Page last updated: 2024-09-04

tariquidar and pilocarpine

tariquidar has been researched along with pilocarpine in 3 studies

Compound Research Comparison

Studies
(tariquidar)
Trials
(tariquidar)
Recent Studies (post-2010)
(tariquidar)
Studies
(pilocarpine)
Trials
(pilocarpine)
Recent Studies (post-2010) (pilocarpine)
210161387,3343401,528

Protein Interaction Comparison

ProteinTaxonomytariquidar (IC50)pilocarpine (IC50)
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)3.0267
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)3.84
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)3.84
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)3.84
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)3.84

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bankstahl, JP; Bethmann, K; Hoffmann, K; Löscher, W1
Bankstahl, JP; Löscher, W1
Bankstahl, JP; Bankstahl, M; Ding, XQ; Kuntner, C; Langer, O; Löscher, W; Meier, M; Müller, M; Stanek, J; Wanek, T1

Other Studies

3 other study(ies) available for tariquidar and pilocarpine

ArticleYear
Glutamate is critically involved in seizure-induced overexpression of P-glycoprotein in the brain.
    Neuropharmacology, 2008, Volume: 54, Issue:6

    Topics: Animals; Apoptosis; ATP Binding Cassette Transporter, Subfamily B, Member 1; Brain Chemistry; Capillaries; Dizocilpine Maleate; Epilepsy, Temporal Lobe; Excitatory Amino Acid Antagonists; Female; Glutamic Acid; Image Processing, Computer-Assisted; Immunohistochemistry; Muscarinic Agonists; Nerve Degeneration; Pilocarpine; Quinolines; Rats; Rats, Wistar; Seizures; Status Epilepticus

2008
Resistance to antiepileptic drugs and expression of P-glycoprotein in two rat models of status epilepticus.
    Epilepsy research, 2008, Volume: 82, Issue:1

    Topics: Amygdala; Animals; Anticonvulsants; ATP Binding Cassette Transporter, Subfamily B; Diazepam; Disease Models, Animal; Drug Resistance; Electric Stimulation; Endothelium, Vascular; Female; Gene Expression Regulation; Genes, MDR; Hippocampus; Phenobarbital; Phenytoin; Pilocarpine; Quinolines; Rats; Rats, Sprague-Dawley; Status Epilepticus

2008
A novel positron emission tomography imaging protocol identifies seizure-induced regional overactivity of P-glycoprotein at the blood-brain barrier.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Jun-15, Volume: 31, Issue:24

    Topics: Analysis of Variance; Animals; Area Under Curve; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blood-Brain Barrier; Calcium Channel Blockers; Carbon Isotopes; Computer Simulation; Disease Models, Animal; Female; Gene Expression Regulation; Heterocyclic Compounds; Magnetic Resonance Imaging; Models, Chemical; Organometallic Compounds; Pilocarpine; Positron-Emission Tomography; Quinolines; Rats; Rats, Sprague-Dawley; Scopolamine; Seizures; Time Factors; Verapamil

2011