Page last updated: 2024-08-16

terbutaline and prazosin

terbutaline has been researched along with prazosin in 23 studies

Research

Studies (23)

TimeframeStudies, this research(%)All Research%
pre-19903 (13.04)18.7374
1990's5 (21.74)18.2507
2000's7 (30.43)29.6817
2010's8 (34.78)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Lombardo, F; Obach, RS; Waters, NJ1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Du-Cuny, L; Mash, EA; Meuillet, EJ; Moses, S; Powis, G; Song, Z; Zhang, S1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Campillo, NE; Guerra, A; Páez, JA1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Sugden, D1
Barnes, PJ; Gold, WM; Phillips, MJ1
Gustafsson, B; Olsson, OA1
Harris, WH; Moore, LA; Yamashiro, S1
Andersson, KE; Colstrup, H; Lose, G; Thind, P2
Bültmann, R; Driessen, B; Gonçalves, J; Starke, K1
Thind, P1
Gyires, K; Kató, E; Lipták, L; Mátyus, P; Rónai, AZ; Shujaa, N1
Segal, S; Wang, SY1
Djouma, E; Dooley, PC; Grills, BL; McDonald, AC; McDonald, SJ; Schuijers, JA; Ward, AR1

Reviews

2 review(s) available for terbutaline and prazosin

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
The significance of smooth and striated muscles in the sphincter function of the urethra in healthy women.
    Neurourology and urodynamics, 1995, Volume: 14, Issue:6

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adult; Autonomic Nervous System; Carbachol; Elasticity; Female; Humans; Muscle Contraction; Muscle, Skeletal; Muscle, Smooth; Nerve Block; Norepinephrine; Prazosin; Pressure; Reference Values; Terbutaline; Urethra; Urinary Bladder; Urinary Catheterization; Urination; Viscosity

1995

Other Studies

21 other study(ies) available for terbutaline and prazosin

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Computational modeling of novel inhibitors targeting the Akt pleckstrin homology domain.
    Bioorganic & medicinal chemistry, 2009, Oct-01, Volume: 17, Issue:19

    Topics: Antineoplastic Agents; Blood Proteins; Caco-2 Cells; Cell Membrane Permeability; Computer Simulation; Drug Discovery; Drug Screening Assays, Antitumor; Humans; Models, Molecular; Phosphoproteins; Protein Binding; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-akt; Quantitative Structure-Activity Relationship

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Beta-adrenergic regulation of cyclic GMP in rat pinealocytes.
    Biochemical and biophysical research communications, 1990, Mar-16, Volume: 167, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Cells, Cultured; Cyclic AMP; Cyclic GMP; Epinephrine; Isoproterenol; Kinetics; Norepinephrine; Pineal Gland; Prazosin; Rats; Rats, Inbred Strains; Terbutaline

1990
Characterization of purified dog mastocytoma cells. Autonomic membrane receptors and pharmacologic modulation of histamine release.
    The American review of respiratory disease, 1985, Volume: 132, Issue:5

    Topics: Acetylcholine; Animals; Cyclic AMP; Dihydroalprenolol; Dogs; Histamine Release; In Vitro Techniques; Isoproterenol; Mast-Cell Sarcoma; Phenylephrine; Prazosin; Propranolol; Quinuclidinyl Benzilate; Radioligand Assay; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Cholinergic; Terbutaline

1985
The effect of D2343 in transmurally stimulated rabbit isthmus muscle.
    Acta pharmacologica et toxicologica, 1985, Volume: 56, Issue:5

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Fallopian Tubes; Female; In Vitro Techniques; Muscle Contraction; Octopamine; Prazosin; Rabbits; Terbutaline

1985
The receptors responsible for heat production in brown adipose tissue in the young rabbit.
    Canadian journal of physiology and pharmacology, 1986, Volume: 64, Issue:2

    Topics: Adipose Tissue, Brown; Albuterol; Animals; Body Temperature Regulation; Hot Temperature; Isoproterenol; Norepinephrine; Phentolamine; Prazosin; Rabbits; Receptors, Adrenergic; Skin Temperature; Terbutaline

1986
The urethral resistance to rapid dilation: an analysis of the effect of autonomic receptor stimulation and blockade and of pudendal nerve blockade in healthy females.
    Scandinavian journal of urology and nephrology, 1995, Volume: 29, Issue:1

    Topics: Adult; Atropine; Autonomic Nervous System; Carbachol; Female; Humans; Middle Aged; Nerve Block; Norepinephrine; Prazosin; Propranolol; Terbutaline; Time Factors; Urethra

1995
The effect of pharmacological stimulation and blockade of autonomic receptors and of pudendal blockade on urethral stress relaxation in healthy women.
    British journal of urology, 1994, Volume: 74, Issue:1

    Topics: Adult; Atropine; Blood Pressure; Carbachol; Female; Heart Rate; Humans; Middle Aged; Muscle Relaxation; Nerve Block; Norepinephrine; Prazosin; Pressure; Propranolol; Stimulation, Chemical; Terbutaline; Urethra; Urinary Bladder

1994
Opposite modulation of noradrenaline and ATP release in guinea-pig vas deferens through prejunctional beta-adrenoceptors: evidence for the beta 2 subtype.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:5

    Topics: Adenosine Triphosphate; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Imidazoles; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Norepinephrine; Prazosin; Propanolamines; Receptors, Adrenergic, beta-2; Suramin; Terbutaline; Vas Deferens

1996
alpha2B-adrenoceptor agonist ST-91 antagonizes beta2-adrenoceptor-mediated relaxation in rat mesenteric artery rings.
    European journal of pharmacology, 2008, Feb-12, Volume: 580, Issue:3

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic beta-2 Receptor Antagonists; Analysis of Variance; Animals; Aorta; Clonidine; Dose-Response Relationship, Drug; In Vitro Techniques; Isoproterenol; Male; Mesenteric Arteries; Phenylephrine; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta-2; Terbutaline; Vas Deferens; Vasodilation; Xylazine; Yohimbine

2008
The effect of maternal catecholamines on the caliber of gravid uterine microvessels.
    Anesthesia and analgesia, 2008, Volume: 106, Issue:3

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Analgesia, Obstetrical; Animals; Arterioles; Catecholamines; Dose-Response Relationship, Drug; Epinephrine; Female; Gravidity; Norepinephrine; Prazosin; Pregnancy; Propranolol; Rats; Rats, Sprague-Dawley; Regional Blood Flow; Terbutaline; Uterus; Vasoconstriction; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents

2008
α(1) adrenergic receptor agonist, phenylephrine, actively contracts early rat rib fracture callus ex vivo.
    Journal of orthopaedic research : official publication of the Orthopaedic Research Society, 2011, Volume: 29, Issue:5

    Topics: Adrenergic alpha-1 Receptor Agonists; Animals; Biomechanical Phenomena; Bony Callus; Fracture Healing; Phenylephrine; Prazosin; Rats; Receptors, Adrenergic, beta-2; Rib Fractures; Terbutaline

2011