Page last updated: 2024-09-04

tariquidar and rhodamine 123

tariquidar has been researched along with rhodamine 123 in 9 studies

Compound Research Comparison

Studies
(tariquidar)
Trials
(tariquidar)
Recent Studies (post-2010)
(tariquidar)
Studies
(rhodamine 123)
Trials
(rhodamine 123)
Recent Studies (post-2010) (rhodamine 123)
210161381,76010424

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (33.33)29.6817
2010's6 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Berridge, G; Callaghan, R; Charlton, P; Higgins, CF; Martin, C; Mistry, P1
Ambudkar, SV; Barnett, D; Bates, SE; Finley, EM; Fojo, T; Oldham, RK; Robey, RW; Shukla, S1
Davies, HA; Lopez-Ramirez, MA; Loughlin, AJ; Male, AD; Male, DK; Reddy, PS; Romero, IA; Tai, LM1
Mongayt, D; Patel, NR; Rathi, A; Torchilin, VP1
Li, H; Shen, GL; Sun, HX; Yuan, M; Zhuang, XM1
Baum, L; Chanteux, H; Kwan, P; Zhang, C; Zuo, Z1
Christlieb, M; Marighetti, F; Pajeva, IK; Steggemann, K; Sterz, K; Wiese, M1
Jara, GE; Pierini, AB; Vera, DM1
Bi, X; Cui, J; Gao, Y; Huang, W; Li, Z; Liu, C; Qian, H; Shi, W; Wang, G1

Trials

1 trial(s) available for tariquidar and rhodamine 123

ArticleYear
Inhibition of P-glycoprotein (ABCB1)- and multidrug resistance-associated protein 1 (ABCC1)-mediated transport by the orally administered inhibitor, CBT-1((R)).
    Biochemical pharmacology, 2008, Mar-15, Volume: 75, Issue:6

    Topics: Adenosine Triphosphatases; Alkaloids; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Biological Factors; Biological Transport; Cell Line; Cell Line, Tumor; Cyclosporins; Depsipeptides; Fluorescent Dyes; Fluorouracil; Humans; Insecta; Multidrug Resistance-Associated Proteins; Neoplasms; Paclitaxel; Prazosin; Quinolines; Rhodamine 123; Verapamil; Vinblastine

2008

Other Studies

8 other study(ies) available for tariquidar and rhodamine 123

ArticleYear
Communication between multiple drug binding sites on P-glycoprotein.
    Molecular pharmacology, 2000, Volume: 58, Issue:3

    Topics: Acridines; Allosteric Regulation; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Benzylidene Compounds; Binding, Competitive; Cell Membrane; CHO Cells; Cricetinae; Drug Interactions; Isoquinolines; Kinetics; Nicardipine; Paclitaxel; Quinolines; Radioligand Assay; Radiopharmaceuticals; Rhodamine 123; Tetrahydroisoquinolines; Tritium; Vinblastine

2000
Polarized P-glycoprotein expression by the immortalised human brain endothelial cell line, hCMEC/D3, restricts apical-to-basolateral permeability to rhodamine 123.
    Brain research, 2009, Oct-06, Volume: 1292

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Blood-Brain Barrier; Brain; Capillary Permeability; Cell Line; Cell Membrane; Cell Membrane Permeability; Cells, Cultured; Central Nervous System Agents; Endothelial Cells; Fluorescent Dyes; Humans; Models, Biological; Quinolines; Rhodamine 123; Vinblastine

2009
Reversal of multidrug resistance by co-delivery of tariquidar (XR9576) and paclitaxel using long-circulating liposomes.
    International journal of pharmaceutics, 2011, Sep-15, Volume: 416, Issue:1

    Topics: Antineoplastic Agents, Phytogenic; Antineoplastic Combined Chemotherapy Protocols; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line, Tumor; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Humans; Liposomes; Molecular Targeted Therapy; Paclitaxel; Particle Size; Quinolines; Rhodamine 123; Surface Properties

2011
[Evaluation of P-glycoprotein mediated in vitro loperamide biliary excretion with sandwich-cultured rat hepatocytes model].
    Yao xue xue bao = Acta pharmaceutica Sinica, 2012, Volume: 47, Issue:4

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biliary Tract; Cells, Cultured; Chromatography, High Pressure Liquid; Cyclosporine; Hepatocytes; Loperamide; Male; Quinidine; Quinolines; Rats; Rats, Sprague-Dawley; Rhodamine 123; Tandem Mass Spectrometry

2012
Potential role for human P-glycoprotein in the transport of lacosamide.
    Epilepsia, 2013, Volume: 54, Issue:7

    Topics: Acetamides; Animals; Anticonvulsants; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Calcium Channel Blockers; Cell Line; Digoxin; Dogs; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gene Expression Regulation; Humans; Lacosamide; Quinolines; Rhodamine 123; RNA, Messenger; Swine; Time Factors; Transfection; Tritium; Verapamil

2013
Interactions of the multidrug resistance modulators tariquidar and elacridar and their analogues with P-glycoprotein.
    ChemMedChem, 2013, Volume: 8, Issue:10

    Topics: Acridines; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Binding Sites; Cell Line, Tumor; Drug Resistance, Multiple; Humans; Mice; Molecular Docking Simulation; Protein Binding; Protein Structure, Tertiary; Quinolines; Rhodamine 123; Structure-Activity Relationship; Substrate Specificity; Tetrahydroisoquinolines

2013
Binding of modulators to mouse and human multidrug resistance P-glycoprotein. A computational study.
    Journal of molecular graphics & modelling, 2013, Volume: 46

    Topics: Amino Acid Motifs; Animals; ATP Binding Cassette Transporter, Subfamily B; Binding Sites; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Hydrophobic and Hydrophilic Interactions; Mice; Molecular Docking Simulation; Molecular Dynamics Simulation; Protein Binding; Protein Structure, Secondary; Protein Structure, Tertiary; Quinolines; Rhodamine 123; Thermodynamics

2013
Design, synthesis and biological evaluation of novel tetrahydroisoquinoline derivatives as P-glycoprotein-mediated multidrug resistance inhibitors.
    Bioorganic & medicinal chemistry, 2018, 05-15, Volume: 26, Issue:9

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Cell Survival; Doxorubicin; Drug Resistance, Neoplasm; Fluorescent Dyes; Humans; Isoquinolines; K562 Cells; Molecular Docking Simulation; Quinolines; Rhodamine 123; Structure-Activity Relationship

2018