Page last updated: 2024-09-02

tadalafil and glyburide

tadalafil has been researched along with glyburide in 4 studies

Compound Research Comparison

Studies
(tadalafil)
Trials
(tadalafil)
Recent Studies (post-2010)
(tadalafil)
Studies
(glyburide)
Trials
(glyburide)
Recent Studies (post-2010) (glyburide)
1,7423921,0896,5546201,344

Protein Interaction Comparison

ProteinTaxonomytadalafil (IC50)glyburide (IC50)
ATP-binding cassette sub-family C member 9Homo sapiens (human)0.22
Bile salt export pumpRattus norvegicus (Norway rat)5.7
Bile salt export pumpHomo sapiens (human)5.5333
Cytochrome P450 2C9 Homo sapiens (human)1.602
ATP-binding cassette sub-family C member 8Homo sapiens (human)0.0043
ATP-sensitive inward rectifier potassium channel 11Homo sapiens (human)0.1121
NACHT, LRR and PYD domains-containing protein 3 Mus musculus (house mouse)10
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)1.8

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (25.00)29.6817
2010's3 (75.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Chan, CL; Dalan, R; Gardner, D; Kao, SL; Lee, KO; Lee, M; Lim, CC; Pratt, E; Tan, B1
Datla, PV; Kodali, B; Pappula, N1

Reviews

1 review(s) available for tadalafil and glyburide

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

3 other study(ies) available for tadalafil and glyburide

ArticleYear
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
An unusual outbreak of hypoglycemia.
    The New England journal of medicine, 2009, Feb-12, Volume: 360, Issue:7

    Topics: Adult; Aged; Aged, 80 and over; Carbolines; Chromatography, High Pressure Liquid; Disease Outbreaks; Drug Contamination; Erectile Dysfunction; Glyburide; Humans; Hypoglycemia; Hypoglycemic Agents; Illicit Drugs; Male; Middle Aged; Phosphodiesterase Inhibitors; Piperazines; Plant Extracts; Purines; Sildenafil Citrate; Singapore; Sulfones; Tadalafil; Young Adult

2009
Selective and rapid determination of tadalafil and finasteride using solid phase extraction by high performance liquid chromatography and tandem mass spectrometry.
    Journal of pharmaceutical and biomedical analysis, 2018, Apr-15, Volume: 152

    Topics: Calibration; Chromatography, High Pressure Liquid; Finasteride; Glyburide; Humans; Reproducibility of Results; Solid Phase Extraction; Tadalafil; Tandem Mass Spectrometry

2018