tacrine and memoquin

tacrine has been researched along with memoquin in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (42.86)29.6817
2010's4 (57.14)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andrisano, V; Banzi, R; Bartolini, M; Bergamini, C; Bolognesi, ML; Cattaneo, A; Cavalli, A; Fato, R; Hrelia, P; Lenaz, G; Melchiorre, C; Minarini, A; Recanatini, M; Rosini, M; Tarozzi, A; Tumiatti, V1
Bolognesi, ML; Cavalli, A; Melchiorre, C; Minarini, A; Recanatini, M; Rosini, M; Tumiatti, V1
Andrisano, V; Bartolini, M; Bolognesi, ML; De Simone, A; Pinto, A; Prati, F; Simoni, E1
Andrisano, V; Bartolini, M; Bergamini, C; Bolognesi, ML; Fato, R; Garcia, GE; Korabecny, J; Kuca, K; Lamba, D; Monti, B; Nepovimova, E; Peña-Altamira, LE; Pesaresi, A; Roberti, M; Samez, S; Uliassi, E1
Andrisano, V; Bartolini, M; Chen, L; De Simone, A; Egea, J; Kang, D; Lamba, D; Lopez, MG; Lou, Y; Pesaresi, A; Samez, S; Stojan, J; Xu, C; Xu, Y; Zha, X; Zhang, L1
Andrisano, V; Bartolini, M; Bolognesi, ML; Melchiorre, C; Minarini, A; Rosini, M; Tumiatti, V1
Bolognesi, ML; Melchiorre, C; Minarini, A; Rosini, M; Simoni, E; Tumiatti, V1

Reviews

3 review(s) available for tacrine and memoquin

ArticleYear
Multi-target-directed ligands to combat neurodegenerative diseases.
    Journal of medicinal chemistry, 2008, Feb-14, Volume: 51, Issue:3

    Topics: Acetylcholinesterase; Alzheimer Disease; Amyloid beta-Peptides; Antioxidants; Binding Sites; Calcium Channel Blockers; Chelating Agents; Cholinesterase Inhibitors; Humans; Huntington Disease; Ligands; Multiple Sclerosis; Neurodegenerative Diseases; Neurofibrillary Tangles; Neurotransmitter Agents; Parkinson Disease; Plaque, Amyloid

2008
MTDL design strategy in the context of Alzheimer's disease: from lipocrine to memoquin and beyond.
    Current pharmaceutical design, 2009, Volume: 15, Issue:6

    Topics: Alkanes; Alzheimer Disease; Animals; Carbazoles; Cholinesterase Inhibitors; Drug Delivery Systems; Drug Design; Ethylamines; Humans; Ligands; Tacrine; Thioctic Acid

2009
Multitarget-directed ligands: innovative chemical probes and therapeutic tools against Alzheimer's disease.
    Current topics in medicinal chemistry, 2011, Volume: 11, Issue:22

    Topics: Acetylcholinesterase; Alkanes; Alzheimer Disease; Amyloid beta-Peptides; Animals; Enzyme Inhibitors; Ethylamines; Humans; Ligands; Tacrine; Thioctic Acid

2011

Other Studies

4 other study(ies) available for tacrine and memoquin

ArticleYear
Novel class of quinone-bearing polyamines as multi-target-directed ligands to combat Alzheimer's disease.
    Journal of medicinal chemistry, 2007, Oct-04, Volume: 50, Issue:20

    Topics: Acetylcholinesterase; Alzheimer Disease; Amyloid beta-Peptides; Antioxidants; Binding Sites; Butyrylcholinesterase; Cell Line; Cholinesterase Inhibitors; Humans; Ligands; Models, Molecular; NAD(P)H Dehydrogenase (Quinone); Oxidative Stress; Polyamines; Protein Binding; Quinones; Reactive Oxygen Species; Structure-Activity Relationship; Substrate Specificity

2007
Quinones bearing non-steroidal anti-inflammatory fragments as multitarget ligands for Alzheimer's disease.
    Bioorganic & medicinal chemistry letters, 2013, Dec-01, Volume: 23, Issue:23

    Topics: Alzheimer Disease; Amyloid; Animals; Anti-Inflammatory Agents, Non-Steroidal; Cholinesterase Inhibitors; Humans; Ligands; Mice; Models, Molecular; Protein Binding; Quinones; Structure-Activity Relationship

2013
Multitarget drug design strategy: quinone-tacrine hybrids designed to block amyloid-β aggregation and to exert anticholinesterase and antioxidant effects.
    Journal of medicinal chemistry, 2014, Oct-23, Volume: 57, Issue:20

    Topics: Acetylcholinesterase; Amyloid beta-Peptides; Animals; Antioxidants; Blood-Brain Barrier; Chemistry Techniques, Synthetic; Cholinesterase Inhibitors; Crystallography, X-Ray; Drug Design; Drug Evaluation, Preclinical; Hep G2 Cells; Humans; Inhibitory Concentration 50; Models, Molecular; Molecular Targeted Therapy; Neurons; Oxidative Stress; Quinones; Rats, Wistar; Tacrine

2014
Novel Tacrine-Benzofuran Hybrids as Potent Multitarget-Directed Ligands for the Treatment of Alzheimer's Disease: Design, Synthesis, Biological Evaluation, and X-ray Crystallography.
    Journal of medicinal chemistry, 2016, Jan-14, Volume: 59, Issue:1

    Topics: Alzheimer Disease; Amyloid Precursor Protein Secretases; Animals; Aspartic Acid Endopeptidases; Behavior, Animal; Benzofurans; Cell Line; Cell Survival; Chemical and Drug Induced Liver Injury; Cholinesterase Inhibitors; Crystallography, X-Ray; Drug Design; Humans; Male; Mice; Mice, Inbred ICR; Models, Molecular; Nootropic Agents; Structure-Activity Relationship; Tacrine; Torpedo

2016