Page last updated: 2024-09-02

tadalafil and metoclopramide

tadalafil has been researched along with metoclopramide in 2 studies

Compound Research Comparison

Studies
(tadalafil)
Trials
(tadalafil)
Recent Studies (post-2010)
(tadalafil)
Studies
(metoclopramide)
Trials
(metoclopramide)
Recent Studies (post-2010) (metoclopramide)
1,7423921,0895,0441,216623

Protein Interaction Comparison

ProteinTaxonomytadalafil (IC50)metoclopramide (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)2.383
MyeloperoxidaseHomo sapiens (human)0.35
Alpha-2A adrenergic receptorHomo sapiens (human)2.721
Cytochrome P450 2D6Homo sapiens (human)0.8
D(2) dopamine receptorHomo sapiens (human)0.127
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)7.8
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)7.8
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)7.7
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)7.7
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)7.7
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)7.8
5-hydroxytryptamine receptor 2AHomo sapiens (human)3.675
5-hydroxytryptamine receptor 2CHomo sapiens (human)2.383
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)7.8
5-hydroxytryptamine receptor 1DRattus norvegicus (Norway rat)7.8
5-hydroxytryptamine receptor 1FRattus norvegicus (Norway rat)7.8
D(3) dopamine receptorHomo sapiens (human)0.2
5-hydroxytryptamine receptor 3ARattus norvegicus (Norway rat)0.88
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.63
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)7.8
D(2) dopamine receptorRattus norvegicus (Norway rat)0.6237
5-hydroxytryptamine receptor 3BRattus norvegicus (Norway rat)0.88

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1

Reviews

1 review(s) available for tadalafil and metoclopramide

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

1 other study(ies) available for tadalafil and metoclopramide

ArticleYear
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013