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tert-butylbicyclophosphorothionate and chlorine

tert-butylbicyclophosphorothionate has been researched along with chlorine in 129 studies

Research

Studies (129)

TimeframeStudies, this research(%)All Research%
pre-199070 (54.26)18.7374
1990's57 (44.19)18.2507
2000's2 (1.55)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ehrmann, ML; Mileson, BE; Schwartz, RD1
Golovko, AI; Sofronov, GA1
Belfiore, S; Giusti, L; Lucacchini, A; Martini, C1
Corda, MG; Giorgi, O; Orlandi, M1
Blakeman, DP; Carter, DB; Hamilton, BJ; Im, HK; Im, WB; Jacobsen, EJ; Petke, JD; Pregenzer, JF1
Biggio, G; Concas, A; Foddi, MC; Ghiani, CA; Melis, MA; Motzo, C; Sanna, E; Serra, M1
Bergendorff, O; Hansen, SK; Nielsen, MP; Rutherford, DM; Sterner, O; Witt, MR1
Miledi, R; Polenzani, L; Woodward, RM1
Biggio, G; Concas, A; Maciocco, E; Mascia, MP; Santoro, G1
Biggio, G; Colombo, G; Cossu, A; Follesa, P; Sanna, E; Serra, M1
Banerjee, PK; Depaulis, A; Hechler, V; Snead, OC; Vergnes, M1
Galpern, WR; Greenblatt, DJ; Lumpkin, M; Miller, LG; Shader, RI2
Gee, KW; Lan, NC1
Bloomquist, JR; Grubs, RE; Knipple, DC; Soderlund, DM1
Biggio, G; Concas, A; Sanna, E; Serra, M2
Chesley, S; Greenblatt, DJ; Lopez, F; Miller, LG; Schatzki, A; Shader, RI1
Buckingham, SD; Lummis, SC; Rauh, JJ; Sattelle, DB1
Chesley, S; Greenblatt, DJ; Lopez, F; Miller, LG; Schatzki, A; Shader, RI; Thompson, ML1
Biggio, G; Concas, A; Sanna, E; Santoro, G; Serra, M2
Biggio, G; Concas, A; Foddi, C; Sanna, E; Serra, M1
Niles, L1
Blakeman, DP; Im, WB1
Badyshtov, BA; Gordey, ML; Nagovitsina, YA; Seredenin, SB1
de Costa, BR; Lewin, AH; Rice, KC; Schoenheimer, JA; Skolnick, P1
Belelli, D; Gee, KW; McCauley, L1
Desarmenien, M; Feltz, P; Hamann, M; Piguet, P; Vanderheyden, P1
Niles, LP; Peace, CH1
Gardier, RW; Higgins, GM1
Barnard, EA; Devine, J; Macdonald, RL; Moss, SJ; Nayeem, N; Porter, NM; Smart, TG; Stephenson, FA1
Gee, KW; Lawrence, LJ; Yamamura, HI2
Braestrup, C; Honore, T; Nielsen, M1
Casida, JE; Lawrence, LJ1
Casida, JE; Seifert, J1
Barnes, EM; Tehrani, MH; Vaidyanathaswamy, R; Verkade, JG1
Barker, JL; Harrison, NL; Majewska, MD; Paul, SM; Schwartz, RD1
Havoundjian, H; Paul, SM; Skolnick, P3
Barnard, EA; Bilbe, G; Brown, DA; Constanti, A; Moss, S; Smart, TG; Van Renterghem, C1
Havoundjian, H; Skolnick, P; Trullas, R1
Braunwalder, A; Loo, P; Wood, PL1
Allan, AM; Bleck, V; Harris, RA; Huidobro-Toro, JP1
Barnard, EA; Bilbe, G; Houamed, K; Moss, SJ; Smart, TG; Van Renterghem, C1
Cole, RJ; Eldefrawi, AT; Eldefrawi, ME; Gant, DB; Valdes, JJ1
Majewska, MD1
Marvizón, JC; Skolnick, P1
McIntyre, TD; Skolnick, P; Trullas, R2
Greenblatt, DJ; Miller, LG; Roy, RB; Shader, RI; Summer, WR1
Eldefrawi, AT; Eldefrawi, ME; Matsumoto, K1
Moody, EJ; Paul, SM; Skolnick, P; Suzdak, PD1
Devaud, LL; Murray, TF1
Casida, JE; Palmer, CJ1
Danielou, G; Lloyd, KG; Thuret, F1
Atsoggiu, T; Biggio, G; Concas, A; Pepitoni, S; Toffano, G1
Bleck, V; Harris, RA; Lewin, E; Peris, J; Zahniser, NR2
Greenblatt, DJ; Kaplan, GB; Lopez, F; Miller, LG; Shader, RI1
Greenblatt, DJ; Lopez, F; Miller, LG; Roy, RB; Wecker, L1
de Costa, BR; Lewin, AH; Rice, KC; Skolnick, P1
Biggio, G; Cau, A; Corda, MG; Laudani, U; Longoni, B; Paci, S; Salvadori, S1
Gaver, A; Greenblatt, DJ; Lopez, F; Miller, LG; Roy, RB; Shader, RI1
Olsen, RW; Ransom, RW; Turner, DM; Yang, JS1
Paul, SM; Schwartz, RD; Seale, TW; Skolnick, P1
Belelli, D; Gee, KW; Joy, DS1
Evoniuk, G; Moody, EJ; Skolnick, P1
Erdö, SL; Wolff, JR1
Abel, MS; Blume, AJ; Garrett, KM2
Lopez, F; Miller, LG; Roy, RB; Weill, CL1
Culp, S; Liljequist, S; Tabakoff, B1
Allan, AM; Buck, KJ; Harris, RA1
Ticku, MK1
Carida, JE; Cole, LM; Palmer, CJ1
Bolger, MB; Brinton, RE; Coirini, H; Gee, KW; McEwen, BS1
Maksay, G; Ticku, MK2
Allan, AM; Daniell, LC; Harris, RA; Nixon, C1
Atsoggiu, T; Concas, A; Serra, M1
Gaver, A; Miller, LG; Roy, RB; Weill, CL1
Casida, JE; Ikeda, M; Laird, H; Malatynska, E; Obata, T; Palmer, CJ; Yamamura, HI1
Abalis, IM; Eldefrawi, AT; Eldefrawi, ME1
Biggio, G; Concas, A; Corda, MG; Serra, M1
Casida, JE; Gee, KW; Lawrence, LJ; Palmer, CJ; Wang, X; Yamamura, HI1
Bloomquist, JR; Soderlund, DM1
Maksay, G; Simonyi, M1
Haefely, W; Möhler, H; Richards, JG; Schoch, P1
Havoundjian, H; Skolnick, P1
Havoundjian, H; Paul, S; Skolnick, P; Trullas, R; Zamir, N1
Majewska, MD; Schwartz, RD1
Barker, JL; Harrington, JW; Harrison, NL; Majewska, MD1
Eldefrawi, AT; Eldefrawi, ME; Gant, DB1
Erdö, SL; Maksay, G1
Brinton, RE; Chang, WC; Gee, KW; McEwen, BS1
Allan, AM; Harris, RA1
Braunwalder, A; Cheney, DL; Loo, P; Wood, PL1
Snowman, AM; Snyder, SH; Trifiletti, RR1
Burke, TR; Rice, KC; Skolnick, P; Weissman, BA1
Carter, DB; Dillon, GH; Im, WB; McKinley, DD1
Carter, DB; Hamilton, BJ; Im, HK; Im, WB; Jacobsen, EJ; Pregenzer, JF1
Ticku, MK; Yu, R1
Burnham, WM; Lôscher, W; Nobrega, JN; Richter, A1
Biggio, G; Concas, A; Cuccheddu, T; Maciocco, E; Santoro, G; Serra, M1
Allan, AM; Harris, RA; McQuilkin, SJ; Mihic, SJ; Whatley, VJ1
Samochocki, M; Strosznajder, J2
Harris, RA; Klein, RL; McQuilkin, SJ; Sanna, E; Whiting, PJ1
Moore, FL; Murray, TF; Orchinik, M1
Corda, MG; Driscoll, P; Escorihuela, RM; Giorgi, O; Lecca, D; Orlandi, M1
Maksay, G1
Biggio, G; Concas, A; Dazzi, L; Maciocco, E; Mascia, MP; Ongini, E; Santoro, G1
Liu, CC; Snead, OC1
Deutsch, SI; Hitri, A; Lukacs, LG; Park, CH1
Harris, BD; Moody, EJ; Skolnick, P1
Carter, DB; Hamilton, BJ; Im, HK; Im, WB; Pregenzer, JF1
Belonga, KL; Carter, DB; Im, HK; Im, WB; Jacobsen, EJ; Petke, JD; Sethy, VH; Stelzer, LS; Tang, AH; TenBrink, RE; VonVoigtlander, PF1
Masonis, AE; McCarthy, MP1
Sousa, A; Ticku, MK1
Ahrens, R; Galeffi, F; Jordan, G; Sah, R; Schwartz-Bloom, RD1
Galofré, M; García, DA; Suñol, C; Vendrell, I1
Eshleman, AJ; Murray, TF1
Frandsen, A; Pomés, A; Rodríguez-Farré, E; Sanfeliu, C; Schousboe, A; Suñol, C1
Chatterjee, SS; Dimpfel, W; Nöldner, M; Ticku, MK1
Ho, IK; Ito, Y1
Cooper, RL; Meacham, CA; Shafer, TJ; Ward, TR1

Reviews

4 review(s) available for tert-butylbicyclophosphorothionate and chlorine

ArticleYear
Interactions of pyrethroid insecticides with chloride ionophore-associated binding sites.
    Neurotoxicology, 1985,Summer, Volume: 6, Issue:2

    Topics: Animals; Benzodiazepinones; Brain; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Drug Interactions; Guinea Pigs; Ion Channels; Picrotoxin; Pyrethrins; Radioligand Assay; Rats; Receptors, GABA-A; Sesterterpenes

1985
Structure-activity correlations for interactions of bicyclophosphorus esters and some polychlorocycloalkane and pyrethroid insecticides with the brain-specific t-butylbicyclophosphorothionate receptor.
    Environmental health perspectives, 1985, Volume: 61

    Topics: Animals; Binding, Competitive; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Hexachlorocyclohexane; In Vitro Techniques; Insecticides; Ion Channels; Male; Microsomes, Liver; Pyrethrins; Rats; Receptors, GABA-A; Structure-Activity Relationship; Sulfur Radioisotopes; Synaptic Membranes

1985
2,6,7-Trioxabicyclo[2.2.2]octanes: chemistry, toxicology and action at the GABA-gated chloride channel.
    Advances in biochemical psychopharmacology, 1988, Volume: 45

    Topics: Animals; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Convulsants; gamma-Aminobutyric Acid; Hydrolysis; Insecta; Ion Channels; Ligands; Structure-Activity Relationship

1988
Benzodiazepine receptors resolved.
    Experientia, 1986, Feb-15, Volume: 42, Issue:2

    Topics: Animals; Antibodies, Monoclonal; Autoradiography; Benzodiazepines; Benzodiazepinones; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Chlorides; Clonazepam; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Histocytochemistry; Humans; Immunologic Techniques; Ionophores; Muscimol; Neurons; Radioisotopes; Radioligand Assay; Receptors, GABA-A; Spinal Cord; Synapses; Tissue Distribution

1986

Other Studies

125 other study(ies) available for tert-butylbicyclophosphorothionate and chlorine

ArticleYear
Alterations in the gamma-aminobutyric acid-gated chloride channel following transient forebrain ischemia in the gerbil.
    Journal of neurochemistry, 1992, Volume: 58, Issue:2

    Topics: Animals; Autoradiography; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; gamma-Aminobutyric Acid; Gerbillinae; Ion Channel Gating; Ischemic Attack, Transient; Male; Membrane Proteins; Motor Activity; Muscimol

1992
[3H-tert-butylbicyclo-ortho-benzoate--a new ligand for chloride ion channel of GABA-A receptor].
    Biulleten' eksperimental'noi biologii i meditsiny, 1992, Volume: 113, Issue:2

    Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; In Vitro Techniques; Ligands; Male; Radioligand Assay; Rats; Receptors, GABA-A; Synaptic Membranes; Tritium

1992
Sex steroid hormones and GABAA receptor complex modulation.
    Advances in biochemical psychopharmacology, 1992, Volume: 47

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Epoxy Compounds; Female; Gonadal Steroid Hormones; Guinea Pigs; In Vitro Techniques; Menstruation; Progesterone; Receptors, GABA-A; Synaptosomes

1992
Decrease in GABAA receptor function induced by pentylenetetrazol kindling in the rat: role of N-methyl-D-aspartate (NMDA) receptors.
    Advances in biochemical psychopharmacology, 1992, Volume: 47

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Dizocilpine Maleate; Down-Regulation; Isoniazid; Kindling, Neurologic; Male; Pentylenetetrazole; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate

1992
Characterization of functional interactions of imidazoquinoxaline derivatives with benzodiazepine-gamma-aminobutyric acidA receptors.
    Molecular pharmacology, 1992, Volume: 42, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Chlorides; Chlorine; Cloning, Molecular; Drug Interactions; Electrophysiology; Flunitrazepam; GABA-A Receptor Antagonists; Kinetics; Male; Membrane Proteins; Models, Chemical; Molecular Conformation; Oxadiazoles; Quinoxalines; Radioisotopes; Rats; Rats, Inbred Strains; Receptors, GABA-A; Structure-Activity Relationship; Synaptosomes; Tritium

1992
Pharmacology of gamma-aminobutyric acidA receptor complex after the in vivo administration of the anxioselective and anticonvulsant beta-carboline derivative abecarnil.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 263, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Chlorides; Exploratory Behavior; gamma-Aminobutyric Acid; In Vitro Techniques; Isoniazid; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Stress, Physiological

1992
Isolation and identification from Salvia officinalis of two diterpenes which inhibit t-butylbicyclophosphoro[35S]thionate binding to chloride channel of rat cerebrocortical membranes in vitro.
    Neuroscience letters, 1992, Feb-03, Volume: 135, Issue:2

    Topics: Abietanes; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Diterpenes; Ion Channels; Kinetics; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Phenanthrenes; Plant Extracts; Plants, Medicinal; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, GABA-A

1992
Characterization of bicuculline/baclofen-insensitive gamma-aminobutyric acid receptors expressed in Xenopus oocytes. I. Effects of Cl- channel inhibitors.
    Molecular pharmacology, 1992, Volume: 42, Issue:1

    Topics: Animals; Baclofen; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Cerebral Cortex; Chloride Channels; Chlorides; Cloning, Molecular; Ion Channels; Membrane Proteins; Ovum; Picrotoxin; Rats; Receptors, GABA-A; Retina; RNA; Xenopus

1992
The general anesthetic propofol: a biochemical tool to study the function of the GABA-coupled chloride channel.
    Clinical neuropharmacology, 1992, Volume: 15 Suppl 1 Pt A

    Topics: Anesthetics; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; gamma-Aminobutyric Acid; Ion Channels; Male; Pentobarbital; Pregnanediones; Propofol; Rats; Rats, Inbred Strains

1992
GABAA and NMDA receptor function during chronic administration of ethanol.
    Advances in biochemical psychopharmacology, 1992, Volume: 47

    Topics: Alcoholic Intoxication; Animals; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Dizocilpine Maleate; Ethanol; Hippocampus; Ion Channels; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Substance Withdrawal Syndrome

1992
The GABAA receptor complex in experimental absence seizures in rat: an autoradiographic study.
    Neuroscience letters, 1992, Jun-08, Volume: 140, Issue:1

    Topics: Animals; Autoradiography; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; Convulsants; Epilepsy, Absence; Flunitrazepam; GABA-A Receptor Antagonists; Ion Channels; Ionophores; Male; Membrane Proteins; Muscimol; Organ Specificity; Pyramidal Tracts; Pyridazines; Rats; Rats, Wistar; Receptors, GABA-A; Sulfur Radioisotopes; Tritium

1992
Chronic benzodiazepine administration. VII. Behavioral tolerance and withdrawal and receptor alterations associated with clonazepam administration.
    Psychopharmacology, 1991, Volume: 104, Issue:2

    Topics: Animals; Behavior, Animal; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Clonazepam; Convulsants; Drug Tolerance; Flumazenil; Male; Mice; Motor Activity; Muscimol; Receptors, GABA-A; Substance Withdrawal Syndrome

1991
Gamma-aminobutyric acidA receptor complexes in rat frontal cortex and spinal cord show differential responses to steroid modulation.
    Molecular pharmacology, 1991, Volume: 40, Issue:6

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Desoxycorticosterone; Diazepam; gamma-Aminobutyric Acid; Ionophores; Male; Pentobarbital; Pregnanediol; Pregnanolone; Rats; Rats, Inbred Strains; Receptors, GABA-A; Spinal Cord; Steroids; Sulfur Radioisotopes

1991
Prolonged exposure to GABA activates GABA-gated chloride channels in the presence of channel-blocking convulsants.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1991, Volume: 99, Issue:3

    Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; Convulsants; Endrin; GABA Antagonists; gamma-Aminobutyric Acid; Ion Channel Gating; Kinetics; Male; Membrane Proteins; Mice; Mice, Inbred ICR; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sesterterpenes; Xenopus

1991
In vivo administration of ethanol enhances the function of the gamma-aminobutyric acid-dependent chloride channel in the rat cerebral cortex.
    Journal of neurochemistry, 1990, Volume: 54, Issue:2

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Diazepam; Ethanol; gamma-Aminobutyric Acid; Ion Channels; Isoniazid; Male; Rats; Rats, Inbred Strains

1990
Chronic administration of benzodiazepines--V. Rapid onset of behavioral and neurochemical alterations after discontinuation of alprazolam.
    Neuropharmacology, 1990, Volume: 29, Issue:3

    Topics: Alprazolam; Animals; Behavior, Animal; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Down-Regulation; Drug Tolerance; Ion Channels; Male; Mice; Motor Activity; Muscimol; Receptors, GABA-A; Substance Withdrawal Syndrome; Sulfur Radioisotopes

1990
Blocking actions of heptachlor at an insect central nervous system GABA receptor.
    Proceedings of the Royal Society of London. Series B, Biological sciences, 1990, May-22, Volume: 240, Issue:1297

    Topics: Animals; Binding, Competitive; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Chloride Channels; Chlorides; Cockroaches; Electrophysiology; gamma-Aminobutyric Acid; Ganglia; Heptachlor; Houseflies; Ion Channels; Membrane Potentials; Membrane Proteins; Motor Neurons; Nervous System Physiological Phenomena; Rats; Receptors, GABA-A

1990
Chronic morphine administration augments benzodiazepine binding and GABAA receptor function.
    Psychopharmacology, 1990, Volume: 101, Issue:4

    Topics: Animals; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Chlorine; Flunitrazepam; In Vitro Techniques; Ion Channels; Male; Mice; Morphine; Muscimol; Naltrexone; Radioisotopes; Receptors, GABA-A; Sulfur Radioisotopes

1990
The action of stress and anxiolytic and anxiogenic benzodiazepine receptors ligands on [35S] T-butylbicyclophosphorothionate binding in the rat cerebral cortex.
    Annali dell'Istituto superiore di sanita, 1990, Volume: 26, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Cerebral Cortex; Chlorides; Drug Interactions; Ion Channel Gating; Ion Channels; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological

1990
Ex vivo binding of t-[35S )butylbicyclophosphorothionate: a biochemical tool to study the pharmacology of ethanol at the gamma-aminobutyric acid-coupled chloride channel.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 256, Issue:3

    Topics: Animals; Azides; Benzodiazepines; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Diazepam; Drug Interactions; Ethanol; gamma-Aminobutyric Acid; Ion Channels; Isoniazid; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sulfur Radioisotopes

1991
Failure of gamma-hydroxybutyrate to alter the function of the GABAA receptor complex in the rat cerebral cortex.
    Psychopharmacology, 1991, Volume: 104, Issue:3

    Topics: Animals; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Diazepam; Flunitrazepam; In Vitro Techniques; Ion Channels; Isoniazid; Male; Nerve Tissue Proteins; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sodium Oxybate; Synaptic Transmission

1991
Melatonin interaction with the benzodiazepine-GABA receptor complex in the CNS.
    Advances in experimental medicine and biology, 1991, Volume: 294

    Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Cerebral Cortex; Chlorides; Diazepam; gamma-Aminobutyric Acid; Humans; Ion Channel Gating; Ion Channels; Melatonin; Muscimol; Prosencephalon; Rats; Receptors, GABA-A; Serotonin; Synaptosomes

1991
Correlation between gamma-aminobutyric acidA receptor ligand-induced changes in t-butylbicyclophosphoro[35S]thionate binding and 36Cl- uptake in rat cerebrocortical membranes.
    Molecular pharmacology, 1991, Volume: 39, Issue:3

    Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cerebral Cortex; Chloride Channels; Chlorides; Desoxycorticosterone; Diazepam; Ethanol; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Ligands; Membrane Proteins; Pentobarbital; Pregnanolone; Rats; Receptors, GABA-A; Synaptosomes

1991
Neurochemical action of the general anaesthetic propofol on the chloride ion channel coupled with GABAA receptors.
    Brain research, 1991, Mar-01, Volume: 542, Issue:2

    Topics: Anesthetics; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; Flunitrazepam; Male; Membrane Proteins; Muscimol; Propofol; Rats; Rats, Inbred Strains; Receptors, GABA-A

1991
Pharmacogenetic analysis of mechanisms of emotional stress: effects of benzodiazepines.
    Annali dell'Istituto superiore di sanita, 1990, Volume: 26, Issue:1

    Topics: Adrenocorticotropic Hormone; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Corticosterone; Diazepam; Exploratory Behavior; Hybridization, Genetic; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Motor Activity; Receptors, GABA-A; Stress, Psychological

1990
Novel site-directed affinity ligands for GABA-gated chloride channels: synthesis, characterization, and molecular modeling of 1-(isothiocyanatophenyl)-4-tert-butyl-2,6,7-trioxabicyclo[2.2.2]octanes .
    Journal of medicinal chemistry, 1991, Volume: 34, Issue:5

    Topics: Animals; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chemical Phenomena; Chemistry; Chlorides; Convulsants; gamma-Aminobutyric Acid; Ion Channel Gating; Ligands; Male; Models, Molecular; Rats; Rats, Inbred Strains

1991
Heterotropic cooperativity between putative recognition sites for progesterone metabolites and the atypical benzodiazepine Ro 5-4864.
    Journal of neurochemistry, 1990, Volume: 55, Issue:1

    Topics: Animals; Benzodiazepinones; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Convulsants; gamma-Aminobutyric Acid; Male; Pregnanediol; Pregnanolone; Progesterone; Rats; Rats, Inbred Strains

1990
Electrophysiological study of tert-butylbicyclophosphorothionate-induced block of spontaneous chloride channels.
    Molecular pharmacology, 1990, Volume: 37, Issue:4

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cell Membrane; Cells, Cultured; Chloride Channels; Chlorides; Convulsants; Electrophysiology; Ion Channel Gating; Kinetics; Membrane Proteins; Pituitary Gland; Swine

1990
Allosteric modulation of t-[35S]butylbicyclophosphorothionate binding in rat brain by melatonin.
    Brain research bulletin, 1990, Volume: 24, Issue:4

    Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chloride Channels; Chlorides; Male; Melatonin; Membrane Proteins; Rats; Rats, Inbred Strains; Receptors, GABA-A

1990
Chronic benzodiazepine administration. VI. A partial agonist produces behavioral effects without tolerance or receptor alterations.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:1

    Topics: Animals; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Dose-Response Relationship, Drug; Drug Tolerance; Male; Mice; Motor Activity; Pyridazines; Receptors, GABA-A

1990
gamma-Aminobutyric acid antagonism produced by an organophosphate-containing combustion product.
    Toxicology and applied pharmacology, 1990, Volume: 105, Issue:1

    Topics: Animals; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Convulsants; Flurothyl; GABA Antagonists; Gas Chromatography-Mass Spectrometry; In Vitro Techniques; Male; Mice; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, GABA-A

1990
Cloned GABA receptors are maintained in a stable cell line: allosteric and channel properties.
    European journal of pharmacology, 1990, Jul-31, Volume: 189, Issue:1

    Topics: Animals; Antibodies, Monoclonal; Barbiturates; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Cell Line; Chlorides; Clone Cells; Convulsants; DNA; gamma-Aminobutyric Acid; Membrane Potentials; Muscimol; Neurons; Plasmids; Receptors, GABA-A; Spinal Cord; Transfection

1990
Radiation inactivation of brain [35S]t-butylbicyclophosphorothionate binding sites reveals complicated molecular arrangements of the GABA/benzodiazepine receptor chloride channel complex.
    Biochemical pharmacology, 1985, Oct-15, Volume: 34, Issue:20

    Topics: Animals; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Cerebellum; Cerebral Cortex; Chlorides; Etazolate; Etomidate; In Vitro Techniques; Ion Channels; Molecular Weight; Muscimol; Organophosphorus Compounds; Radioligand Assay; Rats; Receptors, GABA-A; Sulfur Radioisotopes

1985
Basic neuroproteins modulate TBPS recognition site.
    European journal of pharmacology, 1986, Mar-11, Volume: 122, Issue:1

    Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Calcium Chloride; Cattle; Chlorides; gamma-Aminobutyric Acid; Ion Channels; Membranes; Nerve Tissue Proteins; Rats; Receptors, GABA-A

1986
Interaction of t-butylbicyclophosphorothionate with gamma-aminobutyric acid-gated chloride channels in cultured cerebral neurons.
    Journal of neurochemistry, 1986, Volume: 46, Issue:5

    Topics: Animals; Anions; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cell Membrane; Cells, Cultured; Chick Embryo; Chlorides; gamma-Aminobutyric Acid; Ion Channels; Kinetics; Neurons

1986
Steroid hormone metabolites are barbiturate-like modulators of the GABA receptor.
    Science (New York, N.Y.), 1986, May-23, Volume: 232, Issue:4753

    Topics: 20-alpha-Dihydroprogesterone; Animals; Binding, Competitive; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Chlorides; Desoxycorticosterone; Drug Synergism; Flunitrazepam; Hippocampus; In Vitro Techniques; Ion Channels; Progesterone; Rats; Receptors, GABA-A; Spinal Cord

1986
The permeability of gamma-aminobutyric acid-gated chloride channels is described by the binding of a "cage" convulsant, t-butylbicyclophosphoro[35S]thionate.
    Proceedings of the National Academy of Sciences of the United States of America, 1986, Volume: 83, Issue:23

    Topics: Animals; Anions; Anura; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cerebral Cortex; Chlorides; gamma-Aminobutyric Acid; Ganglia, Spinal; Ion Channels; Male; Neurons; Permeability; Rats

1986
GABA receptors induced in Xenopus oocytes by chick brain mRNA: evaluation of TBPS as a use-dependent channel-blocker.
    Brain research, 1987, Volume: 388, Issue:1

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chick Embryo; Chlorides; Female; GABA Antagonists; Ion Channels; Oocytes; Protein Biosynthesis; Receptors, GABA-A; RNA, Messenger

1987
Stress-induced changes in t-[35S]butylbicyclophosphorothionate binding to gamma-aminobutyric acid-gated chloride channels are mimicked by in vitro occupation of benzodiazepine receptors.
    Journal of neurochemistry, 1987, Volume: 49, Issue:3

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cerebral Cortex; Chlorides; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Ion Channels; Kinetics; Male; Membranes; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological; Swimming

1987
Benzodiazepine receptor modulation of [35S]TBPS binding to the chloride channel. Noncompetitive inhibition of classical benzodiazepines and competitive inhibition of the partial agonist, CGS 9895, by CGS 8216.
    Neuropharmacology, 1987, Volume: 26, Issue:7A

    Topics: Animals; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Ion Channels; Pyrazoles; Rats; Receptors, GABA-A; Sulfur Radioisotopes

1987
Neurochemical actions of anesthetic drugs on the gamma-aminobutyric acid receptor-chloride channel complex.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 242, Issue:3

    Topics: Alcohols; Anesthetics; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; gamma-Aminobutyric Acid; Ion Channels; Male; Mice; Mice, Inbred DBA; Receptors, GABA-A; Structure-Activity Relationship

1987
Functional expression in the Xenopus oocyte of messenger ribonucleic acids encoding brain neurotransmitter receptors: further characterisation of the implanted GABA receptor.
    Neuropharmacology, 1987, Volume: 26, Issue:7B

    Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chick Embryo; Chlorides; Cloning, Molecular; DNA; Dose-Response Relationship, Drug; Flunitrazepam; gamma-Aminobutyric Acid; Gene Expression Regulation; Glycosylation; Ion Channels; Oocytes; Poly A; Receptors, GABA-A; RNA; RNA, Messenger; Xenopus

1987
Action of tremorgenic mycotoxins on GABAA receptor.
    Life sciences, 1987, Nov-09, Volume: 41, Issue:19

    Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Electric Organ; Flunitrazepam; In Vitro Techniques; Ion Channels; Male; Muscimol; Mycotoxins; Rats; Rats, Inbred Strains; Receptors, GABA-A; Torpedo; Tremor

1987
Antagonist-type interaction of glucocorticoids with the GABA receptor-coupled chloride channel.
    Brain research, 1987, Aug-25, Volume: 418, Issue:2

    Topics: Animals; Bicuculline; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Frontal Lobe; Glucocorticoids; Ion Channels; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes

1987
Enhancement of t-[35S]butylbicyclophosphorothionate and [3H]strychnine binding by monovalent anions reveals similarities between gamma-aminobutyric acid- and glycine-gated chloride channels.
    Journal of neurochemistry, 1988, Volume: 50, Issue:5

    Topics: Animals; Anions; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cell Membrane; Cell Membrane Permeability; Chlorides; gamma-Aminobutyric Acid; Glycine; Ion Channels; Male; Medulla Oblongata; Rats; Rats, Inbred Strains; Spinal Cord; Strychnine; Sulfur Radioisotopes; Tritium

1988
Differences in the biophysical properties of the benzodiazepine/gamma-aminobutyric acid receptor chloride channel complex in the long-sleep and short-sleep mouse lines.
    Journal of neurochemistry, 1988, Volume: 51, Issue:2

    Topics: Animals; Azides; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Flunitrazepam; gamma-Aminobutyric Acid; Heart; Ion Channels; Male; Mice; Mice, Mutant Strains; Receptors, GABA-A; Sleep

1988
Chronic benzodiazepine administration. II. Discontinuation syndrome is associated with upregulation of gamma-aminobutyric acidA receptor complex binding and function.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:1

    Topics: Animals; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Drug Tolerance; Flumazenil; Flunitrazepam; Ion Channels; Lorazepam; Male; Mice; Motor Activity; Muscimol; Receptors, GABA-A; Time Factors

1988
Action of polychlorocycloalkane insecticides on binding of [35S]t-butylbicyclophosphorothionate to Torpedo electric organ membranes and stereospecificity of the binding site.
    Toxicology and applied pharmacology, 1988, Sep-15, Volume: 95, Issue:2

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Electric Organ; Hexachlorocyclohexane; Ion Channels; Receptors, GABA-A; Stereoisomerism; Torpedo

1988
Modulation of the benzodiazepine/gamma-aminobutyric acid receptor chloride channel complex by inhalation anesthetics.
    Journal of neurochemistry, 1988, Volume: 51, Issue:5

    Topics: Anesthesia, Inhalation; Anesthetics; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Enflurane; Ether; Halothane; Ion Channels; Male; Methoxyflurane; Muscimol; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes

1988
Involvement of peripheral-type benzodiazepine receptors in the proconvulsant actions of pyrethroid insecticides.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 247, Issue:1

    Topics: Animals; Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Dose-Response Relationship, Drug; In Vitro Techniques; Ion Channels; Isoquinolines; Male; Pyrethrins; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stereoisomerism

1988
Differentiation of activities within the GABAA-chloride ionophore complex by means of 35-S-TBPS binding.
    Advances in biochemical psychopharmacology, 1988, Volume: 45

    Topics: Allosteric Regulation; Animals; Anti-Anxiety Agents; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Convulsants; Hypnotics and Sedatives; Ion Channels; Ionophores; Rats; Receptors, GABA-A

1988
Aging reduces the GABA-dependent 36Cl- flux in rat brain membrane vesicles.
    Life sciences, 1988, Volume: 43, Issue:22

    Topics: Aging; Animals; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Cerebellum; Cerebral Cortex; Chlorides; gamma-Aminobutyric Acid; Hippocampus; Ion Channels; Male; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
Asymmetrical activation of GABA-gated chloride channels in cerebral cortex.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 30, Issue:4

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Flumazenil; Functional Laterality; Ion Channels; Kinetics; Male; Organ Specificity; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
Chemical kindling decreases GABA-activated chloride channels of mouse brain.
    European journal of pharmacology, 1989, Jan-24, Volume: 160, Issue:1

    Topics: Animals; Autoradiography; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; gamma-Aminobutyric Acid; Ion Channels; Kindling, Neurologic; Male; Mice; Mice, Inbred ICR; Muscimol; Sulfur Radioisotopes

1989
Diazepam sensitizes mice to FG 7142 and reduces muscimol-stimulated 36Cl- flux.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 33, Issue:2

    Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Chlorides; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Ion Channels; Kindling, Neurologic; Mice; Mice, Inbred ICR; Muscimol

1989
Interaction of caffeine with the GABAA receptor complex: alterations in receptor function but not ligand binding.
    European journal of pharmacology, 1989, Dec-05, Volume: 172, Issue:6

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Caffeine; Cerebral Cortex; Chlorides; In Vitro Techniques; Ion Channels; Kinetics; Ligands; Male; Mice; Muscimol; Receptors, GABA-A; Sulfur Radioisotopes; Synaptosomes

1989
Dietary choline intake modulates benzodiazepine receptor binding and gamma-aminobutyric acidA receptor function in mouse brain.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:1

    Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; Choline; Diet; Flumazenil; Male; Membrane Proteins; Mice; Motor Activity; Receptors, GABA-A

1989
meta- and para-isothiocyanato-t-butylbicycloorthobenzoate: irreversible ligands of the gamma-aminobutyric acid-regulated chloride ionophore.
    Molecular pharmacology, 1989, Volume: 35, Issue:2

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chloride Channels; Chlorides; gamma-Aminobutyric Acid; In Vitro Techniques; Isothiocyanates; Ligands; Male; Membrane Proteins; Rats; Rats, Inbred Strains; Structure-Activity Relationship; Thiocyanates

1989
Distribution and pharmacological properties of the GABAA/benzodiazepine/chloride ionophore receptor complex in the brain of the fish Anguilla anguilla.
    Journal of neurochemistry, 1989, Volume: 52, Issue:4

    Topics: Anguilla; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Flunitrazepam; gamma-Aminobutyric Acid; Ionophores; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A; Tissue Distribution

1989
Chronic benzodiazepine administration. III. Upregulation of gamma-aminobutyric acidA receptor binding and function associated with chronic benzodiazepine antagonist administration.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:3

    Topics: Animals; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Chlorides; Flumazenil; Male; Membrane Proteins; Mice; Motor Activity; Receptors, GABA-A

1989
Steroid anesthetics and naturally occurring analogs modulate the gamma-aminobutyric acid receptor complex at a site distinct from barbiturates.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:3

    Topics: Anesthetics; Animals; Barbiturates; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; In Vitro Techniques; Male; Muscimol; Pregnanediones; Rats; Rats, Inbred Strains; Receptors, GABA-A; Steroids; Structure-Activity Relationship

1989
Differential seizure sensitivities to picrotoxinin in two inbred strains of mice (DBA/2J and BALB/c ByJ): parallel changes in GABA receptor-mediated chloride flux and receptor binding.
    Brain research, 1989, Feb-27, Volume: 481, Issue:1

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Dose-Response Relationship, Drug; Frontal Lobe; Male; Mice; Mice, Inbred BALB C; Mice, Inbred DBA; Muscimol; Pentobarbital; Picrotoxin; Receptors, GABA-A; Seizures; Species Specificity; Synaptosomes

1989
Complex interactions between pregnenolone sulfate and the t-butylbicyclophosphorothionate-labeled chloride ionophore in rat brain.
    Brain research, 1989, Mar-13, Volume: 482, Issue:1

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cerebral Cortex; Chloride Channels; Chlorides; Drug Interactions; Ionophores; Kinetics; Male; Membrane Proteins; Pregnenolone; Rats; Rats, Inbred Strains; Receptors, GABA-A

1989
Ultraviolet irradiation selectively disrupts the gamma-aminobutyric acid/benzodiazepine receptor-linked chloride ionophore.
    Molecular pharmacology, 1989, Volume: 35, Issue:5

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Chloride Channels; Chlorides; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Membrane Proteins; Rats; Rats, Inbred Strains; Receptors, GABA-A; Ultraviolet Rays

1989
Age-related loss of t-[35S]butylbicyclophosphorothionate binding to the gamma-aminobutyric acidA receptor-coupled chloride ionophore in rat cerebral cortex.
    Journal of neurochemistry, 1989, Volume: 53, Issue:2

    Topics: Aging; Animals; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cerebral Cortex; Chlorides; Female; Ionophores; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sulfur Radioisotopes

1989
Effect of halide ions on t-[35S]butylbicyclophosphorothionate binding.
    Journal of neurochemistry, 1989, Volume: 53, Issue:3

    Topics: Animals; Anions; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Bromides; Chlorides; Fluorides; Halogens; Iodides; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A

1989
Differential effects of iodide and chloride on allosteric interactions of the GABAA receptor.
    Journal of neurochemistry, 1989, Volume: 53, Issue:3

    Topics: Allosteric Regulation; Animals; Anions; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Chlorides; Diazepam; gamma-Aminobutyric Acid; Iodides; Male; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A

1989
Persistent alterations in GABAA receptor binding and function after prenatal lorazepam administration in the chick.
    Brain research bulletin, 1989, Volume: 23, Issue:3

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chick Embryo; Chickens; Chlorides; Female; Flunitrazepam; Lorazepam; Muscimol; Pregnancy; Prenatal Exposure Delayed Effects; Radioligand Assay; Receptors, GABA-A

1989
The effect of ethanol on 35S-TBPS binding to mouse brain membranes in the presence of chloride.
    Pharmacology & toxicology, 1989, Volume: 65, Issue:5

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Benzodiazepinones; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Diazepam; Drug Tolerance; Ethanol; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred C57BL; Pentobarbital; Substance-Related Disorders; Sulfur Radioisotopes

1989
Fluidization of brain membranes by A2C does not produce anesthesia and does not augment muscimol-stimulated 36Cl- influx.
    European journal of pharmacology, 1989, Feb-07, Volume: 160, Issue:3

    Topics: Anesthesia; Animals; Benzyl Alcohols; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Chlorine; gamma-Aminobutyric Acid; Male; Membrane Fluidity; Membranes; Mice; Mice, Inbred ICR; Muscimol; Radioisotopes; Stearates; Stearic Acids; Synaptosomes; Temperature

1989
Behavioral and functional studies indicate a role for GABAAergic transmission in the actions of ethanol.
    Alcohol and alcoholism (Oxford, Oxfordshire). Supplement, 1987, Volume: 1

    Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Chlorides; Ethanol; Flunitrazepam; Male; Mice; Mice, Inbred C57BL; Picrotoxin; Rats; Receptors, GABA-A; Seizures; Spinal Cord

1987
(+/-)-4-tert-butyl-3-cyano-1-(4-ethynylphenyl)-2,6,7-trioxabi cyclo[2.2.2]octane: synthesis of a remarkably potent GABAA receptor antagonist.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:6

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; GABA Antagonists; Mice; Rats; Receptors, GABA-A

1988
Steroid modulation of the chloride ionophore in rat brain: structure-activity requirements, regional dependence and mechanism of action.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:2

    Topics: Androstane-3,17-diol; Animals; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Female; In Vitro Techniques; Ionophores; Kinetics; Male; Mice; Pregnanes; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Structure-Activity Relationship; Sulfur Radioisotopes; Uterus

1988
CNS depressants accelerate the dissociation of 35S-TBPS binding and GABA enhances their displacing potencies.
    Life sciences, 1988, Volume: 43, Issue:16

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cerebral Cortex; Chloride Channels; Chlorides; Convulsants; gamma-Aminobutyric Acid; Hypnotics and Sedatives; In Vitro Techniques; Membrane Proteins; Rats; Receptors, GABA-A

1988
Antagonism of ethanol and pentobarbital actions by benzodiazepine inverse agonists: neurochemical studies.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 247, Issue:3

    Topics: Animals; Azides; Benzodiazepines; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Carbolines; Chloride Channels; Chlorides; Ethanol; Male; Membrane Fluidity; Membrane Proteins; Mice; Mice, Inbred ICR; Pentobarbital; Receptors, GABA-A

1988
[Effect of stress on the function of chloride channels associated with the GABA receptor complex].
    Annali dell'Istituto superiore di sanita, 1988, Volume: 24, Issue:4

    Topics: Animals; Bicuculline; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cerebral Cortex; Chloride Channels; Chlorides; Male; Membrane Proteins; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological

1988
Lorazepam administration during embryonic development alters GABAA receptor binding and function.
    Brain research. Developmental brain research, 1988, Dec-01, Volume: 44, Issue:2

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chick Embryo; Chlorides; Embryonic and Fetal Development; Flunitrazepam; Lorazepam; Receptors, GABA-A; Subcellular Fractions

1988
Modulation of gamma-aminobutyric acid-stimulated chloride influx by bicycloorthocarboxylates, bicyclophosphorus esters, polychlorocycloalkanes and other cage convulsants.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:3

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; Convulsants; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Membrane Proteins; Rats; Rats, Inbred Strains; Structure-Activity Relationship

1988
Actions of avermectin B1a on the gamma-aminobutyric acidA receptor and chloride channels in rat brain.
    Journal of biochemical toxicology, 1986, Volume: 1, Issue:1

    Topics: Animals; Bicuculline; Binding, Competitive; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; Dose-Response Relationship, Drug; Flunitrazepam; Ivermectin; Kinetics; Male; Membrane Proteins; Muscimol; Rats; Receptors, GABA-A

1986
Changes of 36Cl- flux and 35S-TBPS binding induced by stress and gabaergic drugs.
    Advances in biochemical psychopharmacology, 1988, Volume: 45

    Topics: Animals; Anti-Anxiety Agents; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cell Membrane; Cerebral Cortex; Chlorides; Convulsants; gamma-Aminobutyric Acid; Male; Neurons; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological

1988
t-[3H]butylbicycloorthobenzoate: new radioligand probe for the gamma-aminobutyric acid-regulated chloride ionophore.
    Journal of neurochemistry, 1985, Volume: 45, Issue:3

    Topics: Androstanes; Animals; Azasteroids; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chemical Phenomena; Chemistry; Chlorides; gamma-Aminobutyric Acid; Hydrogen-Ion Concentration; Ionophores; Kinetics; Male; Rats; Receptors, GABA-A; Temperature

1985
GABA, depressants and chloride ions affect the rate of dissociation of 35S-t-butylbicyclophosphorothionate binding.
    Life sciences, 1985, Dec-09, Volume: 37, Issue:23

    Topics: Animals; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Central Nervous System Depressants; Cerebral Cortex; Chlorides; Convulsants; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Neurotoxic insecticides inhibit GABA-dependent chloride uptake by mouse brain vesicles.
    Biochemical and biophysical research communications, 1985, Nov-27, Volume: 133, Issue:1

    Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; gamma-Aminobutyric Acid; In Vitro Techniques; Insecticides; Male; Mice; Mice, Inbred ICR; Picrotoxin; Receptors, GABA-A

1985
Benzodiazepine anticonvulsants accelerate and beta-carboline convulsants decelerate the kinetics of [35S]TBPS binding at the chloride ionophore.
    European journal of pharmacology, 1985, Nov-05, Volume: 117, Issue:2

    Topics: Animals; Anticonvulsants; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Chlorides; Convulsants; Flunitrazepam; In Vitro Techniques; Ionophores; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Membranes

1985
Acute, stress-induced changes in the benzodiazepine/gamma-aminobutyric acid receptor complex are confined to the chloride ionophore.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:3

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bromides; Cerebral Cortex; Chlorides; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Iodides; Ionophores; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological; Sulfur Radioisotopes; Swimming; Tritium

1986
Rapid, stress-induced modification of the benzodiazepine receptor-coupled chloride ionophore.
    Brain research, 1986, Jun-11, Volume: 375, Issue:2

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Flunitrazepam; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stimulation, Chemical; Stress, Physiological; Swimming; Temperature

1986
Modulation of the chloride ionophore by benzodiazepine receptor ligands: influence of gamma-aminobutyric acid and ligand efficacy.
    Molecular pharmacology, 1986, Volume: 30, Issue:3

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Cerebral Cortex; Chlorides; Clonazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Ionophores; Kinetics; Ligands; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sulfur Radioisotopes; Tritium

1986
A quantitative relationship between Cl- enhanced [3H]flunitrazepam and [35S]t-butylbicyclophosphorothionate binding to the benzodiazepine/GABA receptor chloride ionophore complex.
    Brain research, 1986, Volume: 387, Issue:3

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cerebral Cortex; Chlorides; Flunitrazepam; In Vitro Techniques; Male; Phospholipases A; Phospholipases A2; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stimulation, Chemical

1986
Environmentally-induced modification of the benzodiazepine/GABA receptor coupled chloride ionophore.
    Psychopharmacology, 1987, Volume: 91, Issue:3

    Topics: Animals; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Environment; Flunitrazepam; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological; Swimming

1987
Pregnenolone-sulfate: an endogenous antagonist of the gamma-aminobutyric acid receptor complex in brain?
    Brain research, 1987, Feb-24, Volume: 404, Issue:1-2

    Topics: Adrenal Glands; Animals; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Male; Muscimol; Picrotoxin; Pregnenolone; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stimulation, Chemical

1987
Structure-activity relationships for steroid interaction with the gamma-aminobutyric acidA receptor complex.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:1

    Topics: Animals; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Desoxycorticosterone; Electric Conductivity; Ethanol; Evoked Potentials; Flunitrazepam; Muscimol; Pregnanes; Progesterone; Rats; Rats, Inbred Strains; Receptors, GABA-A; Steroids; Structure-Activity Relationship

1987
Cyclodiene insecticides inhibit GABAA receptor-regulated chloride transport.
    Toxicology and applied pharmacology, 1987, Volume: 88, Issue:3

    Topics: Animals; Bicuculline; Biological Transport; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Insecticides; Male; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A

1987
[35S]TBPS binding to membranes of the female sex organs: modulation of chloride ionophore by GABA and pentobarbital.
    European journal of pharmacology, 1988, Mar-01, Volume: 147, Issue:2

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Convulsants; Fallopian Tubes; Female; gamma-Aminobutyric Acid; Genitalia, Female; In Vitro Techniques; Ionophores; Membranes; Ovary; Pentobarbital; Rats; Rats, Inbred Strains; Uterus

1988
GABA-dependent modulation of the Cl- ionophore by steroids in rat brain.
    European journal of pharmacology, 1987, Apr-29, Volume: 136, Issue:3

    Topics: Animals; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Cholesterol; gamma-Aminobutyric Acid; In Vitro Techniques; Ionophores; Male; Rats; Rats, Inbred Strains; Steroids

1987
Gamma-aminobutyric acid and alcohol actions: neurochemical studies of long sleep and short sleep mice.
    Life sciences, 1986, Nov-24, Volume: 39, Issue:21

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Cerebellum; Chlorides; Diencephalon; Drug Synergism; Ethanol; Female; gamma-Aminobutyric Acid; Hippocampus; Mice; Muscimol; Pentobarbital; Sleep; Telencephalon

1986
In vitro characterization of agonist, antagonist, inverse agonist and agonist/antagonist benzodiazepines.
    Progress in neuro-psychopharmacology & biological psychiatry, 1984, Volume: 8, Issue:4-6

    Topics: Animals; Benzodiazepines; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Etazolate; Ion Channels; Muscimol; Rats; Receptors, GABA-A

1984
Solubilization and anionic regulation of cerebral sedative/convulsant receptors labeled with [35S] tert-butylbicyclophosphorothionate (TBPS).
    Biochemical and biophysical research communications, 1984, Apr-30, Volume: 120, Issue:2

    Topics: Animals; Anions; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cell Membrane; Cerebral Cortex; Chlorides; Cholic Acids; Detergents; Ion Channels; Male; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Solubility

1984
Alkyl-substituted gamma-butyrolactones inhibit [35S]TBPS binding to a GABA linked chloride ionophore.
    European journal of pharmacology, 1984, Oct-01, Volume: 105, Issue:1-2

    Topics: 4-Butyrolactone; Animals; Barbiturates; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Furans; gamma-Aminobutyric Acid; In Vitro Techniques; Ionophores; Male; Membranes; Picrotoxin; Rats; Rats, Inbred Strains

1984
Enhancement by GABA of the association rate of picrotoxin and tert-butylbicyclophosphorothionate to the rat cloned alpha 1 beta 2 gamma 2 GABAA receptor subtype.
    British journal of pharmacology, 1995, Volume: 115, Issue:3

    Topics: Animals; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Chlorides; Cloning, Molecular; Dose-Response Relationship, Drug; Drug Interactions; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Ion Channels; Kidney; Kinetics; Patch-Clamp Techniques; Picrotoxin; Rats; Receptors, GABA-A

1995
Characterization of U-97775 as a GABAA receptor ligand of dual functionality in cloned rat GABAA receptor subtypes.
    British journal of pharmacology, 1995, Volume: 115, Issue:1

    Topics: Animals; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Chlorides; Electrophysiology; Flumazenil; Humans; Imidazoles; Ligands; Quinoxalines; Rats; Receptors, GABA-A; Recombinant Proteins

1995
Chronic neurosteroid treatment produces functional heterologous uncoupling at the gamma-aminobutyric acid type A/benzodiazepine receptor complex in mammalian cortical neurons.
    Molecular pharmacology, 1995, Volume: 47, Issue:3

    Topics: Androstanes; Animals; Azasteroids; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Cerebral Cortex; Chlorides; Chlorine; Convulsants; Drug Interactions; GABA Antagonists; gamma-Aminobutyric Acid; Kinetics; Mice; Mice, Inbred C57BL; Neurons; Pregnanolone; Radioisotopes; Radioligand Assay; Receptors, GABA-A; Sulfur Radioisotopes; Time Factors; Tritium

1995
Alterations in the brain GABAA/benzodiazepine receptor-chloride ionophore complex in a genetic model of paroxysmal dystonia: a quantitative autoradiographic analysis.
    Neuroscience, 1995, Volume: 64, Issue:1

    Topics: Animals; Autoradiography; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Cricetinae; Dystonia; Flunitrazepam; Ionophores; Male; Models, Genetic; Muscimol; Radiography; Receptors, GABA-A

1995
The effect of cyclopyrrolones on GABAA receptor function is different from that of benzodiazepines.
    Naunyn-Schmiedeberg's archives of pharmacology, 1994, Volume: 350, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Benzodiazepines; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Chlorine; Flumazenil; Hypnotics and Sedatives; Kinetics; Male; Mice; Mice, Inbred Strains; Muscimol; Naphthyridines; Piperazines; Radioisotopes; Receptors, GABA-A; Sulfur Compounds; Sulfur Radioisotopes; Tritium

1994
Gamma-aminobutyric acidA receptor function is inhibited by microtubule depolymerization.
    The Journal of biological chemistry, 1994, Jul-29, Volume: 269, Issue:30

    Topics: Animals; Biological Transport; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Chlorides; Colchicine; Convulsants; Dose-Response Relationship, Drug; Flunitrazepam; Histones; Humans; Lumicolchicines; Membranes; Mice; Microtubules; Muscimol; Nocodazole; Paclitaxel; Phosphorylation; Receptors, GABA-A; Vinblastine; Xenopus

1994
Age-related changes of GABA-activated chloride channel properties in brain cortex synaptic plasma membrane: evidence for phospholipase involvement.
    Journal of neurochemistry, 1994, Volume: 63, Issue:4

    Topics: Aging; Animals; Arachidonic Acid; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Chlorides; Convulsants; Diglycerides; gamma-Aminobutyric Acid; Kinetics; Muscimol; Phospholipases; Picrotoxin; Rats; Rats, Wistar; Sulfur Radioisotopes; Synaptic Membranes; Synaptosomes

1994
Effects of 5-HT3 receptor antagonists on binding and function of mouse and human GABAA receptors.
    European journal of pharmacology, 1994, Jul-15, Volume: 268, Issue:2

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Flumazenil; Flunitrazepam; Humans; Indazoles; Indoles; Male; Mice; Mice, Inbred ICR; Receptors, GABA-A; Serotonin Antagonists; Tropanes; Tropisetron; Xenopus laevis

1994
Steroid modulation of GABAA receptors in an amphibian brain.
    Brain research, 1994, May-23, Volume: 646, Issue:2

    Topics: Animals; Autoradiography; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Chlorides; Convulsants; Corticosterone; Flunitrazepam; Kinetics; Male; Mammals; Neurons; Pregnanolone; Pregnenolone; Rats; Receptors, GABA-A; Salamandridae; Species Specificity; Steroids; Sulfur Radioisotopes; Synaptosomes; Tritium

1994
GABAergic and dopaminergic transmission in the brain of Roman high-avoidance and Roman low-avoidance rats.
    Brain research, 1994, Feb-28, Volume: 638, Issue:1-2

    Topics: Amygdala; Animals; Avoidance Learning; Benzazepines; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Cerebral Cortex; Chlorides; Convulsants; Corpus Striatum; Dopamine; Emotions; Flunitrazepam; gamma-Aminobutyric Acid; Hippocampus; Kinetics; Male; Nucleus Accumbens; Organ Specificity; Prefrontal Cortex; Rats; Rats, Mutant Strains; Receptors, Dopamine D1; Species Specificity; Synaptic Transmission

1994
Modulatory action of arachidonic acid on GABAA/chloride channel receptor function in adult and aged brain cortex membranes.
    Neurochemistry international, 1993, Volume: 23, Issue:3

    Topics: Aging; Animals; Arachidonic Acid; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Cerebral Cortex; Chloride Channels; Chlorides; Convulsants; Docosahexaenoic Acids; Fatty Acids, Nonesterified; Kinetics; Male; Muscimol; Rats; Rats, Wistar; Receptors, GABA-A; Stearic Acids; Synaptic Membranes; Synaptosomes

1993
Partial and full agonists/inverse agonists affect [35S]TBPS binding at different occupancies of central benzodiazepine receptors.
    European journal of pharmacology, 1993, Aug-15, Volume: 246, Issue:3

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Convulsants; Ionophores; Radioligand Assay; Rats; Receptors, GABA-A; Sulfur Radioisotopes

1993
Anticonvulsant doses of 2-chloro-N6-cyclopentyladenosine, an adenosine A1 receptor agonist, reduce GABAergic transmission in different areas of the mouse brain.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 267, Issue:2

    Topics: Adenosine; Animals; Anticonvulsants; Behavior, Animal; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Depression, Chemical; Diazepam; Dose-Response Relationship, Drug; Flunitrazepam; gamma-Aminobutyric Acid; Isoniazid; Male; Mice; Mice, Inbred Strains; Purinergic P1 Receptor Antagonists; Receptors, GABA; Receptors, Purinergic P1; Seizures; Sulfur Radioisotopes; Synaptic Transmission; Tritium; Xanthines

1993
GABAA receptor function in the gamma-hydroxybutyrate model of generalized absence seizures.
    Neuropharmacology, 1993, Volume: 32, Issue:4

    Topics: Aminocaproates; Animals; Anticonvulsants; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Chlorine; Convulsants; Electroencephalography; Epilepsy, Absence; Flunitrazepam; In Vitro Techniques; Kinetics; Male; Muscimol; Radioisotopes; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sodium Oxybate; Synaptosomes; Vigabatrin

1993
Swim stress selectively alters the specific binding of a benzodiazepine antagonist in mice.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 45, Issue:2

    Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Flumazenil; Flurazepam; In Vitro Techniques; Kinetics; Male; Mice; Receptors, GABA-A; Stress, Physiological; Swimming; Tissue Distribution

1993
Stereospecific actions of the inhalation anesthetic isoflurane at the GABAA receptor complex.
    Brain research, 1993, Jun-25, Volume: 615, Issue:1

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Flunitrazepam; In Vitro Techniques; Isoflurane; Male; Mice; Receptors, GABA-A; Stereoisomerism; Sulfur Radioisotopes

1993
U-89843A is a novel allosteric modulator of gamma-aminobutyric acidA receptors.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 275, Issue:3

    Topics: Allosteric Regulation; Animals; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Chloride Channel Agonists; Chlorides; GABA Modulators; Humans; Male; Mice; Pyrimidines; Pyrroles; Rats; Receptors, GABA-A

1995
High-affinity partial agonist imidazo[1,5-a]quinoxaline amides, carbamates, and ureas at the gamma-aminobutyric acid A/benzodiazepine receptor complex.
    Journal of medicinal chemistry, 1996, Jan-05, Volume: 39, Issue:1

    Topics: Animals; Anxiety; Benzodiazepines; Binding, Competitive; Brain; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Flunitrazepam; GABA Agonists; GABA Antagonists; Molecular Conformation; Molecular Structure; Oxadiazoles; Pentylenetetrazole; Quinoxalines; Rats; Receptors, GABA-A

1996
Effects of the androgenic/anabolic steroid stanozolol on GABAA receptor function: GABA-stimulated 36Cl- influx and [35S] TBPS binding.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 279, Issue:1

    Topics: Anabolic Agents; Animals; Brain; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Stanozolol

1996
Interactions of the neurosteroid dehydroepiandrosterone sulfate with the GABA(A) receptor complex reveals that it may act via the picrotoxin site.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 282, Issue:2

    Topics: Animals; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Cerebellum; Cerebral Cortex; Chlorides; Dehydroepiandrosterone; Dehydroepiandrosterone Sulfate; gamma-Aminobutyric Acid; In Vitro Techniques; Ion Transport; Male; Mice; Mice, Inbred C57BL; Picrotoxin; Protein Binding; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

1997
Modulation of the GABA(A)-gated chloride channel by reactive oxygen species.
    Journal of neurochemistry, 2002, Volume: 80, Issue:3

    Topics: Animals; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Hippocampus; Hydrogen Peroxide; Ion Channel Gating; Microscopy, Confocal; Organ Culture Techniques; Oxidants; Oxidative Stress; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Receptors, GABA-A; Sulfur Radioisotopes; Synaptic Transmission

2002
GABA released from cultured cortical neurons influences the modulation of t-[(35)S]butylbicyclophosphorothionate binding at the GABAA receptor Effects of thymol.
    European journal of pharmacology, 2008, Dec-14, Volume: 600, Issue:1-3

    Topics: Allosteric Regulation; Anesthetics, Intravenous; Animals; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Cell Survival; Cells, Cultured; Cerebral Cortex; Chlorides; gamma-Aminobutyric Acid; Mice; Propofol; Receptors, GABA-A; Thymol

2008
Pyrethroid insecticides indirectly inhibit GABA-dependent 36Cl- influx in synaptoneurosomes from the trout brain.
    Neuropharmacology, 1991, Volume: 30, Issue:12A

    Topics: Animals; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorine; Depression, Chemical; gamma-Aminobutyric Acid; In Vitro Techniques; Insecticides; Nerve Tissue Proteins; Nitriles; Pyrethrins; Salmon; Synaptosomes; Tetrodotoxin; Veratridine

1991
Lindane cytotoxicity in cultured neocortical neurons is ameliorated by GABA and flunitrazepam.
    Journal of neuroscience research, 1994, Dec-15, Volume: 39, Issue:6

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Cell Survival; Cells, Cultured; Cerebral Cortex; Chloride Channels; Chlorine; Convulsants; Flunitrazepam; gamma-Aminobutyric Acid; Hexachlorocyclohexane; Mice; Neurons; Potassium; Receptors, GABA

1994
Effects of the anticonvulsant losigamone and its isomers on the GABAA receptor system.
    Epilepsia, 1995, Volume: 36, Issue:10

    Topics: Animals; Anticonvulsants; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Cerebral Cortex; Chloride Channels; Chlorine; Convulsants; Dose-Response Relationship, Drug; Epilepsy; Female; Furans; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Isomerism; Male; Mice; Mice, Inbred C57BL; Radioisotopes; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

1995
Studies on picrotoxin binding sites of GABAA receptors in rat cortical synaptoneurosomes.
    Brain research bulletin, 1994, Volume: 33, Issue:4

    Topics: Animals; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorine; Desoxycorticosterone; Diazepam; In Vitro Techniques; Male; Membranes; Muscimol; Pentobarbital; Picrotoxin; Radioisotopes; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Steroids; Synaptosomes

1994
Effects of the chlorotriazine herbicide, cyanazine, on GABA(A) receptors in cortical tissue from rat brain.
    Toxicology, 1999, Dec-20, Volume: 142, Issue:1

    Topics: Animals; Azides; Benzodiazepines; Binding Sites; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Chlorine; GABA Agonists; Herbicides; Male; Muscimol; Radioisotopes; Rats; Rats, Long-Evans; Receptors, GABA-A; Synaptosomes; Triazines

1999