Page last updated: 2024-08-24

tenocyclidine and piperidines

tenocyclidine has been researched along with piperidines in 31 studies

Research

Studies (31)

TimeframeStudies, this research(%)All Research%
pre-19909 (29.03)18.7374
1990's15 (48.39)18.2507
2000's6 (19.35)29.6817
2010's1 (3.23)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lemaire, S; Rogers, C1
Britt, M; Paschetto, KA; Powel, RJ; Pullan, LM; Stumpo, RJ1
Ando, K; Kawamoto, I; Matsuda, Y; Sano, H; Toki, S; Yoshida, M1
Drian, MJ; Kamenka, JM; Pirat, JL; Privat, A1
de Costa, BR; Jacobson, AE; Mattson, MV; Monn, JA; Reid, AA; Rice, KC; Rothman, RB; Thurkauf, A1
Compton, RP; Hood, WF; Monahan, JB1
Carter, CJ; Lloyd, KG; Scatton, B; Zivkovic, B1
Boksa, P; Chaudieu, I; Mount, H; Quirion, R1
Lemaire, S; Rogers, CA1
Byrd, JC; Paleos, GA; Yang, ZW1
ffrench-Mullen, JM; Pieniek, M; Rogawski, MA; Suzuki, S1
Culp, SG; De Souza, EB; Wolfe, SA1
Aanonsen, LM; Seybold, VS1
Denavit-Saubié, M; Foutz, AS1
Bertin, J; Carter, C; Dupont, R; Duverger, D; Frost, J; Gaudilliere, B; Gotti, B; MacKenzie, ET; Rousseau, J; Scatton, B1
Arbilla, S; Benavides, J; Carter, C; Legendre, P; Lloyd, KG; MacKenzie, ET; Noel, F; Thuret, F; Vincent, JD; Zivkovic, B1
Gundlach, AL; Largent, BL; Snyder, SH2
Bobker, DH; Campbell, BG; Leslie, FM; Mefford, IN; Weber, E1
Hashimoto, A; Maeda, M; Nishikawa, T; Orita, K; Sasaki, S; Umezu, K; Yugami, T1
Jacobsen, P; Klockgether, T; Löschmann, PA; Turski, L1
Cordon, JJ; Coughenour, LL1
Baldet, P; Levallois, C; Privat, A; Valence, C1
Camarasa, J; Camins, A; Canudas, AM; Escubedo, E; Pallas, M; Pubill, D; Sureda, FX1
Hirbec, H; Kamenka, JM; Mausset, AL; Privat, A; Vignon, J1
Sun, W; Wessinger, WD1
Kopjar, N; Petek, MJ; Radić, B; Vrdoljak, AL; Zeljezić, D1
Bloomquist, JR; Geldenhuys, WJ; Malan, SF; Van der Schyf, CJ1
Berend, S; Kopjar, N; Mladinić, M; Petek, MJ; Radić, B; Vrdoljak, AL; Zeljezić, D1
Kristie, TM; Liang, Y; Narayanan, A; Peng, H; Vogel, JL1
Mrsić, G; Petek, MJ; Vrdoljak, AL1

Other Studies

31 other study(ies) available for tenocyclidine and piperidines

ArticleYear
Characterization of [3H]desmethylimipramine binding in bovine adrenal medulla: interactions with sigma- and (or) phencyclidine-receptor ligands.
    Canadian journal of physiology and pharmacology, 1992, Volume: 70, Issue:11

    Topics: Adrenal Medulla; Animals; Binding Sites; Cattle; Desipramine; Dextromethorphan; Dizocilpine Maleate; Phenazocine; Phencyclidine; Piperidines; Potassium Chloride; Receptors, Opioid, delta; Receptors, Phencyclidine; Tranquilizing Agents

1992
Neomycin is an agonist at a polyamine site on the N-methyl-D-aspartate receptor.
    Journal of neurochemistry, 1992, Volume: 59, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; Biguanides; Magnesium; Male; Neomycin; Phencyclidine; Piperazines; Piperidines; Polyamines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spermidine; Synaptic Membranes; Tritium

1992
ES-242-2, -3, -4, -5, -6, -7, and -8, novel bioxanthracenes produced by Verticillium sp., which act on the N-methyl-D-aspartate receptor.
    The Journal of antibiotics, 1992, Volume: 45, Issue:7

    Topics: Animals; Brain; In Vitro Techniques; Kainic Acid; Mitosporic Fungi; Phencyclidine; Piperidines; Pyrans; Rats; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship; Tritium

1992
Non-competitive antagonists of N-methyl-D-aspartate prevent spontaneous neuronal death in primary cultures of embryonic rat cortex.
    Journal of neuroscience research, 1991, Volume: 29, Issue:1

    Topics: Animals; Cell Survival; Cells, Cultured; Cerebral Cortex; Cyclohexanes; Cyclohexenes; Dizocilpine Maleate; Embryo, Mammalian; Female; N-Methylaspartate; Neurons; Phencyclidine; Piperidines; Pregnancy; Rats; Rats, Inbred Strains

1991
Specificity of phencyclidine-like drugs and benzomorphan opiates for two high affinity phencyclidine binding sites in guinea pig brain.
    Neuropharmacology, 1990, Volume: 29, Issue:9

    Topics: Analgesics; Animals; Benzomorphans; Brain; Dioxolanes; Dizocilpine Maleate; Guinea Pigs; In Vitro Techniques; Kinetics; Ligands; Narcotics; Phencyclidine; Piperidines; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Phencyclidine; Structure-Activity Relationship

1990
N-methyl-D-aspartate recognition site ligands modulate activity at the coupled glycine recognition site.
    Journal of neurochemistry, 1990, Volume: 54, Issue:3

    Topics: Animals; Aspartic Acid; Binding Sites; Binding, Competitive; Glutamates; Glutamic Acid; Glycine; Ligands; N-Methylaspartate; Phencyclidine; Pipecolic Acids; Piperidines

1990
Ifenprodil and SL 82.0715 as cerebral antiischemic agents. III. Evidence for antagonistic effects at the polyamine modulatory site within the N-methyl-D-aspartate receptor complex.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Aspartic Acid; Binding Sites; Binding, Competitive; Brain; Cells, Cultured; Drug Interactions; Female; Glycine; Male; N-Methylaspartate; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Spermidine; Spermine; Spinal Cord

1990
Phencyclidine and related compounds evoked [3H]dopamine release from rat mesencephalic cell cultures by a mechanism independent of the phencyclidine receptor, sigma binding site, or dopamine uptake site.
    Canadian journal of physiology and pharmacology, 1990, Volume: 68, Issue:9

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anticonvulsants; Binding Sites; Cells, Cultured; Dioxolanes; Dizocilpine Maleate; Dopamine; Dose-Response Relationship, Drug; Guanidines; Mesencephalon; N-Methylaspartate; Neurotransmitter Uptake Inhibitors; Phencyclidine; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Phencyclidine; Sigma Factor; Tritium

1990
Characterization of (+)-[3H]3-PPP and [3H]TCP binding sites in membrane preparations of bovine adrenal medulla.
    Progress in clinical and biological research, 1990, Volume: 328

    Topics: Adrenal Medulla; Animals; Binding Sites; Binding, Competitive; Cattle; In Vitro Techniques; Membranes; Phencyclidine; Piperidines; Receptors, Opioid; Receptors, sigma

1990
Ontogeny of PCP and sigma receptors in rat brain.
    Brain research. Developmental brain research, 1990, Feb-01, Volume: 51, Issue:2

    Topics: Aging; Animals; Brain; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma

1990
Phencyclidine selectively blocks the sustained voltage-dependent potassium conductance in PC12 cells.
    Brain research, 1988, Jul-19, Volume: 456, Issue:1

    Topics: Anesthetics; Animals; Dioxolanes; Electric Stimulation; Ion Channels; Membrane Potentials; Phencyclidine; Pheochromocytoma; Piperidines; Potassium; Rats; Tumor Cells, Cultured

1988
Sigma-receptors in endocrine organs: identification, characterization, and autoradiographic localization in rat pituitary, adrenal, testis, and ovary.
    Endocrinology, 1989, Volume: 124, Issue:3

    Topics: Adrenal Glands; Animals; Autoradiography; Brain Chemistry; Cell Membrane; Dibenzocycloheptenes; Dizocilpine Maleate; Female; Haloperidol; Hypophysectomy; Male; Ovary; Phencyclidine; Piperidines; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, sigma; Testis; Tissue Distribution

1989
Phencyclidine and sigma receptors in rat spinal cord: binding characterization and quantitative autoradiography.
    Synapse (New York, N.Y.), 1989, Volume: 4, Issue:1

    Topics: Animals; Autoradiography; Binding, Competitive; Ganglia, Spinal; Male; Narcotic Antagonists; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Spinal Cord

1989
Differentiation of phencyclidine and sigma receptor types affecting the central inspiratory termination mechanism in cat.
    Life sciences, 1989, Volume: 45, Issue:14

    Topics: Animals; Brain Stem; Cats; Decerebrate State; Dextrorphan; Dibenzocycloheptenes; Dizocilpine Maleate; Guanidines; Phencyclidine; Phrenic Nerve; Piperidines; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Respiration

1989
Ifenprodil and SL 82.0715 as cerebral anti-ischemic agents. I. Evidence for efficacy in models of focal cerebral ischemia.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 247, Issue:3

    Topics: Animals; Aspartic Acid; Brain Ischemia; Cats; Female; Male; Models, Cardiovascular; N-Methylaspartate; Phencyclidine; Piperidines; Rats; Rats, Inbred F344; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Vasoconstriction

1988
Ifenprodil and SL 82.0715 as cerebral anti-ischemic agents. II. Evidence for N-methyl-D-aspartate receptor antagonist properties.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 247, Issue:3

    Topics: Animals; Aspartic Acid; Brain Ischemia; Cells, Cultured; Cerebellum; Corpus Striatum; Cyclic GMP; Dopamine; Harmaline; In Vitro Techniques; Mice; N-Methylaspartate; Phencyclidine; Piperazines; Piperidines; Rats; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Spinal Cord

1988
Phencyclidine and sigma opiate receptors in brain: biochemical and autoradiographical differentiation.
    European journal of pharmacology, 1985, Jul-31, Volume: 113, Issue:3

    Topics: Autoradiography; Brain; Humans; In Vitro Techniques; Membranes; Phenazocine; Phencyclidine; Piperidines; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Phencyclidine

1985
Pharmacological and autoradiographic discrimination of sigma and phencyclidine receptor binding sites in brain with (+)-[3H]SKF 10,047, (+)-[3H]-3-[3-hydroxyphenyl]-N-(1-propyl)piperidine and [3H]-1-[1-(2-thienyl)cyclohexyl]piperidine.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:2

    Topics: Animals; Autoradiography; Binding, Competitive; Brain Chemistry; In Vitro Techniques; Kinetics; Male; Phenazocine; Phencyclidine; Piperidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Stereoisomerism

1986
Both the sigma receptor-specific ligand (+)3-PPP and the PCP receptor-specific ligand TCP act in the mouse vas deferens via augmentation of electrically evoked norepinephrine release.
    European journal of pharmacology, 1987, Jun-26, Volume: 138, Issue:3

    Topics: Animals; Electric Stimulation; In Vitro Techniques; Male; Mice; Muscle Contraction; Norepinephrine; Phencyclidine; Piperidines; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Receptors, sigma; Vas Deferens

1987
Synthesis and evaluation of 1-(1-[5-(2'-[18F]fluoroethyl)-2-thienyl]-cyclohexyl)piperidine as a potential in vivo radioligand for the NMDA receptor-channel complex.
    Nuclear medicine and biology, 1993, Volume: 20, Issue:7

    Topics: Animals; Fluorine Radioisotopes; Male; Phencyclidine; Piperidines; Radioligand Assay; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Thiophenes; Tissue Distribution; Tomography, Emission-Computed

1993
The antiparkinsonian agent budipine is an N-methyl-D-aspartate antagonist.
    Journal of neural transmission. Parkinson's disease and dementia section, 1993, Volume: 5, Issue:2

    Topics: Amino Acids; Anesthesia; Animals; Antiparkinson Agents; Binding, Competitive; Brain Chemistry; H-Reflex; In Vitro Techniques; Male; Mice; N-Methylaspartate; Phencyclidine; Piperidines; Rats; Receptors, N-Methyl-D-Aspartate; Reflex; Reflex, Monosynaptic; Seizures; Spinal Cord

1993
Characterization of haloperidol and trifluperidol as subtype-selective N-methyl-D-aspartate (NMDA) receptor antagonists using [3H]TCP and [3H]ifenprodil binding in rat brain membranes.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 280, Issue:2

    Topics: Animals; Binding, Competitive; Brain; Cell Membrane; Female; Haloperidol; Illicit Drugs; Kinetics; Oocytes; Phencyclidine; Piperidines; Radioligand Assay; Rats; Receptors, N-Methyl-D-Aspartate; Recombinant Proteins; Trifluperidol; Xenopus

1997
Morphological and morphometric analysis of serotonin-containing neurons in primary dissociated cultures of human rhombencephalon: a study of development.
    Brain research. Developmental brain research, 1997, Apr-18, Volume: 99, Issue:2

    Topics: Cell Differentiation; Cell Size; Cells, Cultured; Cyclohexanes; Cyclohexenes; Excitatory Amino Acid Antagonists; Fetus; Humans; Illicit Drugs; Neurons; Neuroprotective Agents; Phencyclidine; Piperidines; Receptors, N-Methyl-D-Aspartate; Rhombencephalon; Serotonin

1997
Effect of PCP and sigma ligands on both noradrenaline- and electrically-induced contractions and on [3H]-noradrenaline uptake in rat vas deferens.
    Journal of autonomic pharmacology, 1998, Volume: 18, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Dextromethorphan; Dizocilpine Maleate; Dopamine Agonists; Electric Stimulation; Excitatory Amino Acid Antagonists; Ligands; Male; Muscle Contraction; Neuroprotective Agents; Norepinephrine; Phencyclidine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Phencyclidine; Receptors, sigma; Tritium; Vas Deferens

1998
Re-evaluation of phencyclidine low-affinity or "non-NMDA" binding sites.
    Journal of neuroscience research, 2002, May-01, Volume: 68, Issue:3

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Brain Injuries; Cerebellum; Cyclohexanes; Cyclohexenes; Excitatory Amino Acid Antagonists; Glutamic Acid; Male; Neurons; Neuroprotective Agents; Phencyclidine; Piperidines; Radioligand Assay; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Stereoisomerism; Subcellular Fractions; Synapses; Synaptic Transmission; Tritium

2002
Characterization of the non-competitive antagonist binding site of the NMDA receptor in dark Agouti rats.
    Life sciences, 2004, Aug-06, Volume: 75, Issue:12

    Topics: Animals; Binding, Competitive; Brain; Dextromethorphan; Dioxolanes; Dizocilpine Maleate; Dose-Response Relationship, Drug; Female; Ketamine; N-Methylaspartate; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Mutant Strains; Receptors, N-Methyl-D-Aspartate; Scintillation Counting; Tritium

2004
In vitro biological efficiency of tenocyclidine-TCP and its adamantane derivative TAMORF.
    Toxicology in vitro : an international journal published in association with BIBRA, 2006, Volume: 20, Issue:8

    Topics: Adamantane; Cell Survival; Cholinesterase Inhibitors; Cholinesterase Reactivators; Chromosome Aberrations; Comet Assay; Erythrocytes; Gamma Rays; Humans; In Vitro Techniques; Lethal Dose 50; Leukocytes; Lymphocytes; Morpholines; Mutagens; Phencyclidine; Piperidines; Radiation-Protective Agents; Soman; Structure-Activity Relationship; Thiophenes; Trypan Blue

2006
Structure-activity relationships of pentacycloundecylamines at the N-methyl-d-aspartate receptor.
    Bioorganic & medicinal chemistry, 2007, Feb-01, Volume: 15, Issue:3

    Topics: Amines; Animals; Brain; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Ion Channels; Male; Mice; Mice, Inbred ICR; Models, Molecular; Phencyclidine; Piperidines; Radioligand Assay; Receptors, N-Methyl-D-Aspartate; Structure-Activity Relationship; Synaptosomes; Thiophenes

2007
Tenocyclidine treatment in soman-poisoned rats--intriguing results on genotoxicity versus protection.
    Acta biochimica Polonica, 2008, Volume: 55, Issue:1

    Topics: Acetylcholinesterase; Animals; Brain; Cholinesterase Inhibitors; Cholinesterase Reactivators; Cholinesterases; Comet Assay; Leukocytes; Male; Models, Chemical; Mutagens; Phencyclidine; Piperidines; Rats; Rats, Wistar; Soman; Thiophenes

2008
Inhibition of the histone demethylase LSD1 blocks alpha-herpesvirus lytic replication and reactivation from latency.
    Nature medicine, 2009, Volume: 15, Issue:11

    Topics: Animals; Cell Line, Transformed; Chromatin Immunoprecipitation; DNA Replication; Enzyme Activation; Ganglia; Gene Expression Regulation, Viral; Green Fluorescent Proteins; Herpesvirus 1, Human; Herpesvirus 3, Human; Histone Demethylases; Histone Methyltransferases; Histone-Lysine N-Methyltransferase; Host Cell Factor C1; Humans; Lysine; Mice; Monoamine Oxidase Inhibitors; Mutation; Neurons; Pargyline; Phencyclidine; Piperidines; Promoter Regions, Genetic; Reaction Time; RNA, Small Interfering; Simplexvirus; Thiophenes; Time Factors; Transfection; Virus Replication

2009
Qualitative GC-MS assessment of TCP and TAMORF elimination in rats.
    Arhiv za higijenu rada i toksikologiju, 2010, Volume: 61, Issue:1

    Topics: Adamantane; Animals; Gas Chromatography-Mass Spectrometry; Male; Morpholines; Organophosphate Poisoning; Phencyclidine; Piperidines; Rats; Rats, Wistar; Thiophenes

2010