Page last updated: 2024-09-02

tadalafil and mocetinostat

tadalafil has been researched along with mocetinostat in 3 studies

Compound Research Comparison

Studies
(tadalafil)
Trials
(tadalafil)
Recent Studies (post-2010)
(tadalafil)
Studies
(mocetinostat)
Trials
(mocetinostat)
Recent Studies (post-2010) (mocetinostat)
1,7423921,08921,7353908,606

Protein Interaction Comparison

ProteinTaxonomytadalafil (IC50)mocetinostat (IC50)
Histone deacetylase 3Homo sapiens (human)0.7851
Nuclear receptor corepressor 1Homo sapiens (human)0.022
Cytochrome P450 3A4Homo sapiens (human)0.57
Cytochrome P450 2D6Homo sapiens (human)0.102
Cytochrome P450 2C19Homo sapiens (human)0.102
Histone deacetylase 4Homo sapiens (human)0.5717
Histone deacetylase 1Homo sapiens (human)0.3433
Histone deacetylase 7Homo sapiens (human)0.6725
Histone deacetylase 2Homo sapiens (human)0.3537
Histone deacetylase 11 Homo sapiens (human)0.6386
Histone deacetylase 8Homo sapiens (human)0.6725
Histone deacetylase 6Homo sapiens (human)0.5717
Histone deacetylase 5Homo sapiens (human)0.6725
Nuclear receptor corepressor 2Homo sapiens (human)0.045

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Erkasap, N; Erkasap, S; Koken, T; Küçük, A; Ozkurt, M; Tosun, M; Yucel, M1
Akbal, C; Cadirci, S; Cevik, O; Erşahin, M; Reiter, RJ; Sener, G; Sener, TE; Tavukçu, HH; Tinay, I1
Abu-Risha, SE; El-Sisi, AE; Ibrahim, HA; Sokar, SS1

Other Studies

3 other study(ies) available for tadalafil and mocetinostat

ArticleYear
The effects of PDE5 inhibitory drugs on renal ischemia/reperfusion injury in rats.
    Molecular biology reports, 2012, Volume: 39, Issue:10

    Topics: Animals; Apoptosis; Carbolines; Gene Expression; Ischemia; Kidney; Male; Malondialdehyde; Nitric Oxide Synthase Type II; Nitric Oxide Synthase Type III; Oxidative Stress; Peroxidase; Phosphodiesterase 5 Inhibitors; Piperazines; Purines; Rats; Rats, Sprague-Dawley; Reperfusion Injury; Sildenafil Citrate; Sulfones; Tadalafil; Tumor Suppressor Protein p53

2012
Melatonin and tadalafil treatment improves erectile dysfunction after spinal cord injury in rats.
    Clinical and experimental pharmacology & physiology, 2014, Volume: 41, Issue:4

    Topics: Animals; Antioxidants; Carbolines; Erectile Dysfunction; Gene Expression Regulation, Enzymologic; Glutathione; Male; Melatonin; Nitric Oxide Synthase Type III; Peroxidase; Rats; Rats, Wistar; Spinal Cord Injuries; Tadalafil; Vasodilator Agents

2014
Combination of tadalafil and diltiazem attenuates renal ischemia reperfusion-induced acute renal failure in rats.
    Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie, 2016, Volume: 84

    Topics: Acute Kidney Injury; Animals; Apoptosis; Blood Urea Nitrogen; Creatinine; Diltiazem; Drug Therapy, Combination; Intercellular Adhesion Molecule-1; Interleukin-1beta; Kidney; Male; Malondialdehyde; Peroxidase; Rats; Reperfusion Injury; Superoxide Dismutase; Tadalafil; Tumor Necrosis Factor-alpha

2016