Page last updated: 2024-08-16

terfenadine and triprolidine

terfenadine has been researched along with triprolidine in 30 studies

Research

Studies (30)

TimeframeStudies, this research(%)All Research%
pre-199013 (43.33)18.7374
1990's10 (33.33)18.2507
2000's4 (13.33)29.6817
2010's3 (10.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Carrupt, PA; Jolliet, P; Morin, C; Morin, D; Pagliara, A; Rihoux, JP; Testa, B; Tillement, JP; Urien, S1
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Bellman, K; Knegtel, RM; Settimo, L1
Calthrop, JG; Doherty, V; Gibson, JR; Harvey, SG; Kennedy, CT; Sylvester, DG1
Barber, C; Birmingham, AT; Marsden, CA; Swire, FM1
Blog, FB; den Boer, MS; Gibson, JR; Harvey, SG; Jansen, FC; Kuneman, JJ; Starink, TM; van Joost, T; Westerhof, W1
Adams, J; Posner, J; Rolan, PE1
Bruttman, G; Charpin, J; Gervais, P; Grilliat, JP; Michel, FB; Pedrali, P1
Boyle, J; Gibson, JR; Marks, P1
Fleisch, JH; Haisch, KD; Rinkema, LE; Whitesitt, CA1
Cohen, AF; Hamilton, MJ; Peck, AW1
Nicholson, AN; Stone, BM3
Betts, T; Debenham, S; Markman, D; McKevitt, T; Mortiboy, D1
Cohen, AF; Posner, J1
Lang, DG; Wang, CM; Wenger, TL1
O'Hanlon, JF; Ramaekers, JG2
Dunmore, C; Hindmarch, I; Kerr, JS1
Colin, JN; Dry, J; Gillotin, C; Leynadier, F; Murrieta, M; Steru, D1
Dowd, PM; Goldsmith, P1
Edwards, IR; Lindquist, M1
de Abajo, FJ; Rodríguez, LA1
Mattila, MJ; Paakkari, I1
Dunn, N; Mann, RD; Pearce, GL; Shakir, S1
Díaz-Trelles, R; Fernández-Sánchez, MT; Marini, A; Novelli, A; Vega, JA1
Paakkari, I1

Reviews

3 review(s) available for terfenadine and triprolidine

ArticleYear
The new H1 antihistamines. Treatment of urticaria and other clinical problems.
    Dermatologic clinics, 1993, Volume: 11, Issue:1

    Topics: Astemizole; Cetirizine; Dermatitis, Atopic; Histamine H1 Antagonists; Humans; Loratadine; Terfenadine; Triprolidine; Urticaria

1993
Variations among non-sedating antihistamines: are there real differences?
    European journal of clinical pharmacology, 1999, Volume: 55, Issue:2

    Topics: Astemizole; Benzimidazoles; Butyrophenones; Central Nervous System; Cetirizine; Drug Interactions; Heart; Histamine H1 Antagonists; Humans; Hypnotics and Sedatives; Loratadine; Piperidines; Potassium Channel Blockers; Terfenadine; Triprolidine

1999
Cardiotoxicity of new antihistamines and cisapride.
    Toxicology letters, 2002, Feb-28, Volume: 127, Issue:1-3

    Topics: Arrhythmias, Cardiac; Astemizole; Benzimidazoles; Butyrophenones; Cetirizine; Cisapride; Heart Diseases; Histamine H1 Antagonists; Humans; Loratadine; Piperidines; Serotonin Receptor Agonists; Terfenadine; Triprolidine

2002

Trials

13 trial(s) available for terfenadine and triprolidine

ArticleYear
Treatment of itching in atopic eczema with antihistamines with a low sedative profile.
    BMJ (Clinical research ed.), 1989, Jan-14, Volume: 298, Issue:6666

    Topics: Adolescent; Adult; Benzhydryl Compounds; Clinical Trials as Topic; Dermatitis, Atopic; Female; Histamine H1 Antagonists; Humans; Male; Middle Aged; Pruritus; Pyridines; Random Allocation; Terfenadine; Triprolidine

1989
Effects of a sedative and of a non-sedative H1-antihistamine on the event-related potential (ERP) in normal volunteers.
    Psychopharmacology, 1989, Volume: 98, Issue:3

    Topics: Adult; Benzhydryl Compounds; Evoked Potentials; Flicker Fusion; Histamine H1 Antagonists; Humans; Hypnotics and Sedatives; Male; Memory, Short-Term; Psychomotor Performance; Terfenadine; Triprolidine

1989
A comparison of acrivastine versus terfenadine and placebo in the treatment of chronic idiopathic urticaria.
    The Journal of international medical research, 1989, Volume: 17 Suppl 2

    Topics: Adult; Benzhydryl Compounds; Chronic Disease; Clinical Trials as Topic; Double-Blind Method; Female; Histamine H1 Antagonists; Humans; Male; Placebos; Pyridines; Terfenadine; Triprolidine; Urticaria

1989
Comparison of the onset of H1-antagonism with acrivastine and terfenadine by histamine bronchial challenge in volunteers.
    The Journal of international medical research, 1989, Volume: 17 Suppl 2

    Topics: Adult; Aerosols; Benzhydryl Compounds; Female; Forced Expiratory Volume; Histamine; Histamine H1 Antagonists; Humans; Lung; Male; Pyridines; Receptors, Histamine H1; Terfenadine; Triprolidine; Vital Capacity

1989
French multicentre double-blind study to evaluate the efficacy and safety of acrivastine as compared with terfenadine in seasonal allergic rhinitis.
    The Journal of international medical research, 1989, Volume: 17 Suppl 2

    Topics: Adult; Benzhydryl Compounds; Clinical Trials as Topic; Double-Blind Method; Female; France; Histamine H1 Antagonists; Humans; Male; Multicenter Studies as Topic; Pyridines; Random Allocation; Rhinitis, Allergic, Seasonal; Terfenadine; Triprolidine

1989
Acrivastine versus terfenadine in the treatment of symptomatic dermographism--a double-blind, placebo-controlled study.
    The Journal of international medical research, 1989, Volume: 17 Suppl 2

    Topics: Adult; Benzhydryl Compounds; Clinical Trials as Topic; Double-Blind Method; Female; Histamine H1 Antagonists; Humans; Male; Pyridines; Random Allocation; Terfenadine; Triprolidine; Urticaria

1989
The effects of acrivastine (BW825C), diphenhydramine and terfenadine in combination with alcohol on human CNS performance.
    European journal of clinical pharmacology, 1987, Volume: 32, Issue:3

    Topics: Adolescent; Adult; Benzhydryl Compounds; Brain; Diphenhydramine; Double-Blind Method; Drug Synergism; Ethanol; Eye Movements; Female; Histamine H1 Antagonists; Humans; Male; Middle Aged; Psychomotor Performance; Pyridines; Reaction Time; Terfenadine; Triprolidine

1987
Performance studies with the H1-histamine receptor antagonists, astemizole and terfenadine.
    British journal of clinical pharmacology, 1982, Volume: 13, Issue:2

    Topics: Adult; Astemizole; Benzhydryl Compounds; Benzimidazoles; Cognition; Emotions; Female; Histamine H1 Antagonists; Humans; Mental Processes; Motor Skills; Piperidines; Terfenadine; Time Factors; Triprolidine

1982
Effects of two antihistamine drugs on actual driving performance.
    British medical journal (Clinical research ed.), 1984, Jan-28, Volume: 288, Issue:6413

    Topics: Arousal; Automobile Driving; Benzhydryl Compounds; Clinical Trials as Topic; Double-Blind Method; Emotions; Female; Histamine H1 Antagonists; Humans; Pyridines; Terfenadine; Triprolidine

1984
Antihistamine effects on actual driving performance in a standard test: a summary of Dutch experience, 1989-94.
    Allergy, 1995, Volume: 50, Issue:3

    Topics: Automobile Driving; Benzimidazoles; Butyrophenones; Cetirizine; Clemastine; Diphenhydramine; Dose-Response Relationship, Drug; Histamine H1 Antagonists; Humans; Loratadine; Netherlands; Piperidines; Psychomotor Performance; Terfenadine; Triprolidine

1995
Acrivastine, terfenadine and diphenhydramine effects on driving performance as a function of dose and time after dosing.
    European journal of clinical pharmacology, 1994, Volume: 47, Issue:3

    Topics: Administration, Oral; Adult; Automobile Driving; Cross-Over Studies; Diphenhydramine; Dose-Response Relationship, Drug; Drug Interactions; Drug Therapy, Combination; Ephedrine; Female; Humans; Infant, Newborn; Middle Aged; Single-Blind Method; Terfenadine; Triprolidine

1994
The psychomotor and cognitive effects of a new antihistamine, mizolastine, compared to terfenadine, triprolidine and placebo in healthy volunteers.
    European journal of clinical pharmacology, 1994, Volume: 47, Issue:4

    Topics: Adolescent; Adult; Benzimidazoles; Cognition; Histamine H1 Antagonists; Humans; Male; Memory; Placebos; Psychomotor Performance; Terfenadine; Triprolidine

1994
Effects of acrivastine and terfenadine on skin reactivity to histamine.
    Annals of allergy, 1994, Volume: 72, Issue:6

    Topics: Drug Hypersensitivity; Histamine; Histamine H1 Antagonists; Humans; Pruritus; Skin; Skin Tests; Terfenadine; Triprolidine

1994

Other Studies

14 other study(ies) available for terfenadine and triprolidine

ArticleYear
Molecular properties and pharmacokinetic behavior of cetirizine, a zwitterionic H1-receptor antagonist.
    Journal of medicinal chemistry, 1998, Mar-12, Volume: 41, Issue:6

    Topics: Alkanes; Animals; Biological Transport; Blood Proteins; Brain; Cetirizine; Histamine H1 Antagonists; Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydroxyzine; Isomerism; Models, Molecular; Molecular Conformation; Octanols; Rats; Water

1998
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
    Journal of medicinal chemistry, 2008, Jan-24, Volume: 51, Issue:2

    Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase

2008
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Comparison of the accuracy of experimental and predicted pKa values of basic and acidic compounds.
    Pharmaceutical research, 2014, Volume: 31, Issue:4

    Topics: Chemistry, Pharmaceutical; Forecasting; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Random Allocation

2014
Pharmacologic analysis of LY188695 (KB-2413), 1-(2-ethoxyethyl)-2-(4-methyl-1-homopiperazinyl)-benzimidazole difumarate, a potent histamine1 receptor antagonist.
    Agents and actions, 1987, Volume: 20, Issue:1-2

    Topics: Animals; Benzhydryl Compounds; Benzimidazoles; Bronchial Provocation Tests; Chlorpheniramine; Diphenhydramine; Guinea Pigs; Histamine H1 Antagonists; Lung; Male; Muscle, Smooth; Promethazine; Pyrilamine; Terfenadine; Triprolidine

1987
Antihistamines: impaired performance and the tendency to sleep.
    European journal of clinical pharmacology, 1986, Volume: 30, Issue:1

    Topics: Adult; Benzhydryl Compounds; Diazepam; Female; Flicker Fusion; Histamine Antagonists; Humans; Psychomotor Performance; Sleep; Terfenadine; Theophylline; Triprolidine; Visual Acuity

1986
Effects of two antihistamine drugs on actual driving performance.
    British medical journal (Clinical research ed.), 1984, Mar-24, Volume: 288, Issue:6421

    Topics: Automobile Driving; Benzhydryl Compounds; Female; Histamine H1 Antagonists; Humans; Pyridines; Terfenadine; Triprolidine

1984
The H1-antagonist mequitazine: studies on performance and visual function.
    European journal of clinical pharmacology, 1983, Volume: 25, Issue:4

    Topics: Adult; Benzhydryl Compounds; Double-Blind Method; Female; Flicker Fusion; Humans; Phenothiazines; Psychomotor Performance; Terfenadine; Triprolidine; Visual Acuity

1983
Terfenadine alters action potentials in isolated canine Purkinje fibers more than acrivastine.
    Journal of cardiovascular pharmacology, 1993, Volume: 22, Issue:3

    Topics: Action Potentials; Animals; Dogs; Dose-Response Relationship, Drug; Female; Histamine H1 Antagonists; In Vitro Techniques; Male; Purkinje Fibers; Terfenadine; Triprolidine

1993
Risks of non-sedating antihistamines.
    Lancet (London, England), 1997, May-03, Volume: 349, Issue:9061

    Topics: Adverse Drug Reaction Reporting Systems; Astemizole; Cetirizine; Histamine H1 Antagonists; Humans; Loratadine; Terfenadine; Triprolidine

1997
Risk of ventricular arrhythmias associated with nonsedating antihistamine drugs.
    British journal of clinical pharmacology, 1999, Volume: 47, Issue:3

    Topics: Adolescent; Adult; Aged; Arrhythmias, Cardiac; Astemizole; Case-Control Studies; Cetirizine; Child; Child, Preschool; Cohort Studies; Cytochrome P-450 Enzyme Inhibitors; Enzyme Inhibitors; Female; Histamine H1 Antagonists; Humans; Infant; Infant, Newborn; Information Systems; Loratadine; Male; Middle Aged; Risk Factors; Tachycardia, Ventricular; Terfenadine; Triprolidine

1999
Sedation with "non-sedating" antihistamines: four prescription-event monitoring studies in general practice.
    BMJ (Clinical research ed.), 2000, Apr-29, Volume: 320, Issue:7243

    Topics: Adolescent; Adult; Adverse Drug Reaction Reporting Systems; Aged; Cetirizine; Child; Child, Preschool; Consciousness Disorders; Female; Histamine H1 Antagonists; Humans; Infant; Infant, Newborn; Loratadine; Male; Middle Aged; Product Surveillance, Postmarketing; Sleep Stages; Terfenadine; Triprolidine

2000
Antihistamine terfenadine potentiates NMDA receptor-mediated calcium influx, oxygen radical formation, and neuronal death.
    Brain research, 2000, Oct-13, Volume: 880, Issue:1-2

    Topics: Animals; Biological Transport; Calcium; Cell Death; Cell Survival; Cells, Cultured; Cerebellum; Chlorpheniramine; Cyclic GMP; Dizocilpine Maleate; Drug Synergism; Glutamic Acid; Histamine; Histamine H1 Antagonists; N-Methylaspartate; Neurons; Piperazines; Receptors, N-Methyl-D-Aspartate; Signal Transduction; Terfenadine; Triprolidine

2000