Page last updated: 2024-09-04

tariquidar and xr 9577

tariquidar has been researched along with xr 9577 in 2 studies

Compound Research Comparison

Studies
(tariquidar)
Trials
(tariquidar)
Recent Studies (post-2010)
(tariquidar)
Studies
(xr 9577)
Trials
(xr 9577)
Recent Studies (post-2010) (xr 9577)
21016138805

Protein Interaction Comparison

ProteinTaxonomytariquidar (IC50)xr 9577 (IC50)
ATP-dependent translocase ABCB1Mus musculus (house mouse)0.3181
ATP-dependent translocase ABCB1Homo sapiens (human)0.4002
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)0.7516

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Globisch, C; Müller, H; Pajeva, IK; Wiese, M1
Müller, H; Pick, A; Wiese, M1

Other Studies

2 other study(ies) available for tariquidar and xr 9577

ArticleYear
Functional assay and structure-activity relationships of new third-generation P-glycoprotein inhibitors.
    Bioorganic & medicinal chemistry, 2008, Mar-01, Volume: 16, Issue:5

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line, Tumor; Humans; Ligands; Models, Molecular; Molecular Structure; ortho-Aminobenzoates; Quantitative Structure-Activity Relationship

2008
Structure-activity relationships of new inhibitors of breast cancer resistance protein (ABCG2).
    Bioorganic & medicinal chemistry, 2008, Sep-01, Volume: 16, Issue:17

    Topics: ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Breast Neoplasms; Crystallography, X-Ray; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Female; Humans; Models, Molecular; Molecular Structure; Neoplasm Proteins; Phthalic Acids; Quantitative Structure-Activity Relationship; Quinolines; Reproducibility of Results; Stereoisomerism; Time Factors; Tumor Cells, Cultured

2008