Page last updated: 2024-09-02

tadalafil and cilostazol

tadalafil has been researched along with cilostazol in 6 studies

Compound Research Comparison

Studies
(tadalafil)
Trials
(tadalafil)
Recent Studies (post-2010)
(tadalafil)
Studies
(cilostazol)
Trials
(cilostazol)
Recent Studies (post-2010) (cilostazol)
1,7423921,0891,508302848

Protein Interaction Comparison

ProteinTaxonomytadalafil (IC50)cilostazol (IC50)
Cytochrome P450 2C9 Homo sapiens (human)10
cGMP-inhibited 3',5'-cyclic phosphodiesterase BHomo sapiens (human)0.4367
cGMP-inhibited 3',5'-cyclic phosphodiesterase AHomo sapiens (human)0.3285

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (50.00)24.3611
2020's3 (50.00)2.80

Authors

AuthorsStudies
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Huang, YY; Li, Z; Luo, HB; Wu, D; Wu, Y1
Chai, S; Chen, S; Deng, L; Du, K; Shen, R; Sun, H; Sun, T; Xi, M; Xie, M1
Albers, HJ; Coenen, DM; Cosemans, JMEM; Hagué, P; Heinzmann, ACA; Koenen, RR; Kuijpers, MJE; Nagy, M; Oggero, S; Perretti, M; van der Meer, AD; Vanderwinden, JM1
Amin, A; Habib, HA; Heeba, GH; Othman, EM; Zahran, ME1

Reviews

3 review(s) available for tadalafil and cilostazol

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Novel Phosphodiesterase Inhibitors for Cognitive Improvement in Alzheimer's Disease.
    Journal of medicinal chemistry, 2018, 07-12, Volume: 61, Issue:13

    Topics: Alzheimer Disease; Animals; Cognition; Humans; Phosphodiesterase Inhibitors

2018
Therapeutic potential of phosphodiesterase inhibitors for cognitive amelioration in Alzheimer's disease.
    European journal of medicinal chemistry, 2022, Mar-15, Volume: 232

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Alzheimer Disease; Animals; Cognition; Cyclic GMP; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases

2022

Other Studies

3 other study(ies) available for tadalafil and cilostazol

ArticleYear
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Inhibition of Phosphodiesterase 3A by Cilostazol Dampens Proinflammatory Platelet Functions.
    Cells, 2021, 08-05, Volume: 10, Issue:8

    Topics: Animals; Anti-Inflammatory Agents; Blood Coagulation; Blood Platelets; Cells, Cultured; Chemokines; Cilostazol; Cyclic Nucleotide Phosphodiesterases, Type 3; Fibrin; Fibrinolytic Agents; Humans; Inflammation Mediators; Mice, Inbred C57BL; Mice, Knockout; Phosphodiesterase 3 Inhibitors; Phosphodiesterase 5 Inhibitors; Platelet Activation; Platelet Adhesiveness; Signal Transduction; Tadalafil

2021
Mechanistic Protective Effect of Cilostazol in Cisplatin-Induced Testicular Damage via Regulation of Oxidative Stress and TNF-α/NF-κB/Caspase-3 Pathways.
    International journal of molecular sciences, 2023, Aug-10, Volume: 24, Issue:16

    Topics: Animals; Caspase 3; Cilostazol; Cisplatin; Inflammation; Male; NF-kappa B; Oxidative Stress; Pentoxifylline; Phosphodiesterase 3 Inhibitors; Rats; Semen; Tadalafil; Tumor Necrosis Factor-alpha

2023