Page last updated: 2024-08-26

tandospirone and buspirone

tandospirone has been researched along with buspirone in 24 studies

Research

Studies (24)

TimeframeStudies, this research(%)All Research%
pre-19903 (12.50)18.7374
1990's16 (66.67)18.2507
2000's4 (16.67)29.6817
2010's1 (4.17)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Abou-Gharbia, M; Andree, TH; Moyer, JA; Muth, EA; Patel, UR; Webb, MB1
Audinot, V; Chaput, C; Conte, C; Gavaudan, S; Millan, MJ; Newman-Tancredi, A; Touzard, M; Verrièle, L1
Byrnes, JJ; Greenblatt, DJ; Miller, LG; Shemer, A; Thompson, ML1
Moon, SL; Taylor, DP1
Blier, P; Chaput, Y; Curet, O; de Montigny, C1
Lucki, I1
Fischette, C; Hamik, A; Oksenberg, D; Peroutka, SJ1
Boyer, WF; Feighner, JP1
Hirose, A; Kumasaka, Y; Nakamura, M; Shimizu, H; Tanaka, H; Tatsuno, T1
Gondoh, Y; Nishimura, H; Tanaka, M; Tsuda, A1
Matheson, GK; Michel, C; Pfeifer, DM; Weiberg, MB1
Evans, SM; Griffiths, RR; Troisi, JR1
Kuribara, H1
Ator, NA; Griffiths, RR; Sannerud, CA1
Kellar, KJ; Lumpkin, MD; Mulroney, SE; Shemer, A; Skudlarek, C1
Clemente, J; Quartermain, D; Shemer, A1
Bauer, C; Blackbourne, J; Gage, D; Guthrie, D; Knowles, A; Matheson, GK; Michel, C; Weinzapfel, D1
Abe, M; Egawa, M; Nakai, H; Saito, K; Tabata, R1
Yamawaki, S1
Kato, S; Nisijima, K; Ohtuka, K; Shioda, K; Yamauchi, Y1
Inoue, T; Izumi, T; Koyama, T; Masui, T; Nishikawa, H1
Ertugrul, A; Jayathilake, K; Meltzer, HY; Park, S; Roy, A; Sumiyoshi, T1
Bert, B; Bubenikova-Valesova, V; Horacek, J; Sumiyoshi, T1
He, S; Hu, W; Jia, M; Jiang, X; Wang, L; Xie, H1

Reviews

5 review(s) available for tandospirone and buspirone

ArticleYear
Buspirone and related compounds as alternative anxiolytics.
    Neuropeptides, 1991, Volume: 19 Suppl

    Topics: Animals; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepines; Binding Sites; Buspirone; Humans; Isoindoles; Piperazines; Pyrimidines; Receptors, Serotonin; Structure-Activity Relationship

1991
Behavioral studies of serotonin receptor agonists as antidepressant drugs.
    The Journal of clinical psychiatry, 1991, Volume: 52 Suppl

    Topics: Animals; Anti-Anxiety Agents; Antidepressive Agents; Behavior, Animal; Buspirone; Clinical Trials as Topic; Depressive Disorder; Humans; Isoindoles; Piperazines; Pyrimidines; Rats; Receptors, Serotonin

1991
Serotonin-1A anxiolytics: an overview.
    Psychopathology, 1989, Volume: 22 Suppl 1

    Topics: Animals; Anti-Anxiety Agents; Anxiety Disorders; Brain; Buspirone; Clinical Trials as Topic; Double-Blind Method; Humans; Isoindoles; Piperazines; Pyrimidines; Receptors, Serotonin

1989
The use and development of anxiolytics in Japan.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 1999, Volume: 9 Suppl 6

    Topics: Anti-Anxiety Agents; Anxiety; Benzodiazepines; Buspirone; Drug Utilization; GABA-A Receptor Agonists; Humans; Isoindoles; Japan; Piperazines; Pyrimidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists

1999
Serotonin1A receptors in the pathophysiology of schizophrenia: development of novel cognition-enhancing therapeutics.
    Advances in therapy, 2008, Volume: 25, Issue:10

    Topics: Animals; Behavior; Brain; Buspirone; Cognition Disorders; Humans; Isoindoles; Piperazines; Polymorphism, Genetic; Pyrimidines; Receptor, Serotonin, 5-HT1A; Schizophrenia; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists

2008

Trials

4 trial(s) available for tandospirone and buspirone

ArticleYear
Buspirone and related compounds as alternative anxiolytics.
    Neuropeptides, 1991, Volume: 19 Suppl

    Topics: Animals; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepines; Binding Sites; Buspirone; Humans; Isoindoles; Piperazines; Pyrimidines; Receptors, Serotonin; Structure-Activity Relationship

1991
Serotonin-1A anxiolytics: an overview.
    Psychopathology, 1989, Volume: 22 Suppl 1

    Topics: Animals; Anti-Anxiety Agents; Anxiety Disorders; Brain; Buspirone; Clinical Trials as Topic; Double-Blind Method; Humans; Isoindoles; Piperazines; Pyrimidines; Receptors, Serotonin

1989
Tandospirone and alprazolam: comparison of behavioral effects and abuse liability in humans.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 271, Issue:2

    Topics: Adult; Alprazolam; Anti-Anxiety Agents; Buspirone; Cross-Over Studies; Dose-Response Relationship, Drug; Double-Blind Method; Humans; Isoindoles; Male; Piperazines; Psychomotor Performance; Pyrimidines; Serotonin Receptor Agonists; Substance-Related Disorders

1994
Effect of buspirone, a serotonin1A partial agonist, on cognitive function in schizophrenia: a randomized, double-blind, placebo-controlled study.
    Schizophrenia research, 2007, Volume: 95, Issue:1-3

    Topics: Adult; Ambulatory Care; Antipsychotic Agents; Buspirone; Cognition Disorders; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Isoindoles; Male; Neuropsychological Tests; Piperazines; Placebos; Pyrimidines; Schizophrenia; Schizophrenic Psychology; Serotonin Receptor Agonists; Treatment Outcome

2007

Other Studies

17 other study(ies) available for tandospirone and buspirone

ArticleYear
Polycyclic aryl- and heteroarylpiperazinyl imides as 5-HT1A receptor ligands and potential anxiolytic agents: synthesis and structure-activity relationship studies.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:7

    Topics: Animals; Anti-Anxiety Agents; Apomorphine; Avoidance Learning; Behavior, Animal; Brain; Chemical Phenomena; Chemistry; Imides; Male; Piperazines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Serotonin; Stereotyped Behavior; Structure-Activity Relationship

1988
Agonist and antagonist actions of antipsychotic agents at 5-HT1A receptors: a [35S]GTPgammaS binding study.
    European journal of pharmacology, 1998, Aug-21, Volume: 355, Issue:2-3

    Topics: Animals; Antipsychotic Agents; CHO Cells; Cricetinae; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Agents; Sulfur Radioisotopes

1998
Kinetics, brain uptake, and receptor binding of tandospirone and its metabolite 1-(2-pyrimidinyl)-piperazine.
    Journal of clinical psychopharmacology, 1992, Volume: 12, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Brain; Brain Chemistry; Buspirone; Cerebral Cortex; Isoindoles; Male; Mice; Motor Activity; Piperazines; Pyrimidines; Receptors, GABA-A; Receptors, Serotonin

1992
Tandospirone and its metabolite, 1-(2-pyrimidinyl)-piperazine--II. Effects of acute administration of 1-PP and long-term administration of tandospirone on noradrenergic neurotransmission.
    Neuropharmacology, 1991, Volume: 30, Issue:7

    Topics: Animals; Anti-Anxiety Agents; Brain; Buspirone; Clonidine; Electric Stimulation; GABA Antagonists; Isoindoles; Male; Neurons; Norepinephrine; Piperazines; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha

1991
Analysis of tandospirone (SM-3997) interactions with neurotransmitter receptor binding sites.
    Biological psychiatry, 1990, Jul-15, Volume: 28, Issue:2

    Topics: Adenylyl Cyclases; Animals; Anti-Anxiety Agents; Binding, Competitive; Brain; Buspirone; Isoindoles; Male; Piperazines; Pyrimidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Dopamine; Receptors, Serotonin

1990
Effects of the putative anxiolytic SM-3997 on central monoaminergic systems.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 32, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Biogenic Monoamines; Brain; Brain Chemistry; Buspirone; Dopamine; Imipramine; Isoindoles; Male; Norepinephrine; Piperazines; Pyrimidines; Rats; Rats, Inbred Strains; Serotonin

1989
Atypical anxiolytic profile of buspirone and a related drug, SM-3997, in a modified forced swim test employing straw suspension.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 46, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Buspirone; Immobilization; Isoindoles; Male; Piperazines; Pyrimidines; Rats; Rats, Sprague-Dawley; Swimming

1993
The effects of azapirones on serotonin1A neurons of the dorsal raphe.
    General pharmacology, 1994, Volume: 25, Issue:4

    Topics: Animals; Buspirone; Dose-Response Relationship, Drug; Isoindoles; Male; Piperazines; Pyrimidines; Raphe Nuclei; Rats; Receptors, Serotonin; Serotonin Receptor Agonists

1994
Effects of SUN 8399, a potent and selective 5-HT1A agonist, on conflict behavior and ambulatory activity in mice: comparison with those of buspirone, tandospirone and diazepam.
    Japanese journal of pharmacology, 1994, Volume: 64, Issue:4

    Topics: Animals; Behavior, Animal; Buspirone; Conflict, Psychological; Diazepam; Drug Interactions; Isoindoles; Male; Mice; Mice, Inbred Strains; Motor Activity; Oxazepines; Piperazines; Pyrimidines; Serotonin Receptor Agonists

1994
Behavioral pharmacology of tandospirone in baboons: chronic administration and withdrawal, self-injection and drug discrimination.
    Drug and alcohol dependence, 1993, Volume: 32, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Arousal; Buspirone; Cocaine; Discrimination Learning; Dose-Response Relationship, Drug; Eating; Flumazenil; Isoindoles; Lorazepam; Male; Motor Skills; Neurologic Examination; Papio; Pentobarbital; Piperazines; Pyrimidines; Reinforcement Schedule; Self Administration; Serotonin Receptor Agonists; Substance Withdrawal Syndrome; Substance-Related Disorders

1993
Tandospirone stimulates prolactin secretion in the rat by an action at serotonin-1A receptors.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 268, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Buspirone; Dose-Response Relationship, Drug; Isoindoles; Male; Metergoline; Piperazines; Prolactin; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Receptor Agonists

1994
5-HT1A agonists disrupt memory of fear conditioning in mice.
    Biological psychiatry, 1993, Feb-15, Volume: 33, Issue:4

    Topics: Analysis of Variance; Animals; Buspirone; Conditioning, Psychological; Dextroamphetamine; Extinction, Psychological; Fear; Isoindoles; Male; Memory; Mice; Piperazines; Pyrimidines; Retention, Psychology; Serotonin Receptor Agonists

1993
Modification of hypothalamic-pituitary-adrenocortical activity by serotonergic agents in the rat.
    Pharmacology, 1997, Volume: 55, Issue:2

    Topics: Adrenal Cortex; Animals; Behavior, Animal; Buspirone; Carbolines; Corticosterone; Dose-Response Relationship, Drug; Isoindoles; Male; Piperazines; Pituitary Gland; Pyridines; Pyrimidines; Rats; Serotonin Receptor Agonists

1997
Effect of 5-[3-[((2S)-1,4-benzodioxan-2-ylmethyl)amino]propoxy]-1,3-benzodioxole HCl (MKC-242), a novel 5-HT1A-receptor agonist, on aggressive behavior and marble burying behavior in mice.
    Japanese journal of pharmacology, 1998, Volume: 76, Issue:3

    Topics: Aggression; Animals; Anti-Anxiety Agents; Anxiety; Buspirone; Diazepam; Dioxanes; Dioxoles; Disease Models, Animal; Drug Evaluation, Preclinical; Isoindoles; Male; Mice; Mice, Inbred ICR; Obsessive Behavior; Piperazines; Pyrimidines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists

1998
Use of a serotonin 1A receptor agonist to treat restless legs syndrome.
    Journal of clinical psychopharmacology, 2006, Volume: 26, Issue:6

    Topics: Adult; Buspirone; Female; Humans; Isoindoles; Male; Middle Aged; Piperazines; Pyrimidines; Restless Legs Syndrome; Serotonin 5-HT1 Receptor Agonists; Serotonin Receptor Agonists

2006
Effects of cytochrome P450 (CYP) 3A4 inhibitors on the anxiolytic action of tandospirone in rat contextual conditioned fear.
    Progress in neuro-psychopharmacology & biological psychiatry, 2007, May-09, Volume: 31, Issue:4

    Topics: Administration, Oral; Analysis of Variance; Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Buspirone; Conditioning, Classical; Disease Models, Animal; Dose-Response Relationship, Drug; Fear; Isoindoles; Male; Motor Activity; Piperazines; Pyrimidines; Rats; Rats, Sprague-Dawley

2007
Simultaneous determination of tandospirone and its active metabolite, 1-[2-pyrimidyl]-piperazine in rat plasma by LC-MS/MS and its application to a pharmacokinetic study.
    Biomedical chromatography : BMC, 2019, Volume: 33, Issue:7

    Topics: Animals; Buspirone; Chromatography, High Pressure Liquid; Drug Stability; Female; Isoindoles; Limit of Detection; Linear Models; Male; Piperazines; Pyrimidines; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Tandem Mass Spectrometry

2019