tbc-11251 has been researched along with enkephalin, d-penicillamine (2,5)- in 1 studies
Studies (tbc-11251) | Trials (tbc-11251) | Recent Studies (post-2010) (tbc-11251) | Studies (enkephalin, d-penicillamine (2,5)-) | Trials (enkephalin, d-penicillamine (2,5)-) | Recent Studies (post-2010) (enkephalin, d-penicillamine (2,5)-) |
---|---|---|---|---|---|
167 | 32 | 58 | 1,314 | 0 | 73 |
Protein | Taxonomy | tbc-11251 (IC50) | enkephalin, d-penicillamine (2,5)- (IC50) |
---|---|---|---|
Mu-type opioid receptor | Homo sapiens (human) | 0.0016 | |
Delta-type opioid receptor | Homo sapiens (human) | 0.0011 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 1 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Brouwer, K; Gorczynski, R; Hartman, JC; Mandagere, A; Melvin, L | 1 |
1 other study(ies) available for tbc-11251 and enkephalin, d-penicillamine (2,5)-
Article | Year |
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Evaluation of the endothelin receptor antagonists ambrisentan, darusentan, bosentan, and sitaxsentan as substrates and inhibitors of hepatobiliary transporters in sandwich-cultured human hepatocytes.
Topics: Adolescent; Adult; Aged; Antihypertensive Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Bosentan; Cell Culture Techniques; Cells, Cultured; Endothelin Receptor Antagonists; Enkephalin, D-Penicillamine (2,5)-; Estradiol; Female; Hepatocytes; Humans; Isoxazoles; Male; Middle Aged; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Organic Anion Transporters; Organic Anion Transporters, Sodium-Dependent; Phenylpropionates; Pyridazines; Pyrimidines; Sulfonamides; Symporters; Taurocholic Acid; Thiophenes; Young Adult | 2010 |