Page last updated: 2024-09-05

tbc-11251 and enalapril

tbc-11251 has been researched along with enalapril in 3 studies

Compound Research Comparison

Studies
(tbc-11251)
Trials
(tbc-11251)
Recent Studies (post-2010)
(tbc-11251)
Studies
(enalapril)
Trials
(enalapril)
Recent Studies (post-2010) (enalapril)
16732586,3111,924859

Protein Interaction Comparison

ProteinTaxonomytbc-11251 (IC50)enalapril (IC50)
Angiotensin-converting enzyme Homo sapiens (human)0.3536
Angiotensin-converting enzymeOryctolagus cuniculus (rabbit)2.7083
Type-2 angiotensin II receptorRattus norvegicus (Norway rat)1.2
Angiotensin-converting enzymeRattus norvegicus (Norway rat)0.14
Angiotensin-converting enzyme 2 Homo sapiens (human)0.14

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's2 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Clark, AL; Cleland, JG; Coletta, AP; Lammiman, M; Loh, H; Nasir, M; Witte, KK1

Reviews

2 review(s) available for tbc-11251 and enalapril

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Clinical trials update from the European Society of Cardiology meeting 2005: CARE-HF extension study, ESSENTIAL, CIBIS-III, S-ICD, ISSUE-2, STRIDE-2, SOFA, IMAGINE, PREAMI, SIRIUS-II and ACTIVE.
    European journal of heart failure, 2005, Volume: 7, Issue:6

    Topics: Cardiac Pacing, Artificial; Cardiology; Congresses as Topic; Defibrillators, Implantable; Enalapril; Enoximone; Europe; Female; Follow-Up Studies; Heart Failure; Humans; Isoxazoles; Male; Randomized Controlled Trials as Topic; Risk Assessment; Severity of Illness Index; Societies, Medical; Survival Analysis; Thiophenes; Treatment Outcome

2005

Other Studies

1 other study(ies) available for tbc-11251 and enalapril

ArticleYear
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010