Page last updated: 2024-09-04

tariquidar and midazolam

tariquidar has been researched along with midazolam in 2 studies

Compound Research Comparison

Studies
(tariquidar)
Trials
(tariquidar)
Recent Studies (post-2010)
(tariquidar)
Studies
(midazolam)
Trials
(midazolam)
Recent Studies (post-2010) (midazolam)
210161389,8343,1913,301

Protein Interaction Comparison

ProteinTaxonomytariquidar (IC50)midazolam (IC50)
Cytochrome P450 3A4Homo sapiens (human)2.7427

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's1 (50.00)2.80

Authors

AuthorsStudies
Kurnik, D; Wilkinson, GR; Wood, AJ1
da Costa César, I; de Araújo, LL; de Castro, WV; de Lima Nascimento, M; de Oliveira, FM; Derendorf, H; do Carmo Vieira, M; do Nascimento, SB; Duarte-Almeida, JM; Siqueira, JM1

Trials

1 trial(s) available for tariquidar and midazolam

ArticleYear
The erythromycin breath test reflects P-glycoprotein function independently of cytochrome P450 3A activity.
    Clinical pharmacology and therapeutics, 2006, Volume: 80, Issue:3

    Topics: Adult; Area Under Curve; ATP Binding Cassette Transporter, Subfamily B, Member 1; Breath Tests; Cross-Over Studies; Cytochrome P-450 CYP3A; Double-Blind Method; Enzyme Inhibitors; Erythromycin; GABA Modulators; Humans; Infusions, Intravenous; Injections, Intravenous; Liver; Male; Metabolic Clearance Rate; Midazolam; Quinolines; Reproducibility of Results; Time Factors

2006

Other Studies

1 other study(ies) available for tariquidar and midazolam

ArticleYear
Evaluation of the Effects of Maytenus ilicifolia on the Activities of Cytochrome P450 3A and P-glycoprotein.
    Current drug metabolism, 2020, Volume: 21, Issue:4

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Caco-2 Cells; Cell Line; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Drug Interactions; Humans; Ketoconazole; Male; Maytenus; Midazolam; Plant Extracts; Quinolines; Rats; Rats, Wistar; Terfenadine

2020