Page last updated: 2024-09-04

tariquidar and imatinib mesylate

tariquidar has been researched along with imatinib mesylate in 3 studies

Compound Research Comparison

Studies
(tariquidar)
Trials
(tariquidar)
Recent Studies (post-2010)
(tariquidar)
Studies
(imatinib mesylate)
Trials
(imatinib mesylate)
Recent Studies (post-2010) (imatinib mesylate)
2101613811,4779605,773

Protein Interaction Comparison

ProteinTaxonomytariquidar (IC50)imatinib mesylate (IC50)
Tyrosine-protein kinase ABL1Homo sapiens (human)0.31
Mast/stem cell growth factor receptor KitHomo sapiens (human)0.1

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's2 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Figg, WD; Gardner, ER; Smith, NF; Sparreboom, A1
Klinkhammer, W; Pick, A; Wiese, M1
Alcantara, LM; Ayong, LS; Franco, CH; Franzoi, KD; Freitas-Junior, LH; Kim, J; Lee, S; Moraes, CB1

Other Studies

3 other study(ies) available for tariquidar and imatinib mesylate

ArticleYear
Influence of the dual ABCB1 and ABCG2 inhibitor tariquidar on the disposition of oral imatinib in mice.
    Journal of experimental & clinical cancer research : CR, 2009, Jul-10, Volume: 28

    Topics: Administration, Oral; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Benzamides; Imatinib Mesylate; Male; Mice; Mice, Inbred BALB C; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Quinolines

2009
Specific inhibitors of the breast cancer resistance protein (BCRP).
    ChemMedChem, 2010, Sep-03, Volume: 5, Issue:9

    Topics: Adenosine; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Benzamides; Binding Sites; Breast Neoplasms; Cell Line, Tumor; Chlorophyll; Diketopiperazines; Drug Resistance, Multiple; Female; Heterocyclic Compounds, 4 or More Rings; Humans; Imatinib Mesylate; Indoles; Neoplasm Proteins; Novobiocin; Piperazines; Pyrimidines; Quinolines; Structure-Activity Relationship

2010
Chemosensitization potential of P-glycoprotein inhibitors in malaria parasites.
    Experimental parasitology, 2013, Volume: 134, Issue:2

    Topics: Antimalarials; Artemisinins; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzamides; Boron Compounds; Chloroquine; Chlorpheniramine; Dibenzocycloheptenes; Drug Interactions; Drug Resistance, Multiple; Erythrocytes; Fluorescent Dyes; Gefitinib; Humans; Imatinib Mesylate; Mefloquine; Piperazines; Plasmodium falciparum; Protein Kinase Inhibitors; Pyrimidines; Quinazolines; Quinolines

2013