tert-butylbicyclophosphorothionate has been researched along with chlorine in 129 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 70 (54.26) | 18.7374 |
1990's | 57 (44.19) | 18.2507 |
2000's | 2 (1.55) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Ehrmann, ML; Mileson, BE; Schwartz, RD | 1 |
Golovko, AI; Sofronov, GA | 1 |
Belfiore, S; Giusti, L; Lucacchini, A; Martini, C | 1 |
Corda, MG; Giorgi, O; Orlandi, M | 1 |
Blakeman, DP; Carter, DB; Hamilton, BJ; Im, HK; Im, WB; Jacobsen, EJ; Petke, JD; Pregenzer, JF | 1 |
Biggio, G; Concas, A; Foddi, MC; Ghiani, CA; Melis, MA; Motzo, C; Sanna, E; Serra, M | 1 |
Bergendorff, O; Hansen, SK; Nielsen, MP; Rutherford, DM; Sterner, O; Witt, MR | 1 |
Miledi, R; Polenzani, L; Woodward, RM | 1 |
Biggio, G; Concas, A; Maciocco, E; Mascia, MP; Santoro, G | 1 |
Biggio, G; Colombo, G; Cossu, A; Follesa, P; Sanna, E; Serra, M | 1 |
Banerjee, PK; Depaulis, A; Hechler, V; Snead, OC; Vergnes, M | 1 |
Galpern, WR; Greenblatt, DJ; Lumpkin, M; Miller, LG; Shader, RI | 2 |
Gee, KW; Lan, NC | 1 |
Bloomquist, JR; Grubs, RE; Knipple, DC; Soderlund, DM | 1 |
Biggio, G; Concas, A; Sanna, E; Serra, M | 2 |
Chesley, S; Greenblatt, DJ; Lopez, F; Miller, LG; Schatzki, A; Shader, RI | 1 |
Buckingham, SD; Lummis, SC; Rauh, JJ; Sattelle, DB | 1 |
Chesley, S; Greenblatt, DJ; Lopez, F; Miller, LG; Schatzki, A; Shader, RI; Thompson, ML | 1 |
Biggio, G; Concas, A; Sanna, E; Santoro, G; Serra, M | 2 |
Biggio, G; Concas, A; Foddi, C; Sanna, E; Serra, M | 1 |
Niles, L | 1 |
Blakeman, DP; Im, WB | 1 |
Badyshtov, BA; Gordey, ML; Nagovitsina, YA; Seredenin, SB | 1 |
de Costa, BR; Lewin, AH; Rice, KC; Schoenheimer, JA; Skolnick, P | 1 |
Belelli, D; Gee, KW; McCauley, L | 1 |
Desarmenien, M; Feltz, P; Hamann, M; Piguet, P; Vanderheyden, P | 1 |
Niles, LP; Peace, CH | 1 |
Gardier, RW; Higgins, GM | 1 |
Barnard, EA; Devine, J; Macdonald, RL; Moss, SJ; Nayeem, N; Porter, NM; Smart, TG; Stephenson, FA | 1 |
Gee, KW; Lawrence, LJ; Yamamura, HI | 2 |
Braestrup, C; Honore, T; Nielsen, M | 1 |
Casida, JE; Lawrence, LJ | 1 |
Casida, JE; Seifert, J | 1 |
Barnes, EM; Tehrani, MH; Vaidyanathaswamy, R; Verkade, JG | 1 |
Barker, JL; Harrison, NL; Majewska, MD; Paul, SM; Schwartz, RD | 1 |
Havoundjian, H; Paul, SM; Skolnick, P | 3 |
Barnard, EA; Bilbe, G; Brown, DA; Constanti, A; Moss, S; Smart, TG; Van Renterghem, C | 1 |
Havoundjian, H; Skolnick, P; Trullas, R | 1 |
Braunwalder, A; Loo, P; Wood, PL | 1 |
Allan, AM; Bleck, V; Harris, RA; Huidobro-Toro, JP | 1 |
Barnard, EA; Bilbe, G; Houamed, K; Moss, SJ; Smart, TG; Van Renterghem, C | 1 |
Cole, RJ; Eldefrawi, AT; Eldefrawi, ME; Gant, DB; Valdes, JJ | 1 |
Majewska, MD | 1 |
Marvizón, JC; Skolnick, P | 1 |
McIntyre, TD; Skolnick, P; Trullas, R | 2 |
Greenblatt, DJ; Miller, LG; Roy, RB; Shader, RI; Summer, WR | 1 |
Eldefrawi, AT; Eldefrawi, ME; Matsumoto, K | 1 |
Moody, EJ; Paul, SM; Skolnick, P; Suzdak, PD | 1 |
Devaud, LL; Murray, TF | 1 |
Casida, JE; Palmer, CJ | 1 |
Danielou, G; Lloyd, KG; Thuret, F | 1 |
Atsoggiu, T; Biggio, G; Concas, A; Pepitoni, S; Toffano, G | 1 |
Bleck, V; Harris, RA; Lewin, E; Peris, J; Zahniser, NR | 2 |
Greenblatt, DJ; Kaplan, GB; Lopez, F; Miller, LG; Shader, RI | 1 |
Greenblatt, DJ; Lopez, F; Miller, LG; Roy, RB; Wecker, L | 1 |
de Costa, BR; Lewin, AH; Rice, KC; Skolnick, P | 1 |
Biggio, G; Cau, A; Corda, MG; Laudani, U; Longoni, B; Paci, S; Salvadori, S | 1 |
Gaver, A; Greenblatt, DJ; Lopez, F; Miller, LG; Roy, RB; Shader, RI | 1 |
Olsen, RW; Ransom, RW; Turner, DM; Yang, JS | 1 |
Paul, SM; Schwartz, RD; Seale, TW; Skolnick, P | 1 |
Belelli, D; Gee, KW; Joy, DS | 1 |
Evoniuk, G; Moody, EJ; Skolnick, P | 1 |
Erdö, SL; Wolff, JR | 1 |
Abel, MS; Blume, AJ; Garrett, KM | 2 |
Lopez, F; Miller, LG; Roy, RB; Weill, CL | 1 |
Culp, S; Liljequist, S; Tabakoff, B | 1 |
Allan, AM; Buck, KJ; Harris, RA | 1 |
Ticku, MK | 1 |
Carida, JE; Cole, LM; Palmer, CJ | 1 |
Bolger, MB; Brinton, RE; Coirini, H; Gee, KW; McEwen, BS | 1 |
Maksay, G; Ticku, MK | 2 |
Allan, AM; Daniell, LC; Harris, RA; Nixon, C | 1 |
Atsoggiu, T; Concas, A; Serra, M | 1 |
Gaver, A; Miller, LG; Roy, RB; Weill, CL | 1 |
Casida, JE; Ikeda, M; Laird, H; Malatynska, E; Obata, T; Palmer, CJ; Yamamura, HI | 1 |
Abalis, IM; Eldefrawi, AT; Eldefrawi, ME | 1 |
Biggio, G; Concas, A; Corda, MG; Serra, M | 1 |
Casida, JE; Gee, KW; Lawrence, LJ; Palmer, CJ; Wang, X; Yamamura, HI | 1 |
Bloomquist, JR; Soderlund, DM | 1 |
Maksay, G; Simonyi, M | 1 |
Haefely, W; Möhler, H; Richards, JG; Schoch, P | 1 |
Havoundjian, H; Skolnick, P | 1 |
Havoundjian, H; Paul, S; Skolnick, P; Trullas, R; Zamir, N | 1 |
Majewska, MD; Schwartz, RD | 1 |
Barker, JL; Harrington, JW; Harrison, NL; Majewska, MD | 1 |
Eldefrawi, AT; Eldefrawi, ME; Gant, DB | 1 |
Erdö, SL; Maksay, G | 1 |
Brinton, RE; Chang, WC; Gee, KW; McEwen, BS | 1 |
Allan, AM; Harris, RA | 1 |
Braunwalder, A; Cheney, DL; Loo, P; Wood, PL | 1 |
Snowman, AM; Snyder, SH; Trifiletti, RR | 1 |
Burke, TR; Rice, KC; Skolnick, P; Weissman, BA | 1 |
Carter, DB; Dillon, GH; Im, WB; McKinley, DD | 1 |
Carter, DB; Hamilton, BJ; Im, HK; Im, WB; Jacobsen, EJ; Pregenzer, JF | 1 |
Ticku, MK; Yu, R | 1 |
Burnham, WM; Lôscher, W; Nobrega, JN; Richter, A | 1 |
Biggio, G; Concas, A; Cuccheddu, T; Maciocco, E; Santoro, G; Serra, M | 1 |
Allan, AM; Harris, RA; McQuilkin, SJ; Mihic, SJ; Whatley, VJ | 1 |
Samochocki, M; Strosznajder, J | 2 |
Harris, RA; Klein, RL; McQuilkin, SJ; Sanna, E; Whiting, PJ | 1 |
Moore, FL; Murray, TF; Orchinik, M | 1 |
Corda, MG; Driscoll, P; Escorihuela, RM; Giorgi, O; Lecca, D; Orlandi, M | 1 |
Maksay, G | 1 |
Biggio, G; Concas, A; Dazzi, L; Maciocco, E; Mascia, MP; Ongini, E; Santoro, G | 1 |
Liu, CC; Snead, OC | 1 |
Deutsch, SI; Hitri, A; Lukacs, LG; Park, CH | 1 |
Harris, BD; Moody, EJ; Skolnick, P | 1 |
Carter, DB; Hamilton, BJ; Im, HK; Im, WB; Pregenzer, JF | 1 |
Belonga, KL; Carter, DB; Im, HK; Im, WB; Jacobsen, EJ; Petke, JD; Sethy, VH; Stelzer, LS; Tang, AH; TenBrink, RE; VonVoigtlander, PF | 1 |
Masonis, AE; McCarthy, MP | 1 |
Sousa, A; Ticku, MK | 1 |
Ahrens, R; Galeffi, F; Jordan, G; Sah, R; Schwartz-Bloom, RD | 1 |
Galofré, M; García, DA; Suñol, C; Vendrell, I | 1 |
Eshleman, AJ; Murray, TF | 1 |
Frandsen, A; Pomés, A; Rodríguez-Farré, E; Sanfeliu, C; Schousboe, A; Suñol, C | 1 |
Chatterjee, SS; Dimpfel, W; Nöldner, M; Ticku, MK | 1 |
Ho, IK; Ito, Y | 1 |
Cooper, RL; Meacham, CA; Shafer, TJ; Ward, TR | 1 |
4 review(s) available for tert-butylbicyclophosphorothionate and chlorine
Article | Year |
---|---|
Interactions of pyrethroid insecticides with chloride ionophore-associated binding sites.
Topics: Animals; Benzodiazepinones; Brain; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Drug Interactions; Guinea Pigs; Ion Channels; Picrotoxin; Pyrethrins; Radioligand Assay; Rats; Receptors, GABA-A; Sesterterpenes | 1985 |
Structure-activity correlations for interactions of bicyclophosphorus esters and some polychlorocycloalkane and pyrethroid insecticides with the brain-specific t-butylbicyclophosphorothionate receptor.
Topics: Animals; Binding, Competitive; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Hexachlorocyclohexane; In Vitro Techniques; Insecticides; Ion Channels; Male; Microsomes, Liver; Pyrethrins; Rats; Receptors, GABA-A; Structure-Activity Relationship; Sulfur Radioisotopes; Synaptic Membranes | 1985 |
2,6,7-Trioxabicyclo[2.2.2]octanes: chemistry, toxicology and action at the GABA-gated chloride channel.
Topics: Animals; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Convulsants; gamma-Aminobutyric Acid; Hydrolysis; Insecta; Ion Channels; Ligands; Structure-Activity Relationship | 1988 |
Benzodiazepine receptors resolved.
Topics: Animals; Antibodies, Monoclonal; Autoradiography; Benzodiazepines; Benzodiazepinones; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Chlorides; Clonazepam; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Histocytochemistry; Humans; Immunologic Techniques; Ionophores; Muscimol; Neurons; Radioisotopes; Radioligand Assay; Receptors, GABA-A; Spinal Cord; Synapses; Tissue Distribution | 1986 |
125 other study(ies) available for tert-butylbicyclophosphorothionate and chlorine
Article | Year |
---|---|
Alterations in the gamma-aminobutyric acid-gated chloride channel following transient forebrain ischemia in the gerbil.
Topics: Animals; Autoradiography; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; gamma-Aminobutyric Acid; Gerbillinae; Ion Channel Gating; Ischemic Attack, Transient; Male; Membrane Proteins; Motor Activity; Muscimol | 1992 |
[3H-tert-butylbicyclo-ortho-benzoate--a new ligand for chloride ion channel of GABA-A receptor].
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; In Vitro Techniques; Ligands; Male; Radioligand Assay; Rats; Receptors, GABA-A; Synaptic Membranes; Tritium | 1992 |
Sex steroid hormones and GABAA receptor complex modulation.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Epoxy Compounds; Female; Gonadal Steroid Hormones; Guinea Pigs; In Vitro Techniques; Menstruation; Progesterone; Receptors, GABA-A; Synaptosomes | 1992 |
Decrease in GABAA receptor function induced by pentylenetetrazol kindling in the rat: role of N-methyl-D-aspartate (NMDA) receptors.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Dizocilpine Maleate; Down-Regulation; Isoniazid; Kindling, Neurologic; Male; Pentylenetetrazole; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate | 1992 |
Characterization of functional interactions of imidazoquinoxaline derivatives with benzodiazepine-gamma-aminobutyric acidA receptors.
Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Chlorides; Chlorine; Cloning, Molecular; Drug Interactions; Electrophysiology; Flunitrazepam; GABA-A Receptor Antagonists; Kinetics; Male; Membrane Proteins; Models, Chemical; Molecular Conformation; Oxadiazoles; Quinoxalines; Radioisotopes; Rats; Rats, Inbred Strains; Receptors, GABA-A; Structure-Activity Relationship; Synaptosomes; Tritium | 1992 |
Pharmacology of gamma-aminobutyric acidA receptor complex after the in vivo administration of the anxioselective and anticonvulsant beta-carboline derivative abecarnil.
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Chlorides; Exploratory Behavior; gamma-Aminobutyric Acid; In Vitro Techniques; Isoniazid; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Stress, Physiological | 1992 |
Isolation and identification from Salvia officinalis of two diterpenes which inhibit t-butylbicyclophosphoro[35S]thionate binding to chloride channel of rat cerebrocortical membranes in vitro.
Topics: Abietanes; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Diterpenes; Ion Channels; Kinetics; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Phenanthrenes; Plant Extracts; Plants, Medicinal; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1992 |
Characterization of bicuculline/baclofen-insensitive gamma-aminobutyric acid receptors expressed in Xenopus oocytes. I. Effects of Cl- channel inhibitors.
Topics: Animals; Baclofen; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Cerebral Cortex; Chloride Channels; Chlorides; Cloning, Molecular; Ion Channels; Membrane Proteins; Ovum; Picrotoxin; Rats; Receptors, GABA-A; Retina; RNA; Xenopus | 1992 |
The general anesthetic propofol: a biochemical tool to study the function of the GABA-coupled chloride channel.
Topics: Anesthetics; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; gamma-Aminobutyric Acid; Ion Channels; Male; Pentobarbital; Pregnanediones; Propofol; Rats; Rats, Inbred Strains | 1992 |
GABAA and NMDA receptor function during chronic administration of ethanol.
Topics: Alcoholic Intoxication; Animals; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Dizocilpine Maleate; Ethanol; Hippocampus; Ion Channels; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Substance Withdrawal Syndrome | 1992 |
The GABAA receptor complex in experimental absence seizures in rat: an autoradiographic study.
Topics: Animals; Autoradiography; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; Convulsants; Epilepsy, Absence; Flunitrazepam; GABA-A Receptor Antagonists; Ion Channels; Ionophores; Male; Membrane Proteins; Muscimol; Organ Specificity; Pyramidal Tracts; Pyridazines; Rats; Rats, Wistar; Receptors, GABA-A; Sulfur Radioisotopes; Tritium | 1992 |
Chronic benzodiazepine administration. VII. Behavioral tolerance and withdrawal and receptor alterations associated with clonazepam administration.
Topics: Animals; Behavior, Animal; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Clonazepam; Convulsants; Drug Tolerance; Flumazenil; Male; Mice; Motor Activity; Muscimol; Receptors, GABA-A; Substance Withdrawal Syndrome | 1991 |
Gamma-aminobutyric acidA receptor complexes in rat frontal cortex and spinal cord show differential responses to steroid modulation.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Desoxycorticosterone; Diazepam; gamma-Aminobutyric Acid; Ionophores; Male; Pentobarbital; Pregnanediol; Pregnanolone; Rats; Rats, Inbred Strains; Receptors, GABA-A; Spinal Cord; Steroids; Sulfur Radioisotopes | 1991 |
Prolonged exposure to GABA activates GABA-gated chloride channels in the presence of channel-blocking convulsants.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; Convulsants; Endrin; GABA Antagonists; gamma-Aminobutyric Acid; Ion Channel Gating; Kinetics; Male; Membrane Proteins; Mice; Mice, Inbred ICR; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sesterterpenes; Xenopus | 1991 |
In vivo administration of ethanol enhances the function of the gamma-aminobutyric acid-dependent chloride channel in the rat cerebral cortex.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Diazepam; Ethanol; gamma-Aminobutyric Acid; Ion Channels; Isoniazid; Male; Rats; Rats, Inbred Strains | 1990 |
Chronic administration of benzodiazepines--V. Rapid onset of behavioral and neurochemical alterations after discontinuation of alprazolam.
Topics: Alprazolam; Animals; Behavior, Animal; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Down-Regulation; Drug Tolerance; Ion Channels; Male; Mice; Motor Activity; Muscimol; Receptors, GABA-A; Substance Withdrawal Syndrome; Sulfur Radioisotopes | 1990 |
Blocking actions of heptachlor at an insect central nervous system GABA receptor.
Topics: Animals; Binding, Competitive; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Chloride Channels; Chlorides; Cockroaches; Electrophysiology; gamma-Aminobutyric Acid; Ganglia; Heptachlor; Houseflies; Ion Channels; Membrane Potentials; Membrane Proteins; Motor Neurons; Nervous System Physiological Phenomena; Rats; Receptors, GABA-A | 1990 |
Chronic morphine administration augments benzodiazepine binding and GABAA receptor function.
Topics: Animals; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Chlorine; Flunitrazepam; In Vitro Techniques; Ion Channels; Male; Mice; Morphine; Muscimol; Naltrexone; Radioisotopes; Receptors, GABA-A; Sulfur Radioisotopes | 1990 |
The action of stress and anxiolytic and anxiogenic benzodiazepine receptors ligands on [35S] T-butylbicyclophosphorothionate binding in the rat cerebral cortex.
Topics: Animals; Anti-Anxiety Agents; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Cerebral Cortex; Chlorides; Drug Interactions; Ion Channel Gating; Ion Channels; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological | 1990 |
Ex vivo binding of t-[35S )butylbicyclophosphorothionate: a biochemical tool to study the pharmacology of ethanol at the gamma-aminobutyric acid-coupled chloride channel.
Topics: Animals; Azides; Benzodiazepines; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Diazepam; Drug Interactions; Ethanol; gamma-Aminobutyric Acid; Ion Channels; Isoniazid; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sulfur Radioisotopes | 1991 |
Failure of gamma-hydroxybutyrate to alter the function of the GABAA receptor complex in the rat cerebral cortex.
Topics: Animals; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Diazepam; Flunitrazepam; In Vitro Techniques; Ion Channels; Isoniazid; Male; Nerve Tissue Proteins; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sodium Oxybate; Synaptic Transmission | 1991 |
Melatonin interaction with the benzodiazepine-GABA receptor complex in the CNS.
Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Cerebral Cortex; Chlorides; Diazepam; gamma-Aminobutyric Acid; Humans; Ion Channel Gating; Ion Channels; Melatonin; Muscimol; Prosencephalon; Rats; Receptors, GABA-A; Serotonin; Synaptosomes | 1991 |
Correlation between gamma-aminobutyric acidA receptor ligand-induced changes in t-butylbicyclophosphoro[35S]thionate binding and 36Cl- uptake in rat cerebrocortical membranes.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cerebral Cortex; Chloride Channels; Chlorides; Desoxycorticosterone; Diazepam; Ethanol; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Ligands; Membrane Proteins; Pentobarbital; Pregnanolone; Rats; Receptors, GABA-A; Synaptosomes | 1991 |
Neurochemical action of the general anaesthetic propofol on the chloride ion channel coupled with GABAA receptors.
Topics: Anesthetics; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; Flunitrazepam; Male; Membrane Proteins; Muscimol; Propofol; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1991 |
Pharmacogenetic analysis of mechanisms of emotional stress: effects of benzodiazepines.
Topics: Adrenocorticotropic Hormone; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Corticosterone; Diazepam; Exploratory Behavior; Hybridization, Genetic; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Motor Activity; Receptors, GABA-A; Stress, Psychological | 1990 |
Novel site-directed affinity ligands for GABA-gated chloride channels: synthesis, characterization, and molecular modeling of 1-(isothiocyanatophenyl)-4-tert-butyl-2,6,7-trioxabicyclo[2.2.2]octanes .
Topics: Animals; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chemical Phenomena; Chemistry; Chlorides; Convulsants; gamma-Aminobutyric Acid; Ion Channel Gating; Ligands; Male; Models, Molecular; Rats; Rats, Inbred Strains | 1991 |
Heterotropic cooperativity between putative recognition sites for progesterone metabolites and the atypical benzodiazepine Ro 5-4864.
Topics: Animals; Benzodiazepinones; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Convulsants; gamma-Aminobutyric Acid; Male; Pregnanediol; Pregnanolone; Progesterone; Rats; Rats, Inbred Strains | 1990 |
Electrophysiological study of tert-butylbicyclophosphorothionate-induced block of spontaneous chloride channels.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cell Membrane; Cells, Cultured; Chloride Channels; Chlorides; Convulsants; Electrophysiology; Ion Channel Gating; Kinetics; Membrane Proteins; Pituitary Gland; Swine | 1990 |
Allosteric modulation of t-[35S]butylbicyclophosphorothionate binding in rat brain by melatonin.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chloride Channels; Chlorides; Male; Melatonin; Membrane Proteins; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1990 |
Chronic benzodiazepine administration. VI. A partial agonist produces behavioral effects without tolerance or receptor alterations.
Topics: Animals; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Dose-Response Relationship, Drug; Drug Tolerance; Male; Mice; Motor Activity; Pyridazines; Receptors, GABA-A | 1990 |
gamma-Aminobutyric acid antagonism produced by an organophosphate-containing combustion product.
Topics: Animals; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Convulsants; Flurothyl; GABA Antagonists; Gas Chromatography-Mass Spectrometry; In Vitro Techniques; Male; Mice; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1990 |
Cloned GABA receptors are maintained in a stable cell line: allosteric and channel properties.
Topics: Animals; Antibodies, Monoclonal; Barbiturates; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Cell Line; Chlorides; Clone Cells; Convulsants; DNA; gamma-Aminobutyric Acid; Membrane Potentials; Muscimol; Neurons; Plasmids; Receptors, GABA-A; Spinal Cord; Transfection | 1990 |
Radiation inactivation of brain [35S]t-butylbicyclophosphorothionate binding sites reveals complicated molecular arrangements of the GABA/benzodiazepine receptor chloride channel complex.
Topics: Animals; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Cerebellum; Cerebral Cortex; Chlorides; Etazolate; Etomidate; In Vitro Techniques; Ion Channels; Molecular Weight; Muscimol; Organophosphorus Compounds; Radioligand Assay; Rats; Receptors, GABA-A; Sulfur Radioisotopes | 1985 |
Basic neuroproteins modulate TBPS recognition site.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Calcium Chloride; Cattle; Chlorides; gamma-Aminobutyric Acid; Ion Channels; Membranes; Nerve Tissue Proteins; Rats; Receptors, GABA-A | 1986 |
Interaction of t-butylbicyclophosphorothionate with gamma-aminobutyric acid-gated chloride channels in cultured cerebral neurons.
Topics: Animals; Anions; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cell Membrane; Cells, Cultured; Chick Embryo; Chlorides; gamma-Aminobutyric Acid; Ion Channels; Kinetics; Neurons | 1986 |
Steroid hormone metabolites are barbiturate-like modulators of the GABA receptor.
Topics: 20-alpha-Dihydroprogesterone; Animals; Binding, Competitive; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Chlorides; Desoxycorticosterone; Drug Synergism; Flunitrazepam; Hippocampus; In Vitro Techniques; Ion Channels; Progesterone; Rats; Receptors, GABA-A; Spinal Cord | 1986 |
The permeability of gamma-aminobutyric acid-gated chloride channels is described by the binding of a "cage" convulsant, t-butylbicyclophosphoro[35S]thionate.
Topics: Animals; Anions; Anura; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cerebral Cortex; Chlorides; gamma-Aminobutyric Acid; Ganglia, Spinal; Ion Channels; Male; Neurons; Permeability; Rats | 1986 |
GABA receptors induced in Xenopus oocytes by chick brain mRNA: evaluation of TBPS as a use-dependent channel-blocker.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chick Embryo; Chlorides; Female; GABA Antagonists; Ion Channels; Oocytes; Protein Biosynthesis; Receptors, GABA-A; RNA, Messenger | 1987 |
Stress-induced changes in t-[35S]butylbicyclophosphorothionate binding to gamma-aminobutyric acid-gated chloride channels are mimicked by in vitro occupation of benzodiazepine receptors.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cerebral Cortex; Chlorides; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Ion Channels; Kinetics; Male; Membranes; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological; Swimming | 1987 |
Benzodiazepine receptor modulation of [35S]TBPS binding to the chloride channel. Noncompetitive inhibition of classical benzodiazepines and competitive inhibition of the partial agonist, CGS 9895, by CGS 8216.
Topics: Animals; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Ion Channels; Pyrazoles; Rats; Receptors, GABA-A; Sulfur Radioisotopes | 1987 |
Neurochemical actions of anesthetic drugs on the gamma-aminobutyric acid receptor-chloride channel complex.
Topics: Alcohols; Anesthetics; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; gamma-Aminobutyric Acid; Ion Channels; Male; Mice; Mice, Inbred DBA; Receptors, GABA-A; Structure-Activity Relationship | 1987 |
Functional expression in the Xenopus oocyte of messenger ribonucleic acids encoding brain neurotransmitter receptors: further characterisation of the implanted GABA receptor.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chick Embryo; Chlorides; Cloning, Molecular; DNA; Dose-Response Relationship, Drug; Flunitrazepam; gamma-Aminobutyric Acid; Gene Expression Regulation; Glycosylation; Ion Channels; Oocytes; Poly A; Receptors, GABA-A; RNA; RNA, Messenger; Xenopus | 1987 |
Action of tremorgenic mycotoxins on GABAA receptor.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Electric Organ; Flunitrazepam; In Vitro Techniques; Ion Channels; Male; Muscimol; Mycotoxins; Rats; Rats, Inbred Strains; Receptors, GABA-A; Torpedo; Tremor | 1987 |
Antagonist-type interaction of glucocorticoids with the GABA receptor-coupled chloride channel.
Topics: Animals; Bicuculline; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Frontal Lobe; Glucocorticoids; Ion Channels; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes | 1987 |
Enhancement of t-[35S]butylbicyclophosphorothionate and [3H]strychnine binding by monovalent anions reveals similarities between gamma-aminobutyric acid- and glycine-gated chloride channels.
Topics: Animals; Anions; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cell Membrane; Cell Membrane Permeability; Chlorides; gamma-Aminobutyric Acid; Glycine; Ion Channels; Male; Medulla Oblongata; Rats; Rats, Inbred Strains; Spinal Cord; Strychnine; Sulfur Radioisotopes; Tritium | 1988 |
Differences in the biophysical properties of the benzodiazepine/gamma-aminobutyric acid receptor chloride channel complex in the long-sleep and short-sleep mouse lines.
Topics: Animals; Azides; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Flunitrazepam; gamma-Aminobutyric Acid; Heart; Ion Channels; Male; Mice; Mice, Mutant Strains; Receptors, GABA-A; Sleep | 1988 |
Chronic benzodiazepine administration. II. Discontinuation syndrome is associated with upregulation of gamma-aminobutyric acidA receptor complex binding and function.
Topics: Animals; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Drug Tolerance; Flumazenil; Flunitrazepam; Ion Channels; Lorazepam; Male; Mice; Motor Activity; Muscimol; Receptors, GABA-A; Time Factors | 1988 |
Action of polychlorocycloalkane insecticides on binding of [35S]t-butylbicyclophosphorothionate to Torpedo electric organ membranes and stereospecificity of the binding site.
Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Electric Organ; Hexachlorocyclohexane; Ion Channels; Receptors, GABA-A; Stereoisomerism; Torpedo | 1988 |
Modulation of the benzodiazepine/gamma-aminobutyric acid receptor chloride channel complex by inhalation anesthetics.
Topics: Anesthesia, Inhalation; Anesthetics; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Enflurane; Ether; Halothane; Ion Channels; Male; Methoxyflurane; Muscimol; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes | 1988 |
Involvement of peripheral-type benzodiazepine receptors in the proconvulsant actions of pyrethroid insecticides.
Topics: Animals; Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Dose-Response Relationship, Drug; In Vitro Techniques; Ion Channels; Isoquinolines; Male; Pyrethrins; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stereoisomerism | 1988 |
Differentiation of activities within the GABAA-chloride ionophore complex by means of 35-S-TBPS binding.
Topics: Allosteric Regulation; Animals; Anti-Anxiety Agents; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Convulsants; Hypnotics and Sedatives; Ion Channels; Ionophores; Rats; Receptors, GABA-A | 1988 |
Aging reduces the GABA-dependent 36Cl- flux in rat brain membrane vesicles.
Topics: Aging; Animals; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Cerebellum; Cerebral Cortex; Chlorides; gamma-Aminobutyric Acid; Hippocampus; Ion Channels; Male; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1988 |
Asymmetrical activation of GABA-gated chloride channels in cerebral cortex.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Flumazenil; Functional Laterality; Ion Channels; Kinetics; Male; Organ Specificity; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1988 |
Chemical kindling decreases GABA-activated chloride channels of mouse brain.
Topics: Animals; Autoradiography; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; gamma-Aminobutyric Acid; Ion Channels; Kindling, Neurologic; Male; Mice; Mice, Inbred ICR; Muscimol; Sulfur Radioisotopes | 1989 |
Diazepam sensitizes mice to FG 7142 and reduces muscimol-stimulated 36Cl- flux.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Chlorides; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Ion Channels; Kindling, Neurologic; Mice; Mice, Inbred ICR; Muscimol | 1989 |
Interaction of caffeine with the GABAA receptor complex: alterations in receptor function but not ligand binding.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Caffeine; Cerebral Cortex; Chlorides; In Vitro Techniques; Ion Channels; Kinetics; Ligands; Male; Mice; Muscimol; Receptors, GABA-A; Sulfur Radioisotopes; Synaptosomes | 1989 |
Dietary choline intake modulates benzodiazepine receptor binding and gamma-aminobutyric acidA receptor function in mouse brain.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; Choline; Diet; Flumazenil; Male; Membrane Proteins; Mice; Motor Activity; Receptors, GABA-A | 1989 |
meta- and para-isothiocyanato-t-butylbicycloorthobenzoate: irreversible ligands of the gamma-aminobutyric acid-regulated chloride ionophore.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chloride Channels; Chlorides; gamma-Aminobutyric Acid; In Vitro Techniques; Isothiocyanates; Ligands; Male; Membrane Proteins; Rats; Rats, Inbred Strains; Structure-Activity Relationship; Thiocyanates | 1989 |
Distribution and pharmacological properties of the GABAA/benzodiazepine/chloride ionophore receptor complex in the brain of the fish Anguilla anguilla.
Topics: Anguilla; Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Flunitrazepam; gamma-Aminobutyric Acid; Ionophores; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A; Tissue Distribution | 1989 |
Chronic benzodiazepine administration. III. Upregulation of gamma-aminobutyric acidA receptor binding and function associated with chronic benzodiazepine antagonist administration.
Topics: Animals; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Chlorides; Flumazenil; Male; Membrane Proteins; Mice; Motor Activity; Receptors, GABA-A | 1989 |
Steroid anesthetics and naturally occurring analogs modulate the gamma-aminobutyric acid receptor complex at a site distinct from barbiturates.
Topics: Anesthetics; Animals; Barbiturates; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; In Vitro Techniques; Male; Muscimol; Pregnanediones; Rats; Rats, Inbred Strains; Receptors, GABA-A; Steroids; Structure-Activity Relationship | 1989 |
Differential seizure sensitivities to picrotoxinin in two inbred strains of mice (DBA/2J and BALB/c ByJ): parallel changes in GABA receptor-mediated chloride flux and receptor binding.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Dose-Response Relationship, Drug; Frontal Lobe; Male; Mice; Mice, Inbred BALB C; Mice, Inbred DBA; Muscimol; Pentobarbital; Picrotoxin; Receptors, GABA-A; Seizures; Species Specificity; Synaptosomes | 1989 |
Complex interactions between pregnenolone sulfate and the t-butylbicyclophosphorothionate-labeled chloride ionophore in rat brain.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cerebral Cortex; Chloride Channels; Chlorides; Drug Interactions; Ionophores; Kinetics; Male; Membrane Proteins; Pregnenolone; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1989 |
Ultraviolet irradiation selectively disrupts the gamma-aminobutyric acid/benzodiazepine receptor-linked chloride ionophore.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Chloride Channels; Chlorides; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Membrane Proteins; Rats; Rats, Inbred Strains; Receptors, GABA-A; Ultraviolet Rays | 1989 |
Age-related loss of t-[35S]butylbicyclophosphorothionate binding to the gamma-aminobutyric acidA receptor-coupled chloride ionophore in rat cerebral cortex.
Topics: Aging; Animals; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cerebral Cortex; Chlorides; Female; Ionophores; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sulfur Radioisotopes | 1989 |
Effect of halide ions on t-[35S]butylbicyclophosphorothionate binding.
Topics: Animals; Anions; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Bromides; Chlorides; Fluorides; Halogens; Iodides; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1989 |
Differential effects of iodide and chloride on allosteric interactions of the GABAA receptor.
Topics: Allosteric Regulation; Animals; Anions; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Chlorides; Diazepam; gamma-Aminobutyric Acid; Iodides; Male; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1989 |
Persistent alterations in GABAA receptor binding and function after prenatal lorazepam administration in the chick.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chick Embryo; Chickens; Chlorides; Female; Flunitrazepam; Lorazepam; Muscimol; Pregnancy; Prenatal Exposure Delayed Effects; Radioligand Assay; Receptors, GABA-A | 1989 |
The effect of ethanol on 35S-TBPS binding to mouse brain membranes in the presence of chloride.
Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Benzodiazepinones; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Diazepam; Drug Tolerance; Ethanol; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred C57BL; Pentobarbital; Substance-Related Disorders; Sulfur Radioisotopes | 1989 |
Fluidization of brain membranes by A2C does not produce anesthesia and does not augment muscimol-stimulated 36Cl- influx.
Topics: Anesthesia; Animals; Benzyl Alcohols; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Chlorine; gamma-Aminobutyric Acid; Male; Membrane Fluidity; Membranes; Mice; Mice, Inbred ICR; Muscimol; Radioisotopes; Stearates; Stearic Acids; Synaptosomes; Temperature | 1989 |
Behavioral and functional studies indicate a role for GABAAergic transmission in the actions of ethanol.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Chlorides; Ethanol; Flunitrazepam; Male; Mice; Mice, Inbred C57BL; Picrotoxin; Rats; Receptors, GABA-A; Seizures; Spinal Cord | 1987 |
(+/-)-4-tert-butyl-3-cyano-1-(4-ethynylphenyl)-2,6,7-trioxabi cyclo[2.2.2]octane: synthesis of a remarkably potent GABAA receptor antagonist.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; GABA Antagonists; Mice; Rats; Receptors, GABA-A | 1988 |
Steroid modulation of the chloride ionophore in rat brain: structure-activity requirements, regional dependence and mechanism of action.
Topics: Androstane-3,17-diol; Animals; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Female; In Vitro Techniques; Ionophores; Kinetics; Male; Mice; Pregnanes; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Structure-Activity Relationship; Sulfur Radioisotopes; Uterus | 1988 |
CNS depressants accelerate the dissociation of 35S-TBPS binding and GABA enhances their displacing potencies.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cerebral Cortex; Chloride Channels; Chlorides; Convulsants; gamma-Aminobutyric Acid; Hypnotics and Sedatives; In Vitro Techniques; Membrane Proteins; Rats; Receptors, GABA-A | 1988 |
Antagonism of ethanol and pentobarbital actions by benzodiazepine inverse agonists: neurochemical studies.
Topics: Animals; Azides; Benzodiazepines; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Carbolines; Chloride Channels; Chlorides; Ethanol; Male; Membrane Fluidity; Membrane Proteins; Mice; Mice, Inbred ICR; Pentobarbital; Receptors, GABA-A | 1988 |
[Effect of stress on the function of chloride channels associated with the GABA receptor complex].
Topics: Animals; Bicuculline; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cerebral Cortex; Chloride Channels; Chlorides; Male; Membrane Proteins; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological | 1988 |
Lorazepam administration during embryonic development alters GABAA receptor binding and function.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chick Embryo; Chlorides; Embryonic and Fetal Development; Flunitrazepam; Lorazepam; Receptors, GABA-A; Subcellular Fractions | 1988 |
Modulation of gamma-aminobutyric acid-stimulated chloride influx by bicycloorthocarboxylates, bicyclophosphorus esters, polychlorocycloalkanes and other cage convulsants.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; Convulsants; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Membrane Proteins; Rats; Rats, Inbred Strains; Structure-Activity Relationship | 1988 |
Actions of avermectin B1a on the gamma-aminobutyric acidA receptor and chloride channels in rat brain.
Topics: Animals; Bicuculline; Binding, Competitive; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; Dose-Response Relationship, Drug; Flunitrazepam; Ivermectin; Kinetics; Male; Membrane Proteins; Muscimol; Rats; Receptors, GABA-A | 1986 |
Changes of 36Cl- flux and 35S-TBPS binding induced by stress and gabaergic drugs.
Topics: Animals; Anti-Anxiety Agents; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cell Membrane; Cerebral Cortex; Chlorides; Convulsants; gamma-Aminobutyric Acid; Male; Neurons; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological | 1988 |
t-[3H]butylbicycloorthobenzoate: new radioligand probe for the gamma-aminobutyric acid-regulated chloride ionophore.
Topics: Androstanes; Animals; Azasteroids; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chemical Phenomena; Chemistry; Chlorides; gamma-Aminobutyric Acid; Hydrogen-Ion Concentration; Ionophores; Kinetics; Male; Rats; Receptors, GABA-A; Temperature | 1985 |
GABA, depressants and chloride ions affect the rate of dissociation of 35S-t-butylbicyclophosphorothionate binding.
Topics: Animals; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Central Nervous System Depressants; Cerebral Cortex; Chlorides; Convulsants; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1985 |
Neurotoxic insecticides inhibit GABA-dependent chloride uptake by mouse brain vesicles.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; gamma-Aminobutyric Acid; In Vitro Techniques; Insecticides; Male; Mice; Mice, Inbred ICR; Picrotoxin; Receptors, GABA-A | 1985 |
Benzodiazepine anticonvulsants accelerate and beta-carboline convulsants decelerate the kinetics of [35S]TBPS binding at the chloride ionophore.
Topics: Animals; Anticonvulsants; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Chlorides; Convulsants; Flunitrazepam; In Vitro Techniques; Ionophores; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Membranes | 1985 |
Acute, stress-induced changes in the benzodiazepine/gamma-aminobutyric acid receptor complex are confined to the chloride ionophore.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bromides; Cerebral Cortex; Chlorides; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Iodides; Ionophores; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological; Sulfur Radioisotopes; Swimming; Tritium | 1986 |
Rapid, stress-induced modification of the benzodiazepine receptor-coupled chloride ionophore.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Flunitrazepam; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stimulation, Chemical; Stress, Physiological; Swimming; Temperature | 1986 |
Modulation of the chloride ionophore by benzodiazepine receptor ligands: influence of gamma-aminobutyric acid and ligand efficacy.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Cerebral Cortex; Chlorides; Clonazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Ionophores; Kinetics; Ligands; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sulfur Radioisotopes; Tritium | 1986 |
A quantitative relationship between Cl- enhanced [3H]flunitrazepam and [35S]t-butylbicyclophosphorothionate binding to the benzodiazepine/GABA receptor chloride ionophore complex.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cerebral Cortex; Chlorides; Flunitrazepam; In Vitro Techniques; Male; Phospholipases A; Phospholipases A2; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stimulation, Chemical | 1986 |
Environmentally-induced modification of the benzodiazepine/GABA receptor coupled chloride ionophore.
Topics: Animals; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Environment; Flunitrazepam; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological; Swimming | 1987 |
Pregnenolone-sulfate: an endogenous antagonist of the gamma-aminobutyric acid receptor complex in brain?
Topics: Adrenal Glands; Animals; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Male; Muscimol; Picrotoxin; Pregnenolone; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stimulation, Chemical | 1987 |
Structure-activity relationships for steroid interaction with the gamma-aminobutyric acidA receptor complex.
Topics: Animals; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Desoxycorticosterone; Electric Conductivity; Ethanol; Evoked Potentials; Flunitrazepam; Muscimol; Pregnanes; Progesterone; Rats; Rats, Inbred Strains; Receptors, GABA-A; Steroids; Structure-Activity Relationship | 1987 |
Cyclodiene insecticides inhibit GABAA receptor-regulated chloride transport.
Topics: Animals; Bicuculline; Biological Transport; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Insecticides; Male; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1987 |
[35S]TBPS binding to membranes of the female sex organs: modulation of chloride ionophore by GABA and pentobarbital.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Convulsants; Fallopian Tubes; Female; gamma-Aminobutyric Acid; Genitalia, Female; In Vitro Techniques; Ionophores; Membranes; Ovary; Pentobarbital; Rats; Rats, Inbred Strains; Uterus | 1988 |
GABA-dependent modulation of the Cl- ionophore by steroids in rat brain.
Topics: Animals; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Cholesterol; gamma-Aminobutyric Acid; In Vitro Techniques; Ionophores; Male; Rats; Rats, Inbred Strains; Steroids | 1987 |
Gamma-aminobutyric acid and alcohol actions: neurochemical studies of long sleep and short sleep mice.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Cerebellum; Chlorides; Diencephalon; Drug Synergism; Ethanol; Female; gamma-Aminobutyric Acid; Hippocampus; Mice; Muscimol; Pentobarbital; Sleep; Telencephalon | 1986 |
In vitro characterization of agonist, antagonist, inverse agonist and agonist/antagonist benzodiazepines.
Topics: Animals; Benzodiazepines; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Etazolate; Ion Channels; Muscimol; Rats; Receptors, GABA-A | 1984 |
Solubilization and anionic regulation of cerebral sedative/convulsant receptors labeled with [35S] tert-butylbicyclophosphorothionate (TBPS).
Topics: Animals; Anions; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cell Membrane; Cerebral Cortex; Chlorides; Cholic Acids; Detergents; Ion Channels; Male; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Solubility | 1984 |
Alkyl-substituted gamma-butyrolactones inhibit [35S]TBPS binding to a GABA linked chloride ionophore.
Topics: 4-Butyrolactone; Animals; Barbiturates; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Furans; gamma-Aminobutyric Acid; In Vitro Techniques; Ionophores; Male; Membranes; Picrotoxin; Rats; Rats, Inbred Strains | 1984 |
Enhancement by GABA of the association rate of picrotoxin and tert-butylbicyclophosphorothionate to the rat cloned alpha 1 beta 2 gamma 2 GABAA receptor subtype.
Topics: Animals; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Chlorides; Cloning, Molecular; Dose-Response Relationship, Drug; Drug Interactions; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Ion Channels; Kidney; Kinetics; Patch-Clamp Techniques; Picrotoxin; Rats; Receptors, GABA-A | 1995 |
Characterization of U-97775 as a GABAA receptor ligand of dual functionality in cloned rat GABAA receptor subtypes.
Topics: Animals; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Chlorides; Electrophysiology; Flumazenil; Humans; Imidazoles; Ligands; Quinoxalines; Rats; Receptors, GABA-A; Recombinant Proteins | 1995 |
Chronic neurosteroid treatment produces functional heterologous uncoupling at the gamma-aminobutyric acid type A/benzodiazepine receptor complex in mammalian cortical neurons.
Topics: Androstanes; Animals; Azasteroids; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Cerebral Cortex; Chlorides; Chlorine; Convulsants; Drug Interactions; GABA Antagonists; gamma-Aminobutyric Acid; Kinetics; Mice; Mice, Inbred C57BL; Neurons; Pregnanolone; Radioisotopes; Radioligand Assay; Receptors, GABA-A; Sulfur Radioisotopes; Time Factors; Tritium | 1995 |
Alterations in the brain GABAA/benzodiazepine receptor-chloride ionophore complex in a genetic model of paroxysmal dystonia: a quantitative autoradiographic analysis.
Topics: Animals; Autoradiography; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Cricetinae; Dystonia; Flunitrazepam; Ionophores; Male; Models, Genetic; Muscimol; Radiography; Receptors, GABA-A | 1995 |
The effect of cyclopyrrolones on GABAA receptor function is different from that of benzodiazepines.
Topics: Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Benzodiazepines; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Chlorine; Flumazenil; Hypnotics and Sedatives; Kinetics; Male; Mice; Mice, Inbred Strains; Muscimol; Naphthyridines; Piperazines; Radioisotopes; Receptors, GABA-A; Sulfur Compounds; Sulfur Radioisotopes; Tritium | 1994 |
Gamma-aminobutyric acidA receptor function is inhibited by microtubule depolymerization.
Topics: Animals; Biological Transport; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Chlorides; Colchicine; Convulsants; Dose-Response Relationship, Drug; Flunitrazepam; Histones; Humans; Lumicolchicines; Membranes; Mice; Microtubules; Muscimol; Nocodazole; Paclitaxel; Phosphorylation; Receptors, GABA-A; Vinblastine; Xenopus | 1994 |
Age-related changes of GABA-activated chloride channel properties in brain cortex synaptic plasma membrane: evidence for phospholipase involvement.
Topics: Aging; Animals; Arachidonic Acid; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Chlorides; Convulsants; Diglycerides; gamma-Aminobutyric Acid; Kinetics; Muscimol; Phospholipases; Picrotoxin; Rats; Rats, Wistar; Sulfur Radioisotopes; Synaptic Membranes; Synaptosomes | 1994 |
Effects of 5-HT3 receptor antagonists on binding and function of mouse and human GABAA receptors.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Flumazenil; Flunitrazepam; Humans; Indazoles; Indoles; Male; Mice; Mice, Inbred ICR; Receptors, GABA-A; Serotonin Antagonists; Tropanes; Tropisetron; Xenopus laevis | 1994 |
Steroid modulation of GABAA receptors in an amphibian brain.
Topics: Animals; Autoradiography; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Chlorides; Convulsants; Corticosterone; Flunitrazepam; Kinetics; Male; Mammals; Neurons; Pregnanolone; Pregnenolone; Rats; Receptors, GABA-A; Salamandridae; Species Specificity; Steroids; Sulfur Radioisotopes; Synaptosomes; Tritium | 1994 |
GABAergic and dopaminergic transmission in the brain of Roman high-avoidance and Roman low-avoidance rats.
Topics: Amygdala; Animals; Avoidance Learning; Benzazepines; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Cerebral Cortex; Chlorides; Convulsants; Corpus Striatum; Dopamine; Emotions; Flunitrazepam; gamma-Aminobutyric Acid; Hippocampus; Kinetics; Male; Nucleus Accumbens; Organ Specificity; Prefrontal Cortex; Rats; Rats, Mutant Strains; Receptors, Dopamine D1; Species Specificity; Synaptic Transmission | 1994 |
Modulatory action of arachidonic acid on GABAA/chloride channel receptor function in adult and aged brain cortex membranes.
Topics: Aging; Animals; Arachidonic Acid; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Cerebral Cortex; Chloride Channels; Chlorides; Convulsants; Docosahexaenoic Acids; Fatty Acids, Nonesterified; Kinetics; Male; Muscimol; Rats; Rats, Wistar; Receptors, GABA-A; Stearic Acids; Synaptic Membranes; Synaptosomes | 1993 |
Partial and full agonists/inverse agonists affect [35S]TBPS binding at different occupancies of central benzodiazepine receptors.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Convulsants; Ionophores; Radioligand Assay; Rats; Receptors, GABA-A; Sulfur Radioisotopes | 1993 |
Anticonvulsant doses of 2-chloro-N6-cyclopentyladenosine, an adenosine A1 receptor agonist, reduce GABAergic transmission in different areas of the mouse brain.
Topics: Adenosine; Animals; Anticonvulsants; Behavior, Animal; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Depression, Chemical; Diazepam; Dose-Response Relationship, Drug; Flunitrazepam; gamma-Aminobutyric Acid; Isoniazid; Male; Mice; Mice, Inbred Strains; Purinergic P1 Receptor Antagonists; Receptors, GABA; Receptors, Purinergic P1; Seizures; Sulfur Radioisotopes; Synaptic Transmission; Tritium; Xanthines | 1993 |
GABAA receptor function in the gamma-hydroxybutyrate model of generalized absence seizures.
Topics: Aminocaproates; Animals; Anticonvulsants; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Chlorine; Convulsants; Electroencephalography; Epilepsy, Absence; Flunitrazepam; In Vitro Techniques; Kinetics; Male; Muscimol; Radioisotopes; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sodium Oxybate; Synaptosomes; Vigabatrin | 1993 |
Swim stress selectively alters the specific binding of a benzodiazepine antagonist in mice.
Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Flumazenil; Flurazepam; In Vitro Techniques; Kinetics; Male; Mice; Receptors, GABA-A; Stress, Physiological; Swimming; Tissue Distribution | 1993 |
Stereospecific actions of the inhalation anesthetic isoflurane at the GABAA receptor complex.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Flunitrazepam; In Vitro Techniques; Isoflurane; Male; Mice; Receptors, GABA-A; Stereoisomerism; Sulfur Radioisotopes | 1993 |
U-89843A is a novel allosteric modulator of gamma-aminobutyric acidA receptors.
Topics: Allosteric Regulation; Animals; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Chloride Channel Agonists; Chlorides; GABA Modulators; Humans; Male; Mice; Pyrimidines; Pyrroles; Rats; Receptors, GABA-A | 1995 |
High-affinity partial agonist imidazo[1,5-a]quinoxaline amides, carbamates, and ureas at the gamma-aminobutyric acid A/benzodiazepine receptor complex.
Topics: Animals; Anxiety; Benzodiazepines; Binding, Competitive; Brain; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Flunitrazepam; GABA Agonists; GABA Antagonists; Molecular Conformation; Molecular Structure; Oxadiazoles; Pentylenetetrazole; Quinoxalines; Rats; Receptors, GABA-A | 1996 |
Effects of the androgenic/anabolic steroid stanozolol on GABAA receptor function: GABA-stimulated 36Cl- influx and [35S] TBPS binding.
Topics: Anabolic Agents; Animals; Brain; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Stanozolol | 1996 |
Interactions of the neurosteroid dehydroepiandrosterone sulfate with the GABA(A) receptor complex reveals that it may act via the picrotoxin site.
Topics: Animals; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Cerebellum; Cerebral Cortex; Chlorides; Dehydroepiandrosterone; Dehydroepiandrosterone Sulfate; gamma-Aminobutyric Acid; In Vitro Techniques; Ion Transport; Male; Mice; Mice, Inbred C57BL; Picrotoxin; Protein Binding; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A | 1997 |
Modulation of the GABA(A)-gated chloride channel by reactive oxygen species.
Topics: Animals; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Hippocampus; Hydrogen Peroxide; Ion Channel Gating; Microscopy, Confocal; Organ Culture Techniques; Oxidants; Oxidative Stress; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Receptors, GABA-A; Sulfur Radioisotopes; Synaptic Transmission | 2002 |
GABA released from cultured cortical neurons influences the modulation of t-[(35)S]butylbicyclophosphorothionate binding at the GABAA receptor Effects of thymol.
Topics: Allosteric Regulation; Anesthetics, Intravenous; Animals; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Cell Survival; Cells, Cultured; Cerebral Cortex; Chlorides; gamma-Aminobutyric Acid; Mice; Propofol; Receptors, GABA-A; Thymol | 2008 |
Pyrethroid insecticides indirectly inhibit GABA-dependent 36Cl- influx in synaptoneurosomes from the trout brain.
Topics: Animals; Brain Chemistry; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorine; Depression, Chemical; gamma-Aminobutyric Acid; In Vitro Techniques; Insecticides; Nerve Tissue Proteins; Nitriles; Pyrethrins; Salmon; Synaptosomes; Tetrodotoxin; Veratridine | 1991 |
Lindane cytotoxicity in cultured neocortical neurons is ameliorated by GABA and flunitrazepam.
Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Cell Survival; Cells, Cultured; Cerebral Cortex; Chloride Channels; Chlorine; Convulsants; Flunitrazepam; gamma-Aminobutyric Acid; Hexachlorocyclohexane; Mice; Neurons; Potassium; Receptors, GABA | 1994 |
Effects of the anticonvulsant losigamone and its isomers on the GABAA receptor system.
Topics: Animals; Anticonvulsants; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Cerebral Cortex; Chloride Channels; Chlorine; Convulsants; Dose-Response Relationship, Drug; Epilepsy; Female; Furans; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Isomerism; Male; Mice; Mice, Inbred C57BL; Radioisotopes; Rats; Rats, Sprague-Dawley; Receptors, GABA-A | 1995 |
Studies on picrotoxin binding sites of GABAA receptors in rat cortical synaptoneurosomes.
Topics: Animals; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorine; Desoxycorticosterone; Diazepam; In Vitro Techniques; Male; Membranes; Muscimol; Pentobarbital; Picrotoxin; Radioisotopes; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Steroids; Synaptosomes | 1994 |
Effects of the chlorotriazine herbicide, cyanazine, on GABA(A) receptors in cortical tissue from rat brain.
Topics: Animals; Azides; Benzodiazepines; Binding Sites; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Chlorine; GABA Agonists; Herbicides; Male; Muscimol; Radioisotopes; Rats; Rats, Long-Evans; Receptors, GABA-A; Synaptosomes; Triazines | 1999 |