Page last updated: 2024-08-16

terfenadine and cimetidine

terfenadine has been researched along with cimetidine in 38 studies

Research

Studies (38)

TimeframeStudies, this research(%)All Research%
pre-19905 (13.16)18.7374
1990's12 (31.58)18.2507
2000's11 (28.95)29.6817
2010's10 (26.32)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Huang, L; Humphreys, JE; Morgan, JB; Polli, JW; Serabjit-Singh, CS; Webster, LO; Wring, SA1
Fischer, H; Huwyler, J; Poli, S; Schwab, D; Tabatabaei, A1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Artursson, P; Bergström, CA; Hoogstraate, J; Matsson, P; Norinder, U; Pedersen, JM1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Fisk, L; Greene, N; Naven, RT; Note, RR; Patel, ML; Pelletier, DJ1
Ekins, S; Williams, AJ; Xu, JJ1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Gilmour, JW; Norval, M; Simpson, TJ1
Nicholson, AN1
Anderson, J; Eiser, NM; Mills, JG1
Duc, J; Pécoud, A1
Araujo, OE; Flowers, FP; Nieves, CH1
Obel, AO1
Barak, V; Fabian, I; Geller-Bernstein, C; Handzel, ZT; Mor, S; Nagler, A1
Bódis, J; Hanf, V; Papenfuss, F; Schwarz, H; Tinneberg, HR; Török, A1
Cantilena, LR; Conner, DP; Honig, PK; Mullin, JC; Wortham, DC; Zamani, K1
Kozlowski, VA; Mattos Filho, TR1
Archer, CB; Brooks, J; Burton, JL; Sansom, JE1
Vere, DW1
Bende, M; Juliusson, S1
Chan, TY; Chan, WK; Ng, PW1
Guengerich, FP1
Pasco, J1
Del Prete, E; Rossi, R; Scharrer, E1
Irman-Florjanc, T1
Sugawara, K; Tateishi, T; Uno, T; Yasui-Furukori, N1
Fu, YL; He, SH; Xie, H1
Andoh, T; Kamimura, K; Kawai, S; Kuraishi, Y; Nakano, T; Nojima, H; Ohtsuka, E1
Horita, S; Inoue, K; Kondo, T; Kusuhara, H; Maeda, K; Matsushima, S; Nakayama, H; Ohta, KY; Sugiyama, Y; Yuasa, H1
Behrens, CJ; Caliskan, G; Fano, S; Heinemann, U1
Fox, EM; Hübner, MP; Mitre, E; Morris, CP1

Reviews

2 review(s) available for terfenadine and cimetidine

ArticleYear
Antihistamines.
    International journal of dermatology, 1986, Volume: 25, Issue:4

    Topics: Animals; Astemizole; Benzhydryl Compounds; Benzimidazoles; Child; Child, Preschool; Cimetidine; Drug Synergism; Guanidines; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Imidazoles; Infant; Infant, Newborn; Kinetics; Pyrimidinones; Ranitidine; Terfenadine

1986
Role of cytochrome P450 enzymes in drug-drug interactions.
    Advances in pharmacology (San Diego, Calif.), 1997, Volume: 43

    Topics: Animals; Beverages; Binding Sites; Cimetidine; Citrus; Cytochrome P-450 CYP2D6; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Drug Interactions; Ethinyl Estradiol; Food-Drug Interactions; Humans; Mixed Function Oxygenases; Pharmaceutical Preparations; Terfenadine

1997

Trials

5 trial(s) available for terfenadine and cimetidine

ArticleYear
Effect of H1- and H2-receptor antagonists on sputum volume and lung function in patients with generalized bronchiectasis.
    British journal of diseases of the chest, 1985, Volume: 79, Issue:3

    Topics: Adult; Aged; Benzhydryl Compounds; Bronchiectasis; Cimetidine; Clinical Trials as Topic; Double-Blind Method; Female; Histamine H1 Antagonists; Humans; Lung; Male; Middle Aged; Sputum; Terfenadine

1985
Effects of H1- and H2-antihistamines on platelet-activating factor and bradykinin-induced inflammatory responses in human skin.
    Clinical and experimental dermatology, 1996, Volume: 21, Issue:1

    Topics: Administration, Oral; Bradykinin; Cimetidine; Codeine; Double-Blind Method; Doxepin; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Platelet Activating Factor; Skin; Terfenadine; Urticaria

1996
Actions of terfenadine and cimetidine on histamine wheal formation.
    British journal of clinical pharmacology, 1995, Volume: 40, Issue:6

    Topics: Adult; Cimetidine; Drug Combinations; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Male; Middle Aged; Terfenadine; Urticaria

1995
Effect of systemically administered H1- and H2-receptor antagonists on nasal blood flow as measured with laser Doppler flowmetry in a provoked allergic reaction.
    Rhinology, 1996, Volume: 34, Issue:1

    Topics: Adult; Allergens; Cimetidine; Cross-Over Studies; Double-Blind Method; Female; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Laser-Doppler Flowmetry; Male; Microcirculation; Nasal Mucosa; Nasal Provocation Tests; Pollen; Premedication; Rhinitis, Allergic, Seasonal; Terfenadine

1996
Different effects of three transporting inhibitors, verapamil, cimetidine, and probenecid, on fexofenadine pharmacokinetics.
    Clinical pharmacology and therapeutics, 2005, Volume: 77, Issue:1

    Topics: Adult; Area Under Curve; Biological Availability; Calcium Channel Blockers; Cimetidine; Drug Interactions; Half-Life; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Male; Probenecid; Terfenadine; Uricosuric Agents; Verapamil

2005

Other Studies

31 other study(ies) available for terfenadine and cimetidine

ArticleYear
Rational use of in vitro P-glycoprotein assays in drug discovery.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 299, Issue:2

    Topics: Adenosine Triphosphatases; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cells, Cultured; Chromatography, Liquid; Enzyme Inhibitors; Fluoresceins; Fluorescent Dyes; Humans; Mass Spectrometry; Pharmacology; Spodoptera

2001
Comparison of in vitro P-glycoprotein screening assays: recommendations for their use in drug discovery.
    Journal of medicinal chemistry, 2003, Apr-24, Volume: 46, Issue:9

    Topics: Adenosine Triphosphatases; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cells, Cultured; Drug Evaluation, Preclinical; Fluoresceins; Fluorescent Dyes; Humans; Indicators and Reagents; Mice; Models, Molecular; Rhodamines; Species Specificity; Swine

2003
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).
    Journal of medicinal chemistry, 2008, Jun-12, Volume: 51, Issue:11

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Antipsychotic Agents; Antiviral Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Cell Line; Computer Simulation; Cytochrome P-450 Enzyme System; Drug-Related Side Effects and Adverse Reactions; Estradiol; Humans; Insecta; Liver; Models, Molecular; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pharmaceutical Preparations; Pharmacology; Structure-Activity Relationship

2008
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Developing structure-activity relationships for the prediction of hepatotoxicity.
    Chemical research in toxicology, 2010, Jul-19, Volume: 23, Issue:7

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Humans; Structure-Activity Relationship; Tetracyclines; Thiophenes

2010
A predictive ligand-based Bayesian model for human drug-induced liver injury.
    Drug metabolism and disposition: the biological fate of chemicals, 2010, Volume: 38, Issue:12

    Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands

2010
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
The effect of histamine receptor antagonists on immunosuppression induced by the cis-isomer of urocanic acid.
    Photodermatology, photoimmunology & photomedicine, 1990, Volume: 7, Issue:6

    Topics: Adenosine Triphosphatases; Animals; Benzhydryl Compounds; Cell Count; Cimetidine; Female; Herpes Simplex; Histamine H1 Antagonists; Hypersensitivity, Delayed; Mice; Skin; Terfenadine; Urocanic Acid

1990
Central effects of H1 and H2 antihistamines.
    Aviation, space, and environmental medicine, 1985, Volume: 56, Issue:4

    Topics: Aerospace Medicine; Benzhydryl Compounds; Central Nervous System; Chlorpheniramine; Cimetidine; Clemastine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Phenothiazines; Promethazine; Psychomotor Performance; Ranitidine; Sleep Stages; Structure-Activity Relationship; Terfenadine; Visual Acuity; Visual Perception

1985
Successful treatment of idiopathic cold urticaria with the association of H1 and H2 antagonists: a case report.
    Annals of allergy, 1986, Volume: 56, Issue:4

    Topics: Adult; Benzhydryl Compounds; Cimetidine; Cold Temperature; Drug Therapy, Combination; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Male; Terfenadine; Urticaria

1986
Practical therapeutics: the use of histamine receptor antagonists in contemporary times.
    East African medical journal, 1984, Volume: 61, Issue:7

    Topics: Astemizole; Benzhydryl Compounds; Benzimidazoles; Child; Cimetidine; Conjunctivitis, Allergic; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Pyrilamine; Rhinitis, Allergic, Seasonal; Terfenadine

1984
Histamine enhances granulocyte-macrophage colony-stimulating factor and interleukin-6 production by human peripheral blood mononuclear cells.
    Journal of leukocyte biology, 1995, Volume: 58, Issue:4

    Topics: Antibodies; Cell Adhesion; Cells, Cultured; Cimetidine; Enzyme-Linked Immunosorbent Assay; Granulocyte-Macrophage Colony-Stimulating Factor; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Interleukin-3; Interleukin-6; Kinetics; Leukocytes, Mononuclear; Pyrilamine; Radioimmunoassay; Ranitidine; Stem Cells; Stimulation, Chemical; Terfenadine

1995
The effect of histamine on progesterone and estradiol secretion of human granulosa cells in serum-free culture.
    Gynecological endocrinology : the official journal of the International Society of Gynecological Endocrinology, 1993, Volume: 7, Issue:4

    Topics: Adult; Cells, Cultured; Cimetidine; Culture Media; Dose-Response Relationship, Drug; Estradiol; Female; Fertilization in Vitro; Follicular Fluid; Granulosa Cells; Histamine; Humans; Progesterone; Terfenadine

1993
Effect of concomitant administration of cimetidine and ranitidine on the pharmacokinetics and electrocardiographic effects of terfenadine.
    European journal of clinical pharmacology, 1993, Volume: 45, Issue:1

    Topics: Adolescent; Adult; Aged; Cimetidine; Drug Administration Schedule; Drug Interactions; Electrocardiography; Female; Humans; Male; Middle Aged; Prospective Studies; Ranitidine; Terfenadine

1993
Effect of H1 and H2 receptor antagonists on the serum activity of gamma-glutamyltransferase during liver regeneration after partial hepatectomy in rats.
    Pharmacology, 1995, Volume: 51, Issue:2

    Topics: Animals; Cimetidine; gamma-Glutamyltransferase; Hepatectomy; Histamine H1 Antagonists; Histamine H2 Antagonists; Liver Regeneration; Male; Rats; Rats, Wistar; Terfenadine

1995
Torsade de pointes during the concomitant use of terfenadine and cimetidine.
    Australian and New Zealand journal of medicine, 1996, Volume: 26, Issue:1

    Topics: Cimetidine; Drug Interactions; Electrocardiography; Enzyme Inhibitors; Female; Humans; Middle Aged; Terfenadine; Torsades de Pointes

1996
What has the patient been taking?
    Australian family physician, 1998, Volume: 27, Issue:6

    Topics: Aged; Anti-Bacterial Agents; Anti-Ulcer Agents; Chlorothiazide; Cimetidine; Diagnosis, Differential; Diuretics; Electrocardiography; Electrolytes; Erythromycin; Female; Histamine H1 Antagonists; Humans; Long QT Syndrome; Sodium Chloride Symporter Inhibitors; Terfenadine; Torsades de Pointes

1998
Effects of histamine H1 receptors on the feeding and drinking patterns in pygmy goats.
    Journal of dairy science, 1998, Volume: 81, Issue:9

    Topics: Animals; Brompheniramine; Cimetidine; Drinking; Eating; Female; Goats; Histamine H1 Antagonists; Histamine H2 Antagonists; Receptors, Histamine H1; Terfenadine

1998
Kinetics of injected histamine in cat plasma after antihistamine prophylaxis.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 2000, Volume: 49 Suppl 1

    Topics: Animals; Cats; Cimetidine; Ethylenediamines; Female; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Kinetics; Male; Terfenadine

2000
Inhibition of tryptase release from human colon mast cells by histamine receptor antagonists.
    Asian Pacific journal of allergy and immunology, 2005, Volume: 23, Issue:1

    Topics: Calcimycin; Cells, Cultured; Cimetidine; Colon; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Imidazoles; Ionophores; Mast Cells; Serine Endopeptidases; Serine Proteinase Inhibitors; Terfenadine; Thiourea; Tryptases

2005
Possible involvement of 5-lipoxygenase metabolite in itch-associated response of mosquito allergy in mice.
    Journal of pharmacological sciences, 2007, Volume: 105, Issue:1

    Topics: Animals; Arachidonate 5-Lipoxygenase; Betamethasone Valerate; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Chromones; Cimetidine; Culicidae; Dose-Response Relationship, Drug; Fatty Acids, Unsaturated; Hydrazines; Hydroxyurea; Hypersensitivity; Indoles; Indomethacin; Ketoprofen; Leukotriene B4; Lipoxygenase Inhibitors; Male; Mice; Mice, Inbred ICR; NG-Nitroarginine Methyl Ester; Phenylpropionates; Phospholipid Ethers; Propionates; Pruritus; Quinolines; Terfenadine

2007
The inhibition of human multidrug and toxin extrusion 1 is involved in the drug-drug interaction caused by cimetidine.
    Drug metabolism and disposition: the biological fate of chemicals, 2009, Volume: 37, Issue:3

    Topics: Cell Line; Cimetidine; Drug Interactions; Humans; Kidney; Organic Cation Transport Proteins; Probenecid; Terfenadine

2009
Histaminergic modulation of acetylcholine-induced γ oscillations in rat hippocampus.
    Neuroreport, 2011, Aug-03, Volume: 22, Issue:11

    Topics: Acetylcholine; Animals; Attention; Cholinesterase Inhibitors; Cimetidine; Dimaprit; Electroencephalography; Hippocampus; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine Release; Hypoxia, Brain; In Vitro Techniques; Male; Microelectrodes; Physostigmine; Pyramidal Tracts; Rats; Rats, Wistar; Terfenadine

2011
Histamine 1 Receptor Blockade Enhances Eosinophil-Mediated Clearance of Adult Filarial Worms.
    PLoS neglected tropical diseases, 2015, Volume: 9, Issue:7

    Topics: Animals; Cimetidine; Cytokines; Eosinophils; Female; Filariasis; Filarioidea; Gene Expression Regulation; Histamine H1 Antagonists; Histamine H2 Antagonists; Immunoglobulin E; Male; Mice; Mice, Inbred BALB C; Receptors, Histamine H1; Sex Ratio; Spleen; Terfenadine

2015