tariquidar has been researched along with l 660,711 in 4 studies
Studies (tariquidar) | Trials (tariquidar) | Recent Studies (post-2010) (tariquidar) | Studies (l 660,711) | Trials (l 660,711) | Recent Studies (post-2010) (l 660,711) |
---|---|---|---|---|---|
210 | 16 | 138 | 45 | 0 | 12 |
Protein | Taxonomy | tariquidar (IC50) | l 660,711 (IC50) |
---|---|---|---|
ATP-binding cassette sub-family C member 3 | Homo sapiens (human) | 9.3 | |
Multidrug resistance-associated protein 4 | Homo sapiens (human) | 8 | |
Solute carrier organic anion transporter family member 2B1 | Homo sapiens (human) | 2.9 | |
Bile salt export pump | Homo sapiens (human) | 3.515 | |
Multidrug resistance-associated protein 1 | Homo sapiens (human) | 2.9733 | |
Canalicular multispecific organic anion transporter 1 | Rattus norvegicus (Norway rat) | 2.62 | |
Canalicular multispecific organic anion transporter 1 | Homo sapiens (human) | 7 | |
Solute carrier organic anion transporter family member 1B3 | Homo sapiens (human) | 6.4 | |
Solute carrier organic anion transporter family member 1B1 | Homo sapiens (human) | 4.4 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (25.00) | 29.6817 |
2010's | 2 (50.00) | 24.3611 |
2020's | 1 (25.00) | 2.80 |
Authors | Studies |
---|---|
Bernhardt, G; Buschauer, A; Egger, M; Fricker, G; König, B; Kühnle, M; Mahringer, A; Müller, C | 1 |
Hsiao, SH; Hsieh, CH; Huang, YH; Hung, TH; Li, YQ; Lu, YJ; Tuo, WC; Wu, CP; Yang, CC | 1 |
Gallus, J; Krapf, MK; Vahdati, S; Wiese, M | 1 |
Ambudkar, SV; Hsiao, SH; Huang, YH; Hung, TH; Li, YQ; Liu, TC; Lusvarghi, S; Wu, CP | 1 |
4 other study(ies) available for tariquidar and l 660,711
Article | Year |
---|---|
Potent and selective inhibitors of breast cancer resistance protein (ABCG2) derived from the p-glycoprotein (ABCB1) modulator tariquidar.
Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Breast Neoplasms; Cell Line, Tumor; Drug Resistance, Multiple; Female; Humans; Inhibitory Concentration 50; Multidrug Resistance-Associated Protein 2; Neoplasm Proteins; Quinolines; Structure-Activity Relationship | 2009 |
Hernandezine, a Bisbenzylisoquinoline Alkaloid with Selective Inhibitory Activity against Multidrug-Resistance-Linked ATP-Binding Cassette Drug Transporter ABCB1.
Topics: Adenosine Triphosphate; Alkaloids; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Benzylisoquinolines; Drug Resistance, Neoplasm; Humans; Molecular Structure | 2016 |
New Inhibitors of Breast Cancer Resistance Protein (ABCG2) Containing a 2,4-Disubstituted Pyridopyrimidine Scaffold.
Topics: Adenosine Triphosphatases; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily G, Member 2; Cell Line, Tumor; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Mice; Molecular Structure; Neoplasm Proteins; Pyridines; Pyrimidines; Structure-Activity Relationship | 2018 |
Licochalcone A Selectively Resensitizes ABCG2-Overexpressing Multidrug-Resistant Cancer Cells to Chemotherapeutic Drugs.
Topics: Adenosine Triphosphatases; Antineoplastic Agents; Apoptosis; ATP Binding Cassette Transporter, Subfamily G, Member 2; Cell Line, Tumor; Chalcones; Computer Simulation; Drug Resistance, Neoplasm; Drug Synergism; Glycyrrhiza; Humans; Molecular Docking Simulation; Neoplasm Proteins; Topotecan | 2020 |