tert-butylbicyclophosphorothionate has been researched along with bicuculline in 51 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 20 (39.22) | 18.7374 |
| 1990's | 25 (49.02) | 18.2507 |
| 2000's | 5 (9.80) | 29.6817 |
| 2010's | 1 (1.96) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Miledi, R; Polenzani, L; Woodward, RM | 1 |
| Biggio, G; Concas, A; Gessa, GL; Peduto, VA; Santoro, G | 1 |
| Lummis, SC; Rauh, JJ; Sattelle, DB; Wong, JF | 1 |
| Blakeman, DP; Im, WB | 1 |
| Abendschein, KH; Dawson, R; Peris, J; Shawley, A | 1 |
| Feltz, P; Zhang, ZW | 1 |
| Barnard, EA; Devine, J; Macdonald, RL; Moss, SJ; Nayeem, N; Porter, NM; Smart, TG; Stephenson, FA | 1 |
| Danielou, G; Lloyd, GK; Thuret, F | 1 |
| Biggio, G; Concas, A; Mascia, MP; Sanna, E; Serra, M | 1 |
| Majewska, MD | 1 |
| Atsoggiu, T; Biggio, G; Concas, A; Pepitoni, S; Toffano, G | 1 |
| Abel, MS; Blume, AJ; Garrett, KM | 1 |
| Moguilewsky, M; Philibert, D; Shu, C; Vincens, M | 1 |
| Peris, J; Wehner, JM; Zahniser, NR | 1 |
| Ho, IK; Hoskins, B; Ito, Y; Lim, DK | 1 |
| Atsoggiu, T; Concas, A; Serra, M | 1 |
| Gallager, DW; Heninger, C | 1 |
| Abalis, IM; Eldefrawi, AT; Eldefrawi, ME | 1 |
| Haefely, W; Möhler, H; Richards, JG; Schoch, P | 1 |
| Concas, A; Gehlert, DR; Wamsley, JK; Yamamura, HI | 1 |
| Gee, KW | 1 |
| Eldefrawi, AT; Eldefrawi, ME; Gant, DB | 1 |
| Crabbe, JC; Feller, DJ; Harris, RA | 1 |
| Liljequist, S; Tabakoff, B | 2 |
| Gallo, V; Guidotti, A; Vaccarino, F; Wise, BC | 1 |
| Ramanjaneyulu, R; Ticku, MK | 2 |
| Snowman, AM; Snyder, SH; Trifiletti, RR | 1 |
| Bymaster, FP; Squires, RF; Threlkeld, PG; Wong, DT | 1 |
| Korpi, ER; Lüddens, H | 1 |
| Chen, DZ; Chen, SH; Katsura, M; Kuriyama, K; Ohkuma, S | 1 |
| Cancedda, E; Corda, MG; Giorgi, O; Lecca, D; Orlandi, M | 1 |
| Belelli, D; Chen, R; Lambert, JJ; Lan, NC; Peters, JA; Reyes, A | 1 |
| Biggio, G; Concas, A; Dazzi, L; Maciocco, E; Mascia, MP; Santoro, G | 1 |
| Cancedda, E; Corda, MG; Giorgi, O | 1 |
| Maksay, G; van Rijn, CM | 1 |
| Finn, DA; Gee, KW | 1 |
| Korpi, ER; Lüddens, H; Seeburg, PH | 1 |
| Harris, CL; Quinn, MR | 1 |
| Biggio, G; Casula, A; Maciocco, E; Murgia, A; Sanna, E; Tuligi, G; Usala, M | 1 |
| Buckingham, SD; Rauh, J; Sattelle, DB; Schnee, M | 1 |
| Brannen, KC; Devaud, LL; Lauder, JM; Liu, J | 1 |
| Olsen, RW; Sapp, DW; Srinivasan, S; Tobin, AJ | 1 |
| Alho, H; Anghelescu, I; Klawe, C; Korpi, ER; Lüddens, H; Mäkelä, R; Oja, SS; Uusi-Oukari, M | 1 |
| Behrends, JC | 1 |
| Gillardin, J; Poisbeau, P; Rybalchenko, V; Schlichter, R; Verleye, M | 1 |
| Gillardin, JM; Neliat, G; Pansart, Y; Schlichter, R; Verleye, M | 1 |
| Chigr, F; M'hamed, SB; Najimi, M | 1 |
| Hartmann, J; Hildmann, O; Kiewert, C; Klein, J; Kumar, V; Naik, RS; Rueda, M | 1 |
| Baptista-Hon, DT; Deeb, TZ; Gallacher, M; Hales, TG; Othman, NA; Perry, DC | 1 |
1 review(s) available for tert-butylbicyclophosphorothionate and bicuculline
| Article | Year |
|---|---|
Benzodiazepine receptors resolved.
Topics: Animals; Antibodies, Monoclonal; Autoradiography; Benzodiazepines; Benzodiazepinones; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Chlorides; Clonazepam; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Histocytochemistry; Humans; Immunologic Techniques; Ionophores; Muscimol; Neurons; Radioisotopes; Radioligand Assay; Receptors, GABA-A; Spinal Cord; Synapses; Tissue Distribution | 1986 |
50 other study(ies) available for tert-butylbicyclophosphorothionate and bicuculline
| Article | Year |
|---|---|
Characterization of bicuculline/baclofen-insensitive gamma-aminobutyric acid receptors expressed in Xenopus oocytes. I. Effects of Cl- channel inhibitors.
Topics: Animals; Baclofen; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Cerebral Cortex; Chloride Channels; Chlorides; Cloning, Molecular; Ion Channels; Membrane Proteins; Ovum; Picrotoxin; Rats; Receptors, GABA-A; Retina; RNA; Xenopus | 1992 |
Biochemical and electrophysiologic evidence that propofol enhances GABAergic transmission in the rat brain.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Dose-Response Relationship, Drug; Flunitrazepam; gamma-Aminobutyric Acid; Male; Membrane Proteins; Propofol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Transmission | 1991 |
Pharmacology of insect GABA receptors.
Topics: Acetylcholine; Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Female; Flunitrazepam; gamma-Aminobutyric Acid; Houseflies; Insecticides; Male; Membrane Proteins; Nervous System; Neurons; Periplaneta; Pregnanes; Receptors, GABA-A; Synapses | 1991 |
Correlation between gamma-aminobutyric acidA receptor ligand-induced changes in t-butylbicyclophosphoro[35S]thionate binding and 36Cl- uptake in rat cerebrocortical membranes.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cerebral Cortex; Chloride Channels; Chlorides; Desoxycorticosterone; Diazepam; Ethanol; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Ligands; Membrane Proteins; Pentobarbital; Pregnanolone; Rats; Receptors, GABA-A; Synaptosomes | 1991 |
Regulation of 35S-TBPS binding by bicuculline is region specific in rat brain.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Cerebral Cortex; Chromatography, High Pressure Liquid; gamma-Aminobutyric Acid; Male; Microsomes; Rats; Rats, Inbred Strains; Substantia Nigra; Sulfur Radioisotopes | 1991 |
Bicuculline blocks nicotinic acetylcholine response in isolated intermediate lobe cells of the pig.
Topics: Animals; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; GABA Antagonists; In Vitro Techniques; Isonicotinic Acids; Membrane Potentials; Pyridazines; Receptors, Nicotinic; Solutions; Swine | 1991 |
Cloned GABA receptors are maintained in a stable cell line: allosteric and channel properties.
Topics: Animals; Antibodies, Monoclonal; Barbiturates; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Cell Line; Chlorides; Clone Cells; Convulsants; DNA; gamma-Aminobutyric Acid; Membrane Potentials; Muscimol; Neurons; Plasmids; Receptors, GABA-A; Spinal Cord; Transfection | 1990 |
The activity of zolpidem and other hypnotics within the gamma-aminobutyric acid (GABAA) receptor supramolecular complex, as determined by 35S-t-butylbicyclophosphorothionate (35S-TBPS) binding to rat cerebral cortex membranes.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Hypnotics and Sedatives; In Vitro Techniques; Male; Pyridines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Zolpidem | 1990 |
Diazepam enhances bicuculline-induced increase of t-[35S]butylbicyclophosphorothionate binding in unwashed membrane preparations from rat cerebral cortex.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cerebral Cortex; Convulsants; Diazepam; gamma-Aminobutyric Acid; Male; Rats; Rats, Inbred Strains; Subcellular Fractions | 1990 |
Antagonist-type interaction of glucocorticoids with the GABA receptor-coupled chloride channel.
Topics: Animals; Bicuculline; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Chlorides; Frontal Lobe; Glucocorticoids; Ion Channels; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes | 1987 |
Aging reduces the GABA-dependent 36Cl- flux in rat brain membrane vesicles.
Topics: Aging; Animals; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Cerebellum; Cerebral Cortex; Chlorides; gamma-Aminobutyric Acid; Hippocampus; Ion Channels; Male; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1988 |
Differential effects of iodide and chloride on allosteric interactions of the GABAA receptor.
Topics: Allosteric Regulation; Animals; Anions; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Chlorides; Diazepam; gamma-Aminobutyric Acid; Iodides; Male; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1989 |
A progesterone metabolite enhances the activity of the GABAA receptor complex at the pituitary level.
Topics: 5-alpha-Dihydroprogesterone; Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; In Vitro Techniques; Male; Membranes; Muscimol; Picrotoxin; Pituitary Gland, Anterior; Pregnanediones; Progesterone; Prolactin; Radioimmunoassay; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1989 |
[35S]TBPS binding sites are decreased in the colliculi of mice with a genetic predisposition to bicuculline-induced seizures.
Topics: Animals; Autoradiography; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Female; Inferior Colliculi; Mice; Receptors, GABA-A; Seizures; Superior Colliculi | 1989 |
Bicuculline up-regulation of GABAA receptors in rat brain.
Topics: Animals; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Corpus Striatum; Flunitrazepam; Frontal Lobe; gamma-Aminobutyric Acid; Male; Muscimol; Octoxynol; Polyethylene Glycols; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra; Synaptic Membranes | 1988 |
[Effect of stress on the function of chloride channels associated with the GABA receptor complex].
Topics: Animals; Bicuculline; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cerebral Cortex; Chloride Channels; Chlorides; Male; Membrane Proteins; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological | 1988 |
Altered gamma-aminobutyric acid/benzodiazepine interaction after chronic diazepam exposure.
Topics: Animals; Benzodiazepines; Bicuculline; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Diazepam; gamma-Aminobutyric Acid; Ionophores; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Time Factors | 1988 |
Actions of avermectin B1a on the gamma-aminobutyric acidA receptor and chloride channels in rat brain.
Topics: Animals; Bicuculline; Binding, Competitive; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; Dose-Response Relationship, Drug; Flunitrazepam; Ivermectin; Kinetics; Male; Membrane Proteins; Muscimol; Rats; Receptors, GABA-A | 1986 |
Effect of benzodiazepine binding site ligands on [35S] t-butylbicyclophosphorothionate ([35S]TBPS) binding to rat brain: an autoradiographic study.
Topics: Animals; Autoradiography; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Clonazepam; Convulsants; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sulfur Radioisotopes | 1986 |
Phenylquinolines PK 8165 and PK 9084 allosterically modulate [35S]t-butylbicyclophosphorothionate binding to a chloride ionophore in rat brain via a novel Ro5 4864 binding site.
Topics: Animals; Anticonvulsants; Benzodiazepinones; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Convulsants; gamma-Aminobutyric Acid; Kinetics; Male; Quinolines; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1987 |
Cyclodiene insecticides inhibit GABAA receptor-regulated chloride transport.
Topics: Animals; Bicuculline; Biological Transport; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Insecticides; Male; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1987 |
Differences in GABA activity between ethanol withdrawal seizure prone and resistant mice.
Topics: Animals; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Ethanol; Female; Flunitrazepam; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred Strains; Pentylenetetrazole; Picrotoxin; Seizures; Substance Withdrawal Syndrome | 1988 |
Bicuculline-pentobarbital interactions on [35S]TBPS binding in various brain areas.
Topics: Animals; Bicuculline; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Dose-Response Relationship, Drug; Drug Interactions; Kinetics; Male; Mice; Mice, Inbred C57BL; Pentobarbital; Tissue Distribution | 1986 |
gamma-Aminobutyric acid- and benzodiazepine-induced modulation of [35S]-t-butylbicyclophosphorothionate binding to cerebellar granule cells.
Topics: Animals; Benzodiazepines; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Cerebellum; Diazepam; gamma-Aminobutyric Acid; Granulocytes; Muscimol; Picrotoxin; Rats; Sulfur Radioisotopes; Temperature | 1985 |
Differential interactions of GABA agonists, depressant and convulsant drugs with [35S]-t-butylbicyclophosphorothionate binding sites in cortex and cerebellum.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Central Nervous System Depressants; Cerebellum; Cerebral Cortex; Convulsants; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Male; Mitochondria; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Synaptic Transmission; Thiocyanates | 1984 |
Anxiolytic cyclopyrrolone drugs allosterically modulate the binding of [35S]t-butylbicyclophosphorothionate to the benzodiazepine/gamma-aminobutyric acid-A receptor/chloride anionophore complex.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Bicuculline; Binding, Competitive; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cell Membrane; Cerebral Cortex; Kinetics; Macromolecular Substances; Male; Naphthyridines; Piperazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sulfur Compounds; Tissue Distribution | 1984 |
Saturable binding of 35S-t-butylbicyclophosphorothionate to the sites linked to the GABA receptor and the interaction with GABAergic agents.
Topics: Animals; Bicuculline; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cerebral Cortex; gamma-Aminobutyric Acid; Male; Muscimol; Picrotoxin; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Sulfur Radioisotopes; Triazines | 1984 |
RO5-4864 inhibits the binding of [35S]t-butylbicyclophosphorothionate to rat brain membranes.
Topics: Androstanes; Animals; Azasteroids; Benzodiazepinones; Bicuculline; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Cell Membrane; Cerebellum; Cerebral Cortex; Dose-Response Relationship, Drug; Flumazenil; Hippocampus; Male; Picrotoxin; Radioligand Assay; Rats | 1984 |
GABA antagonists differentiate between recombinant GABAA/benzodiazepine receptor subtypes.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Embryo, Mammalian; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Kidney; Pyridazines; Rats; Receptors, GABA-A; Recombination, Genetic | 1995 |
GABAA receptor stimulation enhances NMDA-induced Ca2+ influx in mouse cerebral cortical neurons in primary culture.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Cerebral Cortex; Chloride Channels; Dizocilpine Maleate; Dose-Response Relationship, Drug; GABA Agonists; Isonicotinic Acids; Mice; Muscimol; N-Methylaspartate; Neurons; Picrotoxin; Potassium; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate | 1994 |
Allosteric modulation of [35S]TBPS-binding in the cerebral cortex of the rat during postnatal development.
Topics: Aging; Allosteric Regulation; Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Convulsants; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Stereoisomerism; Sulfur Radioisotopes | 1994 |
Cloning and functional expression of a Drosophila gamma-aminobutyric acid receptor.
Topics: Amino Acid Sequence; Animals; Base Sequence; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cloning, Molecular; Convulsants; DNA Primers; DNA, Complementary; Drosophila melanogaster; Female; Flunitrazepam; gamma-Aminobutyric Acid; Gene Expression; Macromolecular Substances; Molecular Sequence Data; Muscimol; Oocytes; Pentobarbital; Picrotoxin; Polymerase Chain Reaction; Receptors, GABA; Receptors, GABA-A; Transcription, Genetic; Xenopus laevis | 1994 |
Effects of propofol, pentobarbital and alphaxalone on t-[35S]butylbicyclophosphorothionate binding in rat cerebral cortex.
Topics: Anesthetics; Animals; Bicuculline; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Diazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Ion Channel Gating; Male; Membranes; Pentobarbital; Pregnanediones; Propofol; Rats; Rats, Sprague-Dawley; Sulfur Radioisotopes | 1994 |
Modulation of 35S-TBPS binding by GABAergic drugs in the cerebral cortex of newborn and adult rats.
Topics: Aging; Animals; Animals, Newborn; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cell Membrane; Cerebral Cortex; Convulsants; Diazepam; gamma-Aminobutyric Acid; Kinetics; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sulfur Radioisotopes | 1993 |
Interconvertible kinetic states of t-butylbicycloorthobenzoate binding sites of the gamma-aminobutyric acidA ionophores.
Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Bicuculline; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Fractionation; Cell Membrane; Cerebral Cortex; Convulsants; gamma-Aminobutyric Acid; Intracellular Membranes; Kinetics; Ligands; Male; Prosencephalon; Rats; Rats, Wistar; Receptors, GABA-A; Sulfur Radioisotopes; Synaptosomes; Tritium | 1993 |
Bicuculline-produced regional differences in the modulation of 35S-TBPS binding by GABA, pentobarbital and diazepam in mouse cerebellum and cortex.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Cerebral Cortex; Diazepam; Dose-Response Relationship, Drug; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Phenobarbital; Receptors, GABA-A | 1993 |
The influence of estrus cycle on neurosteroid potency at the gamma-aminobutyric acidA receptor complex.
Topics: Animals; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Desoxycorticosterone; Estrus; Female; gamma-Aminobutyric Acid; Male; Pregnanolone; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sex Factors | 1993 |
Modulation of GABAA receptor tert-[35S]butylbicyclophosphorothionate binding by antagonists: relationship to patterns of subunit expression.
Topics: Animals; Autoradiography; Bicuculline; Brain; Bridged Bicyclo Compounds, Heterocyclic; GABA Antagonists; Male; Membranes; Pyridazines; Rats; Rats, Wistar; Receptors, GABA; Sulfur Radioisotopes | 1996 |
Taurine allosterically inhibits binding of [35S]-t-butylbicyclophosphorothionate (TBPS) to rat brain synaptic membranes.
Topics: Allosteric Regulation; Animals; Bicuculline; Binding Sites; Brain Stem; Bridged Bicyclo Compounds, Heterocyclic; Clonazepam; Convulsants; gamma-Aminobutyric Acid; Male; Pentobarbital; Rats; Rats, Sprague-Dawley; Sulfur Radioisotopes; Synaptic Membranes; Taurine | 1995 |
Direct activation of GABAA receptors by loreclezole, an anticonvulsant drug with selectivity for the beta-subunit.
Topics: Animals; Anticonvulsants; Bicuculline; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Cerebral Cortex; Chloride Channels; Convulsants; Diazepam; DNA, Complementary; Female; gamma-Aminobutyric Acid; Humans; Kinetics; Macromolecular Substances; Male; Membrane Potentials; Oocytes; Picrotoxin; Propofol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Recombinant Proteins; Triazoles; Xenopus laevis | 1996 |
Pharmacology of skeletal muscle GABA-gated chloride channels in the cockroach Periplaneta americana.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Flunitrazepam; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Ion Channel Gating; Isonicotinic Acids; Male; Motor Neurons; Muscle, Skeletal; Periplaneta; Picrotoxin; Receptors, GABA; Sesterterpenes | 1997 |
Prenatal exposure to neurotoxicants dieldrin or lindane alters tert-butylbicyclophosphorothionate binding to GABA(A) receptors in fetal rat brainstem.
Topics: Animals; Bicuculline; Brain Stem; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Dieldrin; Female; GABA Antagonists; Gestational Age; Hexachlorocyclohexane; Maternal-Fetal Exchange; Nerve Tissue Proteins; Neurotoxins; Pregnancy; Prenatal Exposure Delayed Effects; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A | 1998 |
Biphasic modulation of GABA(A) receptor binding by steroids suggests functional correlates.
Topics: Androstanes; Anesthetics; Animals; Azasteroids; Baculoviridae; Bicuculline; Brain; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Cell Membrane; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression; Pregnanediones; Rats; Receptors, GABA-A; Recombinant Proteins; Spodoptera; Steroids; Sulfur Radioisotopes | 1999 |
Furosemide action on cerebellar GABA(A) receptors in alcohol-sensitive ANT rats.
Topics: Alcoholism; Animals; Azides; Benzodiazepines; Bicuculline; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cerebellum; Drug Combinations; Female; Furosemide; GABA Agonists; GABA Antagonists; Ligands; Male; Pyridazines; Rats; Receptors, GABA-A; Sodium Chloride | 1999 |
Modulation by bicuculline and penicillin of the block by t-butyl-bicyclo-phosphorothionate (TBPS) of GABA(A)-receptor mediated Cl(-)-current responses in rat striatal neurones.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Chloride Channels; Electrophysiology; GABA Antagonists; gamma-Aminobutyric Acid; Kinetics; Neostriatum; Neurons; Patch-Clamp Techniques; Penicillins; Rats; Receptors, GABA-A | 2000 |
Modulation of GABAergic synaptic transmission by the non-benzodiazepine anxiolytic etifoxine.
Topics: Animals; Behavior, Animal; Bicuculline; Binding, Competitive; Brain; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Dose-Response Relationship, Drug; Drinking Behavior; Flumazenil; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hypothalamus; Isoquinolines; Male; Membrane Potentials; Membranes; Neurons; Oxazines; Patch-Clamp Techniques; Posterior Horn Cells; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, GABA-A; Sulfur Radioisotopes; Synaptic Transmission; Tetrodotoxin; Tranquilizing Agents | 2000 |
Functional modulation of gamma-aminobutyric acid(A) receptors by etifoxine and allopregnanolone in rodents.
Topics: Allosteric Site; Animals; Anticonvulsants; Bicuculline; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Convulsants; Drug Interactions; GABA Antagonists; Male; Oxazines; Pregnanolone; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sulfur Radioisotopes | 2001 |
Modulation Of [35S]-tert-butylbicyclophosphorothionate binding by somatostatin in rat hypothalamus.
Topics: Animals; Bicuculline; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Dose-Response Relationship, Drug; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hypothalamus; Male; Muscimol; Pregnanolone; Rats; Rats, Wistar; Receptors, GABA-A; Somatostatin; Sulfur Radioisotopes | 2002 |
Role of GABAergic antagonism in the neuroprotective effects of bilobalide.
Topics: Animals; Area Under Curve; Bicuculline; Brain Edema; Bridged Bicyclo Compounds, Heterocyclic; Choline; Cyclopentanes; Drug Interactions; Excitatory Amino Acid Agonists; Furans; GABA Antagonists; gamma-Aminobutyric Acid; Ginkgolides; Hippocampus; In Vitro Techniques; Male; N-Methylaspartate; Neuroprotective Agents; Nonlinear Dynamics; Picrotoxin; Rats; Rats, Sprague-Dawley; Synaptosomes | 2007 |
Influences on blockade by t-butylbicyclo-phosphoro-thionate of GABA(A) receptor spontaneous gating, agonist activation and desensitization.
Topics: Bicuculline; Binding Sites; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glycine; HEK293 Cells; Humans; Ion Channel Gating; Mutation; Patch-Clamp Techniques; Picrotoxin; Receptors, GABA-A; Receptors, Serotonin, 5-HT3 | 2012 |