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temafloxacin and carbostyril

temafloxacin has been researched along with carbostyril in 185 studies

Research

Studies (185)

TimeframeStudies, this research(%)All Research%
pre-199011 (5.95)18.7374
1990's171 (92.43)18.2507
2000's3 (1.62)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bale, MJ; Erwin, ME; Gerlach, EH; Jones, RN; Koontz, FP; Murray, PR; Washington, JA2
Philip, E; Stein, GE1
Andrews, JM; Ashby, JP; Baldwin, DR; Honeybourne, D; Wise, R1
Erwin, ME; Jones, RN1
Erwin, ME; Gerlach, EH; Jones, RN; Koontz, FP; Murray, PR; Washington, JA1
Finegold, SM; Molitoris, E; Wexler, HM1
Fenoll, A; López de Felipe, F; Martínez-Suárez, JV; Rodríguez-Tudela, JL1
Aubert, G; Dorche, G; Pozzetto, B3
Barry, AL; Fuchs, PC; Pfaller, MA1
Carpentier, P; Granneman, GR; Morrison, PJ; Pernet, AG2
Bergogne-Bérézin, E; Joly-Guillou, ML1
Arai, S; Gohara, Y; Kawashima, T; Kuwano, K; Matsu-Ura, I1
Hornstein, LE1
Ganiats, TG; Norcross, WA1
Coles, S; Millar, E; Nimmo, W; Wyld, P1
Granneman, GR1
Fabian, W; Granneman, GR; Kinzig, M; Kirch, W; Locke, C; Mahr, G; Naber, KG; Nickel, P; Sörgel, F1
Fabian, W; Granneman, GR; Kujath, P; Mahr, G; Nickel, P; Sörgel, F1
Lubowski, TJ; Nightingale, CH; Quintiliani, R; Sweeney, K1
Granneman, GR; Mukherjee, D1
Sörgel, F1
Granneman, GR; Mahr, G; Muth, P; Nickel, P; Sörgel, F; Stephan, U1
Granneman, GR; Locke, C; Sörgel, F; Stephan, U1
Birner, B; Granneman, GR; Mukherjee, D; Sörgel, F; Stephan, U1
Fuhr, U; Granneman, GR; Kinzig, M; Mahr, G; Muth, P; Nickel, P; Patterson, K; Sörgel, F; Stephan, U1
Mant, T; Millar, E; Morrison, P1
Hammerschlag, MR; Hyman, CL; Roblin, PM1
Garcia, I; Pascual, A; Perea, EJ1
Carbon, C; Chauvin, JP; Hazebroucq, J; Léophonte, P; Petitpretz, P1
Appelbaum, PC; Jacobs, MR; Spangler, SK1
Chuah, SK; Gollapudi, S; Hajji, M; Perumal, VK; Thadepalli, H1
Cummings, M; Glatt, AE; McCormack, W1
Appelbaum, PC; Jacobs, MR; Shiman, R; Spangler, SK1
Citron, DM; Goldstein, EJ2
Nix, DE; Symonds, WT1
Azoulay-Dupuis, E; Bauchet, J; Pocidalo, JJ; Vallée, E1
Bresler, L; Didelot, JP; Hazebroucq, J; Jehl, F; Koechlin, C; Merle-Melet, M1
Barrett, MS; Jones, RN1
Carnegie, CM; Lindsay, G; Scorer, HJ1
Bouvet, A; Carbon, C; Cremieux, AC; Devine, C; Maziere, B; Muffat-Joly, M; Pocidalo, JJ; Saleh-Mghir, A; Vallois, JM1
al-Wali, WI; Douglas, CW; Spencer, RC; Wilcox, MH; Winstanley, TG1
Allen, SD; Baker, CN; Barry, AL; Fuchs, PC; Hardy, DJ; Jorgensen, JH; McLaughlin, JC1
Järhult, B1
Cynamon, MH; DeStefano, MS; Klemens, SP1
Gelber, RH; Iranmanesh, A; Murray, L; Siu, P; Tsang, M1
Arakawa, S; Kamidono, S1
Almodovar, E; Burns, JJ; Qadri, SM; Rabea, N; Ueno, Y1
Gootz, TD; Martin, BA1
Bollet, C; de Micco, P; Gevaudan, MJ; Mallet, MN2
Gikas, A; Grosset, J; Perronne, C; Pocidalo, JJ; Truffot-Pernot, C; Vilde, JL1
Forstall, GJ; Knapp, CC; Washington, JA1
Bethune, L; King, A; Phillips, I2
Chodosh, S2
Davey, PG1
Parish, LC; Witkowski, JA1
Neldner, KH1
Jungkind, DL; Parish, LC1
Hardy, DJ2
Iravani, A2
Cox, CE1
Childs, SJ; Cox, CE1
Mogabgab, WJ1
Fuchs, PC1
Segreti, J2
Pernet, AG1
Pankey, GA1
Appelbaum, PC1
Jacobs, MR1
Krasula, RW; Pernet, AG1
Giardina, WJ1
Kinzig, M; Mahr, G; Muth, P; Naber, KG; Sorgel, F1
Wise, R1
Granneman, GR; Guay, DR1
Callens, E; Chauvin, JP; Hazebroucq, J; Ruff, F; Santais, MC1
Granneman, GR; Varga, LL1
Barry, AL; Fuchs, PC3
Norrby, SR; Pernet, AG1
Ball, P1
Amsterdam, D; Beam, TR; Gorzynski, EA; Lawrence, T; Mandell, LA; Rotstein, C1
Finegold, SM; Molitoris, E; Reeves, D; Wexler, HM1
Azoulay-Dupuis, E; Bergogne-Bérézin, E; Pocidalo, JJ; Vallée, E1
Azoulay-Dupuis, E; Bedos, JP; Pocidalo, JJ; Vallée, E1
Dudley, MN1
Andrews, JM; Baldwin, DR; Honeybourne, D; Wise, R1
Kosmidis, J1
Lode, H; Vogel, F1
Bischoff, W; Blenk, H; Boerema, JB; Carpentier, P; Focht, J; Naber, KG; Sylvester, J1
Bille, J; Glauser, MP1
Conejo, MC; García, I; Pascual, A; Perea, EJ1
Acar, J; Baquero, F; Bergan, T; Forsgren, A; Phillips, I; Wiedemann, B1
Pattyn, SR1
Braeckman, R; Craft, JC; Granneman, GR; Kraut, J; Shupien, S1
Chu, DT; Giardina, WJ; Hardy, DJ; Nordeen, CW; Pernet, AG; Plattner, JJ; Swanson, RN1
Adler, LP; Bednarczyk, EM; Berridge, MS; Green, JA; Leisure, GA; Little, D; Miraldi, FD; Nelson, AD; Panacek, EA1
Brun, Y; Chanal, M; Courtieu, AL; Dabernat, H; Derlot, E; Joly-Guillou, ML; Kitzis, MD; Meyran, M; Morel, C; Soussy, CJ1
Blickle, JF; Brogard, JM; Dorner, M; Jehl, F; Koechlin, C; Monteil, H; Westphal, JF1
Back, DJ; Mant, T; Martin, C; Millar, E; Morrison, P; Orme, M; Tjia, J1
Azoulay-Dupuis, E; Bedos, JP; Hardy, DJ; Pocidalo, JJ; Swanson, RN; Vallée, E1
Bottolfsen, KL; Digranes, A; Hardardottir, H1
Chu, DT; Clement, JJ; Hardy, DJ; Shipkowitz, NL; Swanson, RN1
Elrod, L; Linton, CL; Shelat, BP; Wong, CF1
Andrews, JM; Ashby, JP; Cooper, MA; Matthews, RS; Wise, R1
Blicklé, JF; Brogard, JM; Dorner, M; Jehl, F; Koechlin, C; Westphal, JF1
Cremers, HM; Davies, BI; Gubbelmans, HL; Maesen, FP1
Bassanetti, I; Ceralli, M; Giardini, R; Reggio, S; Sansonetti, G1
Inoue, K; Inoue, M; Mitsuhashi, S; Nakanishi, N; Yamaguchi, T1
Hendrickx, AG; Lasley, BL; Lehrer, SB; Tarantal, AF1
Bauer, JF; Elrod, L; Fornnarino, JR; Heathcote, DE; Krogh, SK; Linton, CL; Norris, BJ; Quick, JE1
Bryan, JP; Krieg, RE; Perine, PL; Sheffield, J; Wagner, K; Waters, C1
Andrews, JM; Ashby, JP; Baldwin, DR; Honeybourne, D; Wilkinson, L; Wise, R1
Hessen, MT; Kaye, D; Pitsakis, PG1
Jehl, F; Koechlin, C; Linger, L; Monteil, H1
Allen, W; Gorzynski, EA; Gutman, SI1
Barry, AL; Jones, RN2
Kapell, KS; Kessler, HA; Segreti, J; Trenholme, GM1
Goodman, LJ; Kaplan, RL; Nelson, JA; Segreti, J; Trenholme, GM1
Andrews, JM; Ashby, JP; Nye, K; Shi, YG; Wise, R1
Chin, NX; Figueredo, VM; Neu, HC; Novelli, A1
Bodey, GP; Gooch, G; Ho, DH; LeBlanc, B; Rolston, KV1
Fernandes, PB; Swanson, RN1
Bower, RR; Chu, DT; Fernandes, PB; Hanson, CW; Hardy, DJ; Hensey, DM; Ramer, NR; Swanson, RN1
Cagni, A; Chuard, C; Lew, DP; Schrenzel, J; Vaudaux, PE1
Davey, P; McDonald, T1
Lietman, PS; Norrby, SR1
Kaatz, GW; Larsson, AJ; Moody, JA; Rotschafer, JC; Walker, KJ; Zabinski, RA1
Sanders, CC; Thomson, KS2
Aoki, M; Goldstein, E; Kunii, O; Ono, Y1
Chin, NX; Neu, HC1
Arakawa, S; Ban, Y; Hirose, T; Ito, Y; Kamidono, S; Kawada, Y; Kumamoto, Y; Kumon, H; Ohmori, H; Suzuki, K1
Forsgren, A; Riesbeck, K1
Gale, E; Maguire, RB; Stroncek, DF; Yearlsey, M1
Carbon, C; Cremieux, AC; Jambou, R; Mghir, AS; Muffat-Joly, M; Pocidalo, JJ1
Blum, MD; Graham, DJ; McCloskey, CA1
Kondo, K; Nakashima, M; Uematsu, T; Umemura, K; Yamaguchi, T; Yano, S1
Fine, DH1
Dudley, MN; Gilbert, D; Marchbanks, CR; McGrath, BJ1
Cartwright, FD; Kenny, GE1
Phillips, I; Power, EG1
Gage, TW1
Krinke, AJ; Moody, JA; Rotschafer, JC; Vance-Bryan, K; Walker, KJ; Zabinski, RA1
Foleno, BD; Fu, KP; Lafredo, SC1
Akashi, A; Arai, S; Gohara, Y; Kuwano, K; Nishimoto, M; Oizumi, K; Takeda, K; Yamaguchi, T; Yano, T1
Finch, RG1
Eliopoulos, GM; Ferraro, MJ; Malanoski, GJ; Moellering, RC1
Ikerd, TR; Koletar, SL1
Deamer, RL; Heming, D; James, RE; Koenker, N; Prichard, JG1
Patel, S; Southern, PM1
Brown, WJ; Moosavi, S1
Cho, N; Matsuda, S; Okada, H; Shimizu, T1
Hendrickx, AG; Hummler, H; Richter, WF1
Lietman, PS1
Iakovlev, SV; Iakovlev, VP; Izotova, GN1
Muñiz, AE1
Banno, K; Matsuoka, M; Sato, T1
Goldstein, EJ1
Morrissey, I1
Baumann-Wilschke, I; Förster, C; Rücker, M; Shakibaei, M; Stahlmann, R; Vormann, J1
Peters, G; Schumacher-Perdreau, F1
Baker, WR; Devasthale, PV; Frank, KE; Gentry, EJ; Keschavarz-Shokri, A; Mitscher, LA; Nilius, A; Ravikumar, VT; Shawar, R; Shen, LL1
Baumann-Wilschke, I; Rücker, M; Shakibaei, M; Stahlmann, R1
Fukuda, H; Kawamura, Y1
Gonoi, T; Saraya, A; Seino, S; Yokokura, M1

Reviews

19 review(s) available for temafloxacin and carbostyril

ArticleYear
Pharmacokinetics of temafloxacin after multiple oral administration.
    Clinical pharmacokinetics, 1992, Volume: 22 Suppl 1

    Topics: Administration, Oral; Adult; Anti-Infective Agents; Double-Blind Method; Drug Administration Schedule; Fluoroquinolones; Humans; Middle Aged; Quinolones

1992
Penetration of temafloxacin into body tissues and fluids.
    Clinical pharmacokinetics, 1992, Volume: 22 Suppl 1

    Topics: Administration, Oral; Anti-Infective Agents; Fluoroquinolones; Humans; Quinolones; Tissue Distribution

1992
Lomefloxacin and temafloxacin: two new fluoroquinolone antimicrobials.
    Clinical pharmacy, 1992, Volume: 11, Issue:9

    Topics: Anti-Infective Agents; Bacteria; Bacterial Infections; Drug Interactions; Drug Resistance, Microbial; Fluoroquinolones; Humans; Quinolones

1992
Temafloxacin as prophylactic agent in neutropenic patients.
    The Journal of antimicrobial chemotherapy, 1992, Volume: 30, Issue:3

    Topics: Anti-Infective Agents; Fluoroquinolones; Humans; Neutropenia; Quinolones; Sepsis

1992
Systemic management of cutaneous bacterial infections.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Anti-Infective Agents; Bacterial Infections; Fluoroquinolones; Humans; Quinolones; Skin Diseases, Infectious

1991
Temafloxacin: an overview.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Anti-Infective Agents; Bacterial Infections; Fluoroquinolones; Humans; Male; Microbial Sensitivity Tests; Prostatitis; Quinolones; Respiratory Tract Infections; Sexually Transmitted Diseases, Bacterial; Skin Diseases, Infectious; Urinary Tract Infections

1991
Evaluation of the bactericidal activity of temafloxacin.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Anti-Infective Agents; Bacteria; Fluoroquinolones; Microbial Sensitivity Tests; Quinolones

1991
Comparative pharmacokinetics of ciprofloxacin and temafloxacin in humans: a review.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Aging; Anti-Infective Agents; Ciprofloxacin; Drug Interactions; Fluoroquinolones; Humans; Kidney Diseases; Liver Diseases; Quinolones; Tissue Distribution

1991
Comparative penetration of selected fluoroquinolones into respiratory tract fluids and tissues.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Anti-Infective Agents; Bronchi; Ciprofloxacin; Epithelium; Fluoroquinolones; Humans; Macrophages, Alveolar; Mucous Membrane; Quinolones; Respiratory System

1991
Use of quinolones for the treatment of acute exacerbations of chronic bronchitis.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Acute Disease; Anti-Infective Agents; Bronchitis; Chronic Disease; Ciprofloxacin; Fluoroquinolones; Humans; Ofloxacin; Quinolones

1991
The role of temafloxacin in the community setting: an overview.
    The Journal of antimicrobial chemotherapy, 1991, Volume: 28 Suppl C

    Topics: Anti-Infective Agents; Fluoroquinolones; Humans; Quinolones

1991
A review of the pharmacokinetic profile of temafloxacin.
    The Journal of antimicrobial chemotherapy, 1991, Volume: 28 Suppl C

    Topics: Anti-Infective Agents; Fluoroquinolones; Humans; Quinolones

1991
Postmarketing surveillance of quinolones, 1990 to 1992.
    Drugs, 1993, Volume: 45 Suppl 3

    Topics: Adverse Drug Reaction Reporting Systems; Anti-Bacterial Agents; Anti-Infective Agents; Databases, Factual; Fluoroquinolones; Hospitalization; Humans; Quinolones; Risk Factors

1993
Safety and tolerability of fluoroquinolones.
    Drugs, 1993, Volume: 45 Suppl 3

    Topics: Adverse Drug Reaction Reporting Systems; Animals; Anti-Infective Agents; Dermatitis, Phototoxic; Drug Tolerance; Fluoroquinolones; Humans; Quinine; Quinolones; Safety

1993
Temafloxacin syndrome: review of 95 cases.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 1994, Volume: 18, Issue:6

    Topics: Adult; Adverse Drug Reaction Reporting Systems; Aged; Aged, 80 and over; Anemia, Hemolytic; Anti-Infective Agents; Female; Fluoroquinolones; Hemolysis; Humans; Male; Middle Aged; Quinolones

1994
Fluoroquinolone toxicities. An update.
    Drugs, 1995, Volume: 49 Suppl 2

    Topics: Anti-Infective Agents; Dermatitis, Phototoxic; Fluoroquinolones; Humans; Joint Diseases; Nervous System Diseases; Quinolones

1995
[Pharmacokinetics of fluoroquinolones in patients with renal insufficiency].
    Antibiotiki i khimioterapiia = Antibiotics and chemoterapy [sic], 1995, Volume: 40, Issue:10

    Topics: Anti-Infective Agents; Ciprofloxacin; Fluoroquinolones; Humans; Ofloxacin; Pefloxacin; Quinolones; Renal Insufficiency

1995
An unlikely childhood overdose: temafloxacin.
    Pediatric emergency care, 1996, Volume: 12, Issue:3

    Topics: Animals; Anti-Infective Agents; Child, Preschool; Drug Overdose; Female; Fluoroquinolones; Humans; Quinolones; Urinary Tract Infections

1996
Possible role for the new fluoroquinolones (levofloxacin, grepafloxacin, trovafloxacin, clinafloxacin, sparfloxacin, and DU-6859a) in the treatment of anaerobic infections: review of current information on efficacy and safety.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 1996, Volume: 23 Suppl 1

    Topics: Anti-Infective Agents; Bacteria, Anaerobic; Bacterial Infections; Fluoroquinolones; Humans; Levofloxacin; Naphthyridines; Ofloxacin; Piperazines; Quinolones; Safety; Syndrome

1996

Trials

31 trial(s) available for temafloxacin and carbostyril

ArticleYear
Comparison of three-day temafloxacin with seven-day ciprofloxacin treatment of urinary tract infections in women.
    The Journal of family practice, 1992, Volume: 34, Issue:2

    Topics: Adult; Aged; Anti-Infective Agents; Ciprofloxacin; Female; Fluoroquinolones; Humans; Middle Aged; Quinolones; Urinary Tract Infections

1992
Pharmacokinetics of temafloxacin in patients with liver impairment.
    Clinical pharmacokinetics, 1992, Volume: 22 Suppl 1

    Topics: Adult; Aged; Anti-Infective Agents; Chromatography, High Pressure Liquid; Female; Fluoroquinolones; Humans; Kidney; Liver; Liver Cirrhosis; Male; Middle Aged; Quinolones

1992
The relative bioavailability of temafloxacin administered through a nasogastric tube with and without enteral feeding.
    Clinical pharmacokinetics, 1992, Volume: 22 Suppl 1

    Topics: Administration, Oral; Adult; Anti-Infective Agents; Biological Availability; Enteral Nutrition; Fluoroquinolones; Humans; Male; Middle Aged; Quinolones

1992
Effects of 2 quinolone antibacterials, temafloxacin and enoxacin, on theophylline pharmacokinetics.
    Clinical pharmacokinetics, 1992, Volume: 22 Suppl 1

    Topics: Administration, Oral; Adult; Aminophylline; Anti-Infective Agents; Double-Blind Method; Drug Interactions; Enoxacin; Fluoroquinolones; Humans; Injections, Intravenous; Male; Quinolones; Theophylline

1992
Effect of cimetidine on the pharmacokinetics of temafloxacin.
    Clinical pharmacokinetics, 1992, Volume: 22 Suppl 1

    Topics: Administration, Oral; Anti-Infective Agents; Cimetidine; Drug Interactions; Female; Fluoroquinolones; Humans; Male; Quinolones

1992
Effect of antacid medication on the pharmacokinetics of temafloxacin.
    Clinical pharmacokinetics, 1992, Volume: 22 Suppl 1

    Topics: Adult; Antacids; Anti-Infective Agents; Drug Interactions; Female; Fluoroquinolones; Humans; Male; Quinolones

1992
Effects of temafloxacin and ciprofloxacin on the pharmacokinetics of caffeine.
    Clinical pharmacokinetics, 1992, Volume: 22 Suppl 1

    Topics: Adult; Anti-Infective Agents; Caffeine; Ciprofloxacin; Double-Blind Method; Drug Interactions; Female; Fluoroquinolones; Humans; Male; Quinolones

1992
Efficacy and safety of temafloxacin versus those of amoxicillin in hospitalized adults with community-acquired pneumonia.
    Antimicrobial agents and chemotherapy, 1992, Volume: 36, Issue:4

    Topics: Administration, Oral; Adult; Aged; Amoxicillin; Anti-Infective Agents; Bacteria; Double-Blind Method; Female; Fluoroquinolones; Humans; Male; Middle Aged; Pneumonia; Quinolones

1992
Safety and efficacy of temafloxacin versus ciprofloxacin in lower respiratory tract infections: a randomized, double-blind trial.
    The Journal of antimicrobial chemotherapy, 1992, Volume: 30, Issue:1

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Anti-Infective Agents; Bacteria; Ciprofloxacin; Double-Blind Method; Drug Interactions; Female; Fluoroquinolones; Humans; Male; Middle Aged; Prospective Studies; Quinolones; Respiratory Tract Infections; Theophylline

1992
Assessment of the UTI criteria for bacterial prostatitis in Japan.
    Infection, 1992, Volume: 20 Suppl 3

    Topics: Acute Disease; Administration, Oral; Adolescent; Adult; Aged; Anti-Infective Agents; Bacterial Infections; Chronic Disease; Fluoroquinolones; Humans; Male; Middle Aged; Prostatitis; Quinolones; Treatment Outcome

1992
Temafloxacin compared with ciprofloxacin in mild to moderate lower respiratory tract infections in ambulatory patients. A multicenter, double-blind, randomized study.
    Chest, 1991, Volume: 100, Issue:6

    Topics: Ambulatory Care; Anti-Infective Agents; Ciprofloxacin; Double-Blind Method; Female; Fluoroquinolones; Humans; Lung Diseases, Obstructive; Male; Microbial Sensitivity Tests; Middle Aged; Pneumonia; Quinolones; Respiratory Tract Infections

1991
Efficacy of temafloxacin versus ciprofloxacin or amoxicillin for lower respiratory tract infections in smokers and the elderly.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Age Factors; Aged; Amoxicillin; Anti-Infective Agents; Ciprofloxacin; Double-Blind Method; Female; Fluoroquinolones; Humans; Male; Quinolones; Respiratory Tract Infections; Smoking

1991
Double-blind randomized study of oral temafloxacin and cefadroxil in patients with mild to moderately severe bacterial skin infections.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Anti-Infective Agents; Cefadroxil; Double-Blind Method; Female; Fluoroquinolones; Humans; Male; Middle Aged; Quinolones; Skin Diseases, Infectious; Staphylococcal Skin Infections; Streptococcal Infections

1991
Systemic antimicrobial therapy in skin and skin structure infections: comparison of temafloxacin and ciprofloxacin.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Anti-Infective Agents; Bacterial Infections; Ciprofloxacin; Double-Blind Method; Female; Fluoroquinolones; Humans; Male; Middle Aged; Quinolones; Skin Diseases, Infectious

1991
Treatment of uncomplicated urinary tract infections with temafloxacin.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Adult; Anti-Infective Agents; Double-Blind Method; Female; Fluoroquinolones; Humans; Quinolones; Urinary Tract Infections

1991
Oral temafloxacin compared to norfloxacin for the treatment of complicated urinary tract infections.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Administration, Oral; Adolescent; Adult; Aged; Aged, 80 and over; Anti-Infective Agents; Double-Blind Method; Female; Fluoroquinolones; Humans; Male; Middle Aged; Norfloxacin; Quinolones; Urinary Tract Infections

1991
Treatment of chronic bacterial prostatitis with temafloxacin.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Adult; Aged; Anti-Infective Agents; Bacterial Infections; Double-Blind Method; Fluoroquinolones; Humans; Male; Middle Aged; Prostatitis; Quinolones

1991
Single-dose oral temafloxacin versus parenteral ceftriaxone in the treatment of gonococcal urethritis/cervicitis.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Administration, Oral; Adolescent; Adult; Aged; Anti-Infective Agents; Ceftriaxone; Female; Fluoroquinolones; Gonorrhea; Humans; Injections, Intramuscular; Male; Middle Aged; Quinolones; Urethritis; Uterine Cervicitis

1991
Assessment of adverse events during drug development: experience with temafloxacin.
    The Journal of antimicrobial chemotherapy, 1991, Volume: 28 Suppl C

    Topics: Aged; Anti-Infective Agents; Drug Evaluation; Female; Fluoroquinolones; Humans; Male; Quinolones

1991
A double-blind study of once-daily temafloxacin in the treatment of bacterial lower respiratory tract infections.
    The Journal of antimicrobial chemotherapy, 1991, Volume: 28 Suppl C

    Topics: Adolescent; Adult; Anti-Infective Agents; Bronchitis; Ciprofloxacin; Double-Blind Method; Female; Fluoroquinolones; Humans; Male; Pneumonia; Quinolones; Respiratory Tract Infections

1991
The use of oral temafloxacin compared with a parenteral cephalosporin in hospitalized patients with pneumonia.
    The Journal of antimicrobial chemotherapy, 1991, Volume: 28 Suppl C

    Topics: Administration, Oral; Adolescent; Adult; Aged; Anti-Infective Agents; Cefotaxime; Female; Fluoroquinolones; Humans; Injections, Intravenous; Male; Middle Aged; Pneumonia; Quinolones

1991
An assessment of temafloxacin in the treatment of chronic bacterial prostatitis.
    The Journal of antimicrobial chemotherapy, 1991, Volume: 28 Suppl C

    Topics: Administration, Oral; Anti-Infective Agents; Chronic Disease; Fluoroquinolones; Humans; Male; Prostatitis; Quinolones

1991
Comparison of the effect of temafloxacin, ciprofloxacin, or placebo on cerebral blood flow, glucose, and oxygen metabolism in healthy subjects by means of positron emission tomography.
    Clinical pharmacology and therapeutics, 1991, Volume: 50, Issue:2

    Topics: Adolescent; Adult; Anti-Infective Agents; Brain; Cerebrovascular Circulation; Ciprofloxacin; Deoxyglucose; Double-Blind Method; Fluoroquinolones; Glucose; Humans; Male; Oxygen; Placebos; Prospective Studies; Quinolones; Reference Values; Tomography, Emission-Computed

1991
[In vitro antibacterial activity of a new fluoroquinolone, temafloxacin, against hospital isolates. Results of a multicenter study].
    Pathologie-biologie, 1991, Volume: 39, Issue:5

    Topics: 4-Quinolones; Acinetobacter; Anti-Infective Agents; Bacteria, Anaerobic; Dose-Response Relationship, Drug; Enterobacteriaceae; Fluoroquinolones; Haemophilus; Humans; In Vitro Techniques; Neisseria; Pseudomonas; Quinolones; Staphylococcus; Streptococcus

1991
The lack of interaction between temafloxacin and combined oral contraceptive steroids.
    Contraception, 1991, Volume: 43, Issue:4

    Topics: 4-Quinolones; Adult; Anti-Infective Agents; Contraceptives, Oral, Combined; Drug Interactions; Ethinyl Estradiol; Female; Fluoroquinolones; Follicle Stimulating Hormone; Humans; Levonorgestrel; Luteinizing Hormone; Norgestrel; Progesterone; Quinolones; Radioimmunoassay

1991
Comparative, double-blind, prospective, multicenter trial of temafloxacin versus trimethoprim-sulfamethoxazole in uncomplicated urinary tract infections in women.
    Antimicrobial agents and chemotherapy, 1991, Volume: 35, Issue:9

    Topics: 4-Quinolones; Adult; Anti-Infective Agents; Double-Blind Method; Female; Fluoroquinolones; Humans; Middle Aged; Prospective Studies; Quinolones; Trimethoprim, Sulfamethoxazole Drug Combination; Urinary Tract Infections

1991
Pharmacokinetics of temafloxacin in humans after single oral doses.
    Antimicrobial agents and chemotherapy, 1991, Volume: 35, Issue:3

    Topics: 4-Quinolones; Administration, Oral; Adult; Anti-Infective Agents; Blood Proteins; Chromatography, High Pressure Liquid; Double-Blind Method; Fluoroquinolones; Half-Life; Humans; Male; Quinolones; Random Allocation

1991
Temafloxacin in acute purulent exacerbations of chronic bronchitis.
    The Journal of antimicrobial chemotherapy, 1990, Volume: 26, Issue:2

    Topics: 4-Quinolones; Anti-Infective Agents; Bronchitis; Chronic Disease; Drug Administration Schedule; Fluoroquinolones; Haemophilus influenzae; Humans; Moraxella catarrhalis; Pseudomonas aeruginosa; Quinolones; Sputum; Streptococcus pneumoniae

1990
[Re-examination of the criteria for clinical evaluation on bacterial prostatitis--analysis of the data of the clinical study of temafloxacin].
    Hinyokika kiyo. Acta urologica Japonica, 1994, Volume: 40, Issue:5

    Topics: Acute Disease; Adolescent; Adult; Aged; Anti-Infective Agents; Bacterial Infections; Chronic Disease; Fluoroquinolones; Humans; Male; Middle Aged; Prostatitis; Quinolones

1994
[Experimental and clinical studies of temafloxacin in the field of obstetrics and gynecology].
    The Japanese journal of antibiotics, 1993, Volume: 46, Issue:6

    Topics: Administration, Oral; Adolescent; Adult; Aged; Anti-Infective Agents; Bacteria; Bacterial Infections; Female; Fluoroquinolones; Genital Diseases, Female; Genitalia, Female; Humans; Middle Aged; Quinolones

1993
Analytical chiral separation of a new quinolone compound in biological fluids by high-performance liquid chromatography.
    Journal of chromatography. B, Biomedical applications, 1996, Feb-09, Volume: 676, Issue:1

    Topics: Anti-Infective Agents; Calibration; Chromatography, High Pressure Liquid; Fluoroquinolones; Half-Life; Humans; Hydrogen-Ion Concentration; Indicators and Reagents; Quinolones; Spectrophotometry, Ultraviolet; Stereoisomerism

1996

Other Studies

135 other study(ies) available for temafloxacin and carbostyril

ArticleYear
MIC quality control guidelines for Haemophilus susceptibility tests using cefdinir (FK482), cefepime, cefetamet, cefpirome, ceftibuten, fleroxacin, temafloxacin, clarithromycin, RP59500, and trospectomycin.
    Journal of clinical microbiology, 1992, Volume: 30, Issue:1

    Topics: Anti-Bacterial Agents; Cefdinir; Cefpirome; Ceftibuten; Ceftizoxime; Cephalosporins; Clarithromycin; Erythromycin; Fleroxacin; Fluoroquinolones; Haemophilus; Humans; Microbial Sensitivity Tests; Quality Control; Quinolones; Spectinomycin; Virginiamycin

1992
Studies show new macrolide antibiotics to be superior to some older agents.
    Oncology (Williston Park, N.Y.), 1992, Volume: 6, Issue:1

    Topics: Anti-Bacterial Agents; Anti-Infective Agents; Bacterial Infections; Clarithromycin; Drug Administration Schedule; Erythromycin; Fluoroquinolones; Humans; Quinolones

1992
Disk diffusion quality control guidelines for Haemophilus susceptibility tests using cefdinir, CI-960, fleroxacin, temafloxacin, and trospectomycin.
    Journal of clinical microbiology, 1992, Volume: 30, Issue:3

    Topics: Anti-Bacterial Agents; Cefdinir; Cephalosporins; Fleroxacin; Fluoroquinolones; Haemophilus influenzae; Microbial Sensitivity Tests; Quality Control; Quinolones; Spectinomycin

1992
The distribution of temafloxacin in bronchial epithelial lining fluid, alveolar macrophages and bronchial mucosa.
    The European respiratory journal, 1992, Volume: 5, Issue:4

    Topics: Anti-Infective Agents; Bronchi; Bronchoalveolar Lavage Fluid; Bronchoscopy; Female; Fluoroquinolones; Humans; Macrophages, Alveolar; Male; Middle Aged; Mucous Membrane; Quinolones; Tissue Distribution

1992
Oral temafloxacin approved for U.S. market.
    Clinical pharmacy, 1992, Volume: 11, Issue:5

    Topics: Administration, Oral; Anti-Infective Agents; Bacterial Infections; Fluoroquinolones; Humans; Quinolones; United States; United States Food and Drug Administration

1992
Interpretive criteria for susceptibility testing of CI-960 (PD127391, AM-1091), fleroxacin, lomefloxacin, and temafloxacin against Neisseria gonorrhoeae, including drug stability in GC agar medium.
    Journal of clinical microbiology, 1992, Volume: 30, Issue:5

    Topics: Agar; Anti-Infective Agents; Drug Stability; Fleroxacin; Fluoroquinolones; Microbial Sensitivity Tests; Neisseria gonorrhoeae; Quinolones

1992
MIC and disk diffusion quality control guidelines for Neisseria gonorrhoeae susceptibility tests of cefdinir, cefetamet, CI-960, fleroxacin, lomefloxacin, and temafloxacin.
    Journal of clinical microbiology, 1992, Volume: 30, Issue:5

    Topics: Anti-Infective Agents; Cefdinir; Ceftizoxime; Cephalosporins; Diffusion; Fleroxacin; Fluoroquinolones; Microbial Sensitivity Tests; Neisseria gonorrhoeae; Quality Control; Quinolones

1992
In vitro activities of three of the newer quinolones against anaerobic bacteria.
    Antimicrobial agents and chemotherapy, 1992, Volume: 36, Issue:1

    Topics: Anti-Infective Agents; Bacteria, Anaerobic; Fluoroquinolones; Microbial Sensitivity Tests; Quinolones

1992
Comparative in-vitro activity of four peptide antibiotics against penicillin-resistant Streptococcus pneumoniae isolated from cerebrospinal fluid (CSF).
    The Journal of antimicrobial chemotherapy, 1992, Volume: 29, Issue:3

    Topics: Anti-Bacterial Agents; Anti-Infective Agents; Cerebrospinal Fluid; Daptomycin; Erythromycin; Fluoroquinolones; Glycopeptides; Humans; Microbial Sensitivity Tests; Penicillin Resistance; Peptides; Quinolones; Serotyping; Streptococcus pneumoniae; Teicoplanin; Vancomycin

1992
Emergence of quinolone-imipenem cross-resistance in Pseudomonas aeruginosa after fluoroquinolone therapy.
    The Journal of antimicrobial chemotherapy, 1992, Volume: 29, Issue:3

    Topics: Anti-Infective Agents; Drug Resistance, Microbial; Drug Therapy, Combination; Fluoroquinolones; Humans; Imipenem; Microbial Sensitivity Tests; Mutation; Naphthyridines; Norfloxacin; Pseudomonas aeruginosa; Pseudomonas Infections; Quinolones

1992
Two new fluoroquinolones.
    The Medical letter on drugs and therapeutics, 1992, Jun-12, Volume: 34, Issue:872

    Topics: Anti-Infective Agents; Clinical Trials as Topic; Drug Interactions; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Quinolones; Respiratory Tract Infections; Urinary Tract Infections

1992
Spontaneously occurring staphylococcal mutants resistant to clinically achievable concentrations of ciprofloxacin and temafloxacin.
    European journal of clinical microbiology & infectious diseases : official publication of the European Society of Clinical Microbiology, 1992, Volume: 11, Issue:3

    Topics: Anti-Infective Agents; Ciprofloxacin; Drug Resistance, Microbial; Fluoroquinolones; Microbial Sensitivity Tests; Mutation; Quinolones; Staphylococcus aureus; Staphylococcus epidermidis

1992
Pharmacokinetics of temafloxacin in humans after multiple oral doses.
    Antimicrobial agents and chemotherapy, 1992, Volume: 36, Issue:2

    Topics: Administration, Oral; Adult; Anti-Infective Agents; Chromatography, High Pressure Liquid; Circadian Rhythm; Fluoroquinolones; Glomerular Filtration Rate; Half-Life; Humans; Male; Models, Biological; Quinolones

1992
In-vitro activity of sparfloxacin, pefloxacin, ciprofloxacin and temafloxacin against clinical isolates of Acinetobacter spp.
    The Journal of antimicrobial chemotherapy, 1992, Volume: 29, Issue:4

    Topics: Acinetobacter; Anti-Infective Agents; Ciprofloxacin; Fluoroquinolones; Pefloxacin; Quinolones

1992
[In vitro antimicrobial activities of new quinolone antibiotics against Mycoplasma pneumoniae].
    Nihon saikingaku zasshi. Japanese journal of bacteriology, 1992, Volume: 47, Issue:2

    Topics: Anti-Bacterial Agents; Anti-Infective Agents; Ciprofloxacin; Drug Resistance, Microbial; Enoxacin; Fluoroquinolones; Macrolides; Mycoplasma pneumoniae; Norfloxacin; Ofloxacin; Quinolones; Tetracyclines

1992
Temafloxacin vs ciprofloxacin for UTI.
    The Journal of family practice, 1992, Volume: 35, Issue:1

    Topics: Anti-Infective Agents; Ciprofloxacin; Fluoroquinolones; Humans; Quinolones; Trimethoprim, Sulfamethoxazole Drug Combination; Urinary Tract Infections

1992
Temafloxacin vs ciprofloxacin for UTI.
    The Journal of family practice, 1992, Volume: 35, Issue:1

    Topics: Anti-Infective Agents; Ciprofloxacin; Fluoroquinolones; Humans; Quinolones; Urinary Tract Infections

1992
Temafloxacin: the pharmacokinetic profile of a new quinolone. A seminar-in-print.
    Clinical pharmacokinetics, 1992, Volume: 22 Suppl 1

    Topics: Anti-Infective Agents; Fluoroquinolones; Humans; Quinolones

1992
Temafloxacin does not potentiate the anticoagulant effect of warfarin in healthy subjects.
    Clinical pharmacokinetics, 1992, Volume: 22 Suppl 1

    Topics: Administration, Oral; Adolescent; Adult; Anti-Infective Agents; Blood Coagulation; Drug Interactions; Fluoroquinolones; Humans; Male; Middle Aged; Platelet Count; Prothrombin Time; Quinolones; Warfarin

1992
Hepatobiliary elimination of temafloxacin.
    Clinical pharmacokinetics, 1992, Volume: 22 Suppl 1

    Topics: Administration, Oral; Adult; Aged; Anti-Infective Agents; Bile; Cholecystectomy; Chromatography, High Pressure Liquid; Female; Fluoroquinolones; Humans; Liver; Male; Middle Aged; Quinolones

1992
The effect of food on the bioavailability of temafloxacin. A review of 3 studies.
    Clinical pharmacokinetics, 1992, Volume: 22 Suppl 1

    Topics: Adult; Anti-Infective Agents; Biological Availability; Capsules; Eating; Female; Fluoroquinolones; Humans; Male; Middle Aged; Quinolones; Solutions; Tablets

1992
Absence of drug interaction between temafloxacin and low dose heparin.
    Clinical pharmacokinetics, 1992, Volume: 22 Suppl 1

    Topics: Administration, Oral; Adolescent; Adult; Anti-Infective Agents; Blood Coagulation Factors; Drug Interactions; Fluoroquinolones; Heparin; Humans; Injections, Subcutaneous; Male; Platelet Count; Quinolones

1992
In vitro activities of five quinolones against Chlamydia pneumoniae.
    Antimicrobial agents and chemotherapy, 1992, Volume: 36, Issue:3

    Topics: Anti-Infective Agents; Chlamydophila pneumoniae; Ciprofloxacin; Fleroxacin; Fluoroquinolones; Microbial Sensitivity Tests; Ofloxacin; Quinolones

1992
Entry of lomefloxacin and temafloxacin into human neutrophils, peritoneal macrophages, and tissue culture cells.
    Diagnostic microbiology and infectious disease, 1992, Volume: 15, Issue:5

    Topics: Animals; Anti-Infective Agents; Cell Line; Cell Survival; Cells, Cultured; Fibroblasts; Fluoroquinolones; Humans; Macrophages; Neutrophils; Opsonin Proteins; Peritoneal Dialysis, Continuous Ambulatory; Quinolones; Temperature; Vero Cells

1992
Susceptibilities of penicillin-susceptible and -resistant strains of Streptococcus pneumoniae to RP 59500, vancomycin, erythromycin, PD 131628, sparfloxacin, temafloxacin, win 57273, ofloxacin, and ciprofloxacin.
    Antimicrobial agents and chemotherapy, 1992, Volume: 36, Issue:4

    Topics: Anti-Infective Agents; Ciprofloxacin; Erythromycin; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Naphthyridines; Ofloxacin; Penicillin Resistance; Quinolones; Streptococcus pneumoniae; Vancomycin; Virginiamycin

1992
Evaluation of temafloxacin in a rat model of intra-abdominal abscess.
    The Journal of antimicrobial chemotherapy, 1992, Volume: 29, Issue:6

    Topics: Abdomen; Abscess; Animals; Anti-Infective Agents; Bacteroides fragilis; Bacteroides Infections; Clindamycin; Escherichia coli Infections; Feces; Fluoroquinolones; Gentamicins; Male; Quinolones; Rats; Rats, Inbred Strains

1992
In vitro activity of temafloxacin compared with those of other agents against 100 clinical isolates of Neisseria gonorrhoeae.
    Antimicrobial agents and chemotherapy, 1992, Volume: 36, Issue:5

    Topics: Anti-Infective Agents; Drug Resistance, Microbial; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Neisseria gonorrhoeae; Quinolones

1992
Susceptibilities of 540 anaerobic gram-negative bacilli to amoxicillin, amoxicillin-BRL 42715, amoxicillin-clavulanate, temafloxacin, and clindamycin.
    Antimicrobial agents and chemotherapy, 1992, Volume: 36, Issue:5

    Topics: Amoxicillin; Amoxicillin-Potassium Clavulanate Combination; Anti-Bacterial Agents; Anti-Infective Agents; Clavulanic Acids; Clindamycin; Drug Resistance, Microbial; Drug Therapy, Combination; Fluoroquinolones; Gram-Negative Anaerobic Bacteria; In Vitro Techniques; Lactams; Microbial Sensitivity Tests; Quinolones

1992
Comparative activity of ciprofloxacin, ofloxacin, sparfloxacin, temafloxacin, CI-960, CI-990, and WIN 57273 against anaerobic bacteria.
    Antimicrobial agents and chemotherapy, 1992, Volume: 36, Issue:5

    Topics: Anti-Infective Agents; Bacteria, Anaerobic; Ciprofloxacin; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Naphthyridines; Ofloxacin; Quinolones

1992
Adverse effects prompt withdrawal of temafloxacin.
    Clinical pharmacy, 1992, Volume: 11, Issue:9

    Topics: Anti-Infective Agents; Fluoroquinolones; Humans; Product Surveillance, Postmarketing; Quinolones

1992
Kinetic disposition of temafloxacin and ciprofloxacin in a murine model of pneumococcal pneumonia. Relevance for drug efficacy.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:3

    Topics: Animals; Anti-Infective Agents; Chromatography, High Pressure Liquid; Ciprofloxacin; Female; Fluoroquinolones; Injections, Subcutaneous; Lung; Metabolic Clearance Rate; Mice; Mice, Inbred C57BL; Pneumonia, Pneumococcal; Quinolones

1992
Pharmacokinetics and biliary elimination of temafloxacin in pigs.
    The Journal of antimicrobial chemotherapy, 1992, Volume: 30, Issue:2

    Topics: Animals; Anti-Infective Agents; Bile; Chromatography, High Pressure Liquid; Duodenum; Fluoroquinolones; Intubation, Gastrointestinal; Quinolones; Spectrometry, Fluorescence; Swine

1992
Interpretive criteria for CI-960, fleroxacin and temafloxacin susceptibility tests with Haemophilus influenzae.
    European journal of clinical microbiology & infectious diseases : official publication of the European Society of Clinical Microbiology, 1992, Volume: 11, Issue:5

    Topics: Anti-Infective Agents; Fleroxacin; Fluoroquinolones; Haemophilus influenzae; Microbial Sensitivity Tests; Quinolones

1992
Efficacy of temafloxacin in experimental Streptococcus adjacens endocarditis and autoradiographic diffusion pattern of [14C]temafloxacin in cardiac vegetations.
    Antimicrobial agents and chemotherapy, 1992, Volume: 36, Issue:10

    Topics: Animals; Anti-Infective Agents; Autoradiography; Drug Therapy, Combination; Endocarditis, Bacterial; Female; Fluoroquinolones; Microbial Sensitivity Tests; Penicillin G Procaine; Quinolones; Rabbits; Streptococcal Infections; Tobramycin

1992
Interpretive criteria and quality control parameters for testing susceptibility of Haemophilus influenzae to enoxacin, ofloxacin, and temafloxacin.
    Journal of clinical microbiology, 1992, Volume: 30, Issue:11

    Topics: Anti-Infective Agents; Drug Resistance, Microbial; Enoxacin; Fluoroquinolones; Haemophilus influenzae; Humans; Microbial Sensitivity Tests; Mutation; Ofloxacin; Quality Control; Quinolones

1992
[Quality assurance for drug information].
    Lakartidningen, 1992, Dec-16, Volume: 89, Issue:51-52

    Topics: Anti-Infective Agents; Drug Information Services; Fluoroquinolones; Humans; Quality Assurance, Health Care; Quinolones; Sweden

1992
Activity of clarithromycin against Mycobacterium avium complex infection in beige mice.
    Antimicrobial agents and chemotherapy, 1992, Volume: 36, Issue:11

    Topics: Amikacin; Animals; Anti-Infective Agents; Antitubercular Agents; Clarithromycin; Clofazimine; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Therapy, Combination; Ethambutol; Female; Fluoroquinolones; Humans; Mice; Mice, Inbred C57BL; Mycobacterium avium; Mycobacterium avium Complex; Quinolones; Rifabutin; Rifampin; Rifamycins; Time Factors; Tuberculosis

1992
Activities of various quinolone antibiotics against Mycobacterium leprae in infected mice.
    Antimicrobial agents and chemotherapy, 1992, Volume: 36, Issue:11

    Topics: Animals; Anti-Infective Agents; Female; Fluoroquinolones; Leprosy; Mice; Mice, Inbred BALB C; Mycobacterium leprae; Pefloxacin; Quinolones

1992
Susceptibility of recent clinical isolates to temafloxacin (A-63004) and other antimicrobial agents.
    Drugs under experimental and clinical research, 1992, Volume: 18, Issue:8

    Topics: Anti-Infective Agents; Bacteria; Bacterial Infections; Drug Resistance, Microbial; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Quinolones

1992
Characterization of high-level quinolone resistance in Campylobacter jejuni.
    Antimicrobial agents and chemotherapy, 1991, Volume: 35, Issue:5

    Topics: Anti-Infective Agents; Campylobacter jejuni; Ciprofloxacin; DNA Topoisomerases, Type II; DNA, Superhelical; Drug Resistance, Microbial; Fluoroquinolones; Microbial Sensitivity Tests; Mutation; Nalidixic Acid; Norfloxacin; Quinolones; Topoisomerase II Inhibitors

1991
[Intra-macrophagic activity of antibiotics combinations against Mycobacterium marinum].
    Pathologie-biologie, 1991, Volume: 39, Issue:5

    Topics: Anti-Infective Agents; Antitubercular Agents; Ciprofloxacin; Clarithromycin; Dose-Response Relationship, Drug; Drug Synergism; Drug Therapy, Combination; Erythromycin; Ethambutol; Fluoroquinolones; Humans; In Vitro Techniques; Macrophages; Minocycline; Mycobacterium; Quinolones; Rifabutin; Rifamycins

1991
Activities of sparfloxacin, azithromycin, temafloxacin, and rifapentine compared with that of clarithromycin against multiplication of Mycobacterium avium complex within human macrophages.
    Antimicrobial agents and chemotherapy, 1991, Volume: 35, Issue:7

    Topics: 4-Quinolones; Acquired Immunodeficiency Syndrome; Anti-Bacterial Agents; Azithromycin; Cell Division; Clarithromycin; Erythromycin; Fluoroquinolones; Humans; In Vitro Techniques; Leprostatic Agents; Macrophages; Microbial Sensitivity Tests; Mycobacterium avium Complex; Quinolones; Rifampin

1991
Activity of new quinolones against ciprofloxacin-resistant staphylococci.
    Antimicrobial agents and chemotherapy, 1991, Volume: 35, Issue:8

    Topics: Anti-Infective Agents; Ciprofloxacin; Drug Resistance, Microbial; Fluoroquinolones; Microbial Sensitivity Tests; Naphthyridines; Ofloxacin; Quinolones; Staphylococcus

1991
The in-vitro activity of temafloxacin compared with other antimicrobial agents.
    The Journal of antimicrobial chemotherapy, 1991, Volume: 27, Issue:6

    Topics: Anti-Infective Agents; Bacteria; Ciprofloxacin; Enoxacin; Enterobacteriaceae; Fluoroquinolones; Microbial Sensitivity Tests; Ofloxacin; Quinolones; Species Specificity

1991
Fluoroquinolones in the treatment of human infection: the role of temafloxacin.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Anti-Infective Agents; Bacteria; Bacterial Infections; Fluoroquinolones; Humans; Quinolones

1991
Activity of temafloxacin and other fluoroquinolones against typical and atypical community-acquired respiratory tract pathogens.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Anti-Infective Agents; Bacteria; Ciprofloxacin; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Ofloxacin; Quinolones; Respiratory Tract Infections

1991
In vitro activity of temafloxacin against gram-positive cocci including methicillin-resistant Staphylococcus aureus.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Anti-Infective Agents; Ciprofloxacin; Enterococcus; Fluoroquinolones; Gram-Positive Cocci; Methicillin Resistance; Microbial Sensitivity Tests; Ofloxacin; Quinolones; Staphylococcus aureus; Streptococcus

1991
Fluoroquinolones for the treatment of nongonococcal urethritis/cervicitis.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Anti-Infective Agents; Female; Fluoroquinolones; Gonorrhea; Humans; Male; Quinolones; Sexually Transmitted Diseases, Bacterial; Urethritis; Uterine Cervicitis

1991
Temafloxacin: a safe antibiotic for the elderly, patients with comorbidities, and other special populations.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Age Factors; Aged; Anti-Infective Agents; Bacterial Infections; Drug Interactions; Female; Fluoroquinolones; Humans; Kidney Diseases; Male; Quinolones; Risk Factors; Sex Factors

1991
In vitro activity of temafloxacin against gram-negative bacteria: an overview.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Anti-Infective Agents; Campylobacter; Ciprofloxacin; Enterobacteriaceae; Fluoroquinolones; Gram-Negative Bacteria; Humans; Hydrogen-Ion Concentration; Microbial Sensitivity Tests; Ofloxacin; Quinolones; Respiratory Tract Infections; Sexually Transmitted Diseases, Bacterial

1991
In vitro activity of temafloxacin against pathogens causing sexually transmitted diseases.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Anti-Infective Agents; Chlamydia trachomatis; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Mycoplasma; Neisseria gonorrhoeae; Quinolones; Sexually Transmitted Diseases, Bacterial; Treponema pallidum; Ureaplasma urealyticum

1991
Mechanisms and frequency of resistance to temafloxacin.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Anti-Infective Agents; Bacteria; Drug Resistance, Microbial; Escherichia coli; Fluoroquinolones; Methicillin Resistance; Mutation; Pseudomonas aeruginosa; Quinolones; Staphylococcus aureus

1991
Comparison of organ-specific toxicity of temafloxacin in animals and humans.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Animals; Anti-Infective Agents; Central Nervous System; Eye; Fluoroquinolones; Humans; Joints; Kidney; Mutagens; Organ Specificity; Quinolones; Species Specificity

1991
Assessment of temafloxacin neurotoxicity in rodents.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Animals; Anti-Infective Agents; Central Nervous System; Ciprofloxacin; Enoxacin; Fluoroquinolones; Male; Mice; Mice, Inbred ICR; Motor Activity; Oxolinic Acid; Phenylbutyrates; Quinolones; Rats; Rats, Inbred Strains; Seizures

1991
The influence of age on the pharmacokinetics of temafloxacin.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Absorption; Administration, Oral; Adult; Aged; Aging; Anti-Infective Agents; Chromatography, High Pressure Liquid; Female; Fluoroquinolones; Humans; Male; Quinolones; Sex Factors

1991
Effect of temafloxacin on the pharmacokinetics of theophylline.
    The American journal of medicine, 1991, Dec-30, Volume: 91, Issue:6A

    Topics: Adult; Anti-Infective Agents; Drug Interactions; Female; Fluoroquinolones; Humans; Male; Middle Aged; Quinolones; Theophylline

1991
High-performance liquid chromatographic procedures for the determination of temafloxacin in biological matrices.
    Journal of chromatography, 1991, Jul-17, Volume: 568, Issue:1

    Topics: Anti-Infective Agents; Chromatography, High Pressure Liquid; Fluoroquinolones; Humans; Quinolones

1991
Anti-staphylococcal activity of temafloxacin, ciprofloxacin, ofloxacin and enoxacin.
    The Journal of antimicrobial chemotherapy, 1991, Volume: 28, Issue:5

    Topics: Anti-Infective Agents; Ciprofloxacin; Enoxacin; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Ofloxacin; Oxacillin; Penicillin Resistance; Quinolones; Staphylococcal Infections; Staphylococcus

1991
The in-vitro activity of tosufloxacin, a new fluorinated quinolone, compared with that of ciprofloxacin and temafloxacin.
    The Journal of antimicrobial chemotherapy, 1991, Volume: 28, Issue:5

    Topics: Anti-Infective Agents; Bacteria; Bacteria, Aerobic; Bacteria, Anaerobic; Ciprofloxacin; Fluoroquinolones; Microbial Sensitivity Tests; Naphthyridines; Quinolones

1991
Clinical results using two new antibiotics--clarithromycin and temafloxacin.
    Oncology (Williston Park, N.Y.), 1991, Volume: 5, Issue:10

    Topics: Acquired Immunodeficiency Syndrome; Anti-Infective Agents; Bacterial Infections; Clarithromycin; Erythromycin; Fluoroquinolones; Humans; Opportunistic Infections; Quinolones

1991
Temafloxacin: an in-vitro and clinical assessment.
    The Journal of antimicrobial chemotherapy, 1991, Volume: 28 Suppl C

    Topics: Animals; Anti-Infective Agents; Fluoroquinolones; Humans; In Vitro Techniques; Quinolones

1991
The in-vitro activity of temafloxacin, against gram-positive bacteria.
    The Journal of antimicrobial chemotherapy, 1991, Volume: 28 Suppl C

    Topics: Anti-Infective Agents; Fluoroquinolones; Gram-Positive Bacteria; Microbial Sensitivity Tests; Quinolones

1991
In-vitro activity of temafloxacin against anaerobic bacteria: a comparative study.
    The Journal of antimicrobial chemotherapy, 1991, Volume: 28 Suppl C

    Topics: Anti-Infective Agents; Bacteria, Anaerobic; Fluoroquinolones; Quinolones

1991
Pharmacokinetics of four fluoroquinolones in an animal model of infected lung.
    The Journal of antimicrobial chemotherapy, 1991, Volume: 28 Suppl C

    Topics: Animals; Anti-Infective Agents; Ciprofloxacin; Disease Models, Animal; Fluoroquinolones; Lung Diseases; Mice; Mice, Inbred Strains; Ofloxacin; Pneumococcal Infections; Quinolones; Streptococcus pneumoniae

1991
Comparative activity of fluorinated quinolones in acute and subacute Streptococcus pneumoniae pneumonia models: efficacy of temafloxacin.
    The Journal of antimicrobial chemotherapy, 1991, Volume: 28 Suppl C

    Topics: Acute Disease; Animals; Anti-Infective Agents; Disease Models, Animal; Female; Fluoroquinolones; Mice; Mice, Inbred Strains; Ofloxacin; Pneumonia; Quinolones; Streptococcus pneumoniae

1991
Comparative pharmacokinetic disposition of fluoroquinolones in the lung.
    The Journal of antimicrobial chemotherapy, 1991, Volume: 28 Suppl C

    Topics: Administration, Oral; Anti-Infective Agents; Ciprofloxacin; Fluoroquinolones; Humans; Injections, Intravenous; Lung; Quinolones

1991
In-vitro activity of temafloxacin for gram-positive pathogens.
    The Journal of antimicrobial chemotherapy, 1991, Volume: 28 Suppl C

    Topics: Anti-Infective Agents; Fluoroquinolones; Gram-Positive Bacteria; Quinolones

1991
Fluorometric and high-performance liquid chromatographic measurement of quinolone uptake by human neutrophils.
    European journal of clinical microbiology & infectious diseases : official publication of the European Society of Clinical Microbiology, 1991, Volume: 10, Issue:11

    Topics: Anti-Infective Agents; Chromatography, High Pressure Liquid; Ciprofloxacin; Fleroxacin; Fluorescence; Fluoroquinolones; Humans; Neutrophils; Norfloxacin; Ofloxacin; Quinolones

1991
ESGAB breakpoint determination: temafloxacin.
    European journal of clinical microbiology & infectious diseases : official publication of the European Society of Clinical Microbiology, 1991, Volume: 10, Issue:11

    Topics: Anti-Infective Agents; Bacteria; Bacterial Infections; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Quinolones

1991
Cross-resistance and cross-susceptibility between fluoroquinolone agents.
    European journal of clinical microbiology & infectious diseases : official publication of the European Society of Clinical Microbiology, 1991, Volume: 10, Issue:12

    Topics: Anti-Infective Agents; Ciprofloxacin; Drug Resistance, Microbial; Enoxacin; Enterobacteriaceae; Fleroxacin; Fluoroquinolones; Microbial Sensitivity Tests; Ofloxacin; Predictive Value of Tests; Quinolones

1991
Anti-Mycobacterium leprae activity of several quinolones studied in the mouse.
    International journal of leprosy and other mycobacterial diseases : official organ of the International Leprosy Association, 1991, Volume: 59, Issue:4

    Topics: Animals; Anti-Infective Agents; Ciprofloxacin; Fleroxacin; Fluoroquinolones; Leprosy; Mice; Mycobacterium leprae; Quinolones

1991
Temafloxacin pharmacokinetics in subjects with normal and impaired renal function.
    Antimicrobial agents and chemotherapy, 1991, Volume: 35, Issue:11

    Topics: Adult; Aged; Anti-Infective Agents; Fluoroquinolones; Half-Life; Humans; Kidney Diseases; Male; Middle Aged; Quinolones; Renal Dialysis; Tissue Distribution

1991
[In vitro bactericidal effect of temafloxacin and tosufloxacin against streptococci].
    Pathologie-biologie, 1991, Volume: 39, Issue:10

    Topics: Anti-Infective Agents; Ciprofloxacin; Dose-Response Relationship, Drug; Enterococcus faecalis; Enterococcus faecium; Fluoroquinolones; In Vitro Techniques; Naphthyridines; Pefloxacin; Quinolones; Streptococcus; Streptococcus agalactiae; Streptococcus bovis; Streptococcus pneumoniae; Streptococcus pyogenes; Streptococcus sanguis

1991
[In vitro effect of new fluoroquinolones and betalactamines combinations against enterococci].
    Pathologie-biologie, 1991, Volume: 39, Issue:10

    Topics: Amoxicillin; Anti-Infective Agents; Ciprofloxacin; Dose-Response Relationship, Drug; Drug Therapy, Combination; Enterococcus faecalis; Fluoroquinolones; Imipenem; In Vitro Techniques; Naphthyridines; Piperacillin; Quinolones

1991
Synthesis, antibacterial activities, and pharmacological properties of enantiomers of temafloxacin hydrochloride.
    Journal of medicinal chemistry, 1991, Volume: 34, Issue:1

    Topics: 4-Quinolones; Animals; Anti-Infective Agents; Escherichia coli; Female; Fluoroquinolones; Indicators and Reagents; Mice; Microbial Sensitivity Tests; Molecular Structure; Motor Activity; Pseudomonas aeruginosa; Quinolones; Rats; Staphylococcus aureus; Stereoisomerism; Streptococcus; Structure-Activity Relationship; Topoisomerase II Inhibitors

1991
[Experimental study on the hepatobiliary kinetics and excretion of temafloxacin. Evidence for production of active metabolites by the rabbit liver].
    Pathologie-biologie, 1991, Volume: 39, Issue:5

    Topics: 4-Quinolones; Animals; Anti-Infective Agents; Bile; Chromatography, High Pressure Liquid; Fluoroquinolones; In Vitro Techniques; Liver; Microbiological Techniques; Quinolones; Rabbits

1991
Antipneumococcal activity of ciprofloxacin, ofloxacin, and temafloxacin in an experimental mouse pneumonia model at various stages of the disease.
    The Journal of infectious diseases, 1991, Volume: 163, Issue:2

    Topics: Amoxicillin; Animals; Anti-Infective Agents; Ciprofloxacin; Disease Models, Animal; Erythromycin; Female; Fluoroquinolones; Lung; Mice; Mice, Inbred C57BL; Ofloxacin; Pneumonia, Pneumococcal; Quinolones; Sepsis; Streptococcus pneumoniae

1991
Temafloxacin: in vitro comparison with five other antibacterial agents.
    Chemotherapy, 1991, Volume: 37, Issue:2

    Topics: 4-Quinolones; Anti-Infective Agents; Fluoroquinolones; Microbial Sensitivity Tests; Quinolones; Tobramycin

1991
Activity of temafloxacin against respiratory pathogens.
    Antimicrobial agents and chemotherapy, 1991, Volume: 35, Issue:3

    Topics: Animals; Anti-Infective Agents; Bacterial Infections; Cells, Cultured; Ciprofloxacin; Dose-Response Relationship, Drug; Female; Fluoroquinolones; Gerbillinae; Gram-Positive Bacteria; Guinea Pigs; Male; Mice; Microbial Sensitivity Tests; Ofloxacin; Quinolones; Respiratory Tract Infections

1991
Determination of minor impurities in temafloxacin hydrochloride by high-performance liquid chromatography.
    Journal of chromatography, 1990, Oct-19, Volume: 519, Issue:1

    Topics: 4-Quinolones; Anti-Infective Agents; Chromatography, High Pressure Liquid; Fluoroquinolones; Quinolones

1990
In-vitro activity of sparfloxacin, a new quinolone antimicrobial agent.
    The Journal of antimicrobial chemotherapy, 1990, Volume: 26, Issue:5

    Topics: Anti-Bacterial Agents; Anti-Infective Agents; Bacteria; Blood Proteins; Ciprofloxacin; Fluoroquinolones; Humans; Lactams; Microbial Sensitivity Tests; Protein Binding; Quinolones

1990
Biliary elimination and hepatic disposition of a new fluoroquinolone, temafloxacin: experimental evaluation.
    Drugs under experimental and clinical research, 1990, Volume: 16, Issue:8

    Topics: 4-Quinolones; Animals; Anti-Infective Agents; Bile; Chromatography, Liquid; Fluoroquinolones; In Vitro Techniques; Liver; Metabolic Clearance Rate; Molecular Structure; Perfusion; Quinolones; Rabbits

1990
Correlation between disc potency and zone size in temafloxacin activity in vitro.
    Drugs under experimental and clinical research, 1990, Volume: 16, Issue:12

    Topics: 4-Quinolones; Anti-Infective Agents; Drug Evaluation; Escherichia coli; Fluoroquinolones; Humans; Klebsiella pneumoniae; Microbial Sensitivity Tests; Proteus mirabilis; Pseudomonas aeruginosa; Quinolones; Serratia marcescens; Staphylococcus aureus

1990
In vitro activity of temafloxacin hydrochloride (TA-167 or A-62254), a new fluorinated 4-quinolone.
    Chemotherapy, 1990, Volume: 36, Issue:5

    Topics: 4-Quinolones; Anti-Infective Agents; Bacteria, Aerobic; Fluoroquinolones; Gram-Positive Bacteria; Hydrogen-Ion Concentration; Magnesium; Microbial Sensitivity Tests; Quinolones; Time Factors

1990
Developmental toxicity of temafloxacin hydrochloride in the long-tailed macaque (Macaca fascicularis).
    Teratology, 1990, Volume: 42, Issue:3

    Topics: 4-Quinolones; Animals; Anti-Infective Agents; Appetite; Dose-Response Relationship, Drug; Embryonic and Fetal Development; Female; Fluoroquinolones; Macaca fascicularis; Pregnancy; Quinolones; Teratogens; Vomiting

1990
Determination of temafloxacin, sarafloxacin, and difloxacin in bulk drug and dosage forms by high-performance liquid chromatography.
    Pharmaceutical research, 1990, Volume: 7, Issue:11

    Topics: Anti-Infective Agents; Chromatography, High Pressure Liquid; Ciprofloxacin; Fluoroquinolones; Quinolones; Solubility; Spectrophotometry, Ultraviolet

1990
In vitro activities of tosufloxacin, temafloxacin, and A-56620 against pathogens of diarrhea.
    Antimicrobial agents and chemotherapy, 1990, Volume: 34, Issue:2

    Topics: Anti-Bacterial Agents; Anti-Infective Agents; Bacteria; Ciprofloxacin; Diarrhea; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Naphthyridines; Quinolones

1990
Concentrations of temafloxacin in serum and bronchial mucosa.
    European journal of clinical microbiology & infectious diseases : official publication of the European Society of Clinical Microbiology, 1990, Volume: 9, Issue:6

    Topics: 4-Quinolones; Aged; Aged, 80 and over; Anti-Infective Agents; Bronchi; Female; Fluoroquinolones; Humans; Male; Middle Aged; Mucous Membrane; Quinolones

1990
Oral temafloxacin versus vancomycin for therapy of experimental endocarditis caused by methicillin-resistant Staphylococcus aureus.
    Antimicrobial agents and chemotherapy, 1990, Volume: 34, Issue:6

    Topics: 4-Quinolones; Administration, Oral; Animals; Anti-Infective Agents; Drug Therapy, Combination; Endocarditis, Bacterial; Fluoroquinolones; Male; Methicillin; Microbial Sensitivity Tests; Penicillin Resistance; Quinolones; Rats; Rats, Inbred Strains; Rifampin; Staphylococcal Infections; Vancomycin

1990
High-performance liquid chromatography for the determination of three new fluoroquinolones, fleroxacin, temafloxacin and A-64730, in biological fluids.
    Journal of chromatography, 1989, Jul-21, Volume: 491, Issue:2

    Topics: Anti-Infective Agents; Bile; Chromatography, High Pressure Liquid; Ciprofloxacin; Fleroxacin; Fluoroquinolones; Humans; Molecular Structure; Naphthyridines; Quinolones; Spectrometry, Fluorescence

1989
Comparative antimycobacterial activities of difloxacin, temafloxacin, enoxacin, pefloxacin, reference fluoroquinolones, and a new macrolide, clarithromycin.
    Antimicrobial agents and chemotherapy, 1989, Volume: 33, Issue:4

    Topics: Anti-Bacterial Agents; Anti-Infective Agents; Ciprofloxacin; Clarithromycin; Enoxacin; Erythromycin; Fluoroquinolones; Microbial Sensitivity Tests; Mycobacterium; Pefloxacin; Quinolones

1989
Temafloxacin disk potency and tentative interpretive criteria for susceptibility tests.
    Journal of clinical microbiology, 1989, Volume: 27, Issue:12

    Topics: Anti-Infective Agents; Bacteria; Drug Resistance, Microbial; Enterobacteriaceae; Fluoroquinolones; Microbial Sensitivity Tests; Nalidixic Acid; Quinolones; Regression Analysis

1989
In vitro activities of temafloxacin (A-62254) and four other antibiotics against Chlamydia trachomatis.
    Antimicrobial agents and chemotherapy, 1989, Volume: 33, Issue:1

    Topics: 4-Quinolones; Anti-Infective Agents; Chlamydia trachomatis; Doxycycline; Drug Resistance, Microbial; Fluoroquinolones; Quinolones

1989
In-vitro activities of temafloxacin, tosufloxacin (A-61827) and five other fluoroquinolone agents.
    The Journal of antimicrobial chemotherapy, 1989, Volume: 23, Issue:4

    Topics: 4-Quinolones; Anti-Infective Agents; Bacteria; Fluoroquinolones; Methicillin; Microbial Sensitivity Tests; Naphthyridines; Penicillin Resistance; Quinolones

1989
In vitro activities of lomefloxacin and temafloxacin against pathogens causing diarrhea.
    Antimicrobial agents and chemotherapy, 1989, Volume: 33, Issue:8

    Topics: 4-Quinolones; Anti-Bacterial Agents; Anti-Infective Agents; Bacteria; Diarrhea; Fluoroquinolones; Humans; Quinolones

1989
The in-vitro activity, pharmacokinetics and tissue penetration of temafloxacin.
    The Journal of antimicrobial chemotherapy, 1989, Volume: 24, Issue:3

    Topics: 4-Quinolones; Adult; Anti-Infective Agents; Bacteria; Blister; Exudates and Transudates; Fluoroquinolones; Humans; Male; Quinolones

1989
In vitro activity of temafloxacin, a new difluoro quinolone antimicrobial agent.
    European journal of clinical microbiology & infectious diseases : official publication of the European Society of Clinical Microbiology, 1988, Volume: 7, Issue:1

    Topics: Anti-Bacterial Agents; Cefotaxime; Chemical Phenomena; Chemistry; Ciprofloxacin; Culture Media; Drug Resistance, Microbial; Enterobacteriaceae; Fluoroquinolones; Gram-Negative Bacteria; Hydrogen-Ion Concentration; Imipenem; Magnesium; Ofloxacin; Oxazines; Pseudomonas; Quinolines; Quinolones; Thienamycins

1988
Comparative in vitro activity of the new difluoro-quinolone temafloxacin (A-62254) against bacterial isolates from cancer patients.
    European journal of clinical microbiology & infectious diseases : official publication of the European Society of Clinical Microbiology, 1988, Volume: 7, Issue:5

    Topics: Anti-Infective Agents; Bacteria; Ciprofloxacin; Enterobacteriaceae; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Neoplasms; Quinolones; Staphylococcus; Streptococcus

1988
Correlation of in vitro activities of the fluoroquinolones to their in vivo efficacies.
    Drugs under experimental and clinical research, 1988, Volume: 14, Issue:6

    Topics: Animals; Anti-Infective Agents; Ciprofloxacin; Enoxacin; Fleroxacin; Fluoroquinolones; Mice; Microbial Sensitivity Tests; Naphthyridines; Norfloxacin; Ofloxacin; Pefloxacin; Quinolones

1988
Comparative antibacterial activities of temafloxacin hydrochloride (A-62254) and two reference fluoroquinolones.
    Antimicrobial agents and chemotherapy, 1987, Volume: 31, Issue:11

    Topics: Animals; Anti-Bacterial Agents; Ciprofloxacin; Drug Resistance, Microbial; Female; Fluoroquinolones; Hydrogen-Ion Concentration; Mice; Microbial Sensitivity Tests; Pyelonephritis; Quinolines; Quinolones

1987
Comparison of sparfloxacin, temafloxacin, and ciprofloxacin for prophylaxis and treatment of experimental foreign-body infection by methicillin-resistant Staphylococcus aureus.
    Antimicrobial agents and chemotherapy, 1995, Volume: 39, Issue:8

    Topics: Animals; Anti-Bacterial Agents; Anti-Infective Agents; Ciprofloxacin; Fluoroquinolones; Foreign Bodies; Guinea Pigs; Methicillin Resistance; Microbial Sensitivity Tests; Quinolones; Rats; Staphylococcal Infections; Staphylococcus aureus; Vancomycin

1995
Effect of aerobic and anaerobic environments on antistaphylococcal activities of five fluoroquinolones.
    Antimicrobial agents and chemotherapy, 1995, Volume: 39, Issue:2

    Topics: Anaerobiosis; Anti-Infective Agents; Carbonyl Cyanide m-Chlorophenyl Hydrazone; Ciprofloxacin; Fluoroquinolones; Hydrogen-Ion Concentration; Microbial Sensitivity Tests; Ofloxacin; Quinolones; Staphylococcus aureus

1995
Dissociated resistance among fluoroquinolones.
    Antimicrobial agents and chemotherapy, 1994, Volume: 38, Issue:9

    Topics: Anti-Infective Agents; Ciprofloxacin; Drug Resistance, Microbial; Fluoroquinolones; Gram-Negative Bacteria; Gram-Positive Bacteria; Microbial Sensitivity Tests; Mutation; Ofloxacin; Piperazines; Quinolones

1994
Effect of newer quinolones on the extra- and intra-cellular chemiluminescence response of human polymorphonuclear leucocytes.
    The Journal of antimicrobial chemotherapy, 1994, Volume: 34, Issue:3

    Topics: Anti-Infective Agents; Ciprofloxacin; Extracellular Space; Fluoroquinolones; Humans; Luminescent Measurements; Neutrophils; Ofloxacin; Quinolones; Reactive Oxygen Species; Tetradecanoylphorbol Acetate; Zymosan

1994
In vitro activity of the new fluoroquinolone CP-99,219.
    Antimicrobial agents and chemotherapy, 1994, Volume: 38, Issue:11

    Topics: Anti-Infective Agents; Ciprofloxacin; Fluoroquinolones; Gram-Negative Bacteria; Gram-Positive Bacteria; Microbial Sensitivity Tests; Naphthyridines; Quinolones

1994
Limited effects of temafloxacin compared with ciprofloxacin on T-lymphocyte function.
    Antimicrobial agents and chemotherapy, 1994, Volume: 38, Issue:4

    Topics: Anti-Infective Agents; Autoradiography; Blotting, Northern; Cells, Cultured; Ciprofloxacin; Fluoroquinolones; Gene Expression; Humans; In Vitro Techniques; Interferon-gamma; Interleukin-2; Phytohemagglutinins; Quinolones; RNA, Messenger; T-Lymphocytes; Thymidine

1994
Hemolytic anemia and acute renal failure associated with temafloxacin-dependent antibodies.
    American journal of hematology, 1994, Volume: 46, Issue:4

    Topics: Acute Kidney Injury; Aged; Anemia, Hemolytic; Anti-Infective Agents; Antibodies; Female; Fluoroquinolones; Humans; Male; Middle Aged; Quinolones

1994
Dextranase enhances antibiotic efficacy in experimental viridans streptococcal endocarditis.
    Antimicrobial agents and chemotherapy, 1994, Volume: 38, Issue:5

    Topics: Animals; Anti-Bacterial Agents; Anti-Infective Agents; Dextranase; Drug Synergism; Endocarditis, Bacterial; Female; Fluoroquinolones; Lipopolysaccharides; Microbial Sensitivity Tests; Microscopy, Electron; Quinolones; Rabbits; Streptococcal Infections; Streptococcus sanguis

1994
Measurement of temafloxacin in human scalp hair as an index of drug exposure.
    Journal of pharmaceutical sciences, 1994, Volume: 83, Issue:1

    Topics: Adult; Anti-Infective Agents; Drug Monitoring; Fluoroquinolones; Hair; Humans; Male; Quinolones; Scalp

1994
Microbial identification and antibiotic sensitivity testing, an aid for patients refractory to periodontal therapy. A report of 3 cases.
    Journal of clinical periodontology, 1994, Volume: 21, Issue:2

    Topics: Adult; Aggregatibacter actinomycetemcomitans; Amoxicillin; Anti-Infective Agents; Clindamycin; Drug Resistance, Microbial; Fluoroquinolones; Humans; Male; Microbial Sensitivity Tests; Periodontal Abscess; Periodontitis; Quinolones; Staphylococcus aureus; Tetracycline Resistance

1994
In vitro postantibiotic effect following repeated exposure to imipenem, temafloxacin, and tobramycin.
    Antimicrobial agents and chemotherapy, 1993, Volume: 37, Issue:8

    Topics: Anti-Infective Agents; Fluoroquinolones; Humans; Imipenem; Microbial Sensitivity Tests; Pseudomonas aeruginosa; Quinolones; Time Factors; Tobramycin

1993
Susceptibilities of Mycoplasma hominis, Mycoplasma pneumoniae, and Ureaplasma urealyticum to a new quinolone, OPC 17116.
    Antimicrobial agents and chemotherapy, 1993, Volume: 37, Issue:8

    Topics: Anti-Infective Agents; Fluoroquinolones; Microbial Sensitivity Tests; Mycoplasma; Mycoplasma pneumoniae; Ofloxacin; Piperazines; Quinolones; Ureaplasma urealyticum

1993
Correlation between umuC induction and Salmonella mutagenicity assay for quinolone antimicrobial agents.
    FEMS microbiology letters, 1993, Sep-15, Volume: 112, Issue:3

    Topics: Anti-Infective Agents; Bacterial Proteins; Ciprofloxacin; DNA-Directed DNA Polymerase; Enoxacin; Escherichia coli; Escherichia coli Proteins; Fluoroquinolones; Gene Expression Regulation, Bacterial; Mutagenicity Tests; Nalidixic Acid; Naphthyridines; Norfloxacin; Quinolones; Salmonella typhimurium; SOS Response, Genetics; Species Specificity

1993
New drugs from 1991-1992.
    Texas dental journal, 1993, Volume: 110, Issue:7

    Topics: 1-Naphthylamine; Anti-Bacterial Agents; Anti-Infective Agents; Anticholesteremic Agents; Antineoplastic Agents; Antiviral Agents; Azithromycin; Butanones; Cardiovascular Agents; Clarithromycin; Drug Approval; Drug Combinations; Drug Interactions; Enoxacin; Finasteride; Flumazenil; Fluoroquinolones; Humans; Ketorolac Tromethamine; Lactams; Nabumetone; Pyridines; Quinolones; Sertraline; Tolmetin; Tromethamine; United States; United States Food and Drug Administration; Zolpidem

1993
Evaluation of activity of temafloxacin against Bacteroides fragilis by an in vitro pharmacodynamic system.
    Antimicrobial agents and chemotherapy, 1993, Volume: 37, Issue:11

    Topics: Anaerobiosis; Anti-Infective Agents; Bacteroides fragilis; Cefotetan; Ciprofloxacin; Colony Count, Microbial; Culture Media; Fluoroquinolones; Microbial Sensitivity Tests; Quinolones

1993
Induction of resistance of Streptococcus pneumoniae to quinolones in vitro.
    Chemotherapy, 1993, Volume: 39, Issue:1

    Topics: Anti-Infective Agents; Ciprofloxacin; Drug Resistance, Microbial; Fluoroquinolones; Levofloxacin; Microbial Sensitivity Tests; Norfloxacin; Ofloxacin; Quinolones; Streptococcus pneumoniae

1993
Selection of a fluoroquinolone-class disk for susceptibility tests.
    The American journal of medicine, 1993, Mar-22, Volume: 94, Issue:3A

    Topics: Anti-Infective Agents; Fluoroquinolones; Microbial Sensitivity Tests; Quinolones

1993
Effects of new quinolones on Mycoplasma pneumoniae-infected hamsters.
    Antimicrobial agents and chemotherapy, 1993, Volume: 37, Issue:2

    Topics: Animals; Anti-Infective Agents; Antibodies, Bacterial; Ciprofloxacin; Cricetinae; Female; Fluoroquinolones; Half-Life; Humans; Lung; Mesocricetus; Mycoplasma pneumoniae; Ofloxacin; Pneumonia, Mycoplasma; Quinolones

1993
The withdrawal of temafloxacin. Are there implications for other quinolones?
    Drug safety, 1993, Volume: 8, Issue:1

    Topics: Adult; Adverse Drug Reaction Reporting Systems; Anti-Infective Agents; Drug and Narcotic Control; Fluoroquinolones; Humans; Quinolones; United States; United States Food and Drug Administration

1993
Effect of pH variation on the susceptibility of Helicobacter pylori to three macrolide antimicrobial agents and temafloxacin.
    European journal of clinical microbiology & infectious diseases : official publication of the European Society of Clinical Microbiology, 1993, Volume: 12, Issue:2

    Topics: Anti-Bacterial Agents; Anti-Infective Agents; Azithromycin; Clarithromycin; Drug Resistance, Microbial; Erythromycin; Fluoroquinolones; Helicobacter pylori; Humans; Hydrogen-Ion Concentration; Microbial Sensitivity Tests; Quinolones

1993
In-vitro activity of ciprofloxacin, temafloxacin, azithromycin, clarithromycin and metronidazole against Giardia lamblia.
    The Journal of antimicrobial chemotherapy, 1993, Volume: 31, Issue:4

    Topics: Animals; Anti-Infective Agents; Azithromycin; Ciprofloxacin; Clarithromycin; Erythromycin; Fluoroquinolones; Giardia lamblia; Metronidazole; Microbial Sensitivity Tests; Quinolones

1993
Comparative susceptibilities of 173 aerobic and anaerobic bite wound isolates to sparfloxacin, temafloxacin, clarithromycin, and older agents.
    Antimicrobial agents and chemotherapy, 1993, Volume: 37, Issue:5

    Topics: Animals; Anti-Bacterial Agents; Bacteria, Aerobic; Bacteria, Anaerobic; Bites and Stings; Clarithromycin; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Quinolones; Wound Infection

1993
Temafloxacin-induced hemolytic anemia and renal failure.
    Clinical pharmacy, 1993, Volume: 12, Issue:5

    Topics: Acute Kidney Injury; Anemia, Hemolytic; Anti-Infective Agents; Bacterial Infections; Erythrocytes; Female; Fluoroquinolones; Hemolysis; Humans; Immune Complex Diseases; Middle Aged; Quinolones

1993
In vitro susceptibility of anaerobic bacteria to temafloxacin.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 1993, Volume: 16 Suppl 4

    Topics: Anti-Infective Agents; Bacteria, Anaerobic; Drug Resistance, Microbial; Fluoroquinolones; Humans; In Vitro Techniques; Microbial Sensitivity Tests; Quinolones

1993
Time-kill studies of the activity of temafloxacin against four strains of Bacteroides.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 1993, Volume: 16 Suppl 4

    Topics: Anti-Infective Agents; Bacteroides; Bacteroides fragilis; Drug Resistance, Microbial; Fluoroquinolones; Humans; In Vitro Techniques; Microbial Sensitivity Tests; Quinolones; Species Specificity

1993
In-vitro evaluation of clarithromycin, temafloxacin, and ethambutol in combination against Mycobacterium avium complex.
    The Journal of antimicrobial chemotherapy, 1993, Volume: 31, Issue:5

    Topics: Acquired Immunodeficiency Syndrome; Anti-Infective Agents; Clarithromycin; Drug Synergism; Drug Therapy, Combination; Ethambutol; Evaluation Studies as Topic; Fluoroquinolones; Humans; Macrophages; Microbial Sensitivity Tests; Mycobacterium avium Complex; Mycobacterium avium-intracellulare Infection; Quinolones

1993
Developmental toxicity of fleroxacin and comparative pharmacokinetics of four fluoroquinolones in the cynomolgus macaque (Macaca fascicularis).
    Toxicology and applied pharmacology, 1993, Volume: 122, Issue:1

    Topics: Administration, Oral; Animals; Anti-Infective Agents; Ciprofloxacin; Embryo, Mammalian; Female; Fleroxacin; Fluoroquinolones; Macaca fascicularis; Norfloxacin; Pregnancy; Pregnancy, Animal; Quinolones

1993
Bactericidal index: a new way to assess quinolone bactericidal activity in vitro.
    The Journal of antimicrobial chemotherapy, 1997, Volume: 39, Issue:6

    Topics: Anti-Infective Agents; Ciprofloxacin; Enterococcus faecalis; Fluoroquinolones; Microbial Sensitivity Tests; Naphthyridines; Ofloxacin; Quinolones

1997
Effects of fluoroquinolones and magnesium deficiency in murine limb bud cultures.
    Archives of toxicology, 1998, Volume: 72, Issue:7

    Topics: Animals; Anti-Infective Agents; Ciprofloxacin; Dose-Response Relationship, Drug; Embryo, Mammalian; Embryonic and Fetal Development; Extremities; Fleroxacin; Fluoroquinolones; Magnesium Deficiency; Mice; Microscopy, Electron; Ofloxacin; Pefloxacin; Quinolones

1998
The effects of increasing levels of quinolone resistance on in-vitro activity of four quinolones.
    The Journal of antimicrobial chemotherapy, 1998, Volume: 42, Issue:2

    Topics: Anti-Infective Agents; Ciprofloxacin; Drug Resistance, Microbial; Fluoroquinolones; Gram-Negative Bacteria; Gram-Positive Bacteria; Humans; Microbial Sensitivity Tests; Mutation; Nalidixic Acid; Ofloxacin; Quinolones

1998
In-vitro activity of three fluoroquinolones, cefotaxime and clindamycin against staphylococci.
    Zentralblatt fur Bakteriologie : international journal of medical microbiology, 1995, Volume: 282, Issue:4

    Topics: Aminoglycosides; Anti-Bacterial Agents; Anti-Infective Agents; Cefotaxime; Cephalosporins; Ciprofloxacin; Clindamycin; Fluoroquinolones; Humans; Microbial Sensitivity Tests; Ofloxacin; Quinolones; Staphylococcal Infections; Staphylococcus

1995
A simple, inexpensive apparatus for performance of preparative scale solution phase multiple parallel synthesis of drug analogs. II. Biological evaluation of a retrospective library of quinolone antiinfective agents.
    Combinatorial chemistry & high throughput screening, 1998, Volume: 1, Issue:2

    Topics: Anti-Infective Agents; Chemistry, Pharmaceutical; DNA; DNA Topoisomerases, Type II; Drug Evaluation, Preclinical; Enzyme Inhibitors; Fluoroquinolones; Microbial Sensitivity Tests; Mycobacterium; Quinolones; Reference Values; Solutions; Structure-Activity Relationship; Topoisomerase II Inhibitors

1998
Ultrastructural characterization of murine limb buds after in vitro exposure to grepafloxacin and other fluoroquinolones.
    Archives of toxicology, 2002, Volume: 75, Issue:11-12

    Topics: Abnormalities, Drug-Induced; Animals; Anti-Infective Agents; Calcium; Dose-Response Relationship, Drug; Embryo, Mammalian; Female; Fluoroquinolones; In Vitro Techniques; Levofloxacin; Limb Buds; Magnesium; Male; Mice; Mice, Inbred Strains; Ofloxacin; Piperazines; Pregnancy; Quinolones

2002
[Drug interactions between nonsteroidal anti-inflammatory drug and pazufloxacin mesilate, a new quinolone antibacterial agent for intravenous use: convulsions in mice after intravenous or intracerebroventricular administration].
    The Japanese journal of antibiotics, 2002, Volume: 55, Issue:3

    Topics: Administration, Oral; Animals; Anti-Bacterial Agents; Anti-Infective Agents; Anti-Inflammatory Agents, Non-Steroidal; beta-Alanine; Biphenyl Compounds; Cefazolin; Cilastatin; Cilastatin, Imipenem Drug Combination; Ciprofloxacin; Convulsants; Drug Combinations; Drug Interactions; Enoxacin; Fleroxacin; Fluoroquinolones; Imipenem; Injections, Intravenous; Injections, Intraventricular; Male; Mice; Mice, Inbred ICR; Norfloxacin; Oxazines; Penicillin G; Quinolones; Seizures; Thienamycins

2002
Effects of fluoroquinolones on insulin secretion and beta-cell ATP-sensitive K+ channels.
    European journal of pharmacology, 2004, Aug-16, Volume: 497, Issue:1

    Topics: Adenosine Triphosphate; Animals; Anti-Bacterial Agents; Cells, Cultured; Fluoroquinolones; Gatifloxacin; Insulin; Insulin Secretion; Islets of Langerhans; Levofloxacin; Mice; Ofloxacin; Patch-Clamp Techniques; Potassium Channels; Quinolones

2004