Page last updated: 2024-08-25

talinolol and rifampin

talinolol has been researched along with rifampin in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's7 (46.67)29.6817
2010's7 (46.67)24.3611
2020's1 (6.67)2.80

Authors

AuthorsStudies
Collett, A; Hallifax, D; Tanianis-Hughes, J; Warhurst, G1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Chang, G; Di, L; Huang, Y; Lin, Z; Liston, TE; Scott, DO; Troutman, MD; Umland, JP1
Artursson, P; Mateus, A; Matsson, P1
Bloomer, WD; Papadopoulou, MV; Rosenzweig, HS1
Eslamimehr, S; Franzblau, SG; Kong, Y; Kurosu, M; Lemieux, MR; Mitachi, K; Park, F; Pressly, JD; Siricilla, S; Wang, Y; Yang, D1
Franke, G; Fritz, P; Hachenberg, T; Kauffmann, HM; Knoke, M; Kroemer, HK; Oertel, R; Schrenk, D; Siegmund, W; Terhaag, B; von Richter, O; Warzok, R; Weinbrenner, A; Westphal, K; Zschiesche, M1
Franke, G; Gramatté, T; Hoffmann, A; Klebingat, KJ; Kroemer, HK; Lemma, GL; Siegmund, W; Terhaag, B; Zschiesche, M1
Chiou, WL; Jeong, HY; Ma, C; Wu, TC1
Caliebe, A; Cascorbi, I; Haenisch, S; May, K; Siegmund, W; Wegner, D1
Dazert, E; Lederer, K; Oswald, S; Saljé, K; Siegmund, W; Warzok, R1
Costales, C; Eatemadpour, S; Kimoto, E; Lazzaro, S; Varma, MV; Yamazaki, S1
D'Argenio, DZ; Siegmund, W; Weiss, M1

Trials

1 trial(s) available for talinolol and rifampin

ArticleYear
Induction of P-glycoprotein by rifampin increases intestinal secretion of talinolol in human beings: a new type of drug/drug interaction.
    Clinical pharmacology and therapeutics, 2000, Volume: 68, Issue:4

    Topics: Administration, Oral; Adrenergic beta-Antagonists; Adult; Anti-Arrhythmia Agents; Antihypertensive Agents; Antitubercular Agents; Area Under Curve; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; Duodenum; Endoscopy, Digestive System; Enzyme Induction; Humans; Immunohistochemistry; Infusions, Intravenous; Male; Propanolamines; Reference Values; Reverse Transcriptase Polymerase Chain Reaction; Rifampin; RNA, Messenger; Up-Regulation

2000

Other Studies

14 other study(ies) available for talinolol and rifampin

ArticleYear
Predicting P-glycoprotein effects on oral absorption: correlation of transport in Caco-2 with drug pharmacokinetics in wild-type and mdr1a(-/-) mice in vivo.
    Pharmaceutical research, 2004, Volume: 21, Issue:5

    Topics: Administration, Oral; Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Biological Transport, Active; Caco-2 Cells; Cell Membrane Permeability; Humans; Intestinal Absorption; Mice; Mice, Knockout; Pharmacokinetics; Spectrometry, Mass, Electrospray Ionization

2004
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Species independence in brain tissue binding using brain homogenates.
    Drug metabolism and disposition: the biological fate of chemicals, 2011, Volume: 39, Issue:7

    Topics: Animals; Brain; Dogs; Guinea Pigs; Humans; Macaca fascicularis; Mice; Rats; Species Specificity

2011
A high-throughput cell-based method to predict the unbound drug fraction in the brain.
    Journal of medicinal chemistry, 2014, Apr-10, Volume: 57, Issue:7

    Topics: Animals; Brain; Dialysis; HEK293 Cells; High-Throughput Screening Assays; Humans; Pharmaceutical Preparations; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization

2014
The antitubercular activity of various nitro(triazole/imidazole)-based compounds.
    Bioorganic & medicinal chemistry, 2017, 11-01, Volume: 25, Issue:21

    Topics: Animals; Antitubercular Agents; Cell Line; Chlorocebus aethiops; Dose-Response Relationship, Drug; Humans; Imidazoles; Macrophages; Mice; Microbial Sensitivity Tests; Molecular Structure; Mycobacterium tuberculosis; Nitro Compounds; Structure-Activity Relationship; Triazoles

2017
An antimycobacterial pleuromutilin analogue effective against dormant bacilli.
    Bioorganic & medicinal chemistry, 2018, 09-15, Volume: 26, Issue:17

    Topics: Administration, Oral; Animals; Antitubercular Agents; Area Under Curve; Biological Availability; Caco-2 Cells; Diterpenes; Female; Half-Life; Humans; Inhibitory Concentration 50; Mice; Mice, Inbred BALB C; Microbial Sensitivity Tests; Mycobacterium tuberculosis; Pleuromutilins; Polycyclic Compounds

2018
Stereoselective disposition of talinolol in man.
    Journal of pharmaceutical sciences, 2002, Volume: 91, Issue:2

    Topics: Adrenergic beta-Antagonists; Adult; Area Under Curve; ATP Binding Cassette Transporter, Subfamily B, Member 1; Drug Interactions; Enzyme Inhibitors; Humans; Male; Microsomes, Liver; Molecular Conformation; Propanolamines; Rifampin; Statistics, Nonparametric

2002
Unexpected lack of effect of the rifampin-induced P-glycoprotein on the oral bioavailability of its substrate, talinolol, in humans: implication in phenotyping.
    Journal of pharmaceutical sciences, 2003, Volume: 92, Issue:1

    Topics: Administration, Oral; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Availability; Humans; Phenotype; Propanolamines; Rifampin; Stereoisomerism; Substrate Specificity

2003
Influence of genetic polymorphisms on intestinal expression and rifampicin-type induction of ABCC2 and on bioavailability of talinolol.
    Pharmacogenetics and genomics, 2008, Volume: 18, Issue:4

    Topics: Administration, Oral; Adult; Antihypertensive Agents; Biological Availability; DNA Primers; Duodenum; Female; Gene Frequency; Genotype; Humans; Infusions, Intravenous; Intestinal Mucosa; Intestines; Male; Membrane Transport Proteins; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Nucleic Acid Synthesis Inhibitors; Polymorphism, Single Nucleotide; Propanolamines; Reverse Transcriptase Polymerase Chain Reaction; Rifampin; RNA, Messenger

2008
Effects of rifampicin, dexamethasone, St. John's Wort and Thyroxine on maternal and foetal expression of Abcb1 and organ distribution of talinolol in pregnant rats.
    Basic & clinical pharmacology & toxicology, 2012, Volume: 111, Issue:2

    Topics: Administration, Oral; Animals; ATP Binding Cassette Transporter, Subfamily B; Brain; Dexamethasone; Female; Fetus; Hypericum; Liver; Placenta; Pregnancy; Propanolamines; Rats; Rats, Wistar; Rifampin; RNA, Messenger; Thyroxine

2012
Physiologically-Based Pharmacokinetic Modeling Approach to Predict Rifampin-Mediated Intestinal P-Glycoprotein Induction.
    CPT: pharmacometrics & systems pharmacology, 2019, Volume: 8, Issue:9

    Topics: Administration, Oral; ATP Binding Cassette Transporter, Subfamily B, Member 1; Dabigatran; Digoxin; Drug Interactions; Female; Gene Expression Regulation; Healthy Volunteers; Humans; Intestinal Mucosa; Male; Models, Biological; Propanolamines; Quinidine; Rifampin

2019
Analysis of Complex Absorption After Multiple Dosing: Application to the Interaction Between the P-glycoprotein Substrate Talinolol and Rifampicin.
    Pharmaceutical research, 2022, Volume: 39, Issue:12

    Topics: Adrenergic beta-Antagonists; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Humans; Propanolamines; Rifampin

2022