temafloxacin has been researched along with carbostyril in 185 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 11 (5.95) | 18.7374 |
1990's | 171 (92.43) | 18.2507 |
2000's | 3 (1.62) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bale, MJ; Erwin, ME; Gerlach, EH; Jones, RN; Koontz, FP; Murray, PR; Washington, JA | 2 |
Philip, E; Stein, GE | 1 |
Andrews, JM; Ashby, JP; Baldwin, DR; Honeybourne, D; Wise, R | 1 |
Erwin, ME; Jones, RN | 1 |
Erwin, ME; Gerlach, EH; Jones, RN; Koontz, FP; Murray, PR; Washington, JA | 1 |
Finegold, SM; Molitoris, E; Wexler, HM | 1 |
Fenoll, A; López de Felipe, F; Martínez-Suárez, JV; Rodríguez-Tudela, JL | 1 |
Aubert, G; Dorche, G; Pozzetto, B | 3 |
Barry, AL; Fuchs, PC; Pfaller, MA | 1 |
Carpentier, P; Granneman, GR; Morrison, PJ; Pernet, AG | 2 |
Bergogne-Bérézin, E; Joly-Guillou, ML | 1 |
Arai, S; Gohara, Y; Kawashima, T; Kuwano, K; Matsu-Ura, I | 1 |
Hornstein, LE | 1 |
Ganiats, TG; Norcross, WA | 1 |
Coles, S; Millar, E; Nimmo, W; Wyld, P | 1 |
Granneman, GR | 1 |
Fabian, W; Granneman, GR; Kinzig, M; Kirch, W; Locke, C; Mahr, G; Naber, KG; Nickel, P; Sörgel, F | 1 |
Fabian, W; Granneman, GR; Kujath, P; Mahr, G; Nickel, P; Sörgel, F | 1 |
Lubowski, TJ; Nightingale, CH; Quintiliani, R; Sweeney, K | 1 |
Granneman, GR; Mukherjee, D | 1 |
Sörgel, F | 1 |
Granneman, GR; Mahr, G; Muth, P; Nickel, P; Sörgel, F; Stephan, U | 1 |
Granneman, GR; Locke, C; Sörgel, F; Stephan, U | 1 |
Birner, B; Granneman, GR; Mukherjee, D; Sörgel, F; Stephan, U | 1 |
Fuhr, U; Granneman, GR; Kinzig, M; Mahr, G; Muth, P; Nickel, P; Patterson, K; Sörgel, F; Stephan, U | 1 |
Mant, T; Millar, E; Morrison, P | 1 |
Hammerschlag, MR; Hyman, CL; Roblin, PM | 1 |
Garcia, I; Pascual, A; Perea, EJ | 1 |
Carbon, C; Chauvin, JP; Hazebroucq, J; Léophonte, P; Petitpretz, P | 1 |
Appelbaum, PC; Jacobs, MR; Spangler, SK | 1 |
Chuah, SK; Gollapudi, S; Hajji, M; Perumal, VK; Thadepalli, H | 1 |
Cummings, M; Glatt, AE; McCormack, W | 1 |
Appelbaum, PC; Jacobs, MR; Shiman, R; Spangler, SK | 1 |
Citron, DM; Goldstein, EJ | 2 |
Nix, DE; Symonds, WT | 1 |
Azoulay-Dupuis, E; Bauchet, J; Pocidalo, JJ; Vallée, E | 1 |
Bresler, L; Didelot, JP; Hazebroucq, J; Jehl, F; Koechlin, C; Merle-Melet, M | 1 |
Barrett, MS; Jones, RN | 1 |
Carnegie, CM; Lindsay, G; Scorer, HJ | 1 |
Bouvet, A; Carbon, C; Cremieux, AC; Devine, C; Maziere, B; Muffat-Joly, M; Pocidalo, JJ; Saleh-Mghir, A; Vallois, JM | 1 |
al-Wali, WI; Douglas, CW; Spencer, RC; Wilcox, MH; Winstanley, TG | 1 |
Allen, SD; Baker, CN; Barry, AL; Fuchs, PC; Hardy, DJ; Jorgensen, JH; McLaughlin, JC | 1 |
Järhult, B | 1 |
Cynamon, MH; DeStefano, MS; Klemens, SP | 1 |
Gelber, RH; Iranmanesh, A; Murray, L; Siu, P; Tsang, M | 1 |
Arakawa, S; Kamidono, S | 1 |
Almodovar, E; Burns, JJ; Qadri, SM; Rabea, N; Ueno, Y | 1 |
Gootz, TD; Martin, BA | 1 |
Bollet, C; de Micco, P; Gevaudan, MJ; Mallet, MN | 2 |
Gikas, A; Grosset, J; Perronne, C; Pocidalo, JJ; Truffot-Pernot, C; Vilde, JL | 1 |
Forstall, GJ; Knapp, CC; Washington, JA | 1 |
Bethune, L; King, A; Phillips, I | 2 |
Chodosh, S | 2 |
Davey, PG | 1 |
Parish, LC; Witkowski, JA | 1 |
Neldner, KH | 1 |
Jungkind, DL; Parish, LC | 1 |
Hardy, DJ | 2 |
Iravani, A | 2 |
Cox, CE | 1 |
Childs, SJ; Cox, CE | 1 |
Mogabgab, WJ | 1 |
Fuchs, PC | 1 |
Segreti, J | 2 |
Pernet, AG | 1 |
Pankey, GA | 1 |
Appelbaum, PC | 1 |
Jacobs, MR | 1 |
Krasula, RW; Pernet, AG | 1 |
Giardina, WJ | 1 |
Kinzig, M; Mahr, G; Muth, P; Naber, KG; Sorgel, F | 1 |
Wise, R | 1 |
Granneman, GR; Guay, DR | 1 |
Callens, E; Chauvin, JP; Hazebroucq, J; Ruff, F; Santais, MC | 1 |
Granneman, GR; Varga, LL | 1 |
Barry, AL; Fuchs, PC | 3 |
Norrby, SR; Pernet, AG | 1 |
Ball, P | 1 |
Amsterdam, D; Beam, TR; Gorzynski, EA; Lawrence, T; Mandell, LA; Rotstein, C | 1 |
Finegold, SM; Molitoris, E; Reeves, D; Wexler, HM | 1 |
Azoulay-Dupuis, E; Bergogne-Bérézin, E; Pocidalo, JJ; Vallée, E | 1 |
Azoulay-Dupuis, E; Bedos, JP; Pocidalo, JJ; Vallée, E | 1 |
Dudley, MN | 1 |
Andrews, JM; Baldwin, DR; Honeybourne, D; Wise, R | 1 |
Kosmidis, J | 1 |
Lode, H; Vogel, F | 1 |
Bischoff, W; Blenk, H; Boerema, JB; Carpentier, P; Focht, J; Naber, KG; Sylvester, J | 1 |
Bille, J; Glauser, MP | 1 |
Conejo, MC; García, I; Pascual, A; Perea, EJ | 1 |
Acar, J; Baquero, F; Bergan, T; Forsgren, A; Phillips, I; Wiedemann, B | 1 |
Pattyn, SR | 1 |
Braeckman, R; Craft, JC; Granneman, GR; Kraut, J; Shupien, S | 1 |
Chu, DT; Giardina, WJ; Hardy, DJ; Nordeen, CW; Pernet, AG; Plattner, JJ; Swanson, RN | 1 |
Adler, LP; Bednarczyk, EM; Berridge, MS; Green, JA; Leisure, GA; Little, D; Miraldi, FD; Nelson, AD; Panacek, EA | 1 |
Brun, Y; Chanal, M; Courtieu, AL; Dabernat, H; Derlot, E; Joly-Guillou, ML; Kitzis, MD; Meyran, M; Morel, C; Soussy, CJ | 1 |
Blickle, JF; Brogard, JM; Dorner, M; Jehl, F; Koechlin, C; Monteil, H; Westphal, JF | 1 |
Back, DJ; Mant, T; Martin, C; Millar, E; Morrison, P; Orme, M; Tjia, J | 1 |
Azoulay-Dupuis, E; Bedos, JP; Hardy, DJ; Pocidalo, JJ; Swanson, RN; Vallée, E | 1 |
Bottolfsen, KL; Digranes, A; Hardardottir, H | 1 |
Chu, DT; Clement, JJ; Hardy, DJ; Shipkowitz, NL; Swanson, RN | 1 |
Elrod, L; Linton, CL; Shelat, BP; Wong, CF | 1 |
Andrews, JM; Ashby, JP; Cooper, MA; Matthews, RS; Wise, R | 1 |
Blicklé, JF; Brogard, JM; Dorner, M; Jehl, F; Koechlin, C; Westphal, JF | 1 |
Cremers, HM; Davies, BI; Gubbelmans, HL; Maesen, FP | 1 |
Bassanetti, I; Ceralli, M; Giardini, R; Reggio, S; Sansonetti, G | 1 |
Inoue, K; Inoue, M; Mitsuhashi, S; Nakanishi, N; Yamaguchi, T | 1 |
Hendrickx, AG; Lasley, BL; Lehrer, SB; Tarantal, AF | 1 |
Bauer, JF; Elrod, L; Fornnarino, JR; Heathcote, DE; Krogh, SK; Linton, CL; Norris, BJ; Quick, JE | 1 |
Bryan, JP; Krieg, RE; Perine, PL; Sheffield, J; Wagner, K; Waters, C | 1 |
Andrews, JM; Ashby, JP; Baldwin, DR; Honeybourne, D; Wilkinson, L; Wise, R | 1 |
Hessen, MT; Kaye, D; Pitsakis, PG | 1 |
Jehl, F; Koechlin, C; Linger, L; Monteil, H | 1 |
Allen, W; Gorzynski, EA; Gutman, SI | 1 |
Barry, AL; Jones, RN | 2 |
Kapell, KS; Kessler, HA; Segreti, J; Trenholme, GM | 1 |
Goodman, LJ; Kaplan, RL; Nelson, JA; Segreti, J; Trenholme, GM | 1 |
Andrews, JM; Ashby, JP; Nye, K; Shi, YG; Wise, R | 1 |
Chin, NX; Figueredo, VM; Neu, HC; Novelli, A | 1 |
Bodey, GP; Gooch, G; Ho, DH; LeBlanc, B; Rolston, KV | 1 |
Fernandes, PB; Swanson, RN | 1 |
Bower, RR; Chu, DT; Fernandes, PB; Hanson, CW; Hardy, DJ; Hensey, DM; Ramer, NR; Swanson, RN | 1 |
Cagni, A; Chuard, C; Lew, DP; Schrenzel, J; Vaudaux, PE | 1 |
Davey, P; McDonald, T | 1 |
Lietman, PS; Norrby, SR | 1 |
Kaatz, GW; Larsson, AJ; Moody, JA; Rotschafer, JC; Walker, KJ; Zabinski, RA | 1 |
Sanders, CC; Thomson, KS | 2 |
Aoki, M; Goldstein, E; Kunii, O; Ono, Y | 1 |
Chin, NX; Neu, HC | 1 |
Arakawa, S; Ban, Y; Hirose, T; Ito, Y; Kamidono, S; Kawada, Y; Kumamoto, Y; Kumon, H; Ohmori, H; Suzuki, K | 1 |
Forsgren, A; Riesbeck, K | 1 |
Gale, E; Maguire, RB; Stroncek, DF; Yearlsey, M | 1 |
Carbon, C; Cremieux, AC; Jambou, R; Mghir, AS; Muffat-Joly, M; Pocidalo, JJ | 1 |
Blum, MD; Graham, DJ; McCloskey, CA | 1 |
Kondo, K; Nakashima, M; Uematsu, T; Umemura, K; Yamaguchi, T; Yano, S | 1 |
Fine, DH | 1 |
Dudley, MN; Gilbert, D; Marchbanks, CR; McGrath, BJ | 1 |
Cartwright, FD; Kenny, GE | 1 |
Phillips, I; Power, EG | 1 |
Gage, TW | 1 |
Krinke, AJ; Moody, JA; Rotschafer, JC; Vance-Bryan, K; Walker, KJ; Zabinski, RA | 1 |
Foleno, BD; Fu, KP; Lafredo, SC | 1 |
Akashi, A; Arai, S; Gohara, Y; Kuwano, K; Nishimoto, M; Oizumi, K; Takeda, K; Yamaguchi, T; Yano, T | 1 |
Finch, RG | 1 |
Eliopoulos, GM; Ferraro, MJ; Malanoski, GJ; Moellering, RC | 1 |
Ikerd, TR; Koletar, SL | 1 |
Deamer, RL; Heming, D; James, RE; Koenker, N; Prichard, JG | 1 |
Patel, S; Southern, PM | 1 |
Brown, WJ; Moosavi, S | 1 |
Cho, N; Matsuda, S; Okada, H; Shimizu, T | 1 |
Hendrickx, AG; Hummler, H; Richter, WF | 1 |
Lietman, PS | 1 |
Iakovlev, SV; Iakovlev, VP; Izotova, GN | 1 |
Muñiz, AE | 1 |
Banno, K; Matsuoka, M; Sato, T | 1 |
Goldstein, EJ | 1 |
Morrissey, I | 1 |
Baumann-Wilschke, I; Förster, C; Rücker, M; Shakibaei, M; Stahlmann, R; Vormann, J | 1 |
Peters, G; Schumacher-Perdreau, F | 1 |
Baker, WR; Devasthale, PV; Frank, KE; Gentry, EJ; Keschavarz-Shokri, A; Mitscher, LA; Nilius, A; Ravikumar, VT; Shawar, R; Shen, LL | 1 |
Baumann-Wilschke, I; Rücker, M; Shakibaei, M; Stahlmann, R | 1 |
Fukuda, H; Kawamura, Y | 1 |
Gonoi, T; Saraya, A; Seino, S; Yokokura, M | 1 |
19 review(s) available for temafloxacin and carbostyril
Article | Year |
---|---|
Pharmacokinetics of temafloxacin after multiple oral administration.
Topics: Administration, Oral; Adult; Anti-Infective Agents; Double-Blind Method; Drug Administration Schedule; Fluoroquinolones; Humans; Middle Aged; Quinolones | 1992 |
Penetration of temafloxacin into body tissues and fluids.
Topics: Administration, Oral; Anti-Infective Agents; Fluoroquinolones; Humans; Quinolones; Tissue Distribution | 1992 |
Lomefloxacin and temafloxacin: two new fluoroquinolone antimicrobials.
Topics: Anti-Infective Agents; Bacteria; Bacterial Infections; Drug Interactions; Drug Resistance, Microbial; Fluoroquinolones; Humans; Quinolones | 1992 |
Temafloxacin as prophylactic agent in neutropenic patients.
Topics: Anti-Infective Agents; Fluoroquinolones; Humans; Neutropenia; Quinolones; Sepsis | 1992 |
Systemic management of cutaneous bacterial infections.
Topics: Anti-Infective Agents; Bacterial Infections; Fluoroquinolones; Humans; Quinolones; Skin Diseases, Infectious | 1991 |
Temafloxacin: an overview.
Topics: Anti-Infective Agents; Bacterial Infections; Fluoroquinolones; Humans; Male; Microbial Sensitivity Tests; Prostatitis; Quinolones; Respiratory Tract Infections; Sexually Transmitted Diseases, Bacterial; Skin Diseases, Infectious; Urinary Tract Infections | 1991 |
Evaluation of the bactericidal activity of temafloxacin.
Topics: Anti-Infective Agents; Bacteria; Fluoroquinolones; Microbial Sensitivity Tests; Quinolones | 1991 |
Comparative pharmacokinetics of ciprofloxacin and temafloxacin in humans: a review.
Topics: Aging; Anti-Infective Agents; Ciprofloxacin; Drug Interactions; Fluoroquinolones; Humans; Kidney Diseases; Liver Diseases; Quinolones; Tissue Distribution | 1991 |
Comparative penetration of selected fluoroquinolones into respiratory tract fluids and tissues.
Topics: Anti-Infective Agents; Bronchi; Ciprofloxacin; Epithelium; Fluoroquinolones; Humans; Macrophages, Alveolar; Mucous Membrane; Quinolones; Respiratory System | 1991 |
Use of quinolones for the treatment of acute exacerbations of chronic bronchitis.
Topics: Acute Disease; Anti-Infective Agents; Bronchitis; Chronic Disease; Ciprofloxacin; Fluoroquinolones; Humans; Ofloxacin; Quinolones | 1991 |
The role of temafloxacin in the community setting: an overview.
Topics: Anti-Infective Agents; Fluoroquinolones; Humans; Quinolones | 1991 |
A review of the pharmacokinetic profile of temafloxacin.
Topics: Anti-Infective Agents; Fluoroquinolones; Humans; Quinolones | 1991 |
Postmarketing surveillance of quinolones, 1990 to 1992.
Topics: Adverse Drug Reaction Reporting Systems; Anti-Bacterial Agents; Anti-Infective Agents; Databases, Factual; Fluoroquinolones; Hospitalization; Humans; Quinolones; Risk Factors | 1993 |
Safety and tolerability of fluoroquinolones.
Topics: Adverse Drug Reaction Reporting Systems; Animals; Anti-Infective Agents; Dermatitis, Phototoxic; Drug Tolerance; Fluoroquinolones; Humans; Quinine; Quinolones; Safety | 1993 |
Temafloxacin syndrome: review of 95 cases.
Topics: Adult; Adverse Drug Reaction Reporting Systems; Aged; Aged, 80 and over; Anemia, Hemolytic; Anti-Infective Agents; Female; Fluoroquinolones; Hemolysis; Humans; Male; Middle Aged; Quinolones | 1994 |
Fluoroquinolone toxicities. An update.
Topics: Anti-Infective Agents; Dermatitis, Phototoxic; Fluoroquinolones; Humans; Joint Diseases; Nervous System Diseases; Quinolones | 1995 |
[Pharmacokinetics of fluoroquinolones in patients with renal insufficiency].
Topics: Anti-Infective Agents; Ciprofloxacin; Fluoroquinolones; Humans; Ofloxacin; Pefloxacin; Quinolones; Renal Insufficiency | 1995 |
An unlikely childhood overdose: temafloxacin.
Topics: Animals; Anti-Infective Agents; Child, Preschool; Drug Overdose; Female; Fluoroquinolones; Humans; Quinolones; Urinary Tract Infections | 1996 |
Possible role for the new fluoroquinolones (levofloxacin, grepafloxacin, trovafloxacin, clinafloxacin, sparfloxacin, and DU-6859a) in the treatment of anaerobic infections: review of current information on efficacy and safety.
Topics: Anti-Infective Agents; Bacteria, Anaerobic; Bacterial Infections; Fluoroquinolones; Humans; Levofloxacin; Naphthyridines; Ofloxacin; Piperazines; Quinolones; Safety; Syndrome | 1996 |
31 trial(s) available for temafloxacin and carbostyril
Article | Year |
---|---|
Comparison of three-day temafloxacin with seven-day ciprofloxacin treatment of urinary tract infections in women.
Topics: Adult; Aged; Anti-Infective Agents; Ciprofloxacin; Female; Fluoroquinolones; Humans; Middle Aged; Quinolones; Urinary Tract Infections | 1992 |
Pharmacokinetics of temafloxacin in patients with liver impairment.
Topics: Adult; Aged; Anti-Infective Agents; Chromatography, High Pressure Liquid; Female; Fluoroquinolones; Humans; Kidney; Liver; Liver Cirrhosis; Male; Middle Aged; Quinolones | 1992 |
The relative bioavailability of temafloxacin administered through a nasogastric tube with and without enteral feeding.
Topics: Administration, Oral; Adult; Anti-Infective Agents; Biological Availability; Enteral Nutrition; Fluoroquinolones; Humans; Male; Middle Aged; Quinolones | 1992 |
Effects of 2 quinolone antibacterials, temafloxacin and enoxacin, on theophylline pharmacokinetics.
Topics: Administration, Oral; Adult; Aminophylline; Anti-Infective Agents; Double-Blind Method; Drug Interactions; Enoxacin; Fluoroquinolones; Humans; Injections, Intravenous; Male; Quinolones; Theophylline | 1992 |
Effect of cimetidine on the pharmacokinetics of temafloxacin.
Topics: Administration, Oral; Anti-Infective Agents; Cimetidine; Drug Interactions; Female; Fluoroquinolones; Humans; Male; Quinolones | 1992 |
Effect of antacid medication on the pharmacokinetics of temafloxacin.
Topics: Adult; Antacids; Anti-Infective Agents; Drug Interactions; Female; Fluoroquinolones; Humans; Male; Quinolones | 1992 |
Effects of temafloxacin and ciprofloxacin on the pharmacokinetics of caffeine.
Topics: Adult; Anti-Infective Agents; Caffeine; Ciprofloxacin; Double-Blind Method; Drug Interactions; Female; Fluoroquinolones; Humans; Male; Quinolones | 1992 |
Efficacy and safety of temafloxacin versus those of amoxicillin in hospitalized adults with community-acquired pneumonia.
Topics: Administration, Oral; Adult; Aged; Amoxicillin; Anti-Infective Agents; Bacteria; Double-Blind Method; Female; Fluoroquinolones; Humans; Male; Middle Aged; Pneumonia; Quinolones | 1992 |
Safety and efficacy of temafloxacin versus ciprofloxacin in lower respiratory tract infections: a randomized, double-blind trial.
Topics: Adolescent; Adult; Aged; Aged, 80 and over; Anti-Infective Agents; Bacteria; Ciprofloxacin; Double-Blind Method; Drug Interactions; Female; Fluoroquinolones; Humans; Male; Middle Aged; Prospective Studies; Quinolones; Respiratory Tract Infections; Theophylline | 1992 |
Assessment of the UTI criteria for bacterial prostatitis in Japan.
Topics: Acute Disease; Administration, Oral; Adolescent; Adult; Aged; Anti-Infective Agents; Bacterial Infections; Chronic Disease; Fluoroquinolones; Humans; Male; Middle Aged; Prostatitis; Quinolones; Treatment Outcome | 1992 |
Temafloxacin compared with ciprofloxacin in mild to moderate lower respiratory tract infections in ambulatory patients. A multicenter, double-blind, randomized study.
Topics: Ambulatory Care; Anti-Infective Agents; Ciprofloxacin; Double-Blind Method; Female; Fluoroquinolones; Humans; Lung Diseases, Obstructive; Male; Microbial Sensitivity Tests; Middle Aged; Pneumonia; Quinolones; Respiratory Tract Infections | 1991 |
Efficacy of temafloxacin versus ciprofloxacin or amoxicillin for lower respiratory tract infections in smokers and the elderly.
Topics: Age Factors; Aged; Amoxicillin; Anti-Infective Agents; Ciprofloxacin; Double-Blind Method; Female; Fluoroquinolones; Humans; Male; Quinolones; Respiratory Tract Infections; Smoking | 1991 |
Double-blind randomized study of oral temafloxacin and cefadroxil in patients with mild to moderately severe bacterial skin infections.
Topics: Adolescent; Adult; Aged; Aged, 80 and over; Anti-Infective Agents; Cefadroxil; Double-Blind Method; Female; Fluoroquinolones; Humans; Male; Middle Aged; Quinolones; Skin Diseases, Infectious; Staphylococcal Skin Infections; Streptococcal Infections | 1991 |
Systemic antimicrobial therapy in skin and skin structure infections: comparison of temafloxacin and ciprofloxacin.
Topics: Adolescent; Adult; Aged; Aged, 80 and over; Anti-Infective Agents; Bacterial Infections; Ciprofloxacin; Double-Blind Method; Female; Fluoroquinolones; Humans; Male; Middle Aged; Quinolones; Skin Diseases, Infectious | 1991 |
Treatment of uncomplicated urinary tract infections with temafloxacin.
Topics: Adult; Anti-Infective Agents; Double-Blind Method; Female; Fluoroquinolones; Humans; Quinolones; Urinary Tract Infections | 1991 |
Oral temafloxacin compared to norfloxacin for the treatment of complicated urinary tract infections.
Topics: Administration, Oral; Adolescent; Adult; Aged; Aged, 80 and over; Anti-Infective Agents; Double-Blind Method; Female; Fluoroquinolones; Humans; Male; Middle Aged; Norfloxacin; Quinolones; Urinary Tract Infections | 1991 |
Treatment of chronic bacterial prostatitis with temafloxacin.
Topics: Adult; Aged; Anti-Infective Agents; Bacterial Infections; Double-Blind Method; Fluoroquinolones; Humans; Male; Middle Aged; Prostatitis; Quinolones | 1991 |
Single-dose oral temafloxacin versus parenteral ceftriaxone in the treatment of gonococcal urethritis/cervicitis.
Topics: Administration, Oral; Adolescent; Adult; Aged; Anti-Infective Agents; Ceftriaxone; Female; Fluoroquinolones; Gonorrhea; Humans; Injections, Intramuscular; Male; Middle Aged; Quinolones; Urethritis; Uterine Cervicitis | 1991 |
Assessment of adverse events during drug development: experience with temafloxacin.
Topics: Aged; Anti-Infective Agents; Drug Evaluation; Female; Fluoroquinolones; Humans; Male; Quinolones | 1991 |
A double-blind study of once-daily temafloxacin in the treatment of bacterial lower respiratory tract infections.
Topics: Adolescent; Adult; Anti-Infective Agents; Bronchitis; Ciprofloxacin; Double-Blind Method; Female; Fluoroquinolones; Humans; Male; Pneumonia; Quinolones; Respiratory Tract Infections | 1991 |
The use of oral temafloxacin compared with a parenteral cephalosporin in hospitalized patients with pneumonia.
Topics: Administration, Oral; Adolescent; Adult; Aged; Anti-Infective Agents; Cefotaxime; Female; Fluoroquinolones; Humans; Injections, Intravenous; Male; Middle Aged; Pneumonia; Quinolones | 1991 |
An assessment of temafloxacin in the treatment of chronic bacterial prostatitis.
Topics: Administration, Oral; Anti-Infective Agents; Chronic Disease; Fluoroquinolones; Humans; Male; Prostatitis; Quinolones | 1991 |
Comparison of the effect of temafloxacin, ciprofloxacin, or placebo on cerebral blood flow, glucose, and oxygen metabolism in healthy subjects by means of positron emission tomography.
Topics: Adolescent; Adult; Anti-Infective Agents; Brain; Cerebrovascular Circulation; Ciprofloxacin; Deoxyglucose; Double-Blind Method; Fluoroquinolones; Glucose; Humans; Male; Oxygen; Placebos; Prospective Studies; Quinolones; Reference Values; Tomography, Emission-Computed | 1991 |
[In vitro antibacterial activity of a new fluoroquinolone, temafloxacin, against hospital isolates. Results of a multicenter study].
Topics: 4-Quinolones; Acinetobacter; Anti-Infective Agents; Bacteria, Anaerobic; Dose-Response Relationship, Drug; Enterobacteriaceae; Fluoroquinolones; Haemophilus; Humans; In Vitro Techniques; Neisseria; Pseudomonas; Quinolones; Staphylococcus; Streptococcus | 1991 |
The lack of interaction between temafloxacin and combined oral contraceptive steroids.
Topics: 4-Quinolones; Adult; Anti-Infective Agents; Contraceptives, Oral, Combined; Drug Interactions; Ethinyl Estradiol; Female; Fluoroquinolones; Follicle Stimulating Hormone; Humans; Levonorgestrel; Luteinizing Hormone; Norgestrel; Progesterone; Quinolones; Radioimmunoassay | 1991 |
Comparative, double-blind, prospective, multicenter trial of temafloxacin versus trimethoprim-sulfamethoxazole in uncomplicated urinary tract infections in women.
Topics: 4-Quinolones; Adult; Anti-Infective Agents; Double-Blind Method; Female; Fluoroquinolones; Humans; Middle Aged; Prospective Studies; Quinolones; Trimethoprim, Sulfamethoxazole Drug Combination; Urinary Tract Infections | 1991 |
Pharmacokinetics of temafloxacin in humans after single oral doses.
Topics: 4-Quinolones; Administration, Oral; Adult; Anti-Infective Agents; Blood Proteins; Chromatography, High Pressure Liquid; Double-Blind Method; Fluoroquinolones; Half-Life; Humans; Male; Quinolones; Random Allocation | 1991 |
Temafloxacin in acute purulent exacerbations of chronic bronchitis.
Topics: 4-Quinolones; Anti-Infective Agents; Bronchitis; Chronic Disease; Drug Administration Schedule; Fluoroquinolones; Haemophilus influenzae; Humans; Moraxella catarrhalis; Pseudomonas aeruginosa; Quinolones; Sputum; Streptococcus pneumoniae | 1990 |
[Re-examination of the criteria for clinical evaluation on bacterial prostatitis--analysis of the data of the clinical study of temafloxacin].
Topics: Acute Disease; Adolescent; Adult; Aged; Anti-Infective Agents; Bacterial Infections; Chronic Disease; Fluoroquinolones; Humans; Male; Middle Aged; Prostatitis; Quinolones | 1994 |
[Experimental and clinical studies of temafloxacin in the field of obstetrics and gynecology].
Topics: Administration, Oral; Adolescent; Adult; Aged; Anti-Infective Agents; Bacteria; Bacterial Infections; Female; Fluoroquinolones; Genital Diseases, Female; Genitalia, Female; Humans; Middle Aged; Quinolones | 1993 |
Analytical chiral separation of a new quinolone compound in biological fluids by high-performance liquid chromatography.
Topics: Anti-Infective Agents; Calibration; Chromatography, High Pressure Liquid; Fluoroquinolones; Half-Life; Humans; Hydrogen-Ion Concentration; Indicators and Reagents; Quinolones; Spectrophotometry, Ultraviolet; Stereoisomerism | 1996 |
135 other study(ies) available for temafloxacin and carbostyril
Article | Year |
---|---|
MIC quality control guidelines for Haemophilus susceptibility tests using cefdinir (FK482), cefepime, cefetamet, cefpirome, ceftibuten, fleroxacin, temafloxacin, clarithromycin, RP59500, and trospectomycin.
Topics: Anti-Bacterial Agents; Cefdinir; Cefpirome; Ceftibuten; Ceftizoxime; Cephalosporins; Clarithromycin; Erythromycin; Fleroxacin; Fluoroquinolones; Haemophilus; Humans; Microbial Sensitivity Tests; Quality Control; Quinolones; Spectinomycin; Virginiamycin | 1992 |
Studies show new macrolide antibiotics to be superior to some older agents.
Topics: Anti-Bacterial Agents; Anti-Infective Agents; Bacterial Infections; Clarithromycin; Drug Administration Schedule; Erythromycin; Fluoroquinolones; Humans; Quinolones | 1992 |
Disk diffusion quality control guidelines for Haemophilus susceptibility tests using cefdinir, CI-960, fleroxacin, temafloxacin, and trospectomycin.
Topics: Anti-Bacterial Agents; Cefdinir; Cephalosporins; Fleroxacin; Fluoroquinolones; Haemophilus influenzae; Microbial Sensitivity Tests; Quality Control; Quinolones; Spectinomycin | 1992 |
The distribution of temafloxacin in bronchial epithelial lining fluid, alveolar macrophages and bronchial mucosa.
Topics: Anti-Infective Agents; Bronchi; Bronchoalveolar Lavage Fluid; Bronchoscopy; Female; Fluoroquinolones; Humans; Macrophages, Alveolar; Male; Middle Aged; Mucous Membrane; Quinolones; Tissue Distribution | 1992 |
Oral temafloxacin approved for U.S. market.
Topics: Administration, Oral; Anti-Infective Agents; Bacterial Infections; Fluoroquinolones; Humans; Quinolones; United States; United States Food and Drug Administration | 1992 |
Interpretive criteria for susceptibility testing of CI-960 (PD127391, AM-1091), fleroxacin, lomefloxacin, and temafloxacin against Neisseria gonorrhoeae, including drug stability in GC agar medium.
Topics: Agar; Anti-Infective Agents; Drug Stability; Fleroxacin; Fluoroquinolones; Microbial Sensitivity Tests; Neisseria gonorrhoeae; Quinolones | 1992 |
MIC and disk diffusion quality control guidelines for Neisseria gonorrhoeae susceptibility tests of cefdinir, cefetamet, CI-960, fleroxacin, lomefloxacin, and temafloxacin.
Topics: Anti-Infective Agents; Cefdinir; Ceftizoxime; Cephalosporins; Diffusion; Fleroxacin; Fluoroquinolones; Microbial Sensitivity Tests; Neisseria gonorrhoeae; Quality Control; Quinolones | 1992 |
In vitro activities of three of the newer quinolones against anaerobic bacteria.
Topics: Anti-Infective Agents; Bacteria, Anaerobic; Fluoroquinolones; Microbial Sensitivity Tests; Quinolones | 1992 |
Comparative in-vitro activity of four peptide antibiotics against penicillin-resistant Streptococcus pneumoniae isolated from cerebrospinal fluid (CSF).
Topics: Anti-Bacterial Agents; Anti-Infective Agents; Cerebrospinal Fluid; Daptomycin; Erythromycin; Fluoroquinolones; Glycopeptides; Humans; Microbial Sensitivity Tests; Penicillin Resistance; Peptides; Quinolones; Serotyping; Streptococcus pneumoniae; Teicoplanin; Vancomycin | 1992 |
Emergence of quinolone-imipenem cross-resistance in Pseudomonas aeruginosa after fluoroquinolone therapy.
Topics: Anti-Infective Agents; Drug Resistance, Microbial; Drug Therapy, Combination; Fluoroquinolones; Humans; Imipenem; Microbial Sensitivity Tests; Mutation; Naphthyridines; Norfloxacin; Pseudomonas aeruginosa; Pseudomonas Infections; Quinolones | 1992 |
Two new fluoroquinolones.
Topics: Anti-Infective Agents; Clinical Trials as Topic; Drug Interactions; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Quinolones; Respiratory Tract Infections; Urinary Tract Infections | 1992 |
Spontaneously occurring staphylococcal mutants resistant to clinically achievable concentrations of ciprofloxacin and temafloxacin.
Topics: Anti-Infective Agents; Ciprofloxacin; Drug Resistance, Microbial; Fluoroquinolones; Microbial Sensitivity Tests; Mutation; Quinolones; Staphylococcus aureus; Staphylococcus epidermidis | 1992 |
Pharmacokinetics of temafloxacin in humans after multiple oral doses.
Topics: Administration, Oral; Adult; Anti-Infective Agents; Chromatography, High Pressure Liquid; Circadian Rhythm; Fluoroquinolones; Glomerular Filtration Rate; Half-Life; Humans; Male; Models, Biological; Quinolones | 1992 |
In-vitro activity of sparfloxacin, pefloxacin, ciprofloxacin and temafloxacin against clinical isolates of Acinetobacter spp.
Topics: Acinetobacter; Anti-Infective Agents; Ciprofloxacin; Fluoroquinolones; Pefloxacin; Quinolones | 1992 |
[In vitro antimicrobial activities of new quinolone antibiotics against Mycoplasma pneumoniae].
Topics: Anti-Bacterial Agents; Anti-Infective Agents; Ciprofloxacin; Drug Resistance, Microbial; Enoxacin; Fluoroquinolones; Macrolides; Mycoplasma pneumoniae; Norfloxacin; Ofloxacin; Quinolones; Tetracyclines | 1992 |
Temafloxacin vs ciprofloxacin for UTI.
Topics: Anti-Infective Agents; Ciprofloxacin; Fluoroquinolones; Humans; Quinolones; Trimethoprim, Sulfamethoxazole Drug Combination; Urinary Tract Infections | 1992 |
Temafloxacin vs ciprofloxacin for UTI.
Topics: Anti-Infective Agents; Ciprofloxacin; Fluoroquinolones; Humans; Quinolones; Urinary Tract Infections | 1992 |
Temafloxacin: the pharmacokinetic profile of a new quinolone. A seminar-in-print.
Topics: Anti-Infective Agents; Fluoroquinolones; Humans; Quinolones | 1992 |
Temafloxacin does not potentiate the anticoagulant effect of warfarin in healthy subjects.
Topics: Administration, Oral; Adolescent; Adult; Anti-Infective Agents; Blood Coagulation; Drug Interactions; Fluoroquinolones; Humans; Male; Middle Aged; Platelet Count; Prothrombin Time; Quinolones; Warfarin | 1992 |
Hepatobiliary elimination of temafloxacin.
Topics: Administration, Oral; Adult; Aged; Anti-Infective Agents; Bile; Cholecystectomy; Chromatography, High Pressure Liquid; Female; Fluoroquinolones; Humans; Liver; Male; Middle Aged; Quinolones | 1992 |
The effect of food on the bioavailability of temafloxacin. A review of 3 studies.
Topics: Adult; Anti-Infective Agents; Biological Availability; Capsules; Eating; Female; Fluoroquinolones; Humans; Male; Middle Aged; Quinolones; Solutions; Tablets | 1992 |
Absence of drug interaction between temafloxacin and low dose heparin.
Topics: Administration, Oral; Adolescent; Adult; Anti-Infective Agents; Blood Coagulation Factors; Drug Interactions; Fluoroquinolones; Heparin; Humans; Injections, Subcutaneous; Male; Platelet Count; Quinolones | 1992 |
In vitro activities of five quinolones against Chlamydia pneumoniae.
Topics: Anti-Infective Agents; Chlamydophila pneumoniae; Ciprofloxacin; Fleroxacin; Fluoroquinolones; Microbial Sensitivity Tests; Ofloxacin; Quinolones | 1992 |
Entry of lomefloxacin and temafloxacin into human neutrophils, peritoneal macrophages, and tissue culture cells.
Topics: Animals; Anti-Infective Agents; Cell Line; Cell Survival; Cells, Cultured; Fibroblasts; Fluoroquinolones; Humans; Macrophages; Neutrophils; Opsonin Proteins; Peritoneal Dialysis, Continuous Ambulatory; Quinolones; Temperature; Vero Cells | 1992 |
Susceptibilities of penicillin-susceptible and -resistant strains of Streptococcus pneumoniae to RP 59500, vancomycin, erythromycin, PD 131628, sparfloxacin, temafloxacin, win 57273, ofloxacin, and ciprofloxacin.
Topics: Anti-Infective Agents; Ciprofloxacin; Erythromycin; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Naphthyridines; Ofloxacin; Penicillin Resistance; Quinolones; Streptococcus pneumoniae; Vancomycin; Virginiamycin | 1992 |
Evaluation of temafloxacin in a rat model of intra-abdominal abscess.
Topics: Abdomen; Abscess; Animals; Anti-Infective Agents; Bacteroides fragilis; Bacteroides Infections; Clindamycin; Escherichia coli Infections; Feces; Fluoroquinolones; Gentamicins; Male; Quinolones; Rats; Rats, Inbred Strains | 1992 |
In vitro activity of temafloxacin compared with those of other agents against 100 clinical isolates of Neisseria gonorrhoeae.
Topics: Anti-Infective Agents; Drug Resistance, Microbial; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Neisseria gonorrhoeae; Quinolones | 1992 |
Susceptibilities of 540 anaerobic gram-negative bacilli to amoxicillin, amoxicillin-BRL 42715, amoxicillin-clavulanate, temafloxacin, and clindamycin.
Topics: Amoxicillin; Amoxicillin-Potassium Clavulanate Combination; Anti-Bacterial Agents; Anti-Infective Agents; Clavulanic Acids; Clindamycin; Drug Resistance, Microbial; Drug Therapy, Combination; Fluoroquinolones; Gram-Negative Anaerobic Bacteria; In Vitro Techniques; Lactams; Microbial Sensitivity Tests; Quinolones | 1992 |
Comparative activity of ciprofloxacin, ofloxacin, sparfloxacin, temafloxacin, CI-960, CI-990, and WIN 57273 against anaerobic bacteria.
Topics: Anti-Infective Agents; Bacteria, Anaerobic; Ciprofloxacin; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Naphthyridines; Ofloxacin; Quinolones | 1992 |
Adverse effects prompt withdrawal of temafloxacin.
Topics: Anti-Infective Agents; Fluoroquinolones; Humans; Product Surveillance, Postmarketing; Quinolones | 1992 |
Kinetic disposition of temafloxacin and ciprofloxacin in a murine model of pneumococcal pneumonia. Relevance for drug efficacy.
Topics: Animals; Anti-Infective Agents; Chromatography, High Pressure Liquid; Ciprofloxacin; Female; Fluoroquinolones; Injections, Subcutaneous; Lung; Metabolic Clearance Rate; Mice; Mice, Inbred C57BL; Pneumonia, Pneumococcal; Quinolones | 1992 |
Pharmacokinetics and biliary elimination of temafloxacin in pigs.
Topics: Animals; Anti-Infective Agents; Bile; Chromatography, High Pressure Liquid; Duodenum; Fluoroquinolones; Intubation, Gastrointestinal; Quinolones; Spectrometry, Fluorescence; Swine | 1992 |
Interpretive criteria for CI-960, fleroxacin and temafloxacin susceptibility tests with Haemophilus influenzae.
Topics: Anti-Infective Agents; Fleroxacin; Fluoroquinolones; Haemophilus influenzae; Microbial Sensitivity Tests; Quinolones | 1992 |
Efficacy of temafloxacin in experimental Streptococcus adjacens endocarditis and autoradiographic diffusion pattern of [14C]temafloxacin in cardiac vegetations.
Topics: Animals; Anti-Infective Agents; Autoradiography; Drug Therapy, Combination; Endocarditis, Bacterial; Female; Fluoroquinolones; Microbial Sensitivity Tests; Penicillin G Procaine; Quinolones; Rabbits; Streptococcal Infections; Tobramycin | 1992 |
Interpretive criteria and quality control parameters for testing susceptibility of Haemophilus influenzae to enoxacin, ofloxacin, and temafloxacin.
Topics: Anti-Infective Agents; Drug Resistance, Microbial; Enoxacin; Fluoroquinolones; Haemophilus influenzae; Humans; Microbial Sensitivity Tests; Mutation; Ofloxacin; Quality Control; Quinolones | 1992 |
[Quality assurance for drug information].
Topics: Anti-Infective Agents; Drug Information Services; Fluoroquinolones; Humans; Quality Assurance, Health Care; Quinolones; Sweden | 1992 |
Activity of clarithromycin against Mycobacterium avium complex infection in beige mice.
Topics: Amikacin; Animals; Anti-Infective Agents; Antitubercular Agents; Clarithromycin; Clofazimine; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Therapy, Combination; Ethambutol; Female; Fluoroquinolones; Humans; Mice; Mice, Inbred C57BL; Mycobacterium avium; Mycobacterium avium Complex; Quinolones; Rifabutin; Rifampin; Rifamycins; Time Factors; Tuberculosis | 1992 |
Activities of various quinolone antibiotics against Mycobacterium leprae in infected mice.
Topics: Animals; Anti-Infective Agents; Female; Fluoroquinolones; Leprosy; Mice; Mice, Inbred BALB C; Mycobacterium leprae; Pefloxacin; Quinolones | 1992 |
Susceptibility of recent clinical isolates to temafloxacin (A-63004) and other antimicrobial agents.
Topics: Anti-Infective Agents; Bacteria; Bacterial Infections; Drug Resistance, Microbial; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Quinolones | 1992 |
Characterization of high-level quinolone resistance in Campylobacter jejuni.
Topics: Anti-Infective Agents; Campylobacter jejuni; Ciprofloxacin; DNA Topoisomerases, Type II; DNA, Superhelical; Drug Resistance, Microbial; Fluoroquinolones; Microbial Sensitivity Tests; Mutation; Nalidixic Acid; Norfloxacin; Quinolones; Topoisomerase II Inhibitors | 1991 |
[Intra-macrophagic activity of antibiotics combinations against Mycobacterium marinum].
Topics: Anti-Infective Agents; Antitubercular Agents; Ciprofloxacin; Clarithromycin; Dose-Response Relationship, Drug; Drug Synergism; Drug Therapy, Combination; Erythromycin; Ethambutol; Fluoroquinolones; Humans; In Vitro Techniques; Macrophages; Minocycline; Mycobacterium; Quinolones; Rifabutin; Rifamycins | 1991 |
Activities of sparfloxacin, azithromycin, temafloxacin, and rifapentine compared with that of clarithromycin against multiplication of Mycobacterium avium complex within human macrophages.
Topics: 4-Quinolones; Acquired Immunodeficiency Syndrome; Anti-Bacterial Agents; Azithromycin; Cell Division; Clarithromycin; Erythromycin; Fluoroquinolones; Humans; In Vitro Techniques; Leprostatic Agents; Macrophages; Microbial Sensitivity Tests; Mycobacterium avium Complex; Quinolones; Rifampin | 1991 |
Activity of new quinolones against ciprofloxacin-resistant staphylococci.
Topics: Anti-Infective Agents; Ciprofloxacin; Drug Resistance, Microbial; Fluoroquinolones; Microbial Sensitivity Tests; Naphthyridines; Ofloxacin; Quinolones; Staphylococcus | 1991 |
The in-vitro activity of temafloxacin compared with other antimicrobial agents.
Topics: Anti-Infective Agents; Bacteria; Ciprofloxacin; Enoxacin; Enterobacteriaceae; Fluoroquinolones; Microbial Sensitivity Tests; Ofloxacin; Quinolones; Species Specificity | 1991 |
Fluoroquinolones in the treatment of human infection: the role of temafloxacin.
Topics: Anti-Infective Agents; Bacteria; Bacterial Infections; Fluoroquinolones; Humans; Quinolones | 1991 |
Activity of temafloxacin and other fluoroquinolones against typical and atypical community-acquired respiratory tract pathogens.
Topics: Anti-Infective Agents; Bacteria; Ciprofloxacin; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Ofloxacin; Quinolones; Respiratory Tract Infections | 1991 |
In vitro activity of temafloxacin against gram-positive cocci including methicillin-resistant Staphylococcus aureus.
Topics: Anti-Infective Agents; Ciprofloxacin; Enterococcus; Fluoroquinolones; Gram-Positive Cocci; Methicillin Resistance; Microbial Sensitivity Tests; Ofloxacin; Quinolones; Staphylococcus aureus; Streptococcus | 1991 |
Fluoroquinolones for the treatment of nongonococcal urethritis/cervicitis.
Topics: Anti-Infective Agents; Female; Fluoroquinolones; Gonorrhea; Humans; Male; Quinolones; Sexually Transmitted Diseases, Bacterial; Urethritis; Uterine Cervicitis | 1991 |
Temafloxacin: a safe antibiotic for the elderly, patients with comorbidities, and other special populations.
Topics: Age Factors; Aged; Anti-Infective Agents; Bacterial Infections; Drug Interactions; Female; Fluoroquinolones; Humans; Kidney Diseases; Male; Quinolones; Risk Factors; Sex Factors | 1991 |
In vitro activity of temafloxacin against gram-negative bacteria: an overview.
Topics: Anti-Infective Agents; Campylobacter; Ciprofloxacin; Enterobacteriaceae; Fluoroquinolones; Gram-Negative Bacteria; Humans; Hydrogen-Ion Concentration; Microbial Sensitivity Tests; Ofloxacin; Quinolones; Respiratory Tract Infections; Sexually Transmitted Diseases, Bacterial | 1991 |
In vitro activity of temafloxacin against pathogens causing sexually transmitted diseases.
Topics: Anti-Infective Agents; Chlamydia trachomatis; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Mycoplasma; Neisseria gonorrhoeae; Quinolones; Sexually Transmitted Diseases, Bacterial; Treponema pallidum; Ureaplasma urealyticum | 1991 |
Mechanisms and frequency of resistance to temafloxacin.
Topics: Anti-Infective Agents; Bacteria; Drug Resistance, Microbial; Escherichia coli; Fluoroquinolones; Methicillin Resistance; Mutation; Pseudomonas aeruginosa; Quinolones; Staphylococcus aureus | 1991 |
Comparison of organ-specific toxicity of temafloxacin in animals and humans.
Topics: Animals; Anti-Infective Agents; Central Nervous System; Eye; Fluoroquinolones; Humans; Joints; Kidney; Mutagens; Organ Specificity; Quinolones; Species Specificity | 1991 |
Assessment of temafloxacin neurotoxicity in rodents.
Topics: Animals; Anti-Infective Agents; Central Nervous System; Ciprofloxacin; Enoxacin; Fluoroquinolones; Male; Mice; Mice, Inbred ICR; Motor Activity; Oxolinic Acid; Phenylbutyrates; Quinolones; Rats; Rats, Inbred Strains; Seizures | 1991 |
The influence of age on the pharmacokinetics of temafloxacin.
Topics: Absorption; Administration, Oral; Adult; Aged; Aging; Anti-Infective Agents; Chromatography, High Pressure Liquid; Female; Fluoroquinolones; Humans; Male; Quinolones; Sex Factors | 1991 |
Effect of temafloxacin on the pharmacokinetics of theophylline.
Topics: Adult; Anti-Infective Agents; Drug Interactions; Female; Fluoroquinolones; Humans; Male; Middle Aged; Quinolones; Theophylline | 1991 |
High-performance liquid chromatographic procedures for the determination of temafloxacin in biological matrices.
Topics: Anti-Infective Agents; Chromatography, High Pressure Liquid; Fluoroquinolones; Humans; Quinolones | 1991 |
Anti-staphylococcal activity of temafloxacin, ciprofloxacin, ofloxacin and enoxacin.
Topics: Anti-Infective Agents; Ciprofloxacin; Enoxacin; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Ofloxacin; Oxacillin; Penicillin Resistance; Quinolones; Staphylococcal Infections; Staphylococcus | 1991 |
The in-vitro activity of tosufloxacin, a new fluorinated quinolone, compared with that of ciprofloxacin and temafloxacin.
Topics: Anti-Infective Agents; Bacteria; Bacteria, Aerobic; Bacteria, Anaerobic; Ciprofloxacin; Fluoroquinolones; Microbial Sensitivity Tests; Naphthyridines; Quinolones | 1991 |
Clinical results using two new antibiotics--clarithromycin and temafloxacin.
Topics: Acquired Immunodeficiency Syndrome; Anti-Infective Agents; Bacterial Infections; Clarithromycin; Erythromycin; Fluoroquinolones; Humans; Opportunistic Infections; Quinolones | 1991 |
Temafloxacin: an in-vitro and clinical assessment.
Topics: Animals; Anti-Infective Agents; Fluoroquinolones; Humans; In Vitro Techniques; Quinolones | 1991 |
The in-vitro activity of temafloxacin, against gram-positive bacteria.
Topics: Anti-Infective Agents; Fluoroquinolones; Gram-Positive Bacteria; Microbial Sensitivity Tests; Quinolones | 1991 |
In-vitro activity of temafloxacin against anaerobic bacteria: a comparative study.
Topics: Anti-Infective Agents; Bacteria, Anaerobic; Fluoroquinolones; Quinolones | 1991 |
Pharmacokinetics of four fluoroquinolones in an animal model of infected lung.
Topics: Animals; Anti-Infective Agents; Ciprofloxacin; Disease Models, Animal; Fluoroquinolones; Lung Diseases; Mice; Mice, Inbred Strains; Ofloxacin; Pneumococcal Infections; Quinolones; Streptococcus pneumoniae | 1991 |
Comparative activity of fluorinated quinolones in acute and subacute Streptococcus pneumoniae pneumonia models: efficacy of temafloxacin.
Topics: Acute Disease; Animals; Anti-Infective Agents; Disease Models, Animal; Female; Fluoroquinolones; Mice; Mice, Inbred Strains; Ofloxacin; Pneumonia; Quinolones; Streptococcus pneumoniae | 1991 |
Comparative pharmacokinetic disposition of fluoroquinolones in the lung.
Topics: Administration, Oral; Anti-Infective Agents; Ciprofloxacin; Fluoroquinolones; Humans; Injections, Intravenous; Lung; Quinolones | 1991 |
In-vitro activity of temafloxacin for gram-positive pathogens.
Topics: Anti-Infective Agents; Fluoroquinolones; Gram-Positive Bacteria; Quinolones | 1991 |
Fluorometric and high-performance liquid chromatographic measurement of quinolone uptake by human neutrophils.
Topics: Anti-Infective Agents; Chromatography, High Pressure Liquid; Ciprofloxacin; Fleroxacin; Fluorescence; Fluoroquinolones; Humans; Neutrophils; Norfloxacin; Ofloxacin; Quinolones | 1991 |
ESGAB breakpoint determination: temafloxacin.
Topics: Anti-Infective Agents; Bacteria; Bacterial Infections; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Quinolones | 1991 |
Cross-resistance and cross-susceptibility between fluoroquinolone agents.
Topics: Anti-Infective Agents; Ciprofloxacin; Drug Resistance, Microbial; Enoxacin; Enterobacteriaceae; Fleroxacin; Fluoroquinolones; Microbial Sensitivity Tests; Ofloxacin; Predictive Value of Tests; Quinolones | 1991 |
Anti-Mycobacterium leprae activity of several quinolones studied in the mouse.
Topics: Animals; Anti-Infective Agents; Ciprofloxacin; Fleroxacin; Fluoroquinolones; Leprosy; Mice; Mycobacterium leprae; Quinolones | 1991 |
Temafloxacin pharmacokinetics in subjects with normal and impaired renal function.
Topics: Adult; Aged; Anti-Infective Agents; Fluoroquinolones; Half-Life; Humans; Kidney Diseases; Male; Middle Aged; Quinolones; Renal Dialysis; Tissue Distribution | 1991 |
[In vitro bactericidal effect of temafloxacin and tosufloxacin against streptococci].
Topics: Anti-Infective Agents; Ciprofloxacin; Dose-Response Relationship, Drug; Enterococcus faecalis; Enterococcus faecium; Fluoroquinolones; In Vitro Techniques; Naphthyridines; Pefloxacin; Quinolones; Streptococcus; Streptococcus agalactiae; Streptococcus bovis; Streptococcus pneumoniae; Streptococcus pyogenes; Streptococcus sanguis | 1991 |
[In vitro effect of new fluoroquinolones and betalactamines combinations against enterococci].
Topics: Amoxicillin; Anti-Infective Agents; Ciprofloxacin; Dose-Response Relationship, Drug; Drug Therapy, Combination; Enterococcus faecalis; Fluoroquinolones; Imipenem; In Vitro Techniques; Naphthyridines; Piperacillin; Quinolones | 1991 |
Synthesis, antibacterial activities, and pharmacological properties of enantiomers of temafloxacin hydrochloride.
Topics: 4-Quinolones; Animals; Anti-Infective Agents; Escherichia coli; Female; Fluoroquinolones; Indicators and Reagents; Mice; Microbial Sensitivity Tests; Molecular Structure; Motor Activity; Pseudomonas aeruginosa; Quinolones; Rats; Staphylococcus aureus; Stereoisomerism; Streptococcus; Structure-Activity Relationship; Topoisomerase II Inhibitors | 1991 |
[Experimental study on the hepatobiliary kinetics and excretion of temafloxacin. Evidence for production of active metabolites by the rabbit liver].
Topics: 4-Quinolones; Animals; Anti-Infective Agents; Bile; Chromatography, High Pressure Liquid; Fluoroquinolones; In Vitro Techniques; Liver; Microbiological Techniques; Quinolones; Rabbits | 1991 |
Antipneumococcal activity of ciprofloxacin, ofloxacin, and temafloxacin in an experimental mouse pneumonia model at various stages of the disease.
Topics: Amoxicillin; Animals; Anti-Infective Agents; Ciprofloxacin; Disease Models, Animal; Erythromycin; Female; Fluoroquinolones; Lung; Mice; Mice, Inbred C57BL; Ofloxacin; Pneumonia, Pneumococcal; Quinolones; Sepsis; Streptococcus pneumoniae | 1991 |
Temafloxacin: in vitro comparison with five other antibacterial agents.
Topics: 4-Quinolones; Anti-Infective Agents; Fluoroquinolones; Microbial Sensitivity Tests; Quinolones; Tobramycin | 1991 |
Activity of temafloxacin against respiratory pathogens.
Topics: Animals; Anti-Infective Agents; Bacterial Infections; Cells, Cultured; Ciprofloxacin; Dose-Response Relationship, Drug; Female; Fluoroquinolones; Gerbillinae; Gram-Positive Bacteria; Guinea Pigs; Male; Mice; Microbial Sensitivity Tests; Ofloxacin; Quinolones; Respiratory Tract Infections | 1991 |
Determination of minor impurities in temafloxacin hydrochloride by high-performance liquid chromatography.
Topics: 4-Quinolones; Anti-Infective Agents; Chromatography, High Pressure Liquid; Fluoroquinolones; Quinolones | 1990 |
In-vitro activity of sparfloxacin, a new quinolone antimicrobial agent.
Topics: Anti-Bacterial Agents; Anti-Infective Agents; Bacteria; Blood Proteins; Ciprofloxacin; Fluoroquinolones; Humans; Lactams; Microbial Sensitivity Tests; Protein Binding; Quinolones | 1990 |
Biliary elimination and hepatic disposition of a new fluoroquinolone, temafloxacin: experimental evaluation.
Topics: 4-Quinolones; Animals; Anti-Infective Agents; Bile; Chromatography, Liquid; Fluoroquinolones; In Vitro Techniques; Liver; Metabolic Clearance Rate; Molecular Structure; Perfusion; Quinolones; Rabbits | 1990 |
Correlation between disc potency and zone size in temafloxacin activity in vitro.
Topics: 4-Quinolones; Anti-Infective Agents; Drug Evaluation; Escherichia coli; Fluoroquinolones; Humans; Klebsiella pneumoniae; Microbial Sensitivity Tests; Proteus mirabilis; Pseudomonas aeruginosa; Quinolones; Serratia marcescens; Staphylococcus aureus | 1990 |
In vitro activity of temafloxacin hydrochloride (TA-167 or A-62254), a new fluorinated 4-quinolone.
Topics: 4-Quinolones; Anti-Infective Agents; Bacteria, Aerobic; Fluoroquinolones; Gram-Positive Bacteria; Hydrogen-Ion Concentration; Magnesium; Microbial Sensitivity Tests; Quinolones; Time Factors | 1990 |
Developmental toxicity of temafloxacin hydrochloride in the long-tailed macaque (Macaca fascicularis).
Topics: 4-Quinolones; Animals; Anti-Infective Agents; Appetite; Dose-Response Relationship, Drug; Embryonic and Fetal Development; Female; Fluoroquinolones; Macaca fascicularis; Pregnancy; Quinolones; Teratogens; Vomiting | 1990 |
Determination of temafloxacin, sarafloxacin, and difloxacin in bulk drug and dosage forms by high-performance liquid chromatography.
Topics: Anti-Infective Agents; Chromatography, High Pressure Liquid; Ciprofloxacin; Fluoroquinolones; Quinolones; Solubility; Spectrophotometry, Ultraviolet | 1990 |
In vitro activities of tosufloxacin, temafloxacin, and A-56620 against pathogens of diarrhea.
Topics: Anti-Bacterial Agents; Anti-Infective Agents; Bacteria; Ciprofloxacin; Diarrhea; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Naphthyridines; Quinolones | 1990 |
Concentrations of temafloxacin in serum and bronchial mucosa.
Topics: 4-Quinolones; Aged; Aged, 80 and over; Anti-Infective Agents; Bronchi; Female; Fluoroquinolones; Humans; Male; Middle Aged; Mucous Membrane; Quinolones | 1990 |
Oral temafloxacin versus vancomycin for therapy of experimental endocarditis caused by methicillin-resistant Staphylococcus aureus.
Topics: 4-Quinolones; Administration, Oral; Animals; Anti-Infective Agents; Drug Therapy, Combination; Endocarditis, Bacterial; Fluoroquinolones; Male; Methicillin; Microbial Sensitivity Tests; Penicillin Resistance; Quinolones; Rats; Rats, Inbred Strains; Rifampin; Staphylococcal Infections; Vancomycin | 1990 |
High-performance liquid chromatography for the determination of three new fluoroquinolones, fleroxacin, temafloxacin and A-64730, in biological fluids.
Topics: Anti-Infective Agents; Bile; Chromatography, High Pressure Liquid; Ciprofloxacin; Fleroxacin; Fluoroquinolones; Humans; Molecular Structure; Naphthyridines; Quinolones; Spectrometry, Fluorescence | 1989 |
Comparative antimycobacterial activities of difloxacin, temafloxacin, enoxacin, pefloxacin, reference fluoroquinolones, and a new macrolide, clarithromycin.
Topics: Anti-Bacterial Agents; Anti-Infective Agents; Ciprofloxacin; Clarithromycin; Enoxacin; Erythromycin; Fluoroquinolones; Microbial Sensitivity Tests; Mycobacterium; Pefloxacin; Quinolones | 1989 |
Temafloxacin disk potency and tentative interpretive criteria for susceptibility tests.
Topics: Anti-Infective Agents; Bacteria; Drug Resistance, Microbial; Enterobacteriaceae; Fluoroquinolones; Microbial Sensitivity Tests; Nalidixic Acid; Quinolones; Regression Analysis | 1989 |
In vitro activities of temafloxacin (A-62254) and four other antibiotics against Chlamydia trachomatis.
Topics: 4-Quinolones; Anti-Infective Agents; Chlamydia trachomatis; Doxycycline; Drug Resistance, Microbial; Fluoroquinolones; Quinolones | 1989 |
In-vitro activities of temafloxacin, tosufloxacin (A-61827) and five other fluoroquinolone agents.
Topics: 4-Quinolones; Anti-Infective Agents; Bacteria; Fluoroquinolones; Methicillin; Microbial Sensitivity Tests; Naphthyridines; Penicillin Resistance; Quinolones | 1989 |
In vitro activities of lomefloxacin and temafloxacin against pathogens causing diarrhea.
Topics: 4-Quinolones; Anti-Bacterial Agents; Anti-Infective Agents; Bacteria; Diarrhea; Fluoroquinolones; Humans; Quinolones | 1989 |
The in-vitro activity, pharmacokinetics and tissue penetration of temafloxacin.
Topics: 4-Quinolones; Adult; Anti-Infective Agents; Bacteria; Blister; Exudates and Transudates; Fluoroquinolones; Humans; Male; Quinolones | 1989 |
In vitro activity of temafloxacin, a new difluoro quinolone antimicrobial agent.
Topics: Anti-Bacterial Agents; Cefotaxime; Chemical Phenomena; Chemistry; Ciprofloxacin; Culture Media; Drug Resistance, Microbial; Enterobacteriaceae; Fluoroquinolones; Gram-Negative Bacteria; Hydrogen-Ion Concentration; Imipenem; Magnesium; Ofloxacin; Oxazines; Pseudomonas; Quinolines; Quinolones; Thienamycins | 1988 |
Comparative in vitro activity of the new difluoro-quinolone temafloxacin (A-62254) against bacterial isolates from cancer patients.
Topics: Anti-Infective Agents; Bacteria; Ciprofloxacin; Enterobacteriaceae; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Neoplasms; Quinolones; Staphylococcus; Streptococcus | 1988 |
Correlation of in vitro activities of the fluoroquinolones to their in vivo efficacies.
Topics: Animals; Anti-Infective Agents; Ciprofloxacin; Enoxacin; Fleroxacin; Fluoroquinolones; Mice; Microbial Sensitivity Tests; Naphthyridines; Norfloxacin; Ofloxacin; Pefloxacin; Quinolones | 1988 |
Comparative antibacterial activities of temafloxacin hydrochloride (A-62254) and two reference fluoroquinolones.
Topics: Animals; Anti-Bacterial Agents; Ciprofloxacin; Drug Resistance, Microbial; Female; Fluoroquinolones; Hydrogen-Ion Concentration; Mice; Microbial Sensitivity Tests; Pyelonephritis; Quinolines; Quinolones | 1987 |
Comparison of sparfloxacin, temafloxacin, and ciprofloxacin for prophylaxis and treatment of experimental foreign-body infection by methicillin-resistant Staphylococcus aureus.
Topics: Animals; Anti-Bacterial Agents; Anti-Infective Agents; Ciprofloxacin; Fluoroquinolones; Foreign Bodies; Guinea Pigs; Methicillin Resistance; Microbial Sensitivity Tests; Quinolones; Rats; Staphylococcal Infections; Staphylococcus aureus; Vancomycin | 1995 |
Effect of aerobic and anaerobic environments on antistaphylococcal activities of five fluoroquinolones.
Topics: Anaerobiosis; Anti-Infective Agents; Carbonyl Cyanide m-Chlorophenyl Hydrazone; Ciprofloxacin; Fluoroquinolones; Hydrogen-Ion Concentration; Microbial Sensitivity Tests; Ofloxacin; Quinolones; Staphylococcus aureus | 1995 |
Dissociated resistance among fluoroquinolones.
Topics: Anti-Infective Agents; Ciprofloxacin; Drug Resistance, Microbial; Fluoroquinolones; Gram-Negative Bacteria; Gram-Positive Bacteria; Microbial Sensitivity Tests; Mutation; Ofloxacin; Piperazines; Quinolones | 1994 |
Effect of newer quinolones on the extra- and intra-cellular chemiluminescence response of human polymorphonuclear leucocytes.
Topics: Anti-Infective Agents; Ciprofloxacin; Extracellular Space; Fluoroquinolones; Humans; Luminescent Measurements; Neutrophils; Ofloxacin; Quinolones; Reactive Oxygen Species; Tetradecanoylphorbol Acetate; Zymosan | 1994 |
In vitro activity of the new fluoroquinolone CP-99,219.
Topics: Anti-Infective Agents; Ciprofloxacin; Fluoroquinolones; Gram-Negative Bacteria; Gram-Positive Bacteria; Microbial Sensitivity Tests; Naphthyridines; Quinolones | 1994 |
Limited effects of temafloxacin compared with ciprofloxacin on T-lymphocyte function.
Topics: Anti-Infective Agents; Autoradiography; Blotting, Northern; Cells, Cultured; Ciprofloxacin; Fluoroquinolones; Gene Expression; Humans; In Vitro Techniques; Interferon-gamma; Interleukin-2; Phytohemagglutinins; Quinolones; RNA, Messenger; T-Lymphocytes; Thymidine | 1994 |
Hemolytic anemia and acute renal failure associated with temafloxacin-dependent antibodies.
Topics: Acute Kidney Injury; Aged; Anemia, Hemolytic; Anti-Infective Agents; Antibodies; Female; Fluoroquinolones; Humans; Male; Middle Aged; Quinolones | 1994 |
Dextranase enhances antibiotic efficacy in experimental viridans streptococcal endocarditis.
Topics: Animals; Anti-Bacterial Agents; Anti-Infective Agents; Dextranase; Drug Synergism; Endocarditis, Bacterial; Female; Fluoroquinolones; Lipopolysaccharides; Microbial Sensitivity Tests; Microscopy, Electron; Quinolones; Rabbits; Streptococcal Infections; Streptococcus sanguis | 1994 |
Measurement of temafloxacin in human scalp hair as an index of drug exposure.
Topics: Adult; Anti-Infective Agents; Drug Monitoring; Fluoroquinolones; Hair; Humans; Male; Quinolones; Scalp | 1994 |
Microbial identification and antibiotic sensitivity testing, an aid for patients refractory to periodontal therapy. A report of 3 cases.
Topics: Adult; Aggregatibacter actinomycetemcomitans; Amoxicillin; Anti-Infective Agents; Clindamycin; Drug Resistance, Microbial; Fluoroquinolones; Humans; Male; Microbial Sensitivity Tests; Periodontal Abscess; Periodontitis; Quinolones; Staphylococcus aureus; Tetracycline Resistance | 1994 |
In vitro postantibiotic effect following repeated exposure to imipenem, temafloxacin, and tobramycin.
Topics: Anti-Infective Agents; Fluoroquinolones; Humans; Imipenem; Microbial Sensitivity Tests; Pseudomonas aeruginosa; Quinolones; Time Factors; Tobramycin | 1993 |
Susceptibilities of Mycoplasma hominis, Mycoplasma pneumoniae, and Ureaplasma urealyticum to a new quinolone, OPC 17116.
Topics: Anti-Infective Agents; Fluoroquinolones; Microbial Sensitivity Tests; Mycoplasma; Mycoplasma pneumoniae; Ofloxacin; Piperazines; Quinolones; Ureaplasma urealyticum | 1993 |
Correlation between umuC induction and Salmonella mutagenicity assay for quinolone antimicrobial agents.
Topics: Anti-Infective Agents; Bacterial Proteins; Ciprofloxacin; DNA-Directed DNA Polymerase; Enoxacin; Escherichia coli; Escherichia coli Proteins; Fluoroquinolones; Gene Expression Regulation, Bacterial; Mutagenicity Tests; Nalidixic Acid; Naphthyridines; Norfloxacin; Quinolones; Salmonella typhimurium; SOS Response, Genetics; Species Specificity | 1993 |
New drugs from 1991-1992.
Topics: 1-Naphthylamine; Anti-Bacterial Agents; Anti-Infective Agents; Anticholesteremic Agents; Antineoplastic Agents; Antiviral Agents; Azithromycin; Butanones; Cardiovascular Agents; Clarithromycin; Drug Approval; Drug Combinations; Drug Interactions; Enoxacin; Finasteride; Flumazenil; Fluoroquinolones; Humans; Ketorolac Tromethamine; Lactams; Nabumetone; Pyridines; Quinolones; Sertraline; Tolmetin; Tromethamine; United States; United States Food and Drug Administration; Zolpidem | 1993 |
Evaluation of activity of temafloxacin against Bacteroides fragilis by an in vitro pharmacodynamic system.
Topics: Anaerobiosis; Anti-Infective Agents; Bacteroides fragilis; Cefotetan; Ciprofloxacin; Colony Count, Microbial; Culture Media; Fluoroquinolones; Microbial Sensitivity Tests; Quinolones | 1993 |
Induction of resistance of Streptococcus pneumoniae to quinolones in vitro.
Topics: Anti-Infective Agents; Ciprofloxacin; Drug Resistance, Microbial; Fluoroquinolones; Levofloxacin; Microbial Sensitivity Tests; Norfloxacin; Ofloxacin; Quinolones; Streptococcus pneumoniae | 1993 |
Selection of a fluoroquinolone-class disk for susceptibility tests.
Topics: Anti-Infective Agents; Fluoroquinolones; Microbial Sensitivity Tests; Quinolones | 1993 |
Effects of new quinolones on Mycoplasma pneumoniae-infected hamsters.
Topics: Animals; Anti-Infective Agents; Antibodies, Bacterial; Ciprofloxacin; Cricetinae; Female; Fluoroquinolones; Half-Life; Humans; Lung; Mesocricetus; Mycoplasma pneumoniae; Ofloxacin; Pneumonia, Mycoplasma; Quinolones | 1993 |
The withdrawal of temafloxacin. Are there implications for other quinolones?
Topics: Adult; Adverse Drug Reaction Reporting Systems; Anti-Infective Agents; Drug and Narcotic Control; Fluoroquinolones; Humans; Quinolones; United States; United States Food and Drug Administration | 1993 |
Effect of pH variation on the susceptibility of Helicobacter pylori to three macrolide antimicrobial agents and temafloxacin.
Topics: Anti-Bacterial Agents; Anti-Infective Agents; Azithromycin; Clarithromycin; Drug Resistance, Microbial; Erythromycin; Fluoroquinolones; Helicobacter pylori; Humans; Hydrogen-Ion Concentration; Microbial Sensitivity Tests; Quinolones | 1993 |
In-vitro activity of ciprofloxacin, temafloxacin, azithromycin, clarithromycin and metronidazole against Giardia lamblia.
Topics: Animals; Anti-Infective Agents; Azithromycin; Ciprofloxacin; Clarithromycin; Erythromycin; Fluoroquinolones; Giardia lamblia; Metronidazole; Microbial Sensitivity Tests; Quinolones | 1993 |
Comparative susceptibilities of 173 aerobic and anaerobic bite wound isolates to sparfloxacin, temafloxacin, clarithromycin, and older agents.
Topics: Animals; Anti-Bacterial Agents; Bacteria, Aerobic; Bacteria, Anaerobic; Bites and Stings; Clarithromycin; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Quinolones; Wound Infection | 1993 |
Temafloxacin-induced hemolytic anemia and renal failure.
Topics: Acute Kidney Injury; Anemia, Hemolytic; Anti-Infective Agents; Bacterial Infections; Erythrocytes; Female; Fluoroquinolones; Hemolysis; Humans; Immune Complex Diseases; Middle Aged; Quinolones | 1993 |
In vitro susceptibility of anaerobic bacteria to temafloxacin.
Topics: Anti-Infective Agents; Bacteria, Anaerobic; Drug Resistance, Microbial; Fluoroquinolones; Humans; In Vitro Techniques; Microbial Sensitivity Tests; Quinolones | 1993 |
Time-kill studies of the activity of temafloxacin against four strains of Bacteroides.
Topics: Anti-Infective Agents; Bacteroides; Bacteroides fragilis; Drug Resistance, Microbial; Fluoroquinolones; Humans; In Vitro Techniques; Microbial Sensitivity Tests; Quinolones; Species Specificity | 1993 |
In-vitro evaluation of clarithromycin, temafloxacin, and ethambutol in combination against Mycobacterium avium complex.
Topics: Acquired Immunodeficiency Syndrome; Anti-Infective Agents; Clarithromycin; Drug Synergism; Drug Therapy, Combination; Ethambutol; Evaluation Studies as Topic; Fluoroquinolones; Humans; Macrophages; Microbial Sensitivity Tests; Mycobacterium avium Complex; Mycobacterium avium-intracellulare Infection; Quinolones | 1993 |
Developmental toxicity of fleroxacin and comparative pharmacokinetics of four fluoroquinolones in the cynomolgus macaque (Macaca fascicularis).
Topics: Administration, Oral; Animals; Anti-Infective Agents; Ciprofloxacin; Embryo, Mammalian; Female; Fleroxacin; Fluoroquinolones; Macaca fascicularis; Norfloxacin; Pregnancy; Pregnancy, Animal; Quinolones | 1993 |
Bactericidal index: a new way to assess quinolone bactericidal activity in vitro.
Topics: Anti-Infective Agents; Ciprofloxacin; Enterococcus faecalis; Fluoroquinolones; Microbial Sensitivity Tests; Naphthyridines; Ofloxacin; Quinolones | 1997 |
Effects of fluoroquinolones and magnesium deficiency in murine limb bud cultures.
Topics: Animals; Anti-Infective Agents; Ciprofloxacin; Dose-Response Relationship, Drug; Embryo, Mammalian; Embryonic and Fetal Development; Extremities; Fleroxacin; Fluoroquinolones; Magnesium Deficiency; Mice; Microscopy, Electron; Ofloxacin; Pefloxacin; Quinolones | 1998 |
The effects of increasing levels of quinolone resistance on in-vitro activity of four quinolones.
Topics: Anti-Infective Agents; Ciprofloxacin; Drug Resistance, Microbial; Fluoroquinolones; Gram-Negative Bacteria; Gram-Positive Bacteria; Humans; Microbial Sensitivity Tests; Mutation; Nalidixic Acid; Ofloxacin; Quinolones | 1998 |
In-vitro activity of three fluoroquinolones, cefotaxime and clindamycin against staphylococci.
Topics: Aminoglycosides; Anti-Bacterial Agents; Anti-Infective Agents; Cefotaxime; Cephalosporins; Ciprofloxacin; Clindamycin; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Ofloxacin; Quinolones; Staphylococcal Infections; Staphylococcus | 1995 |
A simple, inexpensive apparatus for performance of preparative scale solution phase multiple parallel synthesis of drug analogs. II. Biological evaluation of a retrospective library of quinolone antiinfective agents.
Topics: Anti-Infective Agents; Chemistry, Pharmaceutical; DNA; DNA Topoisomerases, Type II; Drug Evaluation, Preclinical; Enzyme Inhibitors; Fluoroquinolones; Microbial Sensitivity Tests; Mycobacterium; Quinolones; Reference Values; Solutions; Structure-Activity Relationship; Topoisomerase II Inhibitors | 1998 |
Ultrastructural characterization of murine limb buds after in vitro exposure to grepafloxacin and other fluoroquinolones.
Topics: Abnormalities, Drug-Induced; Animals; Anti-Infective Agents; Calcium; Dose-Response Relationship, Drug; Embryo, Mammalian; Female; Fluoroquinolones; In Vitro Techniques; Levofloxacin; Limb Buds; Magnesium; Male; Mice; Mice, Inbred Strains; Ofloxacin; Piperazines; Pregnancy; Quinolones | 2002 |
[Drug interactions between nonsteroidal anti-inflammatory drug and pazufloxacin mesilate, a new quinolone antibacterial agent for intravenous use: convulsions in mice after intravenous or intracerebroventricular administration].
Topics: Administration, Oral; Animals; Anti-Bacterial Agents; Anti-Infective Agents; Anti-Inflammatory Agents, Non-Steroidal; beta-Alanine; Biphenyl Compounds; Cefazolin; Cilastatin; Cilastatin, Imipenem Drug Combination; Ciprofloxacin; Convulsants; Drug Combinations; Drug Interactions; Enoxacin; Fleroxacin; Fluoroquinolones; Imipenem; Injections, Intravenous; Injections, Intraventricular; Male; Mice; Mice, Inbred ICR; Norfloxacin; Oxazines; Penicillin G; Quinolones; Seizures; Thienamycins | 2002 |
Effects of fluoroquinolones on insulin secretion and beta-cell ATP-sensitive K+ channels.
Topics: Adenosine Triphosphate; Animals; Anti-Bacterial Agents; Cells, Cultured; Fluoroquinolones; Gatifloxacin; Insulin; Insulin Secretion; Islets of Langerhans; Levofloxacin; Mice; Ofloxacin; Patch-Clamp Techniques; Potassium Channels; Quinolones | 2004 |