tacrine and pirenzepine

tacrine has been researched along with pirenzepine in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19904 (26.67)18.7374
1990's5 (33.33)18.2507
2000's4 (26.67)29.6817
2010's2 (13.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Ferrendelli, CA; Hanchett, HE; Hollifield, MA; Lorenzi, MV; Potter, LT1
Flynn, DD; Mash, DC1
Cross, AJ; Green, AR; Hunter, AJ; Jones, JA; Murray, TK1
Pearce, BD; Potter, LT1
Mohr, K; Tränkle, C1
Lau, WM; Szilagyi, M1
Nordberg, A; Svensson, AL; Zhang, X1
Brefel-Courbon, C; Freslon, JL; Lazartigues, E; Montastruc, JL; Pelat, M; Rascol, O; Tellioglu, T; Tran, MA1
Carlson, BB; Salamone, JD; Trevitt, JT2
Braida, D; Ottonello, F; Sala, M; Virag, W1
Gong, ZH; Meyerson, B; Nordberg, A; Svensson, AL; Tian, JY; Zhang, X1
Badia, A; Camps, P; Clos, MV; Formosa, X; Galdeano, C; Muñoz-Torrero, D; Pera, M; Ratia, M; Relat, J; Sola, I; Viayna, E1

Other Studies

15 other study(ies) available for tacrine and pirenzepine

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Tetrahydroaminoacridine and other allosteric antagonists of hippocampal M1 muscarine receptors.
    Molecular pharmacology, 1989, Volume: 35, Issue:5

    Topics: Allosteric Regulation; Aminoacridines; Animals; Ethylmaleimide; Guanylyl Imidodiphosphate; Hippocampus; In Vitro Techniques; N-Methylscopolamine; Parasympatholytics; Pirenzepine; Protein Conformation; Rabbits; Receptors, Muscarinic; Scopolamine Derivatives; Solubility; Tacrine

1989
Multiple in vitro interactions with and differential in vivo regulation of muscarinic receptor subtypes by tetrahydroaminoacridine.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:2

    Topics: Allosteric Regulation; Aminoacridines; Animals; Brain; Cholinesterase Inhibitors; Male; Oxotremorine; Pirenzepine; Potassium Channels; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; Tacrine

1989
The cholinergic pharmacology of tetrahydroaminoacridine in vivo and in vitro.
    British journal of pharmacology, 1989, Volume: 98, Issue:1

    Topics: Aminoacridines; Animals; Behavior, Animal; Brain Chemistry; Cholinesterase Inhibitors; Gallamine Triethiodide; In Vitro Techniques; Male; Mice; Myocardium; N-Methylscopolamine; Nicotine; Oxotremorine; Parasympathetic Nervous System; Physostigmine; Pirenzepine; Rats; Receptors, Muscarinic; Scopolamine Derivatives; Tacrine

1989
Effects of tetrahydroaminoacridine on M1 and M2 muscarine receptors.
    Neuroscience letters, 1988, Jun-07, Volume: 88, Issue:3

    Topics: Acetylcholinesterase; Aminoacridines; Animals; Binding, Competitive; Brain Stem; Butyrylcholinesterase; Hippocampus; Pirenzepine; Quinuclidinyl Benzilate; Rabbits; Receptors, Muscarinic; Scopolamine; Tacrine

1988
Allosteric effects of the alkane-bis-ammonium compound W84 and of tacrine on [3H]pirenzepine binding at M1-receptors in rat cerebral cortex.
    Pharmacology & toxicology, 1994, Volume: 75, Issue:6

    Topics: Allosteric Regulation; Animals; Binding, Competitive; Cerebral Cortex; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Isoindoles; Male; Phthalimides; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Cholinergic; Structure-Activity Relationship; Tacrine

1994
Interaction of tacrine at M1 and M2 cholinoceptors in guinea pig brain.
    Pharmacology, 1993, Volume: 47, Issue:4

    Topics: Animals; Binding Sites; Brain; Diamines; Drug Interactions; Female; Guinea Pigs; Parasympatholytics; Pirenzepine; Receptors, Cholinergic; Tacrine

1993
Biphasic effect of tacrine on acetylcholine release in rat brain via M1 and M2 receptors.
    Brain research, 1996, Jul-08, Volume: 726, Issue:1-2

    Topics: Acetylcholine; Alzheimer Disease; Analysis of Variance; Animals; Atropine; Brain; Cholinesterase Inhibitors; Disease Models, Animal; Male; Muscarinic Antagonists; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Synaptosomes; Tacrine

1996
Pressor and bradycardic effects of tacrine and other acetylcholinesterase inhibitors in the rat.
    European journal of pharmacology, 1998, Nov-13, Volume: 361, Issue:1

    Topics: Adrenergic Antagonists; Animals; Antidiuretic Hormone Receptor Antagonists; Atropine; Atropine Derivatives; Blood Pressure; Carbamates; Cardiovascular Agents; Chlorisondamine; Cholinergic Antagonists; Cholinesterase Inhibitors; Diamines; Diastole; Dose-Response Relationship, Drug; Heart Rate; Male; Phenylcarbamates; Physostigmine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Rivastigmine; Systole; Tacrine

1998
Behavioral assessment of atypical antipsychotics in rats: studies of the effects of olanzapine (Zyprexa).
    Psychopharmacology, 1999, Volume: 145, Issue:3

    Topics: Animals; Antipsychotic Agents; Benzodiazepines; Jaw; Male; Movement; Nootropic Agents; Olanzapine; Pirenzepine; Rats; Rats, Sprague-Dawley; Tacrine

1999
Effects of H1 antagonists on cholinomimetic-induced tremulous jaw movements: studies of diphenhydramine, doxepin, and mepyramine.
    Pharmacology, biochemistry, and behavior, 2000, Volume: 65, Issue:4

    Topics: Animals; Antidepressive Agents, Tricyclic; Antipsychotic Agents; Benzodiazepines; Cholinergic Agents; Clozapine; Diphenhydramine; Dose-Response Relationship, Drug; Doxepin; Histamine H1 Antagonists; Jaw; Male; Movement; Olanzapine; Pirenzepine; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Histamine H1; Receptors, Muscarinic; Tacrine; Tremor

2000
Excitatory and inhibitory effects of second-generation cholinesterase inhibitors on rat gastrointestinal transit.
    Pharmacological research, 2000, Volume: 41, Issue:6

    Topics: Administration, Oral; Animals; Cholinesterase Inhibitors; Donepezil; Dose-Response Relationship, Drug; Gastrointestinal Transit; Hydrocarbons, Brominated; Indans; Male; Physostigmine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptor, Muscarinic M1; Receptors, Muscarinic; Receptors, Nicotinic; Scopolamine; Tacrine

2000
Chronic treatments with tacrine and (-)-nicotine induce different changes of nicotinic and muscarinic acetylcholine receptors in the brain of aged rat.
    Journal of neural transmission (Vienna, Austria : 1996), 2002, Volume: 109, Issue:3

    Topics: Aging; Animals; Binding Sites; Brain; Bridged Bicyclo Compounds, Heterocyclic; Drug Administration Schedule; Male; Nicotine; Nicotinic Agonists; Parasympathomimetics; Pirenzepine; Pyridines; Radioligand Assay; Rats; Receptors, Muscarinic; Receptors, Nicotinic; Tacrine; Tritium

2002
Expanding the multipotent profile of huprine-tacrine heterodimers as disease-modifying anti-Alzheimer agents.
    Neuro-degenerative diseases, 2012, Volume: 10, Issue:1-4

    Topics: Aminoquinolines; Analysis of Variance; Animals; Cell Line, Tumor; Cell Survival; Dose-Response Relationship, Drug; Heterocyclic Compounds, 4 or More Rings; Hippocampus; Humans; Hydrogen Peroxide; Muscarinic Antagonists; Neuroblastoma; Oxidative Stress; Pirenzepine; Protein Binding; Protein Multimerization; Quinuclidinyl Benzilate; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship; Tacrine; Tritium

2012