Page last updated: 2024-08-16

temazepam and diazepam

temazepam has been researched along with diazepam in 105 studies

Research

Studies (105)

TimeframeStudies, this research(%)All Research%
pre-199045 (42.86)18.7374
1990's25 (23.81)18.2507
2000's17 (16.19)29.6817
2010's16 (15.24)24.3611
2020's2 (1.90)2.80

Authors

AuthorsStudies
Collins, RJ; Gall, M; Kamdar, BV1
Babbini, M; Barbaro, AM; Bartoletti, M; Biagi, GL; Borea, PA; Gaiardi, M; Guerra, MC1
Johnston, GA; Maddalena, DJ1
Karplus, M; So, SS1
Topliss, JG; Yoshida, F1
Chang, TK; Ensom, MH; Kiang, TK1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Du-Cuny, L; Huwyler, J; Kansy, M; Wiese, M1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Carmona, AV; Kumari, S; Tiwari, AK; Trippier, PC1
Nicholson, AN; Stone, BM2
Nicholson, AN2
Baars, AM; Hekster, YA; O'Reilly, WJ; van der Kleijn, E; Vree, TB1
Stone, BM1
Allen, MD; Greenblatt, DJ; Orsulak, PJ; Shader, RI; Woo, E1
Clarke, CH; Nicholson, AN1
Kanto, J; Mäenpää, M; Mäntylä, R; Sellman, R; Valovirta, E1
Loeffler, PM1
Beischlag, TV; Inaba, T; Kalow, W; Mahon, WA1
Cobbs, LW1
Lewis, DC; Sullivan, JT; Swift, RM1
Fisher, PB; Fryer, RI; Pestka, S; Solowey, WE; Spector, S1
Guentert, TW; Stebler, T1
Hooper, WD; Mason, SR; Reilly, PE; Thompson, DA1
Dollar, NS; Matthews, NS; Shawley, RV1
Dusci, LJ; Good, SM; Hall, RW; Ilett, KF1
Chenery, RJ; Lockwood, GF; Seddon, T1
Barry, H; Cullen, JH; Harris, D; O'Boyte, CA1
Barry, H; Harris, D; O'Boyle, CA1
Castleden, M; Fancourt, G1
Brook, IM; Hoise, HE; Holmes, A1
Barry, H; Harris, D; O'Boyle, C1
Brook, IM; Hosie, HE; Nimmo, WS1
Klockowski, PM; Levy, G2
Brase, DA; Dewey, WL; Glennon, RA; Young, R1
Dolan, S; Lau, CE; Tang, M1
Igarashi, T; Kitagawa, H; Ohmori, S; Okiyama, M; Ueno, K1
Herschman, HR; Kujubu, DA; Lim, RW; Varnum, BC1
Moroji, T; Motomura, H; Noguchi, T; Sekiguchi, R; Tada, K1
Martin, WR; McNicholas, LF; Pruitt, TA1
Aranko, K1
Meeles, MT; Thys, CP; Tjaden, UR; van der Kaay, M1
Bianchi, MC; Bruni, G; Ghirardi, P; Loreti, P; Ravaccia, F; Tallone, G1
Douglas, JG; Finlayson, ND; Heading, RC; Jarvie, DR; Nimmo, WS; Wanlesss, R1
Amarasekera, K1
El-Hazmi, MA1
Bardhan, KD1
Burt, D; Clark, G; Erwin, D; Major, E; Yate, P1
Löscher, W1
MacKinnon, GL; Parker, WA1
Bittencourt, PR; Richens, A; Smith, AT; Wade, P2
Berlin, RM; Conell, LJ1
Swift, CG1
Arunasalam, K; Cundy, JM1
Booij, LH; Crul, JF; Driessen, JJ; van Egmond, J; Vree, TB1
Coffman, WB; McFarland, SA; Meyer, EA; Mumford, R; Wynn, RL1
Chiba, K; Chiba, T; Hirano, T; Horii, H; Ishizaki, T; Kato, Y1
Holden, JD; Hughes, IM; Tree, A1
Andersson, T; Birkett, DJ; Miners, JO; Veronese, ME1
Robertson, JR1
Pang, KS; St-Pierre, MV1
Garretty, DJ; Hay, AW; Raistrick, D; Wolff, K1
Gunaratna, C; Kissinger, PT1
Gelboin, HV; Gonzalez, FJ; Korzekwa, KR; Shou, M; Yang, SK; Yang, TJ1
Ali, HM; Azzam, RM; Notarianni, LJ1
Ackermann, I; Angermaier, L; Deinl, I; Franzelius, C; Machbert, G1
Carlin, JB; Holm-Knudsen, RJ; McKenzie, IM1
Baillie, TA; Dai, R; Ettore, MW; Mei, Q; Rushmore, TH; Shou, M1
Augustijns, P; Kinget, R; Van den Mooter, G1
Bond, CM; Hickey, F; Matheson, C1
Abou-Mandour, AA; Beckmann, H; Czygan, FC; Kavvadias, D; Riederer, P; Sand, P; Schreier, P1
Mørland, J; Olsen, KM; Skuterud, B; Smith-Kielland, A1
Contel, N; Grossman, S; Liu, Z; Ren, S; Rose, A; Short, J; Unger, S1
Black, M; Oliver, JS; Seymour, A1
Blaton, N; Kinget, R; Van den Mooter, G; Verheyen, S1
Abd-Ellah, MF; Andrews, J; Carlile, DJ; Friedberg, T; Houston, JB; Kenworthy, KE; Randolph, NL1
Djeridane, Y; Touitou, Y1
Fujita, S; Ishizuka, M; Kazusaka, A; Kim, HS; Saito, K; Sakai, N1
Fidecka, S; Listos, J; Malec, D1
Dickson, SJ; Irving, RC1
Acikgöz, A; Bader, A; Giri, S; Karim, N; Schmidt-Heck, W1
Cole, B; Fishbain, DA; Gao, J; Lewis, JE; Rosomoff, RS1
Iannello, C; Mandrioli, R; Matrisciano, F; Mercolini, L; Nicoletti, F; Raggi, MA1
Abe, K; Kobayashi, N; Nakamura, K; Nishiya, Y; Okazaki, O; Okudaira, N1
Acikgöz, A; Bader, A; Giri, S; Maringka, M; Nieber, K1
Bowron, P; Fu, S; Lewis, J; Molnar, A; Wang, H1
Darwish, WS; Hayami, A; Ikenaka, Y; Ishizuka, M; Nakayama, SM1
Liang, C; Ni, C; Rao, Y; Wang, R; Wang, X; Xiong, L; Zhang, Y1
Atayee, RS; Best, BM; Luk, S; Ma, JD1
Bertol, E; Boscolo Berto, R; Favretto, D; Mannaioni, G; Mari, F; Vaiano, F1
Bankstahl, M; Gramer, M; Hausknecht, M; Klein, S; Löscher, W1
Li, J; Liu, H; Wu, L; Zhang, J1
Darwish, WS; Hayami, A; Ikenaka, Y; Ishizuka, M; Kawai, YK; Mizukawa, H; Nakayama, SM; Watanabe, KP1
Jia, J; Jiang, F; Johansen, SS; Linnet, K; Rao, Y; Wang, X; Zhang, Y1
Mangelings, D; Muscat Galea, C; Vander Heyden, Y1
Castro, A; Costa, P; Franco, JM; Melo, P; Quintas, MJ; Tarelho, S; Teixeira, HM1
Downes, MA; Lovett, CJ; Sadler, CW; Vidler, S1
Adhikari, S; Barron, LP; Bhatnagar, A; Bowes, DA; Coronado-Apodaca, KG; Driver, EM; Halden, RU; Kumar, R; Martínez-Ruiz, M; McCall, KL; Melchor-Martínez, EM; Ng, KT; Oyervides-Muñoz, MA; Parra-Saldivar, R; Piper, BJ; Smith, T; Sosa-Hernandez, JE1

Reviews

6 review(s) available for temazepam and diazepam

ArticleYear
UDP-glucuronosyltransferases and clinical drug-drug interactions.
    Pharmacology & therapeutics, 2005, Volume: 106, Issue:1

    Topics: Clinical Trials as Topic; Drug Interactions; Enzyme Activation; Enzyme Induction; Glucuronides; Glucuronosyltransferase; Humans; Pharmaceutical Preparations; Pharmacogenetics; Polymorphism, Genetic

2005
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Amide Bond Bioisosteres: Strategies, Synthesis, and Successes.
    Journal of medicinal chemistry, 2020, 11-12, Volume: 63, Issue:21

    Topics: Amides; Carbamates; Click Chemistry; Drug Design; Pyridines; Structure-Activity Relationship; Triazoles; Urea

2020
Oral benzodiazepines and conscious sedation: a review.
    Journal of oral and maxillofacial surgery : official journal of the American Association of Oral and Maxillofacial Surgeons, 1992, Volume: 50, Issue:9

    Topics: Administration, Oral; Alprazolam; Ambulatory Surgical Procedures; Anti-Anxiety Agents; Conscious Sedation; Diazepam; Flurazepam; Humans; Lorazepam; Midazolam; Oxazepam; Premedication; Receptors, GABA-A; Temazepam; Triazolam

1992
Benzodiazepine withdrawal syndrome: a literature review and evaluation.
    The American journal of drug and alcohol abuse, 1982, Volume: 9, Issue:1

    Topics: Anti-Anxiety Agents; Chlordiazepoxide; Diazepam; Dose-Response Relationship, Drug; Humans; Lorazepam; Nitrazepam; Oxazepam; Substance Withdrawal Syndrome; Substance-Related Disorders; Temazepam; Time Factors

1982
Postural instability as a measure of sedative drug response.
    British journal of clinical pharmacology, 1984, Volume: 18 Suppl 1

    Topics: Adult; Aged; Amitriptyline; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Chlormethiazole; Diazepam; Dose-Response Relationship, Drug; Humans; Hypnotics and Sedatives; Nitrazepam; Posture; Temazepam; Time Factors; Triazolam

1984

Trials

16 trial(s) available for temazepam and diazepam

ArticleYear
Diazepam and 3-hydroxydiazepam (temazepam) and sleep of middle age.
    British journal of clinical pharmacology, 1979, Volume: 7, Issue:5

    Topics: Anti-Anxiety Agents; Diazepam; Humans; Male; Middle Aged; Placebos; Sleep; Sleep Stages; Temazepam; Time Factors

1979
Immediate and residual effects in man of the metabolites of diazepam.
    British journal of clinical pharmacology, 1978, Volume: 6, Issue:4

    Topics: Adult; Choice Behavior; Diazepam; Humans; Male; Motor Skills; Nordazepam; Oxazepam; Placebos; Reaction Time; Temazepam; Time Factors

1978
Differential effect of benzodiazepine sedation in high and low anxious patients in a "real life" stress setting.
    Psychopharmacology, 1986, Volume: 88, Issue:2

    Topics: Adult; Anti-Anxiety Agents; Anxiety; Diazepam; Double-Blind Method; Female; Humans; Male; Models, Neurological; Personality Inventory; Random Allocation; Stress, Psychological; Temazepam; Tooth, Impacted

1986
Sedation in outpatient oral surgery. Comparison of temazepam by mouth and diazepam i.v.
    British journal of anaesthesia, 1986, Volume: 58, Issue:4

    Topics: Administration, Oral; Adolescent; Adult; Anti-Anxiety Agents; Anxiety; Diazepam; Double-Blind Method; Female; Hemodynamics; Humans; Hypnotics and Sedatives; Injections, Intravenous; Male; Patient Acceptance of Health Care; Psychomotor Performance; Temazepam; Tooth Extraction; Tooth, Impacted

1986
Oral sedation with temazepam: controlled comparison of a soft gelatin capsule formulation with intravenous diazepam.
    British dental journal, 1987, Apr-25, Volume: 162, Issue:8

    Topics: Administration, Oral; Adolescent; Adult; Anesthesia, Dental; Anti-Anxiety Agents; Anxiety; Capsules; Diazepam; Double-Blind Method; Female; Humans; Injections, Intravenous; Male; Preanesthetic Medication; Temazepam; Tooth, Impacted

1987
Comparison of sedation with temazepam by mouth and diazemuls i.v. for dental surgery. Variability in absorption may influence clinical effect.
    British journal of anaesthesia, 1988, Volume: 60, Issue:1

    Topics: Administration, Oral; Adolescent; Adult; Anesthesia, Dental; Anti-Anxiety Agents; Anxiety; Diazepam; Female; Humans; Hypnotics and Sedatives; Injections, Intravenous; Intestinal Absorption; Male; Middle Aged; Surgery, Oral; Temazepam

1988
Task-dependent development of cross-tolerance to psychomotor effects of lorazepam in man.
    Acta pharmacologica et toxicologica, 1985, Volume: 56, Issue:5

    Topics: Adult; Alprazolam; Benzodiazepines; Diazepam; Drug Tolerance; Female; Humans; Lorazepam; Male; Nitrazepam; Psychomotor Performance; Temazepam

1985
Sedation for upper gastro-intestinal endoscopy. A comparison of oral temazepam and i.v. diazepam.
    British journal of anaesthesia, 1980, Volume: 52, Issue:8

    Topics: Administration, Oral; Anti-Anxiety Agents; Diazepam; Digestive System; Endoscopy; Female; Humans; Injections, Intravenous; Male; Middle Aged; Premedication; Temazepam

1980
Temazepam as a premedicant in minor surgery.
    Anaesthesia, 1980, Volume: 35, Issue:8

    Topics: Adult; Anti-Anxiety Agents; Anxiety; Blood Pressure; Diazepam; Female; Heart Rate; Humans; Minor Surgical Procedures; Patient Acceptance of Health Care; Preanesthetic Medication; Temazepam

1980
Temazepam as premedication in elderly patients.
    Anaesthesia, 1982, Volume: 37, Issue:4

    Topics: Aged; Anti-Anxiety Agents; Anxiety; Clinical Trials as Topic; Diazepam; Double-Blind Method; Humans; Male; Middle Aged; Preanesthetic Medication; Random Allocation; Temazepam; Time Factors

1982
Benzodiazepines impair smooth pursuit eye movements.
    British journal of clinical pharmacology, 1983, Volume: 15, Issue:2

    Topics: Adult; Anti-Anxiety Agents; Diazepam; Double-Blind Method; Eye Movements; Humans; Male; Random Allocation; Temazepam

1983
Profile of recovery after general anaesthesia.
    British medical journal (Clinical research ed.), 1983, Jun-25, Volume: 286, Issue:6383

    Topics: Anesthesia, General; Anesthesia, Obstetrical; Diazepam; Female; Humans; Pregnancy; Reaction Time; Temazepam; Time Factors

1983
The relationship between peak velocity of saccadic eye movements and serum benzodiazepine concentration.
    British journal of clinical pharmacology, 1981, Volume: 12, Issue:4

    Topics: Adult; Benzodiazepines; Diazepam; Double-Blind Method; Eye Movements; Flurazepam; Humans; Male; Nitrazepam; Nordazepam; Reticular Formation; Saccades; Temazepam

1981
Distress at induction of anaesthesia in children. A survey of incidence, associated factors and recovery characteristics.
    Paediatric anaesthesia, 1998, Volume: 8, Issue:5

    Topics: Adjuvants, Anesthesia; Adolescent; Age Factors; Anesthesia; Anesthesia Recovery Period; Anti-Anxiety Agents; Anxiety; Arousal; Child; Child, Preschool; Diazepam; Female; Humans; Hypnotics and Sedatives; Infant; Male; Midazolam; Preanesthetic Medication; Temazepam

1998
Urinary excretion of diazepam metabolites in healthy volunteers and drug users.
    Scandinavian journal of clinical and laboratory investigation, 2001, Volume: 61, Issue:3

    Topics: Adult; Anti-Anxiety Agents; Chromatography, Gas; Chromatography, High Pressure Liquid; Creatinine; Diazepam; Female; Humans; Male; Middle Aged; Nordazepam; Oxazepam; Substance Abuse Detection; Substance-Related Disorders; Temazepam

2001
Effect of a metabolite of diazepam, 3-hydroxydiazepam (temazepam), on sleep in man.
    British journal of clinical pharmacology, 1976, Volume: 3, Issue:4

    Topics: Adult; Diazepam; Electroencephalography; Humans; Hypnotics and Sedatives; Male; Sleep; Sleep Stages; Temazepam; Time Factors; Young Adult

1976

Other Studies

83 other study(ies) available for temazepam and diazepam

ArticleYear
Pharmacology of some metabolites of triazolam, alprazolam, and diazepam prepared by a simple, one-step oxidation of benzodiazepines.
    Journal of medicinal chemistry, 1978, Volume: 21, Issue:12

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Diazepam; Hydroxylation; Male; Methods; Mice; Oxidation-Reduction; Triazolam; Triazoles

1978
Rm values and structure-activity relationship of benzodiazepines.
    Journal of medicinal chemistry, 1980, Volume: 23, Issue:2

    Topics: Animals; Benzodiazepines; Chromatography, Thin Layer; Conflict, Psychological; Exploratory Behavior; Models, Biological; Rats; Solubility; Structure-Activity Relationship

1980
Prediction of receptor properties and binding affinity of ligands to benzodiazepine/GABAA receptors using artificial neural networks.
    Journal of medicinal chemistry, 1995, Feb-17, Volume: 38, Issue:4

    Topics: Binding Sites; Ligands; Neural Networks, Computer; Predictive Value of Tests; Receptors, GABA-A; Structure-Activity Relationship

1995
Genetic neural networks for quantitative structure-activity relationships: improvements and application of benzodiazepine affinity for benzodiazepine/GABAA receptors.
    Journal of medicinal chemistry, 1996, Dec-20, Volume: 39, Issue:26

    Topics: Algorithms; Benzodiazepines; Models, Genetic; Nerve Net; Protein Binding; Receptors, GABA-A; Structure-Activity Relationship

1996
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Computational aqueous solubility prediction for drug-like compounds in congeneric series.
    European journal of medicinal chemistry, 2008, Volume: 43, Issue:3

    Topics: Benzodiazepines; Computer Simulation; Crystallography, X-Ray; Databases, Factual; Least-Squares Analysis; Models, Chemical; Organic Chemicals; Pharmaceutical Preparations; Principal Component Analysis; Solubility; Sulfonamides; Water

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Hypnotics today.
    The Practitioner, 1979, Volume: 223, Issue:1336

    Topics: Aged; Anti-Anxiety Agents; Diazepam; Electroencephalography; Humans; Sleep; Sleep Initiation and Maintenance Disorders; Temazepam; Triazolam

1979
Simultaneous determination of diazepam and its metabolies N-desmethyldiazepam, oxydiazepam and oxazepam in plasma and urine of man and dog by means of high-performance liquid chromatography.
    Journal of chromatography, 1979, Apr-11, Volume: 162, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Chromatography, High Pressure Liquid; Diazepam; Dogs; Humans; Nordazepam; Oxazepam; Species Specificity; Temazepam

1979
Diazepam and its hydroxylated metabolites: studies on sleep in healthy man.
    British journal of clinical pharmacology, 1979, Volume: 8, Issue:1

    Topics: Adult; Aging; Diazepam; Humans; Hydroxylation; Male; Middle Aged; Oxazepam; Sleep; Sleep, REM; Temazepam

1979
Rapid recovery from massive diazepam overdose.
    JAMA, 1978, Oct-20, Volume: 240, Issue:17

    Topics: Adult; Biotransformation; Diazepam; Female; Half-Life; Humans; Male; Middle Aged; Nordazepam; Oxazepam; Remission, Spontaneous; Suicide, Attempted; Temazepam; Time Factors

1978
Effect of age on the pharmacokinetics of diazepam given in conjunction with spinal anesthesia.
    Anesthesiology, 1979, Volume: 51, Issue:2

    Topics: Adult; Age Factors; Aged; Anesthesia, Spinal; Body Water; Diazepam; Humans; Kinetics; Middle Aged; Nordazepam; Oxazepam; Temazepam

1979
Performance studies with diazepam and its hydroxylated metabolites.
    British journal of clinical pharmacology, 1979, Volume: 8, Issue:1

    Topics: Barbiturates; Diazepam; Flurazepam; Humans; Hydroxylation; Motor Skills; Oxazepam; Temazepam; Time Factors

1979
Diazepam metabolism by rat and human liver in vitro: inhibition by mephenytoin.
    Xenobiotica; the fate of foreign compounds in biological systems, 1992, Volume: 22, Issue:5

    Topics: Animals; Chromatography, Gas; Diazepam; Humans; Hydroxylation; In Vitro Techniques; Kinetics; Liver; Male; Mephenytoin; Methylation; Nordazepam; Polymorphism, Genetic; Rats; Temazepam

1992
Paranoia in a polypharmacy setting.
    Hospital practice (Office ed.), 1992, Aug-15, Volume: 27, Issue:8

    Topics: Carisoprodol; Diazepam; Drug Therapy, Combination; Ephedrine; Haloperidol; Humans; Ibuprofen; Male; Meprobamate; Middle Aged; Phenylpropanolamine; Psychoses, Substance-Induced; Temazepam

1992
Benzodiazepine requirements during alcohol withdrawal syndrome: clinical implications of using a standardized withdrawal scale.
    Journal of clinical psychopharmacology, 1991, Volume: 11, Issue:5

    Topics: Administration, Oral; Adult; Alcohol Withdrawal Delirium; Anti-Anxiety Agents; Chlordiazepoxide; Diazepam; Hospitalization; Humans; Length of Stay; Lorazepam; Neurologic Examination; Oxazepam; Retrospective Studies; Temazepam; Triazolam

1991
Peripheral-acting benzodiazepines inhibit the growth of human melanoma cells and potentiate the antiproliferative activity of recombinant human interferons.
    Journal of interferon research, 1990, Volume: 10, Issue:3

    Topics: Antineoplastic Agents; Benzodiazepines; Cell Division; Diazepam; Drug Synergism; Humans; Interferon Type I; Interferon-gamma; Interferons; Melanoma; Recombinant Proteins; Structure-Activity Relationship; Temazepam; Tumor Cells, Cultured

1990
Determination of diazepam and nordazepam in milk and plasma in the presence of oxazepam and temazepam.
    Journal of chromatography, 1991, Mar-08, Volume: 564, Issue:1

    Topics: Chromatography, High Pressure Liquid; Diazepam; Flurazepam; Humans; Hydrogen-Ion Concentration; Milk, Human; Nordazepam; Oxazepam; Temazepam

1991
Cytochrome P450IIIA enzymes in rat liver microsomes: involvement in C3-hydroxylation of diazepam and nordazepam but not N-dealkylation of diazepam and temazepam.
    Molecular pharmacology, 1990, Volume: 37, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Cytochrome P-450 Enzyme System; Diazepam; Female; Hydroxylation; Kinetics; Male; Microsomes, Liver; Nordazepam; Oxidoreductases, N-Demethylating; Phenobarbital; Rats; Rats, Inbred Strains; Sex Factors; Species Specificity; Substrate Specificity; Temazepam

1990
Halothane-sparing effect of benzodiazepines in ponies.
    The Cornell veterinarian, 1990, Volume: 80, Issue:3

    Topics: Anesthesia; Animals; Anti-Anxiety Agents; Blood Gas Analysis; Blood Pressure; Diazepam; Female; Halothane; Heart Rate; Horses; Male; Positive-Pressure Respiration; Pulmonary Alveoli; Respiration; Temazepam

1990
Excretion of diazepam and its metabolites in human milk during withdrawal from combination high dose diazepam and oxazepam.
    British journal of clinical pharmacology, 1990, Volume: 29, Issue:1

    Topics: Adult; Diazepam; Drug Combinations; Female; Humans; Infant; Milk, Human; Nordazepam; Oxazepam; Substance Withdrawal Syndrome; Substance-Related Disorders; Temazepam

1990
In vitro drug metabolism and pharmacokinetics of diazepam in cynomolgus monkey hepatocytes during culture for six days.
    Biochemical pharmacology, 1989, Aug-15, Volume: 38, Issue:16

    Topics: Animals; Cells, Cultured; Cytochrome P-450 Enzyme System; Diazepam; Liver; Macaca fascicularis; Male; Models, Biological; Nordazepam; Oxazepam; Oxygenases; Temazepam; Time Factors

1989
The use of benzodiazepines with particular reference to the elderly.
    British journal of hospital medicine, 1986, Volume: 35, Issue:5

    Topics: Aged; Anti-Anxiety Agents; Anxiety; Chlordiazepoxide; Diazepam; Humans; Infusions, Parenteral; Kinetics; Sleep Initiation and Maintenance Disorders; Temazepam; Triazolam

1986
Studies in dental sedation and anaesthesia.
    SAAD digest, 1986, Volume: 6, Issue:8

    Topics: Anesthesia, Dental; Anti-Anxiety Agents; Diazepam; Humans; Midazolam; Temazepam

1986
Oral sedation with temazepam: a practical alternative for use in dentistry?
    British dental journal, 1987, Mar-07, Volume: 162, Issue:5

    Topics: Administration, Oral; Adolescent; Adult; Anesthesia, Dental; Anti-Anxiety Agents; Diazepam; Double-Blind Method; Female; Humans; Injections, Intravenous; Male; Middle Aged; Preanesthetic Medication; Random Allocation; Temazepam; Time Factors

1987
Kinetics of drug action in disease states. XXIV. Pharmacodynamics of diazepam and its active metabolites in rats.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Brain; Diazepam; Female; Nordazepam; Oxazepam; Rats; Rats, Inbred Lew; Reflex; Temazepam

1988
Potencies of diazepam metabolites in rats trained to discriminate diazepam.
    Life sciences, 1986, Jul-07, Volume: 39, Issue:1

    Topics: Animals; Conditioning, Operant; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Male; Nordazepam; Oxazepam; Rats; Rats, Inbred Strains; Temazepam

1986
Microsample determination of diazepam and its three metabolites in serum by reversed-phase high-performance liquid chromatography.
    Journal of chromatography, 1987, Apr-24, Volume: 416, Issue:1

    Topics: Animals; Biotransformation; Chlordiazepoxide; Chromatography, High Pressure Liquid; Diazepam; Hydrogen-Ion Concentration; Indicators and Reagents; Nordazepam; Rats; Spectrophotometry, Ultraviolet; Temazepam

1987
Simultaneous determination of diazepam and its active metabolites in rat serum, brain and cerebrospinal fluid by high-performance liquid chromatography.
    Journal of chromatography, 1987, Nov-27, Volume: 422

    Topics: Animals; Brain Chemistry; Chromatography, High Pressure Liquid; Diazepam; Female; Nordazepam; Oxazepam; Postural Balance; Rats; Rats, Inbred Strains; Temazepam

1987
Imipramine treatment alters the pharmacokinetics and pharmacodynamics of diazepam.
    Journal of pharmaceutical sciences, 1987, Volume: 76, Issue:12

    Topics: Animals; Blood Proteins; Brain Chemistry; Diazepam; Drug Interactions; Imipramine; Liver; Male; Nordazepam; Oxazepam; Pentylenetetrazole; Protein Binding; Rats; Rats, Inbred Strains; Temazepam

1987
Induction of transiently expressed genes in PC-12 pheochromocytoma cells.
    Oncogene, 1987, Volume: 1, Issue:3

    Topics: Animals; Benzodiazepines; Cell Differentiation; Cell Division; Cell Line; Cycloheximide; Dexamethasone; Diazepam; Epidermal Growth Factor; Gene Expression Regulation; Nerve Growth Factors; Pheochromocytoma; Potassium; Rats; RNA, Messenger; Temazepam; Tetradecanoylphorbol Acetate

1987
Liquid-chromatographic assay of diazepam and its major metabolites in serum, and application to pharmacokinetic study of high doses of diazepam in schizophrenics.
    Clinical chemistry, 1985, Volume: 31, Issue:10

    Topics: Administration, Oral; Chromatography, High Pressure Liquid; Diazepam; Female; Humans; Kinetics; Nordazepam; Oxazepam; Schizophrenia; Temazepam

1985
N-desmethyldiazepam physical dependence in dogs.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: Analysis of Variance; Animals; Body Weight; Diazepam; Dogs; Drinking; Energy Intake; Female; Lorazepam; Muscle Spasticity; Nordazepam; Oxazepam; Paresthesia; Substance Withdrawal Syndrome; Temazepam; Time Factors

1985
Determination of some benzodiazepines and metabolites in serum, urine and saliva by high-performance liquid chromatography.
    Journal of chromatography, 1980, Feb-08, Volume: 181, Issue:2

    Topics: Anti-Anxiety Agents; Chromatography, High Pressure Liquid; Diazepam; Humans; Mathematics; Nordazepam; Oxazepam; Saliva; Temazepam

1980
Reaction time to acoustic or visual stimuli after administration of camazepam and diazepam in man.
    Arzneimittel-Forschung, 1980, Volume: 30, Issue:6

    Topics: Acoustic Stimulation; Adult; Anti-Anxiety Agents; Diazepam; Double-Blind Method; Humans; Male; Middle Aged; Photic Stimulation; Reaction Time; Temazepam

1980
Aspects of the interaction of thyroxine and its binding serum proteins with 1,4-benzodiazepine tranquillizers.
    Biochemical medicine, 1981, Volume: 26, Issue:2

    Topics: Anti-Anxiety Agents; Autoradiography; Binding, Competitive; Chlordiazepoxide; Diazepam; Electrophoresis, Polyacrylamide Gel; Humans; Male; Nordazepam; Oxazepam; Temazepam; Thyroxine; Thyroxine-Binding Proteins

1981
Sedation for upper gastrointestinal endoscopy.
    British journal of anaesthesia, 1981, Volume: 53, Issue:12

    Topics: Aged; Anti-Anxiety Agents; Diazepam; Gastroscopy; Humans; Temazepam

1981
Rapid gas chromatographic measurement of diazepam and its metabolites desmethyldiazepam, oxazepam, and 3-hydroxydiazepam (temazepam) in small samples of plasma.
    Therapeutic drug monitoring, 1982, Volume: 4, Issue:3

    Topics: Anti-Anxiety Agents; Biotransformation; Chromatography, Gas; Diazepam; Humans; Nordazepam; Oxazepam; Temazepam

1982
Withdrawal after substitution of a short-acting for a long-acting benzodiazepine.
    JAMA, 1983, Nov-25, Volume: 250, Issue:20

    Topics: Anti-Anxiety Agents; Anxiety; Chronic Disease; Delayed-Action Preparations; Diazepam; Flurazepam; Half-Life; Humans; Oxazepam; Sleep Initiation and Maintenance Disorders; Substance Withdrawal Syndrome; Temazepam

1983
In vitro interaction of diazepam and oxazepam with pancuronium and suxamethonium.
    British journal of anaesthesia, 1984, Volume: 56, Issue:10

    Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; In Vitro Techniques; Muscle Contraction; Neuromuscular Junction; Nordazepam; Oxazepam; Pancuronium; Rats; Rats, Inbred Strains; Succinylcholine; Temazepam

1984
Structure activity relationships of selected benzodiazepines as anticonvulsants to local anesthetics.
    Pharmacology and therapeutics in dentistry, 1980, Volume: 5, Issue:1-2

    Topics: Anesthetics, Local; Animals; Anticonvulsants; Benzodiazepines; Diazepam; Lidocaine; Male; Mepivacaine; Mice; Nitrazepam; Nordazepam; Oxazepam; Prilocaine; Seizures; Structure-Activity Relationship; Temazepam

1980
Systematic review of the benzodiazepines. Guidelines for data sheets on diazepam, chlordiazepoxide, medazepam, clorazepate, lorazepam, oxazepam, temazepam, triazolam, nitrazepam, and flurazepam. Committee on the Review of Medicines.
    British medical journal, 1980, Mar-29, Volume: 280, Issue:6218

    Topics: Benzodiazepines; Chlordiazepoxide; Clorazepate Dipotassium; Diazepam; Flurazepam; Humans; Lorazepam; Medazepam; Nitrazepam; Oxazepam; Safety; Substance Withdrawal Syndrome; Substance-Related Disorders; Temazepam; Triazolam

1980
Development and preliminary application of high-performance liquid chromatographic assay of urinary metabolites of diazepam in humans.
    Journal of chromatography. B, Biomedical applications, 1995, Jun-09, Volume: 668, Issue:1

    Topics: Chromatography, High Pressure Liquid; Diazepam; Humans; Nordazepam; Oxazepam; Reference Values; Reproducibility of Results; Temazepam

1995
Benzodiazepine prescribing and withdrawal for 3234 patients in 15 general practices.
    Family practice, 1994, Volume: 11, Issue:4

    Topics: Adult; Age Factors; Aged; Anti-Anxiety Agents; Diazepam; Drug Prescriptions; Drug Utilization; England; Family Practice; Follow-Up Studies; Humans; Lorazepam; Medical Audit; Nitrazepam; Temazepam

1994
Diazepam metabolism by human liver microsomes is mediated by both S-mephenytoin hydroxylase and CYP3A isoforms.
    British journal of clinical pharmacology, 1994, Volume: 38, Issue:2

    Topics: Aryl Hydrocarbon Hydroxylases; Benzoflavones; Cytochrome P-450 CYP2C19; Cytochrome P-450 CYP2E1; Cytochrome P-450 Enzyme System; Diazepam; Humans; In Vitro Techniques; Isoenzymes; Mephenytoin; Microsomes, Liver; Mixed Function Oxygenases; Nordazepam; Temazepam

1994
Misuse of benzodiazepines. Drug users will shift to another preparation.
    BMJ (Clinical research ed.), 1994, Jun-25, Volume: 308, Issue:6945

    Topics: Capsules; Choice Behavior; Diazepam; Humans; Substance Abuse, Intravenous; Temazepam

1994
Concentration-dependent metabolism of diazepam in mouse liver.
    Journal of pharmacokinetics and biopharmaceutics, 1995, Volume: 23, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Biotransformation; Chromatography, High Pressure Liquid; Computer Simulation; Diazepam; Glucuronates; In Vitro Techniques; Liver; Mice; Microsomes, Liver; Oxidation-Reduction; Temazepam

1995
Benzodiazepine misuse by drug addicts.
    Annals of clinical biochemistry, 1997, Volume: 34 ( Pt 1)

    Topics: Alcoholism; Benzodiazepines; Chromatography, High Pressure Liquid; Diazepam; Humans; Narcotics; Nitrazepam; Nordazepam; Substance-Related Disorders; Temazepam

1997
Application of microdialysis to study the in vitro metabolism of drugs in liver microsomes.
    Journal of pharmaceutical and biomedical analysis, 1997, Volume: 16, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Anti-Arrhythmia Agents; Anti-Inflammatory Agents, Non-Steroidal; Chromatography, High Pressure Liquid; Diazepam; Ibuprofen; Kinetics; Microdialysis; Microsomes, Liver; Nordazepam; Rats; Salicylates; Salicylic Acid; Temazepam

1997
Role of cDNA-expressed human cytochromes P450 in the metabolism of diazepam.
    Biochemical pharmacology, 1998, Mar-15, Volume: 55, Issue:6

    Topics: Cytochrome P-450 Enzyme System; Diazepam; DNA, Complementary; Gene Expression Regulation, Enzymologic; Humans; Isoenzymes; Kinetics; Linear Models; Microsomes, Liver; Nordazepam; Temazepam

1998
Rapid and simple chromatographic method for the determination of diazepam and its major metabolites in human plasma and urine.
    Journal of chromatography. B, Biomedical sciences and applications, 1998, Apr-24, Volume: 708, Issue:1-2

    Topics: Calibration; Chromatography, High Pressure Liquid; Clonazepam; Diazepam; Humans; Nordazepam; Oxazepam; Reference Values; Temazepam

1998
Simultaneous extraction of selected benzodiazepines and benzodiazepine-glucuronides from urine by immunoadsorption.
    Journal of analytical toxicology, 1998, Volume: 22, Issue:5

    Topics: Anti-Anxiety Agents; Diazepam; Glucuronates; Humans; Immunosorbent Techniques; Immunosorbents; Lorazepam; Oxazepam; Temazepam

1998
Sigmoidal kinetic model for two co-operative substrate-binding sites in a cytochrome P450 3A4 active site: an example of the metabolism of diazepam and its derivatives.
    The Biochemical journal, 1999, Jun-15, Volume: 340 ( Pt 3)

    Topics: Adult; Allosteric Regulation; Allosteric Site; Antibodies, Monoclonal; Catalysis; Cell Line; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Diazepam; Dose-Response Relationship, Drug; Female; Humans; Kinetics; Male; Microsomes, Liver; Middle Aged; Mixed Function Oxygenases; Models, Chemical; Nordazepam; Oxidation-Reduction; Temazepam

1999
Stability prediction of amorphous benzodiazepines by calculation of the mean relaxation time constant using the Williams-Watts decay function.
    European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V, 1999, Volume: 48, Issue:1

    Topics: Benzodiazepines; Calorimetry, Differential Scanning; Chemical Phenomena; Chemistry, Physical; Crystallization; Diazepam; Drug Stability; Temazepam; Thermodynamics; Time Factors; Triazolam

1999
Prescribing and dispensing for drug misusers in primary care: current practice in Scotland.
    Family practice, 1999, Volume: 16, Issue:4

    Topics: Analgesics, Opioid; Anti-Anxiety Agents; Codeine; Community Pharmacy Services; Diazepam; Drug Prescriptions; Drug Utilization; Humans; Methadone; Narcotics; Practice Patterns, Physicians'; Primary Health Care; Scotland; Substance-Related Disorders; Surveys and Questionnaires; Temazepam

1999
Identification of benzodiazepines in Artemisia dracunculus and Solanum tuberosum rationalizing their endogenous formation in plant tissue.
    Biochemical and biophysical research communications, 2000, Mar-05, Volume: 269, Issue:1

    Topics: Artemisia; Benzodiazepines; Binding, Competitive; Cerebral Cortex; Chromatography, High Pressure Liquid; Diazepam; Humans; In Vitro Techniques; Mass Spectrometry; Plants, Medicinal; Receptors, GABA-A; Solanum tuberosum; Temazepam

2000
The simultaneous determination of diazepam and its three metabolites in dog plasma by high-performance liquid chromatography with mass spectroscopy detection.
    Journal of pharmaceutical and biomedical analysis, 2001, Volume: 26, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Chromatography, High Pressure Liquid; Diazepam; Dogs; Mass Spectrometry; Nordazepam; Oxazepam; Reproducibility of Results; Temazepam

2001
Drug related deaths in the Strathclyde region of Scotland, 1995-1998.
    Forensic science international, 2001, Oct-15, Volume: 122, Issue:1

    Topics: Adolescent; Adult; Cause of Death; Diazepam; Female; Humans; Incidence; Male; Methadone; Middle Aged; Morphine; Prisoners; Scotland; Substance-Related Disorders; Temazepam

2001
Mechanism of increased dissolution of diazepam and temazepam from polyethylene glycol 6000 solid dispersions.
    International journal of pharmaceutics, 2002, Dec-05, Volume: 249, Issue:1-2

    Topics: Chemistry, Pharmaceutical; Delayed-Action Preparations; Diazepam; Particle Size; Polyethylene Glycols; Solubility; Temazepam

2002
Comparative study of the metabolism of drug substrates by human cytochrome P450 3A4 expressed in bacterial, yeast and human lymphoblastoid cells.
    Xenobiotica; the fate of foreign compounds in biological systems, 2002, Volume: 32, Issue:11

    Topics: Adult; Chromatography, High Pressure Liquid; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Dextromethorphan; Diazepam; Dose-Response Relationship, Drug; Escherichia coli; Excitatory Amino Acid Antagonists; Female; GABA Modulators; Humans; Kinetics; Liver; Lymphocytes; Male; Microsomes, Liver; Midazolam; Middle Aged; Protein Binding; Recombinant Proteins; Saccharomyces cerevisiae; Substrate Specificity; Temazepam

2002
Effects of diazepam and its metabolites on nocturnal melatonin secretion in the rat pineal and Harderian glands. A comparative in vivo and in vitro study.
    Chronobiology international, 2003, Volume: 20, Issue:2

    Topics: Animals; Circadian Rhythm; Diazepam; Harderian Gland; In Vitro Techniques; Male; Melatonin; Nordazepam; Oxazepam; Perfusion; Pineal Gland; Rats; Rats, Wistar; Temazepam

2003
Strain differences in diazepam metabolism at its three metabolic sites in sprague-dawley, brown norway, dark agouti, and wistar strain rats.
    Drug metabolism and disposition: the biological fate of chemicals, 2004, Volume: 32, Issue:9

    Topics: Alcohol Oxidoreductases; Animals; Aryl Hydrocarbon Hydroxylases; Blotting, Western; Chromatography, High Pressure Liquid; Cytochrome P-450 CYP3A; Cytochrome P450 Family 2; Diazepam; Hydroxylation; Immune Sera; Kinetics; Male; Membrane Proteins; Microsomes, Liver; NADP; Polymorphism, Genetic; Rats; Rats, Inbred BN; Rats, Inbred Strains; Rats, Mutant Strains; Rats, Sprague-Dawley; Rats, Wistar; Species Specificity; Steroid 16-alpha-Hydroxylase; Temazepam

2004
Influence of adenosine receptor agonists on benzodiazepine withdrawal signs in mice.
    European journal of pharmacology, 2005, Oct-31, Volume: 523, Issue:1-3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Male; Mice; Pentylenetetrazole; Phenethylamines; Purinergic Agonists; Purinergic P1 Receptor Agonists; Purinergic P2 Receptor Agonists; Seizures; Substance Withdrawal Syndrome; Temazepam

2005
The detection of sedatives in hair and nail samples using tandem LC-MS-MS.
    Forensic science international, 2007, Feb-14, Volume: 166, Issue:1

    Topics: Adult; Aged; Aged, 80 and over; Alprazolam; Azabicyclo Compounds; Benzodiazepines; Chromatography, Liquid; Clobazam; Clonazepam; Diazepam; Female; Forensic Pathology; Hair; Humans; Hypnotics and Sedatives; Male; Mass Spectrometry; Midazolam; Middle Aged; Nails; Oxazepam; Piperazines; Predictive Value of Tests; Rape; Temazepam; Triazolam

2007
Two compartment model of diazepam biotransformation in an organotypical culture of primary human hepatocytes.
    Toxicology and applied pharmacology, 2009, Jan-15, Volume: 234, Issue:2

    Topics: Anti-Inflammatory Agents; Antithyroid Agents; Biotransformation; Cell Separation; Chlorodiphenyl (54% Chlorine); Chromatography, High Pressure Liquid; Cytochrome P-450 Enzyme System; Dexamethasone; Diazepam; Enzyme Induction; Hepatocytes; Humans; Hypnotics and Sedatives; Models, Biological; Models, Statistical; Nordazepam; Organ Culture Techniques; Oxazepam; Phenobarbital; Temazepam

2009
Alleged breaches of "standards of medical care" in a patient overdose death possibly related to chronic opioid analgesic therapy, application of the controlled substances model guidelines: case report.
    Pain medicine (Malden, Mass.), 2009, Volume: 10, Issue:3

    Topics: Adult; Analgesics, Opioid; Anti-Anxiety Agents; Antidepressive Agents, Tricyclic; Diazepam; Doxepin; Drug Overdose; Female; Heroin Dependence; Humans; Hydrocodone; Malpractice; Methadone; Nordazepam; Pain; Pain Measurement; Practice Guidelines as Topic; Shoulder; Shoulder Injuries; Temazepam

2009
Simultaneous analysis of diazepam and its metabolites in rat plasma and brain tissue by HPLC-UV and SPE.
    Talanta, 2009, Nov-15, Volume: 80, Issue:1

    Topics: Animals; Brain; Brain Chemistry; Chromatography, High Pressure Liquid; Diazepam; Nordazepam; Oxazepam; Rats; Reproducibility of Results; Solid Phase Extraction; Spectrophotometry, Ultraviolet; Temazepam

2009
Effects of organic solvents on the time-dependent inhibition of CYP3A4 by diazepam.
    Xenobiotica; the fate of foreign compounds in biological systems, 2010, Volume: 40, Issue:1

    Topics: Acetonitriles; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Diazepam; Dimethyl Sulfoxide; GABA Modulators; Humans; Kinetics; Methanol; Microsomes, Liver; Nordazepam; Solvents; Temazepam

2010
Biotransformation of diazepam in a clinically relevant flat membrane bioreactor model using primary porcine hepatocytes.
    Fundamental & clinical pharmacology, 2011, Volume: 25, Issue:3

    Topics: Adult; Animals; Bioreactors; Biotransformation; Cells, Cultured; Culture Media; Culture Media, Serum-Free; Diazepam; Female; Hepatocytes; Humans; Inactivation, Metabolic; Liver, Artificial; Male; Nordazepam; Oxazepam; Swine; Temazepam; Young Adult

2011
Reduction of temazepam to diazepam and lorazepam to delorazepam during enzymatic hydrolysis.
    Analytical and bioanalytical chemistry, 2011, Volume: 400, Issue:1

    Topics: Benzodiazepines; Chromatography, Liquid; Diazepam; Glucuronidase; Humans; Hydrolysis; Lorazepam; Mass Spectrometry; Nordazepam; Reference Standards; Temazepam

2011
In vitro diazepam metabolism in horses.
    The Japanese journal of veterinary research, 2013, Volume: 61 Suppl

    Topics: Animals; Anti-Anxiety Agents; Cytochrome P-450 Enzyme System; Diazepam; Horses; Male; Microsomes, Liver; Rats; Rats, Sprague-Dawley; Temazepam

2013
Direct determination of diazepam and its glucuronide metabolites in human whole blood by μElution solid-phase extraction and liquid chromatography-tandem mass spectrometry.
    Forensic science international, 2013, Dec-10, Volume: 233, Issue:1-3

    Topics: Chromatography, Liquid; Diazepam; Forensic Toxicology; Humans; Hypnotics and Sedatives; Limit of Detection; Nordazepam; Oxazepam; Reproducibility of Results; Solid Phase Extraction; Tandem Mass Spectrometry; Temazepam

2013
Urinary diazepam metabolite distribution in a chronic pain population.
    Journal of analytical toxicology, 2014, Volume: 38, Issue:3

    Topics: Aryl Hydrocarbon Hydroxylases; Chromatography, High Pressure Liquid; Chronic Pain; Cytochrome P-450 CYP2C19; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Diazepam; Drug Interactions; Esomeprazole; Female; Fluoxetine; Humans; Male; Methadone; Nordazepam; Oxazepam; Retrospective Studies; Specimen Handling; Temazepam

2014
A mixed MDPV and benzodiazepine intoxication in a chronic drug abuser: determination of MDPV metabolites by LC-HRMS and discussion of the case.
    Forensic science international, 2014, Volume: 243

    Topics: Adult; Alprazolam; Benzodiazepines; Benzodioxoles; Chlordiazepoxide; Chromatography, Liquid; Diazepam; Humans; Hypnotics and Sedatives; Male; Mass Spectrometry; Nordazepam; Oxazepam; Psychotropic Drugs; Pyrrolidines; Substance-Related Disorders; Synthetic Cathinone; Temazepam

2014
Low doses of ethanol markedly potentiate the anti-seizure effect of diazepam in a mouse model of difficult-to-treat focal seizures.
    Epilepsy research, 2014, Volume: 108, Issue:10

    Topics: Animals; Anticonvulsants; Brain; Diazepam; Disease Models, Animal; Drug Compounding; Drug Synergism; Electroencephalography; Epilepsy, Temporal Lobe; Ethanol; Female; Kainic Acid; Mice; Nordazepam; Oxazepam; Seizures; Solvents; Temazepam; Water

2014
A comparative study of primary secondary amino (PSA) and multi-walled carbon nanotubes (MWCNTs) as QuEChERS absorbents for the rapid determination of diazepam and its major metabolites in fish samples by high-performance liquid chromatography-electrospray
    Journal of the science of food and agriculture, 2016, Jan-30, Volume: 96, Issue:2

    Topics: Adsorption; Animals; Chromatography, High Pressure Liquid; Diazepam; Fishes; Food Contamination; Nanotubes, Carbon; Nordazepam; Oxazepam; Seafood; Sensitivity and Specificity; Spectrometry, Mass, Electrospray Ionization; Tandem Mass Spectrometry; Temazepam

2016
Characterization of equine cytochrome P450: role of CYP3A in the metabolism of diazepam.
    Journal of veterinary pharmacology and therapeutics, 2016, Volume: 39, Issue:5

    Topics: Animals; Chlorocebus aethiops; COS Cells; Cytochrome P-450 CYP3A; Diazepam; Horses; Hypnotics and Sedatives; Male; Microsomes, Liver; Nordazepam; Oxazepam; Phylogeny; Protein Isoforms; Rats; Rats, Sprague-Dawley; Species Specificity; Temazepam

2016
Deposition of diazepam and its metabolites in hair following a single dose of diazepam.
    International journal of legal medicine, 2017, Volume: 131, Issue:1

    Topics: Adult; Asian People; Chromatography, Liquid; Diazepam; Female; Hair; Healthy Volunteers; Humans; Hypnotics and Sedatives; Male; Nordazepam; Oxazepam; Tandem Mass Spectrometry; Temazepam; Young Adult

2017
Investigation of the effect of mobile phase composition on selectivity using a solvent-triangle based approach in achiral SFC.
    Journal of pharmaceutical and biomedical analysis, 2017, Jan-05, Volume: 132

    Topics: 1-Propanol; Acetonitriles; Benzodiazepines; Chromatography, Supercritical Fluid; Diazepam; Drug Contamination; Ethanol; Furans; Hydrogen Bonding; Lorazepam; Methanol; Multivariate Analysis; Organic Chemicals; Oxazepam; Principal Component Analysis; Reproducibility of Results; Silicon Dioxide; Solvents; Temazepam

2017
Pentobarbital in the context of possible suicides: Analysis of a Case.
    Forensic science international, 2017, Volume: 274

    Topics: Adult; Central Nervous System Depressants; Diazepam; Ethanol; Gastrointestinal Contents; Humans; Male; Nordazepam; Oxazepam; Pentobarbital; Suicide; Temazepam

2017
Difficult to sedate case of acute behavioural disturbance secondary to baclofen withdrawal.
    Emergency medicine Australasia : EMA, 2019, Volume: 31, Issue:3

    Topics: Adult; Antipsychotic Agents; Baclofen; Benzodiazepines; Diazepam; Droperidol; Humans; Male; Problem Behavior; Seizures; Substance Withdrawal Syndrome; Temazepam

2019
Occurrence of Z-drugs, benzodiazepines, and ketamine in wastewater in the United States and Mexico during the Covid-19 pandemic.
    The Science of the total environment, 2023, Jan-20, Volume: 857, Issue:Pt 2

    Topics: Alprazolam; Benzodiazepines; Clonazepam; COVID-19; Diazepam; Humans; Ketamine; Lorazepam; Mexico; Nordazepam; Pandemics; Tandem Mass Spectrometry; Temazepam; United States; Wastewater; Zolpidem

2023