tele-methylhistamine and piperidines

tele-methylhistamine has been researched along with piperidines in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19903 (25.00)18.7374
1990's1 (8.33)18.2507
2000's4 (33.33)29.6817
2010's3 (25.00)24.3611
2020's1 (8.33)2.80

Authors

AuthorsStudies
Itoh, Y; Nishibori, M; Oishi, R; Saeki, K1
Garbarg, M; Gros, C; Pollard, H; Schwartz, JC; Trung Tuong, MD1
Oishi, R1
Morisset, S; Schwartz, JC; Traiffort, E1
Oreland, L; Sakurai, E; Singh Jossan, S; Tanaka, Y; Watanabe, T1
Barnes, W; Boyd, D; Hough, L1
Anaclet, C; Arrang, JM; Berrebi-Bertrand, I; Bertaina-Anglade, V; Calmels, TP; Camelin, JC; d'Aniello, F; Ganellin, CR; Gbahou, F; la Rochelle, CD; Landais, L; Lecomte, JM; Ligneau, X; Lin, JS; Parmentier, R; Perrin, D; Rouleau, A; Schunack, W; Schwartz, JC; Stark, H1
Chiba, S; Itateyama, E; Sakata, T; Yoshimatsu, H1
Armand, V; Arrang, JM; Bayard, C; Burban, A; Faucard, R; Vorobjev, V1
Groeber, E; Li, W; Liu, J; Schmidt, CJ; Steenwyk, R; Tella, M; Tingley, FD; Tseng, E; Yang, X; Zhang, Y1
Korosteleva, AS; Potapieva, NN; Shteinikov, VY; Tikhonov, DB; Tikhonova, TB1
Badange, R; Benade, V; Bhyrapuneni, G; Daripelli, S; Jasti, V; Jayarajan, P; Kamuju, V; Mekala, VR; Muddana, NR; Nirogi, R; Petlu, S; Shinde, A; Subramanian, R1

Reviews

1 review(s) available for tele-methylhistamine and piperidines

ArticleYear
[Turnover of brain histamine and its changes by various drugs].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1988, Volume: 92, Issue:5

    Topics: Anesthetics; Animals; Brain; Circadian Rhythm; Dronabinol; Ethanol; Half-Life; Histamine; Methylhistamines; Piperidines; Psychotropic Drugs

1988

Other Studies

11 other study(ies) available for tele-methylhistamine and piperidines

ArticleYear
Effects of the histamine H3-agonist (R)-alpha-methylhistamine and the antagonist thioperamide on histamine metabolism in the mouse and rat brain.
    Journal of neurochemistry, 1989, Volume: 52, Issue:5

    Topics: Amygdala; Animals; Brain; Cerebral Cortex; Histamine; Histamine Antagonists; Kinetics; Male; Methylhistamines; Mice; Pargyline; Piperidines; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H3; Tissue Distribution

1989
Sensitive radioimmunoassays for histamine and tele-methylhistamine in the brain.
    Journal of neurochemistry, 1989, Volume: 53, Issue:6

    Topics: Animals; Brain Chemistry; Cerebral Cortex; Chromatography, High Pressure Liquid; Cross Reactions; Histamine; Histidine Decarboxylase; Male; Methylhistamines; Methylhistidines; Organ Specificity; Pargyline; Piperidines; Radioimmunoassay; Rats; Rats, Inbred Strains; Reference Values; Tritium

1989
Inhibition of histamine versus acetylcholine metabolism as a mechanism of tacrine activity.
    European journal of pharmacology, 1996, Nov-07, Volume: 315, Issue:1

    Topics: Animals; Cerebral Cortex; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Histamine Antagonists; Histamine N-Methyltransferase; Male; Methylhistamines; Mice; Nootropic Agents; Piperidines; Tacrine

1996
Effects of histamine H3-receptor ligands on brain monoamine oxidase in various mammalian species.
    Brain research, 2001, Jul-06, Volume: 906, Issue:1-2

    Topics: Aged; Animals; Binding, Competitive; Dose-Response Relationship, Drug; Histamine; Histamine Agonists; Histamine Antagonists; Humans; Hypothalamus; Imidazoles; Ligands; Macaca; Methylhistamines; Middle Aged; Monoamine Oxidase; Neurons; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Subcellular Fractions; Synaptic Transmission

2001
Dynamics of histamine H(3) receptor antagonists on brain histamine metabolism: do all histamine H(3) receptor antagonists act at a single site?
    European journal of pharmacology, 2001, Nov-16, Volume: 431, Issue:2

    Topics: Analysis of Variance; Animals; Binding Sites; Brain; Histamine; Histamine Antagonists; Imidazoles; Male; Methylhistamines; Mice; Pargyline; Piperidines; Rats; Receptors, Histamine H3; Thiourea

2001
BF2.649 [1-{3-[3-(4-Chlorophenyl)propoxy]propyl}piperidine, hydrochloride], a nonimidazole inverse agonist/antagonist at the human histamine H3 receptor: Preclinical pharmacology.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 320, Issue:1

    Topics: Acetylcholine; Animals; Cats; Dopamine; Electroencephalography; Guinea Pigs; Histamine Agonists; Histamine Antagonists; Histamine Release; Humans; Imidazoles; Male; Methylhistamines; Mice; Mice, Inbred C57BL; Piperidines; Prefrontal Cortex; Receptors, Histamine H3; Scopolamine

2007
Acute central administration of immepip, a histamine H3 receptor agonist, suppresses hypothalamic histamine release and elicits feeding behavior in rats.
    Brain research bulletin, 2009, Apr-06, Volume: 79, Issue:1

    Topics: Analysis of Variance; Animals; Catheterization; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Feeding Behavior; Histamine Agonists; Histamine Release; Hypokinesia; Hypothalamus; Imidazoles; Injections, Intraventricular; Linear Models; Male; Methylhistamines; Piperidines; Rats; Rats, Wistar; Receptors, Histamine H3

2009
Histamine potentiates N-methyl-D-aspartate receptors by interacting with an allosteric site distinct from the polyamine binding site.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 332, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Allosteric Site; Animals; Binding Sites; Calcium; Dizocilpine Maleate; Drug Synergism; Hippocampus; Histamine; In Vitro Techniques; Intracellular Space; Male; Methylhistamines; N-Methylaspartate; Neurons; Norepinephrine; Piperidines; Polyamines; Radioligand Assay; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Spermine; Synaptosomes

2010
Development and validation of a sample stabilization strategy and a UPLC-MS/MS method for the simultaneous quantitation of acetylcholine (ACh), histamine (HA), and its metabolites in rat cerebrospinal fluid (CSF).
    Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 2011, Jul-15, Volume: 879, Issue:22

    Topics: Acetylcholine; Animals; Benzofurans; Cholinesterase Inhibitors; Chromatography, High Pressure Liquid; Donepezil; Drug Stability; Histamine; Hydrophobic and Hydrophilic Interactions; Imidazoles; Indans; Male; Methylhistamines; Piperidines; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Sensitivity and Specificity; Tandem Mass Spectrometry

2011
Ligands of histamine receptors modulate acid-sensing ion channels.
    Biochemical and biophysical research communications, 2017, 09-02, Volume: 490, Issue:4

    Topics: Acid Sensing Ion Channels; Animals; CHO Cells; Cricetulus; Dimaprit; Gene Expression Regulation; Histamine; Histamine Agonists; Histamine Antagonists; Humans; Hydrogen-Ion Concentration; Ligands; Methylhistamines; Patch-Clamp Techniques; Piperidines; Receptors, Histamine; Recombinant Proteins; Signal Transduction

2017
Samelisant (SUVN-G3031), a potent, selective and orally active histamine H3 receptor inverse agonist for the potential treatment of narcolepsy: pharmacological and neurochemical characterisation.
    Psychopharmacology, 2021, Volume: 238, Issue:6

    Topics: Animals; Electroencephalography; Histamine; Histamine Agonists; Humans; Male; Methylhistamines; Mice; Mice, Inbred C57BL; Mice, Knockout; Morpholines; Narcolepsy; Orexins; Piperidines; Rats; Rats, Wistar; Sleep; Wakefulness

2021