tacrine has been researched along with thiourea in 5 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 5 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Ibrar, A; Khan, I; Saeed, F; Shehzadi, SA | 1 |
Drtinova, L; Gazova, Z; Horova, A; Korabecny, J; Kral, J; Kuca, K; Musilek, K; Siposova, K; Soukup, O; Spilovska, K | 1 |
Böhm, S; Danihel, I; Hamulakova, S; Holas, O; Imrich, J; Janovec, L; Kozurkova, M; Kristian, P; Kuca, K; Pohanka, M | 1 |
Hamulakova, S; Hrabinova, M; Janockova, J; Janovec, L; Jun, D; Kuca, K; Sepsova, V; Soukup, O | 1 |
Babkova, K; Brabec, V; Fedorocko, P; Hamulakova, S; Janockova, J; Jendzelovsky, R; Kasparkova, J; Konkolova, E; Korabecny, J; Koval, J; Kozurkova, M; Kuca, K; Kucerova, D; Plsikova, J; Rosocha, J; Soukup, O; Vargova, J | 1 |
1 review(s) available for tacrine and thiourea
Article | Year |
---|---|
Developing hybrid molecule therapeutics for diverse enzyme inhibitory action: Active role of coumarin-based structural leads in drug discovery.
Topics: Aldehyde Reductase; Alkaline Phosphatase; Cholinesterases; Coumarins; Drug Design; Enzymes; Glucosidases; Humans; Molecular Docking Simulation; Monoamine Oxidase | 2018 |
4 other study(ies) available for tacrine and thiourea
Article | Year |
---|---|
7-Methoxytacrine-adamantylamine heterodimers as cholinesterase inhibitors in Alzheimer's disease treatment--synthesis, biological evaluation and molecular modeling studies.
Topics: Acetylcholinesterase; Alzheimer Disease; Amantadine; Cholinesterase Inhibitors; Dimerization; Enzyme Assays; Humans; Inhibitory Concentration 50; Models, Molecular; Molecular Docking Simulation; Reference Standards; Tacrine; Thiourea | 2013 |
Novel tacrine/acridine anticholinesterase inhibitors with piperazine and thiourea linkers.
Topics: Acetylcholinesterase; Acridines; Butyrylcholinesterase; Cholinesterase Inhibitors; Enzyme Activation; Humans; Models, Molecular; Molecular Conformation; Piperazine; Piperazines; Protein Binding; Tacrine; Thiourea | 2014 |
Tacrine-coumarin and Tacrine-7-chloroquinoline Hybrids with Thiourea Linkers: Cholinesterase Inhibition Properties, Kinetic Study, Molecular Docking and Permeability Assay for Blood-brain Barrier.
Topics: Animals; Blood-Brain Barrier; Cholinesterase Inhibitors; Coumarins; Humans; Kinetics; Models, Molecular; Molecular Docking Simulation; Permeability; Structure-Activity Relationship; Tacrine; Thiourea | 2018 |
In vitro investigating of anticancer activity of new 7-MEOTA-tacrine heterodimers.
Topics: A549 Cells; Acridines; Antineoplastic Agents; Cell Proliferation; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Fibroblasts; HL-60 Cells; Humans; Structure-Activity Relationship; Tacrine; Thiourea | 2019 |