tacrine and thiourea

tacrine has been researched along with thiourea in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's5 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ibrar, A; Khan, I; Saeed, F; Shehzadi, SA1
Drtinova, L; Gazova, Z; Horova, A; Korabecny, J; Kral, J; Kuca, K; Musilek, K; Siposova, K; Soukup, O; Spilovska, K1
Böhm, S; Danihel, I; Hamulakova, S; Holas, O; Imrich, J; Janovec, L; Kozurkova, M; Kristian, P; Kuca, K; Pohanka, M1
Hamulakova, S; Hrabinova, M; Janockova, J; Janovec, L; Jun, D; Kuca, K; Sepsova, V; Soukup, O1
Babkova, K; Brabec, V; Fedorocko, P; Hamulakova, S; Janockova, J; Jendzelovsky, R; Kasparkova, J; Konkolova, E; Korabecny, J; Koval, J; Kozurkova, M; Kuca, K; Kucerova, D; Plsikova, J; Rosocha, J; Soukup, O; Vargova, J1

Reviews

1 review(s) available for tacrine and thiourea

ArticleYear
Developing hybrid molecule therapeutics for diverse enzyme inhibitory action: Active role of coumarin-based structural leads in drug discovery.
    Bioorganic & medicinal chemistry, 2018, 07-30, Volume: 26, Issue:13

    Topics: Aldehyde Reductase; Alkaline Phosphatase; Cholinesterases; Coumarins; Drug Design; Enzymes; Glucosidases; Humans; Molecular Docking Simulation; Monoamine Oxidase

2018

Other Studies

4 other study(ies) available for tacrine and thiourea

ArticleYear
7-Methoxytacrine-adamantylamine heterodimers as cholinesterase inhibitors in Alzheimer's disease treatment--synthesis, biological evaluation and molecular modeling studies.
    Molecules (Basel, Switzerland), 2013, Feb-20, Volume: 18, Issue:2

    Topics: Acetylcholinesterase; Alzheimer Disease; Amantadine; Cholinesterase Inhibitors; Dimerization; Enzyme Assays; Humans; Inhibitory Concentration 50; Models, Molecular; Molecular Docking Simulation; Reference Standards; Tacrine; Thiourea

2013
Novel tacrine/acridine anticholinesterase inhibitors with piperazine and thiourea linkers.
    International journal of biological macromolecules, 2014, Volume: 70

    Topics: Acetylcholinesterase; Acridines; Butyrylcholinesterase; Cholinesterase Inhibitors; Enzyme Activation; Humans; Models, Molecular; Molecular Conformation; Piperazine; Piperazines; Protein Binding; Tacrine; Thiourea

2014
Tacrine-coumarin and Tacrine-7-chloroquinoline Hybrids with Thiourea Linkers: Cholinesterase Inhibition Properties, Kinetic Study, Molecular Docking and Permeability Assay for Blood-brain Barrier.
    Current Alzheimer research, 2018, Volume: 15, Issue:12

    Topics: Animals; Blood-Brain Barrier; Cholinesterase Inhibitors; Coumarins; Humans; Kinetics; Models, Molecular; Molecular Docking Simulation; Permeability; Structure-Activity Relationship; Tacrine; Thiourea

2018
In vitro investigating of anticancer activity of new 7-MEOTA-tacrine heterodimers.
    Journal of enzyme inhibition and medicinal chemistry, 2019, Volume: 34, Issue:1

    Topics: A549 Cells; Acridines; Antineoplastic Agents; Cell Proliferation; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Fibroblasts; HL-60 Cells; Humans; Structure-Activity Relationship; Tacrine; Thiourea

2019