Page last updated: 2024-09-04

tariquidar and l 660,711

tariquidar has been researched along with l 660,711 in 4 studies

Compound Research Comparison

Studies
(tariquidar)
Trials
(tariquidar)
Recent Studies (post-2010)
(tariquidar)
Studies
(l 660,711)
Trials
(l 660,711)
Recent Studies (post-2010) (l 660,711)
2101613845012

Protein Interaction Comparison

ProteinTaxonomytariquidar (IC50)l 660,711 (IC50)
ATP-binding cassette sub-family C member 3Homo sapiens (human)9.3
Multidrug resistance-associated protein 4Homo sapiens (human)8
Solute carrier organic anion transporter family member 2B1 Homo sapiens (human)2.9
Bile salt export pumpHomo sapiens (human)3.515
Multidrug resistance-associated protein 1 Homo sapiens (human)2.9733
Canalicular multispecific organic anion transporter 1Rattus norvegicus (Norway rat)2.62
Canalicular multispecific organic anion transporter 1Homo sapiens (human)7
Solute carrier organic anion transporter family member 1B3Homo sapiens (human)6.4
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)4.4

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (25.00)29.6817
2010's2 (50.00)24.3611
2020's1 (25.00)2.80

Authors

AuthorsStudies
Bernhardt, G; Buschauer, A; Egger, M; Fricker, G; König, B; Kühnle, M; Mahringer, A; Müller, C1
Hsiao, SH; Hsieh, CH; Huang, YH; Hung, TH; Li, YQ; Lu, YJ; Tuo, WC; Wu, CP; Yang, CC1
Gallus, J; Krapf, MK; Vahdati, S; Wiese, M1
Ambudkar, SV; Hsiao, SH; Huang, YH; Hung, TH; Li, YQ; Liu, TC; Lusvarghi, S; Wu, CP1

Other Studies

4 other study(ies) available for tariquidar and l 660,711

ArticleYear
Potent and selective inhibitors of breast cancer resistance protein (ABCG2) derived from the p-glycoprotein (ABCB1) modulator tariquidar.
    Journal of medicinal chemistry, 2009, Feb-26, Volume: 52, Issue:4

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Breast Neoplasms; Cell Line, Tumor; Drug Resistance, Multiple; Female; Humans; Inhibitory Concentration 50; Multidrug Resistance-Associated Protein 2; Neoplasm Proteins; Quinolines; Structure-Activity Relationship

2009
Hernandezine, a Bisbenzylisoquinoline Alkaloid with Selective Inhibitory Activity against Multidrug-Resistance-Linked ATP-Binding Cassette Drug Transporter ABCB1.
    Journal of natural products, 2016, 08-26, Volume: 79, Issue:8

    Topics: Adenosine Triphosphate; Alkaloids; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Benzylisoquinolines; Drug Resistance, Neoplasm; Humans; Molecular Structure

2016
New Inhibitors of Breast Cancer Resistance Protein (ABCG2) Containing a 2,4-Disubstituted Pyridopyrimidine Scaffold.
    Journal of medicinal chemistry, 2018, 04-26, Volume: 61, Issue:8

    Topics: Adenosine Triphosphatases; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily G, Member 2; Cell Line, Tumor; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Mice; Molecular Structure; Neoplasm Proteins; Pyridines; Pyrimidines; Structure-Activity Relationship

2018
Licochalcone A Selectively Resensitizes ABCG2-Overexpressing Multidrug-Resistant Cancer Cells to Chemotherapeutic Drugs.
    Journal of natural products, 2020, 05-22, Volume: 83, Issue:5

    Topics: Adenosine Triphosphatases; Antineoplastic Agents; Apoptosis; ATP Binding Cassette Transporter, Subfamily G, Member 2; Cell Line, Tumor; Chalcones; Computer Simulation; Drug Resistance, Neoplasm; Drug Synergism; Glycyrrhiza; Humans; Molecular Docking Simulation; Neoplasm Proteins; Topotecan

2020