 |
| Basile, AS | 1 |
| Biggio, G; Concas, A; Mascia, MP; Sanna, E; Santoro, V; Serra, M | 1 |
| Andrews, JS; Jensen, LH; Kehr, W; Petersen, EN; Rettig, KJ; Schmiechen, R; Schneider, HH; Stephens, DN; Turner, JD; Turski, L | 1 |
| Badyshtov, BA; Gordey, ML; Nagovitsina, YA; Seredenin, SB | 1 |
| Biggio, G; Concas, A; Mascia, MP; Sanna, E; Serra, M | 1 |
| Maggi, A; Perez, J; Zucchi, I | 1 |
| Bleck, V; Harris, RA; Lewin, E; Peris, J; Zahniser, NR | 1 |
| Biggio, G; Concas, A; Corda, MG; Serra, M | 1 |
| Biggio, G; Sanna, E; Serra, M | 1 |
| Abel, MS; Blume, AJ; Garrett, KM | 1 |
| Biggio, G; Pepitoni, S; Sanna, E; Serra, M | 1 |
| Culp, S; Liljequist, S; Tabakoff, B | 1 |
| Böser, S; Klotz, KN; Lohse, MJ; Schwabe, U | 1 |
| Maksay, G; Simonyi, M | 1 |
| Gallager, DW; Heninger, C | 1 |
| Atsoggiu, T; Biggio, G; Concas, A; Serra, M | 1 |
| Schneider, HH; Stephens, DN | 1 |
| Creveling, CR; Daly, JW; Hollingsworth, EB; Lewandowski, G; Waters, JA | 1 |
| Chow, SC; Holan, G; Johnston, GA; Lummis, SC | 1 |
| Crofton, KM; Mailman, RB; Reiter, LW | 1 |
| Gallo, V; Guidotti, A; Vaccarino, F; Wise, BC | 1 |
| Braestrup, C; Tacke, U | 1 |
| Ramanjaneyulu, R; Ticku, MK | 1 |
| Cancedda, E; Corda, MG; Giorgi, O; Lecca, D; Orlandi, M | 1 |
| Biggio, G; Concas, A; Dazzi, L; Maciocco, E; Mascia, MP; Santoro, G | 1 |
| Bishop, M; Carter, ML; Huff, RA; Schwartz, RD; Yu, X | 1 |
| Ho, IK; Ito, Y | 1 |
| Cancedda, E; Corda, MG; Giorgi, O | 1 |
| Biggio, G; Concas, A; Dazzi, L; Maciocco, E; Mascia, MP; Ongini, E; Santoro, G | 1 |
| Korpi, ER; Seeburg, PH | 1 |
| Liljequist, S; Tabakoff, B | 1 |
| Biggio, G; Ghiani, CA; Maciocco, E; Sanna, E; Serra, M; Tuligi, G | 1 |
| Ai, J; Dekermendjian, K; Nielsen, M; Shan, R; Sterner, O; Witt, MR | 1 |
| Biggio, G; Casula, A; Maciocco, E; Murgia, A; Sanna, E; Tuligi, G; Usala, M | 1 |
| Firestone, LL; Homanics, GE; Korpi, ER; Mäkelä, R; Quinlan, JJ; Uusi-Oukari, M; Wisden, W | 1 |
| Korpi, ER; Uusi-Oukari, M; Vekovischeva, O | 1 |
| Daly, JW; Padgett, WL; Shi, D | 1 |
| Biggio, G; Busonero, F; Maciocco, E; Mostallino, MC; Mura, ML; Pisu, MG; Sanna, E; Serra, M; Talani, G | 1 |
47 other study(ies) available for tert-butylbicyclophosphorothionate and diazepam
| Article | Year |
|---|---|
Sex differences in sensitivity to pentylenetetrazol but not in GABAA receptor binding.
Topics: Anesthetics; Animals; Anticonvulsants; Autoradiography; Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Diazepam; Electroshock; Ethanol; Female; Flunitrazepam; Male; Muscimol; Orchiectomy; Ovariectomy; Pentylenetetrazole; Pregnanediones; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Seizures; Sex Characteristics | 1992 |
Central benzodiazepine receptors: in vitro efficacies and potencies of 3-substituted 1,4-benzodiazepine stereoisomers.
Topics: Allosteric Regulation; Animals; Benzodiazepines; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; In Vitro Techniques; Male; Protein Conformation; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stereoisomerism; Structure-Activity Relationship | 1991 |
"In vivo" administration of valproate decreases t-[35S]butylbicyclophosphorothionate binding in the rat brain.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Depression, Chemical; Diazepam; Kinetics; Male; Membranes; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sulfur Radioisotopes; Valproic Acid | 1991 |
Gamma-aminobutyric acidA receptor complexes in rat frontal cortex and spinal cord show differential responses to steroid modulation.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Desoxycorticosterone; Diazepam; gamma-Aminobutyric Acid; Ionophores; Male; Pentobarbital; Pregnanediol; Pregnanolone; Rats; Rats, Inbred Strains; Receptors, GABA-A; Spinal Cord; Steroids; Sulfur Radioisotopes | 1991 |
In vivo administration of ethanol enhances the function of the gamma-aminobutyric acid-dependent chloride channel in the rat cerebral cortex.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Diazepam; Ethanol; gamma-Aminobutyric Acid; Ion Channels; Isoniazid; Male; Rats; Rats, Inbred Strains | 1990 |
Ex vivo binding of t-[35S )butylbicyclophosphorothionate: a biochemical tool to study the pharmacology of ethanol at the gamma-aminobutyric acid-coupled chloride channel.
Topics: Animals; Azides; Benzodiazepines; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Diazepam; Drug Interactions; Ethanol; gamma-Aminobutyric Acid; Ion Channels; Isoniazid; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sulfur Radioisotopes | 1991 |
Failure of gamma-hydroxybutyrate to alter the function of the GABAA receptor complex in the rat cerebral cortex.
Topics: Animals; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Diazepam; Flunitrazepam; In Vitro Techniques; Ion Channels; Isoniazid; Male; Nerve Tissue Proteins; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sodium Oxybate; Synaptic Transmission | 1991 |
Melatonin interaction with the benzodiazepine-GABA receptor complex in the CNS.
Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Cerebral Cortex; Chlorides; Diazepam; gamma-Aminobutyric Acid; Humans; Ion Channel Gating; Ion Channels; Melatonin; Muscimol; Prosencephalon; Rats; Receptors, GABA-A; Serotonin; Synaptosomes | 1991 |
Correlation between gamma-aminobutyric acidA receptor ligand-induced changes in t-butylbicyclophosphoro[35S]thionate binding and 36Cl- uptake in rat cerebrocortical membranes.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cerebral Cortex; Chloride Channels; Chlorides; Desoxycorticosterone; Diazepam; Ethanol; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Ligands; Membrane Proteins; Pentobarbital; Pregnanolone; Rats; Receptors, GABA-A; Synaptosomes | 1991 |
The contribution of endogenous benzodiazepine receptor ligands to the pathogenesis of hepatic encephalopathy.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chromatography, High Pressure Liquid; Diazepam; Flumazenil; Hepatic Encephalopathy; Kinetics; Ligands; Male; Mass Spectrometry; Muscimol; Peripheral Nerves; Rabbits; Radioligand Assay; Receptors, GABA-A; Sulfur Radioisotopes | 1991 |
"Ex vivo" binding of 35S-TBPS as a tool to study the pharmacology of GABAA receptors.
Topics: Alprazolam; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Convulsants; Diazepam; Drug Synergism; Ethanol; In Vitro Techniques; Isoniazid; Male; Protein Conformation; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological; Sulfur Radioisotopes; Valproic Acid | 1990 |
Abecarnil, a metabolically stable, anxioselective beta-carboline acting at benzodiazepine receptors.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Diazepam; Female; Lorazepam; Male; Mice; Motor Activity; Punishment; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1990 |
Pharmacogenetic analysis of mechanisms of emotional stress: effects of benzodiazepines.
Topics: Adrenocorticotropic Hormone; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Corticosterone; Diazepam; Exploratory Behavior; Hybridization, Genetic; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Motor Activity; Receptors, GABA-A; Stress, Psychological | 1990 |
Diazepam enhances bicuculline-induced increase of t-[35S]butylbicyclophosphorothionate binding in unwashed membrane preparations from rat cerebral cortex.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cerebral Cortex; Convulsants; Diazepam; gamma-Aminobutyric Acid; Male; Rats; Rats, Inbred Strains; Subcellular Fractions | 1990 |
Estrogen modulation of the gamma-aminobutyric acid receptor complex in the central nervous system of rat.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; Dose-Response Relationship, Drug; Estrogens; Female; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; RNA; Seizures | 1988 |
Diazepam sensitizes mice to FG 7142 and reduces muscimol-stimulated 36Cl- flux.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Chlorides; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Ion Channels; Kindling, Neurologic; Mice; Mice, Inbred ICR; Muscimol | 1989 |
Enhancement of GABAergic transmission by zolpidem, an imidazopyridine with preferential affinity for type I benzodiazepine receptors.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; gamma-Aminobutyric Acid; Hypnotics and Sedatives; Male; Muscimol; Pyridines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Transmission; Zolpidem | 1989 |
Isoniazid, an inhibitor of GABAergic transmission, enhances [35S]TBPS binding in rat cerebral cortex.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cerebral Cortex; Convulsants; Diazepam; gamma-Aminobutyric Acid; Isoniazid; Male; Membranes; Rats; Rats, Inbred Strains; Sulfur Radioisotopes; Synaptic Transmission | 1989 |
Differential effects of iodide and chloride on allosteric interactions of the GABAA receptor.
Topics: Allosteric Regulation; Animals; Anions; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Chlorides; Diazepam; gamma-Aminobutyric Acid; Iodides; Male; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1989 |
Dramatic increase in nigral t-[35S]butylbicyclophosphorothionate binding sites elicited by the degeneration of the striato-nigral GABAergic pathway: reversal by diazepam.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Corpus Striatum; Diazepam; gamma-Aminobutyric Acid; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra | 1989 |
The effect of ethanol on 35S-TBPS binding to mouse brain membranes in the presence of chloride.
Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Benzodiazepinones; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Diazepam; Drug Tolerance; Ethanol; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred C57BL; Pentobarbital; Substance-Related Disorders; Sulfur Radioisotopes | 1989 |
Affinities of barbiturates for the GABA-receptor complex and A1 adenosine receptors: a possible explanation of their excitatory effects.
Topics: Animals; Barbiturates; Binding, Competitive; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; In Vitro Techniques; Male; Methohexital; Phenylisopropyladenosine; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Purinergic | 1987 |
Nonequilibrium modulation of 35S-TBPS binding by benzodiazepine agonists and antagonists.
Topics: Animals; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Diazepam; Flunitrazepam; In Vitro Techniques; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Structure-Activity Relationship | 1988 |
Altered gamma-aminobutyric acid/benzodiazepine interaction after chronic diazepam exposure.
Topics: Animals; Benzodiazepines; Bicuculline; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Diazepam; gamma-Aminobutyric Acid; Ionophores; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Time Factors | 1988 |
Foot-shock stress and anxiogenic beta-carbolines increase t-[35S]butylbicyclophosphorothionate binding in the rat cerebral cortex, an effect opposite to anxiolytics and gamma-aminobutyric acid mimetics.
Topics: Animals; Anti-Anxiety Agents; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Cell Membrane; Cerebral Cortex; Convulsants; Diazepam; Electroshock; GABA Antagonists; gamma-Aminobutyric Acid; Kinetics; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological | 1988 |
Tolerance to the benzodiazepine diazepam in an animal model of anxiolytic activity.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Diazepam; Drug Tolerance; Female; gamma-Aminobutyric Acid; Lorazepam; Male; Mice; Punishment; Receptors, GABA-A | 1985 |
Anticonvulsant activity of piperidinol and (dialkylamino)alkanol esters.
Topics: Amino Alcohols; Animals; Anticonvulsants; Ataxia; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Diazepam; Electroshock; Esters; Muscimol; Pentylenetetrazole; Phenytoin; Piperidines; Rats; Receptors, GABA-A; Structure-Activity Relationship | 1986 |
gamma-Aminobutyric acid receptor ionophore complexes: differential effects of deltamethrin, dichlorodiphenyltrichloroethane, and some novel insecticides in a rat brain membrane preparation.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; DDT; Diazepam; Insecticides; Ionophores; Male; Muscimol; Nitriles; Pyrethrins; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1987 |
Pyrethroid insecticides and radioligand displacement from the GABA receptor chloride ionophore complex.
Topics: Animals; Binding, Competitive; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; Flunitrazepam; Male; Muscimol; Nitriles; Permethrin; Pyrethrins; Rats; Receptors, GABA-A | 1987 |
gamma-Aminobutyric acid- and benzodiazepine-induced modulation of [35S]-t-butylbicyclophosphorothionate binding to cerebellar granule cells.
Topics: Animals; Benzodiazepines; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Cerebellum; Diazepam; gamma-Aminobutyric Acid; Granulocytes; Muscimol; Picrotoxin; Rats; Sulfur Radioisotopes; Temperature | 1985 |
A study on benzodiazepine receptor binding in audiogenic seizure-susceptible rats.
Topics: Acoustic Stimulation; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Convulsants; Diazepam; Female; Flunitrazepam; In Vitro Techniques; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures | 1984 |
Binding characteristics and interactions of depressant drugs with [35S]t-butylbicyclophosphorothionate, a ligand that binds to the picrotoxinin site.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Convulsants; Diazepam; Etomidate; gamma-Aminobutyric Acid; Male; Membranes; Pentobarbital; Picrotoxin; Psychotropic Drugs; Rats; Rats, Inbred Strains; Sesterterpenes | 1984 |
Allosteric modulation of [35S]TBPS-binding in the cerebral cortex of the rat during postnatal development.
Topics: Aging; Allosteric Regulation; Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Convulsants; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Stereoisomerism; Sulfur Radioisotopes | 1994 |
Effects of propofol, pentobarbital and alphaxalone on t-[35S]butylbicyclophosphorothionate binding in rat cerebral cortex.
Topics: Anesthetics; Animals; Bicuculline; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Diazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Ion Channel Gating; Male; Membranes; Pentobarbital; Pregnanediones; Propofol; Rats; Rats, Sprague-Dawley; Sulfur Radioisotopes | 1994 |
Postischemic diazepam is neuroprotective in the gerbil hippocampus.
Topics: Animals; Body Temperature; Brain Ischemia; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Survival; Diazepam; Gerbillinae; Hippocampus; Male; Motor Activity; Rectum | 1994 |
Studies on picrotoxin binding sites of GABAA receptors in rat cortical synaptoneurosomes.
Topics: Animals; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorine; Desoxycorticosterone; Diazepam; In Vitro Techniques; Male; Membranes; Muscimol; Pentobarbital; Picrotoxin; Radioisotopes; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Steroids; Synaptosomes | 1994 |
Modulation of 35S-TBPS binding by GABAergic drugs in the cerebral cortex of newborn and adult rats.
Topics: Aging; Animals; Animals, Newborn; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cell Membrane; Cerebral Cortex; Convulsants; Diazepam; gamma-Aminobutyric Acid; Kinetics; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sulfur Radioisotopes | 1993 |
Anticonvulsant doses of 2-chloro-N6-cyclopentyladenosine, an adenosine A1 receptor agonist, reduce GABAergic transmission in different areas of the mouse brain.
Topics: Adenosine; Animals; Anticonvulsants; Behavior, Animal; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Depression, Chemical; Diazepam; Dose-Response Relationship, Drug; Flunitrazepam; gamma-Aminobutyric Acid; Isoniazid; Male; Mice; Mice, Inbred Strains; Purinergic P1 Receptor Antagonists; Receptors, GABA; Receptors, Purinergic P1; Seizures; Sulfur Radioisotopes; Synaptic Transmission; Tritium; Xanthines | 1993 |
Natural mutation of GABAA receptor alpha 6 subunit alters benzodiazepine affinity but not allosteric GABA effects.
Topics: Animals; Azides; Benzodiazepines; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Cerebellum; Cloning, Molecular; Convulsants; Diazepam; gamma-Aminobutyric Acid; Granulocytes; Humans; Kidney; Muscimol; Mutation; Picrotoxin; Rats; Receptors, GABA-A; Recombinant Proteins; Transfection | 1993 |
Bicuculline-produced regional differences in the modulation of 35S-TBPS binding by GABA, pentobarbital and diazepam in mouse cerebellum and cortex.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Cerebral Cortex; Diazepam; Dose-Response Relationship, Drug; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Phenobarbital; Receptors, GABA-A | 1993 |
Biochemical evaluations of the effects of loreclezole and propofol on the GABAA receptor in rat brain.
Topics: Anesthetics; Animals; Anticonvulsants; Brain; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; Flunitrazepam; GABA Modulators; gamma-Aminobutyric Acid; Hypnotics and Sedatives; In Vitro Techniques; Male; Muscimol; Pentobarbital; Pregnanediones; Propofol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sulfur Radioisotopes; Triazoles; Tritium | 1996 |
Characterisation of the furanocoumarin phellopterin as a rat brain benzodiazepine receptor partial agonist in vitro.
Topics: Animals; Binding Sites; Brain; Bridged Bicyclo Compounds, Heterocyclic; Coumarins; Diazepam; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; In Vitro Techniques; Male; Rats; Rats, Wistar; Receptors, GABA; Receptors, GABA-A | 1996 |
Direct activation of GABAA receptors by loreclezole, an anticonvulsant drug with selectivity for the beta-subunit.
Topics: Animals; Anticonvulsants; Bicuculline; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Cerebral Cortex; Chloride Channels; Convulsants; Diazepam; DNA, Complementary; Female; gamma-Aminobutyric Acid; Humans; Kinetics; Macromolecular Substances; Male; Membrane Potentials; Oocytes; Picrotoxin; Propofol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Recombinant Proteins; Triazoles; Xenopus laevis | 1996 |
Cerebellar gamma-aminobutyric acid type A receptors: pharmacological subtypes revealed by mutant mouse lines.
Topics: Animals; Azides; Benzodiazepines; Binding Sites; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cerebellum; Convulsants; Diazepam; Diuretics; Furosemide; GABA Agonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Mice; Mice, Inbred C57BL; Mutation; Pregnanolone; Pyridazines; Receptors, GABA-A; Sulfur Radioisotopes; Tritium; Zinc | 1997 |
Tolerance to diazepam-induced motor impairment: a study with GABAA receptor alpha6 subunit knockout mice.
Topics: Animals; Autoradiography; Brain; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; Male; Mice; Mice, Knockout; Motor Activity; Nervous System Diseases; Organ Specificity; Receptors, GABA-A; Sulfur Radioisotopes; Tissue Distribution | 2003 |
Caffeine analogs: effects on ryanodine-sensitive calcium-release channels and GABAA receptors.
Topics: Animals; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Caffeine; Calcium Signaling; Cell Membrane; Cerebral Cortex; Diazepam; Dose-Response Relationship, Drug; Male; Mice; Muscle, Skeletal; Neurons; Rabbits; Radioisotopes; Radioligand Assay; Receptors, GABA-A; Ryanodine; Ryanodine Receptor Calcium Release Channel; Xanthines | 2003 |
Low tolerance and dependence liabilities of etizolam: molecular, functional, and pharmacological correlates.
Topics: Animals; Animals, Newborn; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Cerebral Cortex; Diazepam; Fluorescent Antibody Technique; GABA Modulators; Gene Expression; Hippocampus; Isoniazid; Lorazepam; Male; Membrane Potentials; Mice; Neurons; Patch-Clamp Techniques; Protein Subunits; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; RNA, Messenger; Seizures; Sulfur Radioisotopes; Tranquilizing Agents | 2005 |