Page last updated: 2024-08-24

tenocyclidine and n-methylaspartate

tenocyclidine has been researched along with n-methylaspartate in 53 studies

Research

Studies (53)

TimeframeStudies, this research(%)All Research%
pre-199022 (41.51)18.7374
1990's28 (52.83)18.2507
2000's2 (3.77)29.6817
2010's1 (1.89)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cler, JA; Garland, DJ; Hood, WF; Iyengar, S; Mick, SJ; Monahan, JB; Rao, TS; Sun, ET; Vazquez, ML1
Matsuda, Y; Nonaka, H; Nozawa, M; Toki, S; Tsukuda, E; Yoshida, M1
Bonhaus, DW; McNamara, JO3
Nishikawa, T; Ohi, K; Takahashi, K; Takashima, M1
Bonhaus, DW; Hosford, DA; McNamara, JO1
Drian, MJ; Kamenka, JM; Pirat, JL; Privat, A1
Ben-Ari, Y; Roisin-Lallemand, MP; Tremblay, E1
Fujiwara, M; Fukunaga, R; Kameyama, M; Ninomiya, H; Shimohama, S; Taniguchi, T1
Compton, RP; Hood, WF; Monahan, JB1
Bommarito, M; Johnston, MV; McDonald, JW; Silverstein, FS1
Carter, CJ; Lloyd, KG; Scatton, B; Zivkovic, B1
Boksa, P; Chaudieu, I; Mount, H; Quirion, R1
Ikin, AF; Kloog, Y; Sokolovsky, M1
Baron, BM; Harrison, BL; McDonald, IA; Miller, FP; Palfreyman, MG; Salituro, FG; Schmidt, CJ; Sorensen, SM; White, HS1
Cruz, LJ; Gullak, MF; Mena, EE; Olivera, BM; Pagnozzi, MJ; Richter, KE; Rivier, J1
Nabeshima, T; Ogita, K; Yoneda, Y1
Fagg, GE1
Johnson, KM; Morter, RS; Snell, LD2
Bonhaus, DW; McNamara, JO; Skaryak, L; Yeh, GC1
Belaidi, M; Kamenka, JM; Lerner-Natoli, M; N'Gouemo, P; Rondouin, G1
Iversen, SD; Oles, RJ; Preston, C; Singh, L; Tricklebank, MD1
Johnson, KM; Jones, SM1
Johnston, MV; McDonald, JW; Silverstein, FS1
Jarvis, MF; Murphy, DE; Williams, M1
Johnson, KM; Snell, LD1
Bertin, J; Carter, C; Dupont, R; Duverger, D; Frost, J; Gaudilliere, B; Gotti, B; MacKenzie, ET; Rousseau, J; Scatton, B1
Arbilla, S; Benavides, J; Carter, C; Legendre, P; Lloyd, KG; MacKenzie, ET; Noel, F; Thuret, F; Vincent, JD; Zivkovic, B1
Johnson, KM; Nichtenhauser, R; Rivier, J; Snell, LD; Vale, W; Zukin, RS; Zukin, SR1
Ambar, I; Kloog, Y; Sokolovsky, M1
Astier, H; Tapia-Arancibia, L1
Chu, DC; Greenamyre, JT; Maragos, WF; Penney, JB; Young, AB1
Drejer, J; Honoré, T; Nielsen, M; Olverman, HJ; Watkins, JC1
Johnson, KM; Sacaan, AI; Snell, LD1
Johnson, KM; Snell, LD; Yi, SJ1
Drejer, J; Honoré, T1
Ault, B; DeHaven-Hudkins, DL; Dority, JA; Dung, JS; Earley, WG; Herrmann, JL; Kumar, V; Mallamo, JP; Miller, MS; Subramanyam, C1
Bowe, MA; Nadler, JV1
Ferkany, JW; Karbon, EW; Price, CH; Saab, OH; Sweetnam, PM; Wroblewski, JT1
Kovács, KJ; Larson, AA1
Denavit-Saubié, M; Ghilini, G; Salès, N1
Jacobsen, P; Klockgether, T; Löschmann, PA; Turski, L1
French, ED; Mura, A; Wang, T1
Chen, X; Hurlbert, M; Joseph, DB; Kumar, KN; Michaelis, EK; Michaelis, ML1
Nishikawa, T; Takahashi, K; Umino, A; Yoshida, Y1
Baron, BM; Fadayel, GM; Harrison, BL; Kehne, JH; McCloskey, TC; Murawsky, MK; Nyce, P; Salituro, FG; Schmidt, CJ; Senyah, Y; Siegel, BW; Taylor, VL; van Giersbergen, PL; White, HS1
d'Arbigny, P; Gourdier, B; Hoizey, G; Lamiable, D; Millart, H; Vistelle, R1
Mateu, G; Privat, A; Thibault, J; Vignon, J1
Boireau, A; Bordier, F; Imperato, A; Meunier, M; Monterrat, C1
Sun, W; Wessinger, WD1
Bac, P; Gressens, P; Maurois, P; Pages, N; Stables, JP; Stanicki, D; Vamecq, J; Vanden Eynde, JJ1

Reviews

1 review(s) available for tenocyclidine and n-methylaspartate

ArticleYear
TCP binding: a tool for studying NMDA receptor-mediated neurotransmission in kindling.
    Neuroscience and biobehavioral reviews, 1989,Winter, Volume: 13, Issue:4

    Topics: Animals; Aspartic Acid; Brain; Glycine; Kindling, Neurologic; N-Methylaspartate; Phencyclidine; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter

1989

Other Studies

52 other study(ies) available for tenocyclidine and n-methylaspartate

ArticleYear
Characterization of 3-carboxy-5-phosphono-1,2,3,4-tetrahydroisoquinoline (SC-48981), a potent competitive N-methy-D-aspartate (NMDA) receptor antagonist, in vitro and in vivo.
    Neuroscience letters, 1992, Feb-03, Volume: 135, Issue:2

    Topics: Animals; Binding, Competitive; Cerebellum; Cyclic GMP; Glutamates; Glutamic Acid; Glycine; In Vitro Techniques; Isoquinolines; Male; Mice; N-Methylaspartate; Organophosphorus Compounds; Phencyclidine; Receptors, N-Methyl-D-Aspartate; Tetrahydroisoquinolines

1992
The ES-242s, novel N-methyl-D-aspartate antagonists of microbial origin, interact with both the neurotransmitter recognition site and the ion channel domain.
    The Journal of biological chemistry, 1992, Jul-25, Volume: 267, Issue:21

    Topics: Animals; Binding, Competitive; Biological Transport; Calcium; Cells, Cultured; Cyclic GMP; Dizocilpine Maleate; Hippocampus; Ion Channels; Kinetics; Mice; N-Methylaspartate; Neurons; Neurotransmitter Agents; Phencyclidine; Pipecolic Acids; Pyrans; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Synaptic Membranes

1992
Uncompetitive antagonist binding: a biochemical index of activation of the NMDA receptor-coupled ion channel.
    Epilepsy research. Supplement, 1992, Volume: 8

    Topics: 2-Amino-5-phosphonovalerate; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Binding, Competitive; Culture Techniques; Glutamates; Glutamic Acid; Hippocampus; Ibotenic Acid; Ion Channels; Kainic Acid; N-Methylaspartate; Phencyclidine; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission

1992
N-methyl-D-aspartate receptor participates in neuronal transmission of photic information through the retinohypothalamic tract.
    Neuroendocrinology, 1991, Volume: 53, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; Animals; Arylamine N-Acetyltransferase; Hypothalamus; Light; Male; Melatonin; N-Methylaspartate; Neurons; Phencyclidine; Pineal Gland; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Retina; Suprachiasmatic Nucleus; Synaptic Transmission

1991
A radiohistochemical measure of [3H]TCP binding to the activated NMDA-receptor-gated ion channel in rat brain.
    Brain research, 1990, May-21, Volume: 516, Issue:2

    Topics: Animals; Aspartic Acid; Brain; Glycine; Ion Channels; Male; N-Methylaspartate; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter

1990
Non-competitive antagonists of N-methyl-D-aspartate prevent spontaneous neuronal death in primary cultures of embryonic rat cortex.
    Journal of neuroscience research, 1991, Volume: 29, Issue:1

    Topics: Animals; Cell Survival; Cells, Cultured; Cerebral Cortex; Cyclohexanes; Cyclohexenes; Dizocilpine Maleate; Embryo, Mammalian; Female; N-Methylaspartate; Neurons; Phencyclidine; Piperidines; Pregnancy; Rats; Rats, Inbred Strains

1991
Developmental study of [3H]TCP and [3H]glycine binding sites in the rat hippocampus.
    Brain research. Developmental brain research, 1990, Dec-01, Volume: 57, Issue:1

    Topics: Aging; Animals; Autoradiography; Hippocampus; In Vitro Techniques; Kinetics; Magnesium; N-Methylaspartate; Nerve Tissue Proteins; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Strychnine

1990
[3H]N-[1-(2-thienyl)cyclohexyl]-3,4-piperidine ([3H]TCP) binding in human frontal cortex: decreases in Alzheimer-type dementia.
    Journal of neurochemistry, 1990, Volume: 54, Issue:2

    Topics: Alzheimer Disease; Aspartic Acid; Binding Sites; Frontal Lobe; Glutamates; Glutamic Acid; Humans; Membranes; N-Methylaspartate; Phencyclidine; Reference Values

1990
N-methyl-D-aspartate recognition site ligands modulate activity at the coupled glycine recognition site.
    Journal of neurochemistry, 1990, Volume: 54, Issue:3

    Topics: Animals; Aspartic Acid; Binding Sites; Binding, Competitive; Glutamates; Glutamic Acid; Glycine; Ligands; N-Methylaspartate; Phencyclidine; Pipecolic Acids; Piperidines

1990
Effects of hypoxia-ischemia and MK-801 treatment on the binding of a phencyclidine analogue in the developing rat brain.
    Stroke, 1990, Volume: 21, Issue:2

    Topics: Animals; Animals, Newborn; Aspartic Acid; Autoradiography; Binding Sites; Brain; Brain Ischemia; Dibenzocycloheptenes; Dizocilpine Maleate; Glutamates; Glutamic Acid; Hypoxia; N-Methylaspartate; Phencyclidine; Rats; Rats, Inbred Strains; Tritium

1990
Ifenprodil and SL 82.0715 as cerebral antiischemic agents. III. Evidence for antagonistic effects at the polyamine modulatory site within the N-methyl-D-aspartate receptor complex.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Aspartic Acid; Binding Sites; Binding, Competitive; Brain; Cells, Cultured; Drug Interactions; Female; Glycine; Male; N-Methylaspartate; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Spermidine; Spermine; Spinal Cord

1990
Phencyclidine and related compounds evoked [3H]dopamine release from rat mesencephalic cell cultures by a mechanism independent of the phencyclidine receptor, sigma binding site, or dopamine uptake site.
    Canadian journal of physiology and pharmacology, 1990, Volume: 68, Issue:9

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anticonvulsants; Binding Sites; Cells, Cultured; Dioxolanes; Dizocilpine Maleate; Dopamine; Dose-Response Relationship, Drug; Guanidines; Mesencephalon; N-Methylaspartate; Neurotransmitter Uptake Inhibitors; Phencyclidine; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Phencyclidine; Sigma Factor; Tritium

1990
N-methyl-D-aspartate/phencyclidine receptor complex of rat forebrain: purification and biochemical characterization.
    Biochemistry, 1990, Mar-06, Volume: 29, Issue:9

    Topics: Animals; Aspartic Acid; Brain; Chromatography, Affinity; Electrophoresis, Polyacrylamide Gel; Glutamates; Glycine; Male; Molecular Weight; N-Methylaspartate; Phencyclidine; Rats; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Solubility

1990
Activity of 5,7-dichlorokynurenic acid, a potent antagonist at the N-methyl-D-aspartate receptor-associated glycine binding site.
    Molecular pharmacology, 1990, Volume: 38, Issue:4

    Topics: Animals; Calcium; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Kynurenic Acid; Male; N-Methylaspartate; Norepinephrine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter

1990
Conantokin-G: a novel peptide antagonist to the N-methyl-D-aspartic acid (NMDA) receptor.
    Neuroscience letters, 1990, Oct-16, Volume: 118, Issue:2

    Topics: Amino Acid Sequence; Animals; Conotoxins; Cyclic GMP; Glutamates; Glycine; In Vitro Techniques; Kainic Acid; Molecular Sequence Data; N-Methylaspartate; Peptides, Cyclic; Phencyclidine; Rats; Receptors, N-Methyl-D-Aspartate; Tritium

1990
[3H]thienylcyclohexylpiperidine binding activity in brain synaptic membranes treated with Triton X-100.
    Journal of neurochemistry, 1990, Volume: 55, Issue:5

    Topics: Animals; Brain; Detergents; Drug Synergism; Glutamates; Male; N-Methylaspartate; Octoxynol; Phencyclidine; Polyethylene Glycols; Rats; Rats, Inbred Strains; Synaptic Membranes; Tritium

1990
Phencyclidine and related drugs bind to the activated N-methyl-D-aspartate receptor-channel complex in rat brain membranes.
    Neuroscience letters, 1987, May-06, Volume: 76, Issue:2

    Topics: Amino Acids; Anesthetics, Dissociative; Animals; Aspartic Acid; Brain; Ion Channels; Male; N-Methylaspartate; Narcotics; Phencyclidine; Rats; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Subcellular Fractions

1987
Structural requirements for activation of the glycine receptor that modulates the N-methyl-D-aspartate operated ion channel.
    European journal of pharmacology, 1988, Oct-26, Volume: 156, Issue:1

    Topics: Amino Acids; Animals; Aspartic Acid; Cerebral Cortex; Glycine; Ion Channels; N-Methylaspartate; Phencyclidine; Rats; Receptors, Glycine; Receptors, Neurotransmitter

1988
Glycine regulation of the N-methyl-D-aspartate receptor-gated ion channel in hippocampal membranes.
    Molecular pharmacology, 1989, Volume: 36, Issue:2

    Topics: Allosteric Regulation; Animals; Aspartic Acid; Cell Membrane; Glutamates; Glycine; Hippocampus; In Vitro Techniques; Ion Channels; Kinetics; Male; N-Methylaspartate; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter

1989
[Excitotoxic damage of the hippocampus in the rat: involvement of N-methyl-D-aspartate receptors].
    Comptes rendus des seances de la Societe de biologie et de ses filiales, 1989, Volume: 183, Issue:3

    Topics: Animals; Aspartic Acid; Hippocampus; Illicit Drugs; Kainic Acid; Male; N-Methylaspartate; Phencyclidine; Rats; Rats, Inbred Strains

1989
The behavioural effects of MK-801: a comparison with antagonists acting non-competitively and competitively at the NMDA receptor.
    European journal of pharmacology, 1989, Aug-11, Volume: 167, Issue:1

    Topics: Animals; Anticonvulsants; Aspartic Acid; Behavior, Animal; Binding, Competitive; Dibenzocycloheptenes; Discrimination Learning; Dizocilpine Maleate; Dose-Response Relationship, Drug; Ketamine; Male; Motor Activity; N-Methylaspartate; Phenazocine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Seizures

1989
Effects of amygdaloid kindling on NMDA receptor function and regulation.
    Experimental neurology, 1989, Volume: 106, Issue:1

    Topics: Amygdala; Animals; Aspartic Acid; Brain; Glutamates; Glutamic Acid; Glycine; Hippocampus; Kindling, Neurologic; Male; N-Methylaspartate; Norepinephrine; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter

1989
Neuroprotective effects of MK-801, TCP, PCP and CPP against N-methyl-D-aspartate induced neurotoxicity in an in vivo perinatal rat model.
    Brain research, 1989, Jun-19, Volume: 490, Issue:1

    Topics: Animals; Aspartic Acid; Brain; Dose-Response Relationship, Drug; Female; Male; N-Methylaspartate; Phencyclidine; Piperazines; Rats; Rats, Inbred Strains

1989
Quantitative autoradiographic localization of NMDA receptors in rat brain using [3H]CPP: comparison with [3H]TCP binding sites.
    European journal of pharmacology, 1987, Sep-02, Volume: 141, Issue:1

    Topics: Animals; Aspartic Acid; Autoradiography; Brain; Brain Chemistry; In Vitro Techniques; Ligands; Male; N-Methylaspartate; Phencyclidine; Piperazines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter

1987
Cycloleucine competitively antagonizes the strychnine-insensitive glycine receptor.
    European journal of pharmacology, 1988, Jun-22, Volume: 151, Issue:1

    Topics: Amino Acids; Animals; Aspartic Acid; Binding, Competitive; Cycloleucine; Glycine; In Vitro Techniques; Male; N-Methylaspartate; Phencyclidine; Rats; Receptors, Glycine; Receptors, Neurotransmitter; Strychnine

1988
N-methyl-D-aspartate receptor regulation of uncompetitive antagonist binding in rat brain membranes: kinetic analysis.
    Molecular pharmacology, 1988, Volume: 34, Issue:3

    Topics: Animals; Aspartic Acid; Brain; Glycine; In Vitro Techniques; Kinetics; Male; N-Methylaspartate; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter

1988
Ifenprodil and SL 82.0715 as cerebral anti-ischemic agents. I. Evidence for efficacy in models of focal cerebral ischemia.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 247, Issue:3

    Topics: Animals; Aspartic Acid; Brain Ischemia; Cats; Female; Male; Models, Cardiovascular; N-Methylaspartate; Phencyclidine; Piperidines; Rats; Rats, Inbred F344; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Vasoconstriction

1988
Ifenprodil and SL 82.0715 as cerebral anti-ischemic agents. II. Evidence for N-methyl-D-aspartate receptor antagonist properties.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 247, Issue:3

    Topics: Animals; Aspartic Acid; Brain Ischemia; Cells, Cultured; Cerebellum; Corpus Striatum; Cyclic GMP; Dopamine; Harmaline; In Vitro Techniques; Mice; N-Methylaspartate; Phencyclidine; Piperazines; Piperidines; Rats; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Spinal Cord

1988
An endogenous ligand of the brain sigma/PCP receptor antagonizes NMDA-induced neurotransmitter release.
    Brain research, 1987, Jul-21, Volume: 416, Issue:1

    Topics: Acetylcholine; Animals; Aspartic Acid; Cattle; Corpus Striatum; Dopamine; Hippocampus; In Vitro Techniques; Male; N-Methylaspartate; Neurotransmitter Agents; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Phencyclidine; Tissue Extracts

1987
Solubilization of rat brain phencyclidine receptors in an active binding form that is sensitive to N-methyl-D-aspartate receptor ligands.
    Journal of neurochemistry, 1988, Volume: 51, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Animals; Aspartic Acid; Binding, Competitive; Brain Chemistry; Cell Membrane; Cholic Acid; Cholic Acids; Detergents; Glutamates; Glutamic Acid; Male; N-Methylaspartate; Phencyclidine; Rats; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Phencyclidine; Solubility; Valine

1988
Glutamate stimulates somatostatin release from diencephalic neurons in primary culture.
    Endocrinology, 1988, Volume: 123, Issue:5

    Topics: 2-Amino-5-phosphonovalerate; Animals; Aspartic Acid; Cells, Cultured; Diencephalon; Glutamates; Glutamic Acid; Kainic Acid; Magnesium; N-Methylaspartate; Neurons; Oxadiazoles; Phencyclidine; Potassium; Quisqualic Acid; Rats; Somatostatin; Tetrodotoxin; Valine; Veratridine

1988
High correlation between the localization of [3H]TCP binding and NMDA receptors.
    European journal of pharmacology, 1986, Apr-09, Volume: 123, Issue:1

    Topics: Animals; Aspartic Acid; Autoradiography; Brain; N-Methylaspartate; Phencyclidine; Rats; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter

1986
Molecular target size of NMDA antagonist binding sites.
    European journal of pharmacology, 1987, Apr-07, Volume: 136, Issue:1

    Topics: Animals; Aspartic Acid; Cerebral Cortex; In Vitro Techniques; Ligands; Molecular Weight; N-Methylaspartate; Phencyclidine; Pyrazines; Radioligand Assay; Rats; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter

1987
Equilibrium analysis of [3H]TCP binding: effects of glycine, magnesium and N-methyl-D-aspartate agonists.
    European journal of pharmacology, 1988, Jul-26, Volume: 152, Issue:1-2

    Topics: Animals; Aspartic Acid; Binding, Competitive; Cerebral Cortex; Dialysis; Glycine; In Vitro Techniques; Magnesium; Male; N-Methylaspartate; Phencyclidine; Rats; Rats, Inbred Strains; Synaptosomes

1988
Comparison of the effects of MK-801 and phencyclidine on catecholamine uptake and NMDA-induced norepinephrine release.
    European journal of pharmacology, 1988, Jan-12, Volume: 145, Issue:2

    Topics: Animals; Aspartic Acid; Catecholamines; Dibenzocycloheptenes; Dizocilpine Maleate; Hippocampus; In Vitro Techniques; N-Methylaspartate; Norepinephrine; Phencyclidine; Rats

1988
Phencyclidine analogues inhibit NMDA-stimulated [3H]GABA release from cultured cortex neurons.
    European journal of pharmacology, 1987, Nov-10, Volume: 143, Issue:2

    Topics: Animals; Aspartic Acid; Binding, Competitive; Cerebral Cortex; gamma-Aminobutyric Acid; In Vitro Techniques; N-Methylaspartate; Neurons; Phencyclidine; Rats

1987
Glycine potentiates N-methyl-D-aspartate-induced [3H]TCP binding to rat cortical membranes.
    Neuroscience letters, 1987, Dec-29, Volume: 83, Issue:3

    Topics: Animals; Aspartic Acid; Cell Membrane; Cerebral Cortex; Drug Synergism; Electric Stimulation; Glycine; In Vitro Techniques; Male; N-Methylaspartate; Phencyclidine; Rats; Rats, Inbred Strains

1987
Identification, synthesis, and characterization of a unique class of N-methyl-D-aspartate antagonists. The 6,11-ethanobenzo[b]quinolizinium cation.
    Journal of medicinal chemistry, 1994, Dec-23, Volume: 37, Issue:26

    Topics: Animals; Binding Sites; Ion Channels; Male; Mice; N-Methylaspartate; Neuroprotective Agents; Phencyclidine; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship

1994
Polyamines antagonize N-methyl-D-aspartate-evoked depolarizations, but reduce Mg2+ block.
    European journal of pharmacology, 1995, May-04, Volume: 278, Issue:1

    Topics: Action Potentials; Analysis of Variance; Animals; Binding, Competitive; Chromatography, High Pressure Liquid; Diamines; Drug Interactions; Eflornithine; Female; Hippocampus; Magnesium; Male; N-Methylaspartate; Phencyclidine; Polyamines; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Spermine

1995
The envelope glycoprotein of HIV-1 alters NMDA receptor function.
    The European journal of neuroscience, 1993, Mar-01, Volume: 5, Issue:3

    Topics: Animals; Calcium Channel Blockers; Cells, Cultured; Dizocilpine Maleate; Electrophysiology; HIV Envelope Protein gp120; N-Methylaspartate; Oocytes; Phencyclidine; Pipecolic Acids; Radioligand Assay; Rats; Receptors, N-Methyl-D-Aspartate; Recombinant Proteins; Xenopus

1993
Density of NMDA-coupled and uncoupled 1-[1-(2-[3H]thienyl) cyclohexyl]piperidine recognition sites in the brain and spinal cord: differential effects of NMDA agonists and antagonists.
    Journal of neurochemistry, 1994, Volume: 63, Issue:5

    Topics: Animals; Binding Sites; Brain; Brain Chemistry; Dizocilpine Maleate; Glutamic Acid; Glycine; Haloperidol; Male; Mice; N-Methylaspartate; Phencyclidine; Spinal Cord; Tritium

1994
Autoradiographic localisation of NMDA binding sites in brainstem cardiorespiratory areas of adult and newborn cats.
    Brain research. Developmental brain research, 1993, Sep-17, Volume: 75, Issue:1

    Topics: Aging; Animals; Animals, Newborn; Autoradiography; Binding Sites; Brain Mapping; Brain Stem; Cats; Illicit Drugs; Membrane Potentials; N-Methylaspartate; Neurons; Phencyclidine; Pons; Receptors, N-Methyl-D-Aspartate; Tritium

1993
The antiparkinsonian agent budipine is an N-methyl-D-aspartate antagonist.
    Journal of neural transmission. Parkinson's disease and dementia section, 1993, Volume: 5, Issue:2

    Topics: Amino Acids; Anesthesia; Animals; Antiparkinson Agents; Binding, Competitive; Brain Chemistry; H-Reflex; In Vitro Techniques; Male; Mice; N-Methylaspartate; Phencyclidine; Piperidines; Rats; Receptors, N-Methyl-D-Aspartate; Reflex; Reflex, Monosynaptic; Seizures; Spinal Cord

1993
MK-801, phencyclidine (PCP), and PCP-like drugs increase burst firing in rat A10 dopamine neurons: comparison to competitive NMDA antagonists.
    Synapse (New York, N.Y.), 1993, Volume: 13, Issue:2

    Topics: Action Potentials; Animals; Dizocilpine Maleate; Dopamine; Dose-Response Relationship, Drug; Illicit Drugs; Male; N-Methylaspartate; Neurons; Phencyclidine; Pipecolic Acids; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Stereotaxic Techniques; Tegmentum Mesencephali; Vibrissae

1993
Ethanol-induced inhibition of [3H]thienylcyclohexylpiperidine (TCP) binding to NMDA receptors in brain synaptic membranes and to a purified protein complex.
    Journal of neurochemistry, 1996, Volume: 67, Issue:1

    Topics: Animals; Brain Chemistry; Dizocilpine Maleate; Dopamine Antagonists; Ethanol; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Glycine; Haloperidol; Illicit Drugs; Kinetics; Male; Membrane Proteins; N-Methylaspartate; Phencyclidine; Protein Binding; Proteins; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Sensitivity and Specificity; Spermidine; Synaptic Membranes; Tritium

1996
Evidence for N-methyl-D-aspartate receptor-mediated increase in norepinephrine utilization in the prefrontal cortex of unanesthetized rats.
    Brain research, 1997, Jan-02, Volume: 744, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Adrenergic Agents; Animals; Binding, Competitive; Consciousness; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Male; Microinjections; N-Methylaspartate; Norepinephrine; Oxidopamine; Phencyclidine; Piperazines; Prefrontal Cortex; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Sympathomimetics; Tritium

1997
Pharmacological characterization of MDL 105,519, an NMDA receptor glycine site antagonist.
    European journal of pharmacology, 1997, Apr-04, Volume: 323, Issue:2-3

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Calcium Channels; Cells, Cultured; Cerebellum; Cyclic GMP; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Indoles; Ligands; Male; Mice; Mice, Inbred DBA; Motor Activity; N-Methylaspartate; Phencyclidine; Rats; Rats, Inbred F344; Rats, Wistar; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate; Sodium Channels

1997
Determination of gacyclidine enantiomers in human plasma by gas chromatography-mass spectrometry using selected-ion monitoring.
    Journal of chromatography. B, Biomedical sciences and applications, 1997, Dec-19, Volume: 704, Issue:1-2

    Topics: Calibration; Gas Chromatography-Mass Spectrometry; Humans; Hydrogen-Ion Concentration; Male; Microchemistry; N-Methylaspartate; Phencyclidine; Quality Control; Sensitivity and Specificity; Solvents; Stereoisomerism

1997
Comparison of glutamate and N-methyl-D-aspartate toxicities on rat mesencephalic primary cell cultures.
    International journal of developmental neuroscience : the official journal of the International Society for Developmental Neuroscience, 1997, Volume: 15, Issue:7

    Topics: Animals; Cells, Cultured; Dopamine; Excitatory Amino Acid Antagonists; Glutamic Acid; Logistic Models; N-Methylaspartate; Neurons; Neuroprotective Agents; Phencyclidine; Rats; Rats, Sprague-Dawley; Substantia Nigra

1997
Effects of RPR 118723, a novel antagonist at the glycine site of the NMDA receptor, in vitro.
    European journal of pharmacology, 2000, Aug-04, Volume: 401, Issue:2

    Topics: Animals; Binding, Competitive; Cerebral Cortex; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Glycine; In Vitro Techniques; Male; Membranes; Mice; N-Methylaspartate; Phencyclidine; Pyrazines; Rats; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate; Tritium

2000
Characterization of the non-competitive antagonist binding site of the NMDA receptor in dark Agouti rats.
    Life sciences, 2004, Aug-06, Volume: 75, Issue:12

    Topics: Animals; Binding, Competitive; Brain; Dextromethorphan; Dioxolanes; Dizocilpine Maleate; Dose-Response Relationship, Drug; Female; Ketamine; N-Methylaspartate; Phenazocine; Phencyclidine; Piperidines; Rats; Rats, Mutant Strains; Receptors, N-Methyl-D-Aspartate; Scintillation Counting; Tritium

2004
1,2-ethane bis-1-amino-4-benzamidine is active against several brain insult and seizure challenges through anti-NMDA mechanisms targeting the 3H-TCP binding site and antioxidant action.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:7

    Topics: Animals; Anticonvulsants; Antioxidants; Benzamidines; Binding Sites; Body Temperature; Brain; Mice; Models, Molecular; Molecular Conformation; Motor Activity; N-Methylaspartate; Neuroprotective Agents; Phencyclidine; Receptors, N-Methyl-D-Aspartate; Seizures

2010