tacrine and neostigmine

tacrine has been researched along with neostigmine in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19901 (7.69)18.7374
1990's5 (38.46)18.2507
2000's2 (15.38)29.6817
2010's5 (38.46)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Ahlin, G; Bergström, F; Bredberg, U; Fridén, M; Hammarlund-Udenaes, M; Rehngren, M; Wan, H1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Ji, J; Peng, Y; Rakesh, KP; Wang, S; Xu, M; Zhu, L1
Henriksson, BG; Järbe, TU; Johansson, JO1
Galli, A; Gori, I; Lucherini, M; Mori, F1
Miyamoto, MD; Provan, SD1
Itoh, Y; Nishibori, M; Oishi, R; Saeki, K1
Arnal, F; Coté, LJ; Ginsburg, S; Lawrence, GD; Naini, A; Sano, M1
Dodds, HM; Rivory, LP1
Kaur, J; Zhang, MQ1
Ben-Hur, T; Ben-Menachem, O; Gilboa, A; Pollak, Y; Soreq, H; Yirmiya, R1

Reviews

2 review(s) available for tacrine and neostigmine

ArticleYear
Triazole derivatives as inhibitors of Alzheimer's disease: Current developments and structure-activity relationships.
    European journal of medicinal chemistry, 2019, Oct-15, Volume: 180

    Topics: Acetylcholinesterase; Alzheimer Disease; Butyrylcholinesterase; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Humans; Molecular Structure; Neuroprotective Agents; Structure-Activity Relationship; Triazoles

2019
Molecular modelling and QSAR of reversible acetylcholines-terase inhibitors.
    Current medicinal chemistry, 2000, Volume: 7, Issue:3

    Topics: Alkaloids; Alzheimer Disease; Cholinesterase Inhibitors; Crystallography, X-Ray; Donepezil; Drug Design; Glaucoma; Humans; Indans; Models, Molecular; Myasthenia Gravis; Neostigmine; Physostigmine; Piperidines; Sesquiterpenes; Structure-Activity Relationship; Surface Properties; Tacrine

2000

Other Studies

11 other study(ies) available for tacrine and neostigmine

ArticleYear
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Measurement of unbound drug exposure in brain: modeling of pH partitioning explains diverging results between the brain slice and brain homogenate methods.
    Drug metabolism and disposition: the biological fate of chemicals, 2011, Volume: 39, Issue:3

    Topics: Animals; Biological Transport; Brain; Chemical Phenomena; Dialysis; Hydrogen-Ion Concentration; In Vitro Techniques; Lysosomes; Male; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Tissue Distribution

2011
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Drug discrimination in rats: the effects of phencyclidine and ditran.
    Psychopharmacologia, 1975, Apr-30, Volume: 42, Issue:1

    Topics: Animals; Cues; Cyclohexylamines; Discrimination Learning; Drug Combinations; Fenclonine; Glycolates; Imipramine; Ketamine; Male; Neostigmine; Phencyclidine; Physostigmine; Piperidines; Pyrrolidines; Rats; Tacrine; Tetrabenazine; Yohimbine

1975
In vitro protection of acetylcholinesterase and butyrylcholinesterase by tetrahydroaminoacridine. Comparison with physostigmine.
    Biochemical pharmacology, 1992, Jun-09, Volume: 43, Issue:11

    Topics: Acetylcholinesterase; Binding Sites; Butyrylcholinesterase; Cholinesterase Reactivators; Dose-Response Relationship, Drug; Isoflurophate; Neostigmine; Organophosphorus Compounds; Physostigmine; Tacrine

1992
Tetrahydroaminoacridine and physostigmine have opposing effects on probability of transmitter release at the frog neuromuscular junction.
    Neuroscience letters, 1991, Feb-11, Volume: 123, Issue:1

    Topics: Animals; Evoked Potentials; In Vitro Techniques; Kinetics; Motor Endplate; Neostigmine; Neurotransmitter Agents; Physostigmine; Potassium; Rana pipiens; Skin; Tacrine

1991
9-Amino-1,2,3,4-tetrahydroacridine is a potent inhibitor of histamine N-methyltransferase.
    Japanese journal of pharmacology, 1991, Volume: 55, Issue:4

    Topics: Animals; Brain; Cattle; Histamine; Histamine N-Methyltransferase; In Vitro Techniques; Male; Methylhistamines; Mice; Mice, Inbred Strains; Neostigmine; Physostigmine; Tacrine

1991
Studies on new, centrally active and reversible acetylcholinesterase inhibitors.
    Neurochemical research, 1990, Volume: 15, Issue:6

    Topics: Acetylcholinesterase; Animals; Blood-Brain Barrier; Brain; Cholinesterase Inhibitors; Dopamine; Male; Mice; Neostigmine; Norepinephrine; Pyridostigmine Bromide; Tacrine

1990
The mechanism for the inhibition of acetylcholinesterases by irinotecan (CPT-11).
    Molecular pharmacology, 1999, Volume: 56, Issue:6

    Topics: Acetylcholinesterase; Acylation; Alzheimer Disease; Binding, Competitive; Butyrylcholinesterase; Camptothecin; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Erythrocytes; Humans; Hydrolysis; Irinotecan; Kinetics; Neostigmine; Propidium; Substrate Specificity; Tacrine

1999
Acetylcholinesterase inhibitors reduce brain and blood interleukin-1beta production.
    Annals of neurology, 2005, Volume: 57, Issue:5

    Topics: Animals; Brain Chemistry; Cholinesterase Inhibitors; Hippocampus; Interleukin-1; Lipopolysaccharides; Male; Mice; Mice, Inbred C57BL; Neostigmine; Oligodeoxyribonucleotides; Oligonucleotides; Oligonucleotides, Antisense; Phenylcarbamates; Rivastigmine; Tacrine

2005