Page last updated: 2024-08-17

taurocholic acid and glyburide

taurocholic acid has been researched along with glyburide in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (9.09)18.2507
2000's8 (72.73)29.6817
2010's2 (18.18)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hagenbuch, B; Meier, PJ; Noe, J; St-Pierre, MV1
Funk, C; Gasser, R; Jehle, L; Lazendic, M; Pantze, M; Ponelle, C; Scheuermann, G1
Byrne, JA; Higgins, CF; Linton, KJ; Mieli-Vergani, G; Strautnieks, SS; Thompson, RJ1
Artursson, P; Bergström, CA; Hoogstraate, J; Matsson, P; Norinder, U; Pedersen, JM1
Benet, LZ; Brouwer, KL; Chu, X; Dahlin, A; Evers, R; Fischer, V; Giacomini, KM; Hillgren, KM; Hoffmaster, KA; Huang, SM; Ishikawa, T; Keppler, D; Kim, RB; Lee, CA; Niemi, M; Polli, JW; Sugiyama, Y; Swaan, PW; Tweedie, DJ; Ware, JA; Wright, SH; Yee, SW; Zamek-Gliszczynski, MJ; Zhang, L1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Hanrahan, JW; Linsdell, P1
Fattinger, K; Kullak-Ublick, GA; Madon, J; Meier, PJ; Stieger, B1
Fattinger, K; Funk, C; Meier, PJ; Pantze, M; Reichen, J; Stieger, B; Weber, C1
Burliegh, J; Cai, H; Hanson, J; Kostrubsky, VE; Rose, K; Sahi, J; Sinclair, JF; Strom, SC; Urda, E; Zocharski, P1
Löbenberg, R; Wei, H1

Reviews

1 review(s) available for taurocholic acid and glyburide

ArticleYear
Membrane transporters in drug development.
    Nature reviews. Drug discovery, 2010, Volume: 9, Issue:3

    Topics: Animals; Computer Simulation; Decision Trees; Drug Approval; Drug Discovery; Drug Evaluation, Preclinical; Drug Interactions; Humans; Membrane Transport Proteins; Mice; Mice, Knockout; Prescription Drugs

2010

Other Studies

10 other study(ies) available for taurocholic acid and glyburide

ArticleYear
Characterization of the mouse bile salt export pump overexpressed in the baculovirus system.
    Hepatology (Baltimore, Md.), 2001, Volume: 33, Issue:5

    Topics: Adenosine Triphosphatases; Amino Acid Sequence; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Baculoviridae; Biological Transport; Blotting, Southern; Cell Line; DNA, Complementary; Gene Expression; Insecta; Mice; Molecular Sequence Data; Phosphorylation; Precipitin Tests

2001
Troglitazone-induced intrahepatic cholestasis by an interference with the hepatobiliary export of bile acids in male and female rats. Correlation with the gender difference in troglitazone sulfate formation and the inhibition of the canalicular bile salt
    Toxicology, 2001, Oct-05, Volume: 167, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Biliary Tract; Biological Transport, Active; Cholestasis, Intrahepatic; Chromans; Cytosol; Female; Glyburide; Hypoglycemic Agents; Liver; Male; Rats; Rats, Wistar; Sex Factors; Sulfates; Taurocholic Acid; Thiazoles; Thiazolidinediones; Troglitazone

2001
The human bile salt export pump: characterization of substrate specificity and identification of inhibitors.
    Gastroenterology, 2002, Volume: 123, Issue:5

    Topics: Adenosine Triphosphatases; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Binding, Competitive; Carrier Proteins; Cloning, Molecular; Cyclosporine; DNA, Complementary; Enzyme Inhibitors; Glyburide; Humans; Rifampin; Substrate Specificity

2002
Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).
    Journal of medicinal chemistry, 2008, Jun-12, Volume: 51, Issue:11

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Antipsychotic Agents; Antiviral Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Cell Line; Computer Simulation; Cytochrome P-450 Enzyme System; Drug-Related Side Effects and Adverse Reactions; Estradiol; Humans; Insecta; Liver; Models, Molecular; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pharmaceutical Preparations; Pharmacology; Structure-Activity Relationship

2008
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
Substrates of multidrug resistance-associated proteins block the cystic fibrosis transmembrane conductance regulator chloride channel.
    British journal of pharmacology, 1999, Volume: 126, Issue:6

    Topics: Animals; ATP-Binding Cassette Transporters; Calcium Channel Blockers; Chlorides; CHO Cells; Cholates; Cricetinae; Cystic Fibrosis Transmembrane Conductance Regulator; Dose-Response Relationship, Drug; Electric Stimulation; Estradiol; Glyburide; Membrane Potentials; Multidrug Resistance-Associated Proteins; ortho-Aminobenzoates; Stilbenes; Taurocholic Acid; Taurolithocholic Acid

1999
Drug- and estrogen-induced cholestasis through inhibition of the hepatocellular bile salt export pump (Bsep) of rat liver.
    Gastroenterology, 2000, Volume: 118, Issue:2

    Topics: Adenosine Triphosphate; Animals; Anion Transport Proteins; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Biological Transport; Carrier Proteins; Cell Line; Cyclosporine; Estradiol; Glyburide; Kinetics; Liver; Rats; Recombinant Proteins; Rifampin; Rifamycins; Spodoptera; Taurocholic Acid; Transfection

2000
The endothelin antagonist bosentan inhibits the canalicular bile salt export pump: a potential mechanism for hepatic adverse reactions.
    Clinical pharmacology and therapeutics, 2001, Volume: 69, Issue:4

    Topics: Animals; Antihypertensive Agents; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Bile Canaliculi; Bosentan; Cholestasis, Intrahepatic; Clinical Trials as Topic; Dose-Response Relationship, Drug; Drug Combinations; Endothelin Receptor Antagonists; Glyburide; Humans; Hypertension; Liver; Male; Rats; Rats, Sprague-Dawley; Rats, Wistar; Sulfonamides; Taurocholic Acid

2001
Evaluation of hepatotoxic potential of drugs by inhibition of bile-acid transport in cultured primary human hepatocytes and intact rats.
    Toxicological sciences : an official journal of the Society of Toxicology, 2003, Volume: 76, Issue:1

    Topics: Animals; Bile Acids and Salts; Biological Transport; Cells, Cultured; Culture Media; Drug Evaluation, Preclinical; Drug Synergism; Glyburide; Hepatocytes; Humans; Injections, Intravenous; Liver; Macrolides; Rats; Rats, Sprague-Dawley; Taurocholic Acid; Thiazines; Time Factors

2003
Biorelevant dissolution media as a predictive tool for glyburide a class II drug.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2006, Volume: 29, Issue:1

    Topics: Algorithms; Area Under Curve; Caco-2 Cells; Chemistry, Pharmaceutical; Chromatography, High Pressure Liquid; Computer Simulation; Glyburide; Humans; Hydrogen-Ion Concentration; Hypoglycemic Agents; Permeability; Phosphatidylcholines; Predictive Value of Tests; Solubility; Tablets; Taurocholic Acid

2006