Page last updated: 2024-09-04

tariquidar and doxorubicin hydrochloride

tariquidar has been researched along with doxorubicin hydrochloride in 3 studies

Compound Research Comparison

Studies
(tariquidar)
Trials
(tariquidar)
Recent Studies (post-2010)
(tariquidar)
Studies
(doxorubicin hydrochloride)
Trials
(doxorubicin hydrochloride)
Recent Studies (post-2010) (doxorubicin hydrochloride)
210161382770205

Protein Interaction Comparison

ProteinTaxonomytariquidar (IC50)doxorubicin hydrochloride (IC50)
RNA polymerase beta subunit (EC 2.7.7.6), partialEscherichia coli14.3747
90-kda heat shock protein beta HSP90 beta, partialHomo sapiens (human)0.266
Apoptotic peptidase activating factor 1Homo sapiens (human)21.2
TPA: protein transporter TIM23Saccharomyces cerevisiae S288C12.7
caspase-9 isoform alpha precursorHomo sapiens (human)34.6
caspase-3 isoform a preproproteinHomo sapiens (human)34.6
heat shock protein HSP 90-alpha isoform 2Homo sapiens (human)0.266
14-3-3 protein gammaHomo sapiens (human)0.7812
DNA topoisomerase 2-alphaHomo sapiens (human)0.94

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (66.67)24.3611
2020's1 (33.33)2.80

Authors

AuthorsStudies
Cui, J; Ghaleb, H; Huang, W; Jiao, L; Kairuki, M; Liao, C; Lin, H; Pan, M; Qian, H; Zhou, J1
Bi, X; Cui, J; Gao, Y; Huang, W; Li, Z; Liu, C; Qian, H; Shi, W; Wang, G1
Cai, Z; Ghaleb, H; Huang, W; Jiang, Y; Liu, Y; Qian, H; Qiu, Q; Shi, W; Yin, Z; Zhang, P; Zhou, J; Zou, F1

Other Studies

3 other study(ies) available for tariquidar and doxorubicin hydrochloride

ArticleYear
Synthesis and biological evaluation of JL-A7 derivatives as potent ABCB1 inhibitors.
    Bioorganic & medicinal chemistry, 2017, 08-01, Volume: 25, Issue:15

    Topics: Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B; Carbon-13 Magnetic Resonance Spectroscopy; Cell Line, Tumor; Doxorubicin; Drug Resistance, Multiple; Humans; Isoquinolines; Proton Magnetic Resonance Spectroscopy; Spectrometry, Mass, Electrospray Ionization; Structure-Activity Relationship; Triazoles

2017
Design, synthesis and biological evaluation of novel tetrahydroisoquinoline derivatives as P-glycoprotein-mediated multidrug resistance inhibitors.
    Bioorganic & medicinal chemistry, 2018, 05-15, Volume: 26, Issue:9

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Cell Survival; Doxorubicin; Drug Resistance, Neoplasm; Fluorescent Dyes; Humans; Isoquinolines; K562 Cells; Molecular Docking Simulation; Quinolines; Rhodamine 123; Structure-Activity Relationship

2018
Exploration of novel phthalazinone derivatives as potential efflux transporter inhibitors for reversing multidrug resistance and improving the oral absorption of paclitaxel.
    European journal of medicinal chemistry, 2022, Apr-05, Volume: 233

    Topics: ATP Binding Cassette Transporter, Subfamily G, Member 2; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Neoplasm Proteins; Neoplasms; Paclitaxel

2022